Page last updated: 2024-08-26

u 69593 and quinpirole

u 69593 has been researched along with quinpirole in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (10.00)18.2507
2000's7 (70.00)29.6817
2010's2 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Berzetei-Gurske, IP; Guerrieri, E; Schmidhammer, H; Spetea, M1
Acri, JB; Izenwasser, S; Kunko, PM; Shippenberg, T1
Acri, JB; Shippenberg, T; Thompson, AC1
Butelman, ER; Kreek, MJ1
Bisnaire, L; Graham, D; Hayton, S; Perreault, ML; Simms, J; Szechtman, H1
Foster, JA; Graham, D; Perreault, ML; Scattolon, S; Szechtman, H; Wang, Y1
Perreault, ML; Seeman, P; Szechtman, H1
Fields, HL; Hjelmstad, GO; Ishikawa, J; Margolis, EB; Mitchell, JM1
Beerepoot, P; Lam, V; Luu, A; Siebert, D; Szechtman, H; Tsoi, B1
Andrés, ME; Escobar, AP; España, RA; Fuentealba, JA; González, MP; Gysling, K; Henny, P; Meza, RC; Noches, V1

Other Studies

10 other study(ies) available for u 69593 and quinpirole

ArticleYear
Discovery and pharmacological evaluation of a diphenethylamine derivative (HS665), a highly potent and selective κ opioid receptor agonist.
    Journal of medicinal chemistry, 2012, Nov-26, Volume: 55, Issue:22

    Topics: Acetic Acid; Analgesics; Animals; Drug Discovery; Mice; Nociception; Pain; Phenethylamines; Receptors, Opioid, kappa

2012
Repeated treatment with the selective kappa opioid agonist U-69593 produces a marked depletion of dopamine D2 receptors.
    Synapse (New York, N.Y.), 1998, Volume: 30, Issue:3

    Topics: Animals; Benzazepines; Benzeneacetamides; Carrier Proteins; Caudate Nucleus; Dopamine Plasma Membrane Transport Proteins; Down-Regulation; Drug Administration Schedule; Male; Membrane Glycoproteins; Membrane Transport Proteins; Motor Activity; Nerve Tissue Proteins; Nucleus Accumbens; Putamen; Pyrrolidines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Opioid, kappa; Sulpiride; Synapses; Time Factors

1998
Modulation of pre- and postsynaptic dopamine D2 receptor function by the selective kappa-opioid receptor agonist U69593.
    Synapse (New York, N.Y.), 2001, Mar-15, Volume: 39, Issue:4

    Topics: Animals; Autoreceptors; Benzeneacetamides; Dopamine; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Down-Regulation; Male; Microdialysis; Motor Activity; Neostriatum; Pyrrolidines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Synaptic Transmission

2001
kappa-Opioid receptor agonist-induced prolactin release in primates is blocked by dopamine D(2)-like receptor agonists.
    European journal of pharmacology, 2001, Jul-06, Volume: 423, Issue:2-3

    Topics: Animals; Behavior, Animal; Benzazepines; Benzeneacetamides; Conscious Sedation; Dopamine Agonists; Dose-Response Relationship, Drug; Female; Macaca mulatta; Male; Prolactin; Pyrrolidines; Quinpirole; Receptors, Dopamine D2; Receptors, Opioid, kappa; Tetrahydronaphthalenes

2001
Kappa-opioid agonist U69593 potentiates locomotor sensitization to the D2/D3 agonist quinpirole: pre- and postsynaptic mechanisms.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2006, Volume: 31, Issue:9

    Topics: Algorithms; Analgesics; Animals; Benzeneacetamides; Data Interpretation, Statistical; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Synergism; Male; Motor Activity; Pyrrolidines; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Opioid, kappa; Receptors, Presynaptic; Synapses

2006
Cotreatment with the kappa opioid agonist U69593 enhances locomotor sensitization to the D2/D3 dopamine agonist quinpirole and alters dopamine D2 receptor and prodynorphin mRNA expression in rats.
    Psychopharmacology, 2007, Volume: 194, Issue:4

    Topics: Analgesics; Analysis of Variance; Animals; Autoradiography; Basal Ganglia; Benzeneacetamides; Dopamine Agonists; Dopamine Antagonists; Drug Synergism; Enkephalins; Gene Expression; In Situ Hybridization; Injections; Male; Motor Activity; Protein Precursors; Pyrrolidines; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Opioid, kappa; RNA, Messenger; Sulfur Isotopes; Time Factors

2007
Kappa-opioid receptor stimulation quickens pathogenesis of compulsive checking in the quinpirole sensitization model of obsessive-compulsive disorder (OCD).
    Behavioral neuroscience, 2007, Volume: 121, Issue:5

    Topics: Algorithms; Animals; Benzazepines; Benzeneacetamides; Domperidone; Dopamine Agonists; Dopamine Antagonists; Hyperkinesis; Kinetics; Ligands; Male; Motor Activity; Obsessive-Compulsive Disorder; Pyrrolidines; Quinpirole; Raclopride; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Opioid, kappa; Stereotyped Behavior

2007
Midbrain dopamine neurons: projection target determines action potential duration and dopamine D(2) receptor inhibition.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2008, Sep-03, Volume: 28, Issue:36

    Topics: Action Potentials; Amygdala; Analgesics; Animals; Animals, Newborn; Benzeneacetamides; Dopamine; Dopamine Agonists; Dopamine Antagonists; In Vitro Techniques; Lysine; Male; Neural Inhibition; Neural Pathways; Neurons; Patch-Clamp Techniques; Pyrrolidines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Tyrosine 3-Monooxygenase; Ventral Tegmental Area

2008
Effects of salvinorin A on locomotor sensitization to D2/D3 dopamine agonist quinpirole.
    Neuroscience letters, 2008, Dec-03, Volume: 446, Issue:2-3

    Topics: Analgesics; Animals; Benzeneacetamides; Central Nervous System; Diterpenes, Clerodane; Dopamine; Dopamine Agents; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Drug Resistance; Drug Synergism; Male; Motor Activity; Pyrrolidines; Quinpirole; Rats; Rats, Long-Evans; Receptors, Dopamine D2; Receptors, Dopamine D3; Receptors, Opioid, kappa; Synaptic Transmission

2008
Mechanisms of Kappa Opioid Receptor Potentiation of Dopamine D2 Receptor Function in Quinpirole-Induced Locomotor Sensitization in Rats.
    The international journal of neuropsychopharmacology, 2017, 08-01, Volume: 20, Issue:8

    Topics: Analgesics, Opioid; Animals; Benzeneacetamides; Dopamine; Dopamine Agonists; Extracellular Space; Male; Mice, Inbred C57BL; Motor Activity; Neural Inhibition; Neurons; Nucleus Accumbens; Pyrrolidines; Quinpirole; Rats, Sprague-Dawley; Receptors, Dopamine D2; Receptors, Opioid, kappa; Synapses; Synaptosomes; Tissue Culture Techniques

2017