u 69593 has been researched along with mr 2266 in 9 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 5 (55.56) | 18.7374 |
1990's | 4 (44.44) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bansinath, M; Ramabadran, K; Shukla, VK; Turndorf, H | 1 |
Caliezi, A; Drack, E; Halter, F; Scheurer, U; Varga, L; Wenger, F | 1 |
Frey, HH | 1 |
Kamei, H; Kameyama, T; Nabeshima, T | 1 |
Bansinath, M; Puig, MM; Ramabadran, K; Turndorf, H | 1 |
Berzetei, IP; Duckles, SP; Fong, A; Yamamura, HI | 1 |
Lahti, RA; McCall, JM; Mickelson, MM; Von Voigtlander, PF | 1 |
Desmeules, JA; Guilbaud, G; Kayser, V | 1 |
Bauer, U; Göthert, M; Kathmann, M; Nakazi, M; Schlicker, E | 1 |
9 other study(ies) available for u 69593 and mr 2266
Article | Year |
---|---|
Intracerebroventricular administration of kappa-agonists induces convulsions in mice.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Baclofen; Benzeneacetamides; Benzomorphans; Cerebral Ventricles; Convulsants; Dizocilpine Maleate; Injections, Intraventricular; Ketamine; Mice; Mice, Inbred Strains; Muscimol; Naloxone; Narcotic Antagonists; Narcotics; Pyrroles; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Seizures; Stereoisomerism; Thiophenes | 1991 |
Different motor actions of dynorphins and nonpeptide kappa opioid receptor agonists in the isolated rat colon.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Antihypertensive Agents; Benzeneacetamides; Benzodiazepines; Benzomorphans; Colon; Diuretics; Dynorphins; Gastrointestinal Motility; In Vitro Techniques; Male; Muscle, Smooth; Naloxone; Narcotic Antagonists; Pressure; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa | 1990 |
Effect of mu- and kappa-opioid agonists on the electroconvulsive seizure threshold in mice and antagonism by naloxone and MR 2266.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzeneacetamides; Benzodiazepines; Benzomorphans; Electroshock; Fentanyl; Male; Mice; Morphinans; Morphine; Nalbuphine; Naloxone; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Receptors, Opioid, mu; Seizures | 1988 |
Opioid kappa receptors correlate with the development of conditioned suppression of motility in mice.
Topics: Analgesics; Animals; Benzeneacetamides; Benzomorphans; Conditioning, Operant; Electroshock; Male; Mice; Mice, Inbred Strains; Motor Activity; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa | 1988 |
Stereospecific inhibition of gastrointestinal transit by kappa opioid agonists in mice.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzeneacetamides; Benzomorphans; Gastrointestinal Transit; Male; Mice; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism | 1988 |
Characterization of kappa opioid receptors in the rabbit ear artery.
Topics: Animals; Benzeneacetamides; Benzomorphans; Cyclazocine; Dynorphins; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Muscle, Smooth, Vascular; Narcotic Antagonists; Peptide Fragments; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1988 |
[3H]U-69593 a highly selective ligand for the opioid kappa receptor.
Topics: Analgesics; Animals; Benzeneacetamides; Benzomorphans; Brain; Guinea Pigs; In Vitro Techniques; Ligands; Male; Mice; Naloxone; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa | 1985 |
Selective opioid receptor agonists modulate mechanical allodynia in an animal model of neuropathic pain.
Topics: Analgesics; Animals; Benzeneacetamides; Benzomorphans; Disease Models, Animal; Drug Interactions; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Male; Naloxone; Naltrexone; Narcotic Antagonists; Oligopeptides; Pain; Pain Measurement; Pain Threshold; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Vocalization, Animal | 1993 |
The stereoselective kappa-opioid receptor antagonist Mr 2266 does not exhibit stereoselectivity as an antagonist at the orphan opioid (ORL1) receptor.
Topics: Animals; Benzeneacetamides; Benzomorphans; Cerebral Cortex; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Mice; Narcotic Antagonists; Nociceptin; Nociceptin Receptor; Opioid Peptides; Perfusion; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism | 1999 |