Page last updated: 2024-08-26

u 73122 and guanosine 5'-o-(3-thiotriphosphate)

u 73122 has been researched along with guanosine 5'-o-(3-thiotriphosphate) in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's13 (54.17)18.2507
2000's9 (37.50)29.6817
2010's2 (8.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hahner, L; Harris, RA; McQuilkin, S1
Eusebi, F; Giovannelli, A; Grassi, F; Limatola, C; Mattei, E; Ragozzino, D1
Hicks, JL; Salter, MW1
Barritt, GJ; Berven, LA1
Helliwell, RM; Large, WA1
Geurts, M; Hermans, E; Maloteaux, JM1
Abdel-Latif, AA; Akhtar, RA; Ding, KH; Husain, S; Isales, CM1
Lee, SJ; Shen, SS1
Fayos, BE; Wattenberg, BW1
Bhullar, RP; Fleming, N; Li, L; Mellow, L1
Bell, MI; Lee, K; Richardson, PJ1
Bispham, JR; Hill, SJ; Walker, EM1
Dumont, M; Lemaire, S1
Gudermann, T; Hofmann, T; Obukhov, AG; Plant, TD; Schaefer, M; Schultz, G1
Gailly, P; Hermans, E; Najimi, M1
Behar, J; Biancani, P; Cao, W; Chen, Q; Harnett, KM; Kim, N; Kirber, MT; Sohn, UD1
Bernardi, G; Caputi, L; Guatteo, E; Mercuri, NB; Tozzi, A1
Akaike, A; Kaneko, S; Kanki, H; Kinoshita, M; Mori, Y; Satoh, M1
Cho, H; Earm, YE; Ho, WK; Ryu, SY; Youm, JB1
Gloyna, W; Schmitz, F; Seebeck, J1
Alzheimer, C; Huth, T; Klose, A; Sickmann, T1
Balasubramaniam, A; Park, EA; Parker, MS; Parker, SL; Sah, R; Sallee, FR; Sweatman, T1
Fine, M; Hilgemann, DW; Lariccia, V; Lin, MJ; Llaguno, MC; Magi, S; Yaradanakul, A1
Kyozuka, K; Nakano, T1

Other Studies

24 other study(ies) available for u 73122 and guanosine 5'-o-(3-thiotriphosphate)

ArticleYear
Cerebellar GABAB receptors modulate function of GABAA receptors.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 1991, Volume: 5, Issue:10

    Topics: Animals; Baclofen; Barium; Calcium; Cells, Cultured; Cerebellum; Cerebral Cortex; Chlorine; Dose-Response Relationship, Drug; Estrenes; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Mice; Mice, Inbred ICR; Muscimol; Pyrrolidinones; Receptors, GABA-A; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors; Type C Phospholipases

1991
Acetylcholine-activated inward current induces cytosolic Ca2+ mobilization in mouse C2C12 myotubes.
    Cell calcium, 1995, Volume: 18, Issue:1

    Topics: Acetylcholine; Animals; Calcium; Cell Line; Culture Media; Cytosol; Electrophysiology; Estrenes; Guanosine 5'-O-(3-Thiotriphosphate); Heparin; Inositol 1,4,5-Trisphosphate; Ion Transport; Kinetics; Membrane Potentials; Mice; Muscles; Permeability; Pyrrolidinones

1995
ATP causes release of intracellular Ca2+ via the phospholipase C beta/IP3 pathway in astrocytes from the dorsal spinal cord.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1995, Volume: 15, Issue:4

    Topics: Adenosine Triphosphate; Aluminum Compounds; Animals; Astrocytes; Calcium; Calcium Channel Blockers; Calcium Channels; Calcium-Transporting ATPases; Cells, Cultured; Egtazic Acid; Estrenes; Fetus; Fluorides; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Heparin; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Isoenzymes; Patch-Clamp Techniques; Pyrrolidinones; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Signal Transduction; Spinal Cord; Terpenes; Thapsigargin; Thionucleotides; Time Factors; Type C Phospholipases

1995
Evidence obtained using single hepatocytes for inhibition by the phospholipase C inhibitor U73122 of store-operated Ca2+ inflow.
    Biochemical pharmacology, 1995, May-17, Volume: 49, Issue:10

    Topics: Binding Sites; Calcium; Calcium Channels; Estrenes; Fura-2; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Inositol Phosphates; Liver; Photolysis; Pyrrolidinones; Type C Phospholipases

1995
Alpha 1-adrenoceptor activation of a non-selective cation current in rabbit portal vein by 1,2-diacyl-sn-glycerol.
    The Journal of physiology, 1997, Mar-01, Volume: 499 ( Pt 2)

    Topics: Alkaloids; Animals; Benzophenanthridines; Carcinogens; Cyclohexanones; Diglycerides; Enzyme Inhibitors; Estrenes; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Inositol 1,4,5-Trisphosphate; Lipoprotein Lipase; Norepinephrine; Phenanthridines; Phorbol 12,13-Dibutyrate; Phosphodiesterase Inhibitors; Portal Vein; Pyrrolidinones; Rabbits; Receptors, Adrenergic, alpha-1; Thionucleotides; Type C Phospholipases

1997
Agonist and antagonist modulation of [35S]-GTP gamma S binding in transfected CHO cells expressing the neurotensin receptor.
    British journal of pharmacology, 1997, Volume: 121, Issue:8

    Topics: Animals; CHO Cells; Cricetinae; Estrenes; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Neurotensin; Pyrrolidinones; Rats; Receptors, Neurotensin; Sodium Chloride; Transfection

1997
Inhibition of muscarinic-stimulated polyphosphoinositide hydrolysis and Ca2+ mobilization in cat iris sphincter smooth muscle cells by cAMP-elevating agents.
    Cellular signalling, 1997, Volume: 9, Issue:6

    Topics: Adrenergic beta-Agonists; Animals; Calcium; Carbachol; Cats; Cell Fractionation; Cell Membrane; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; Guanosine 5'-O-(3-Thiotriphosphate); Hydrolysis; Inositol 1,4,5-Trisphosphate; Iris; Isoproterenol; Kinetics; Muscarinic Agonists; Muscarinic Antagonists; Muscle, Smooth; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Phosphates; Phosphodiesterase Inhibitors; Phosphorylation; Pyrrolidinones; Ryanodine; Thapsigargin; Type C Phospholipases

1997
The calcium transient in sea urchin eggs during fertilization requires the production of inositol 1,4,5-trisphosphate.
    Developmental biology, 1998, Jan-15, Volume: 193, Issue:2

    Topics: Animals; Calcium; Cytoplasm; Estrenes; Female; Fertilization; Guanosine 5'-O-(3-Thiotriphosphate); Hydrogen-Ion Concentration; Inositol 1,4,5-Trisphosphate; Male; Ovum; Pyrrolidinones; Sea Urchins; Sperm-Ovum Interactions; Spermatozoa

1998
Regulated exocytosis in vascular endothelial cells can be triggered by intracellular guanine nucleotides and requires a hydrophobic, thiol-sensitive component. Studies of regulated von Willebrand factor secretion from digitonin permeabilized endothelial c
    Endothelium : journal of endothelial cell research, 1997, Volume: 5, Issue:4

    Topics: Alkylating Agents; Animals; Calcium; Cell Membrane Permeability; Cells, Cultured; CHO Cells; Cricetinae; Cricetulus; Cytosol; Digitonin; Dithiothreitol; Endothelium, Vascular; Estrenes; Exocytosis; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Intracellular Fluid; Pyrrolidinones; Secretory Rate; Signal Transduction; Sulfhydryl Compounds; Umbilical Veins; von Willebrand Factor

1997
Activation of phospholipase D by ADP-ribosylation factor in rat submandibular acinar cells.
    Archives of oral biology, 1998, Volume: 43, Issue:3

    Topics: Animals; Anti-Bacterial Agents; Arachidonic Acids; Brefeldin A; Carbachol; Carrier Proteins; Cyclopentanes; Cytosol; Diglycerides; Dose-Response Relationship, Drug; Enzyme Activation; Estrenes; GTP-Binding Proteins; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Hydrolysis; Macrolides; Male; Membrane Lipids; Phosphatidic Acids; Phosphatidylcholines; Phosphodiesterase Inhibitors; Phospholipase D; Poly(ADP-ribose) Polymerases; Protein Synthesis Inhibitors; Pyrrolidinones; ras Proteins; Rats; Rats, Sprague-Dawley; Signal Transduction; Submandibular Gland; Time Factors; Type C Phospholipases

1998
Characterization of the mechanism of action of tachykinins in rat striatal cholinergic interneurons.
    Neuroscience, 1998, Volume: 87, Issue:3

    Topics: 2-Amino-5-phosphonovalerate; Acetylcholine; Animals; Chelating Agents; Corpus Striatum; Diazonium Compounds; Electric Stimulation; Estrenes; Excitatory Amino Acid Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Interneurons; Male; Membrane Potentials; Patch-Clamp Techniques; Phenoxyacetates; Phosphodiesterase Inhibitors; Photochemistry; Piperidines; Pyrrolidinones; Quinoxalines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-1; Substance P; Synaptic Transmission; Tachykinins; Tetrodotoxin

1998
Nonselective effects of the putative phospholipase C inhibitor, U73122, on adenosine A1 receptor-mediated signal transduction events in Chinese hamster ovary cells.
    Biochemical pharmacology, 1998, Dec-01, Volume: 56, Issue:11

    Topics: Animals; Cell Survival; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Estrenes; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Inositol Phosphates; Kinetics; Phosphatidylinositols; Pyrrolidinones; Receptors, Purinergic P1; Recombinant Proteins; Signal Transduction; Transfection; Type C Phospholipases; Xanthines

1998
Characterization of the high affinity [3H]nociceptin binding site in membrane preparations of rat heart: correlations with the non-opioid dynorphin binding site.
    Journal of molecular and cellular cardiology, 1998, Volume: 30, Issue:12

    Topics: Animals; Binding Sites; Dose-Response Relationship, Drug; Dynorphins; Estrenes; Guanosine 5'-O-(3-Thiotriphosphate); Guanylyl Imidodiphosphate; Heart; Hypertension; Male; Myocardium; Neomycin; Nociceptin; Opioid Peptides; Pyrrolidinones; Rats; Rats, Inbred SHR; Reverse Transcriptase Polymerase Chain Reaction; Synaptosomes; Time Factors

1998
Receptor-mediated regulation of the nonselective cation channels TRPC4 and TRPC5.
    The Journal of biological chemistry, 2000, Jun-09, Volume: 275, Issue:23

    Topics: Animals; Brain; Calcium Channels; Calcium Signaling; Cation Transport Proteins; Cell Line; Estrenes; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Ion Channels; Kidney; Manganese; Mice; Phosphodiesterase Inhibitors; Pyrrolidinones; Receptor Protein-Tyrosine Kinases; Receptors, Cell Surface; Recombinant Proteins; Thapsigargin; Transfection; TRPC Cation Channels

2000
Evidence for the dual coupling of the rat neurotensin receptor with pertussis toxin-sensitive and insensitive G-proteins.
    FEBS letters, 2000, Oct-20, Volume: 483, Issue:2-3

    Topics: Animals; Binding, Competitive; Calcium; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Estrenes; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Inositol Phosphates; Neurotensin; Pertussis Toxin; Phosphodiesterase Inhibitors; Protein Binding; Pyrrolidinones; Rats; Receptors, Neurotensin; Tritium; Virulence Factors, Bordetella

2000
Ca2+-induced contraction of cat esophageal circular smooth muscle cells.
    American journal of physiology. Cell physiology, 2001, Volume: 280, Issue:4

    Topics: Adrenergic beta-Antagonists; Alkaloids; Animals; Antibodies; Azepines; Benzophenanthridines; Bridged-Ring Compounds; Calcium; Calcium Signaling; Cats; Dose-Response Relationship, Drug; Enzyme Inhibitors; Esophagus; Estrenes; Female; Guanosine 5'-O-(3-Thiotriphosphate); Isoenzymes; Male; Muscle Contraction; Muscle, Smooth; Myosin Light Chains; Naphthalenes; Norbornanes; Phenanthridines; Phosphodiesterase Inhibitors; Phospholipase D; Phosphorylation; Propranolol; Protein Kinase C; Protein Kinase C-epsilon; Pyrrolidinones; Quercetin; Second Messenger Systems; Thiocarbamates; Thiones; Type C Phospholipases

2001
Group I mGluRs coupled to G proteins are regulated by tyrosine kinase in dopamine neurons of the rat midbrain.
    Journal of neurophysiology, 2001, Volume: 85, Issue:6

    Topics: Animals; Dopamine; Enzyme Activation; Enzyme Inhibitors; Estrenes; Excitatory Amino Acid Antagonists; Female; Genistein; Glycine; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Diphosphate; Male; Membrane Potentials; Mesencephalon; Neurons; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Protein Kinase C; Protein-Tyrosine Kinases; Pyrrolidinones; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Resorcinols; Thionucleotides; Type C Phospholipases; Tyrphostins

2001
Activation of inositol 1,4,5-trisphosphate receptor is essential for the opening of mouse TRP5 channels.
    Molecular pharmacology, 2001, Volume: 60, Issue:5

    Topics: Acetylcholine; Adenosine; Allosteric Regulation; Animals; Calcium; Calcium Channel Agonists; Calcium Channels; Cation Transport Proteins; Electrophysiology; Estrenes; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Heterotrimeric GTP-Binding Proteins; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Macrocyclic Compounds; Mice; Nuclear Proteins; Oligodeoxyribonucleotides, Antisense; Oocytes; Oxazoles; Peptides; Phosphodiesterase Inhibitors; Protein Serine-Threonine Kinases; Pyrrolidinones; Receptor, Muscarinic M1; Receptors, Cytoplasmic and Nuclear; Receptors, Muscarinic; TRPC Cation Channels; Type C Phospholipases; Xenopus laevis

2001
Inhibition of acetylcholine-activated K(+) currents by U73122 is mediated by the inhibition of PIP(2)-channel interaction.
    British journal of pharmacology, 2001, Volume: 134, Issue:5

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Atrial Function; Dose-Response Relationship, Drug; Estrenes; Guanosine 5'-O-(3-Thiotriphosphate); Heart Atria; Membrane Potentials; Mice; Patch-Clamp Techniques; Phosphatidylinositol 4,5-Diphosphate; Phosphodiesterase Inhibitors; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Binding; Pyrrolidinones; Sodium

2001
Inhibition of phospholipase C-independent exocytotic responses in rat peritoneal mast cells by U73122.
    Regulatory peptides, 2005, Feb-15, Volume: 125, Issue:1-3

    Topics: Animals; Bacterial Proteins; Calcium; Cells, Cultured; Dose-Response Relationship, Drug; Estrenes; Exocytosis; Female; Guanosine 5'-O-(3-Thiotriphosphate); Inhibitory Concentration 50; Intercellular Signaling Peptides and Proteins; Male; Mast Cells; Peptides; Peritoneum; Phosphatidylinositol Diacylglycerol-Lyase; Phosphoinositide Phospholipase C; Platelet Aggregation Inhibitors; Protein Kinase Inhibitors; Pyrrolidinones; Rats; Rats, Wistar; Signal Transduction; Streptolysins; Time Factors; Type C Phospholipases; Wasp Venoms

2005
Unexpected suppression of neuronal G protein-activated, inwardly rectifying K+ current by common phospholipase C inhibitor.
    Neuroscience letters, 2008, May-09, Volume: 436, Issue:2

    Topics: Adenosine; Analgesics; Analysis of Variance; Animals; Animals, Newborn; Baclofen; Cells, Cultured; Dose-Response Relationship, Drug; Drug Interactions; Estrenes; G Protein-Coupled Inwardly-Rectifying Potassium Channels; GABA Agonists; Guanosine 5'-O-(3-Thiotriphosphate); Membrane Potentials; Neural Inhibition; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Pyramidal Cells; Pyrrolidinones; Rats; Somatosensory Cortex

2008
Dimers of the neuropeptide Y (NPY) Y2 receptor show asymmetry in agonist affinity and association with G proteins.
    Journal of receptor and signal transduction research, 2008, Volume: 28, Issue:5

    Topics: Animals; CHO Cells; Cricetinae; Cricetulus; Estrenes; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Mice; Phosphodiesterase Inhibitors; Protein Multimerization; Pyrrolidinones; Rabbits; Receptors, Neuropeptide Y

2008
Massive calcium-activated endocytosis without involvement of classical endocytic proteins.
    The Journal of general physiology, 2011, Volume: 137, Issue:1

    Topics: Actin Cytoskeleton; Adenosine Triphosphate; Animals; beta-Cyclodextrins; Calcineurin; Calcium; Cell Membrane; Cells, Cultured; Ceramides; Cholesterol; Clathrin; Cricetinae; Dynamins; Electric Capacitance; Endocytosis; Estrenes; Exocytosis; Guanosine 5'-O-(3-Thiotriphosphate); HEK293 Cells; Humans; Inositol Polyphosphate 5-Phosphatases; Kidney; Lipids; Membrane Proteins; Naphthalenes; Phosphoric Monoester Hydrolases; Polyamines; Pyridinium Compounds; Pyrones; Pyrrolidinones; Quaternary Ammonium Compounds; Sodium-Calcium Exchanger; Sphingomyelin Phosphodiesterase

2011
Soluble sperm extract specifically recapitulates the initial phase of the Ca2+ response in the fertilized oocyte of P. occelata following a G-protein/ PLCĪ² signaling pathway.
    Zygote (Cambridge, England), 2015, Volume: 23, Issue:6

    Topics: Animals; Calcium; Cell Extracts; Embryo, Nonmammalian; Estrenes; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Male; Microinjections; Oocytes; Polychaeta; Pyrrolidinones; Signal Transduction; Solubility; Sperm-Ovum Interactions; Spermatozoa; Type C Phospholipases; Zygote

2015