u 69593 has been researched along with glutamic acid in 15 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 6 (40.00) | 18.2507 |
2000's | 5 (33.33) | 29.6817 |
2010's | 4 (26.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Cheng, J; McCorvy, JD; Tan, L; Yan, W | 1 |
Kuraishi, Y; Oyama, T; Satoh, M; Sugimoto, K; Ueda, M | 1 |
Chavkin, C; Drake, CT; Simmons, ML; Terman, GW | 1 |
Chavkin, C; Terman, GW; Wagner, JJ | 1 |
Ho, IK; Hoshi, K; Ma, T | 1 |
McGinty, JF; Rawls, SM | 1 |
Gray, AM; McGinty, JF; Rawls, SM; Shippenberg, TS | 1 |
Fields, HL; Hjelmstad, GO | 1 |
Bie, B; Pan, ZZ | 1 |
Choi, DH; Jung, EB; Kim, MS; Kim, TY; Lee, J; Moon, SK; Park, C; Park, R | 1 |
Bonci, A; Fields, HL; Hjelmstad, GO; Margolis, EB | 1 |
Bains, JS; Iremonger, KJ | 1 |
Bäckman, CM; Chefer, V; Counotte, DS; O'Donnell, P; Oh, E; Ramamoorthy, S; Schultz-Kuszak, KN; Shippenberg, TS; Tejeda, HA | 1 |
Hanks, AN; Hughes, ZA; Mejias-Aponte, C; O'Donnell, P; Scott, L; Tejeda, HA | 1 |
Diaz, MR; Przybysz, KR; Werner, DF | 1 |
1 review(s) available for u 69593 and glutamic acid
Article | Year |
---|---|
Biased Ligands of G Protein-Coupled Receptors (GPCRs): Structure-Functional Selectivity Relationships (SFSRs) and Therapeutic Potential.
Topics: Animals; Drug Discovery; Humans; Ligands; Receptors, G-Protein-Coupled; Signal Transduction; Structure-Activity Relationship | 2018 |
14 other study(ies) available for u 69593 and glutamic acid
Article | Year |
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Opioidergic inhibition of capsaicin-evoked release of glutamate from rat spinal dorsal horn slices.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzeneacetamides; Capsaicin; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Glutamate Dehydrogenase; Glutamic Acid; In Vitro Techniques; Male; Morphine; Nerve Endings; Neurons, Afferent; Opioid Peptides; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Spinal Cord | 1995 |
Inhibition of glutamate release by presynaptic kappa 1-opioid receptors in the guinea pig dentate gyrus.
Topics: Afferent Pathways; Analgesics; Animals; Autoradiography; Benzeneacetamides; Culture Techniques; Dominance, Cerebral; Glutamic Acid; Guinea Pigs; Hippocampus; Male; Neural Inhibition; Pyrrolidines; Receptors, Opioid, kappa; Synaptic Transmission | 1994 |
Endogenous dynorphins inhibit excitatory neurotransmission and block LTP induction in the hippocampus.
Topics: Action Potentials; Animals; Benzeneacetamides; Dynorphins; Glutamates; Glutamic Acid; Guinea Pigs; Hippocampus; In Vitro Techniques; Naltrexone; Neural Inhibition; Neurotransmitter Agents; Pyrrolidines; Receptors, Opioid, kappa; Synapses; Time Factors | 1993 |
Precipitated kappa-opioid receptor agonist withdrawal increase glutamate in rat locus coeruleus.
Topics: Analgesics; Analysis of Variance; Animals; Aspartic Acid; Benzeneacetamides; Butorphanol; Glutamic Acid; Injections, Intraventricular; Locus Coeruleus; Male; Microdialysis; Naloxone; Narcotic Antagonists; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Substance Withdrawal Syndrome | 1996 |
Kappa receptor activation attenuates L-trans-pyrrolidine-2,4-dicarboxylic acid-evoked glutamate levels in the striatum.
Topics: Animals; Benzeneacetamides; Calcium; Corpus Striatum; Dicarboxylic Acids; Glutamic Acid; Kinetics; Male; Microdialysis; Naltrexone; Neurotransmitter Uptake Inhibitors; Perfusion; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid, kappa | 1998 |
The kappa-opioid agonist, U-69593, decreases acute amphetamine-evoked behaviors and calcium-dependent dialysate levels of dopamine and glutamate in the ventral striatum.
Topics: Amphetamine; Animals; Behavior, Animal; Benzeneacetamides; Calcium; Dopamine; Glutamic Acid; Male; Microdialysis; Naltrexone; Narcotic Antagonists; Neostriatum; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid, kappa | 1999 |
Kappa opioid receptor inhibition of glutamatergic transmission in the nucleus accumbens shell.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzeneacetamides; Dopamine Antagonists; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Male; Neural Inhibition; Neurons; Nucleus Accumbens; Patch-Clamp Techniques; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Receptors, Opioid, kappa; Receptors, Opioid, mu; Synaptic Transmission | 2001 |
Presynaptic mechanism for anti-analgesic and anti-hyperalgesic actions of kappa-opioid receptors.
Topics: Analgesics, Opioid; Animals; Behavior, Animal; Benzeneacetamides; Cells, Cultured; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Hyperalgesia; Male; Patch-Clamp Techniques; Pyrrolidines; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Opioid, kappa; Receptors, Opioid, mu; Receptors, Presynaptic; Synaptic Transmission | 2003 |
Morphine prevents glutamate-induced death of primary rat neonatal astrocytes through modulation of intracellular redox.
Topics: Acetylcysteine; Animals; Animals, Newborn; Apoptosis; Astrocytes; Benzeneacetamides; Benzimidazoles; Bisbenzimidazole; Carbocyanines; Cell Line, Tumor; Cell Nucleus; Cell Survival; Cells, Cultured; Dizocilpine Maleate; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Glutamic Acid; Glutathione; Hydrogen Peroxide; Ion Channels; Microscopy, Fluorescence; Mitochondrial Membrane Transport Proteins; Mitochondrial Permeability Transition Pore; Morphine; Naloxone; Narcotic Antagonists; Neuroglia; Oxidation-Reduction; Oxidative Stress; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Rhodamine 123 | 2004 |
Both kappa and mu opioid agonists inhibit glutamatergic input to ventral tegmental area neurons.
Topics: Analgesics, Opioid; Analysis of Variance; Animals; Benzeneacetamides; Drug Interactions; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Male; Neural Inhibition; Neurons; Patch-Clamp Techniques; Pyrrolidines; Rats; Rats, Sprague-Dawley; Time Factors; Ventral Tegmental Area | 2005 |
Retrograde opioid signaling regulates glutamatergic transmission in the hypothalamus.
Topics: 4-Aminopyridine; Analysis of Variance; Animals; Animals, Genetically Modified; Animals, Newborn; Benzeneacetamides; Calcium; Calcium Channel Blockers; Dendrites; Dynorphins; Electric Stimulation; Enzyme Inhibitors; Glutamic Acid; Green Fluorescent Proteins; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Male; Narcotic Antagonists; Neural Inhibition; Neural Pathways; Neurons; omega-Conotoxin GVIA; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Potassium Channel Blockers; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Signal Transduction; Synaptic Transmission | 2009 |
Prefrontal cortical kappa-opioid receptor modulation of local neurotransmission and conditioned place aversion.
Topics: Analgesics; Animals; Avoidance Learning; Benzeneacetamides; Dicarboxylic Acids; Dopamine; Drug Interactions; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Glutamic Acid; Male; Mice; Mice, Knockout; Microinjections; Miniature Postsynaptic Potentials; Naltrexone; Narcotic Antagonists; Neurotransmitter Uptake Inhibitors; Prefrontal Cortex; Pyramidal Cells; Pyrrolidines; Rats; Receptors, Opioid, kappa; Synaptic Transmission | 2013 |
Prefrontal Cortical Kappa Opioid Receptors Attenuate Responses to Amygdala Inputs.
Topics: Analgesics, Opioid; Animals; Anti-Anxiety Agents; Anxiety; Basolateral Nuclear Complex; Benzeneacetamides; Excitatory Postsynaptic Potentials; Glutamic Acid; Hippocampus; Male; Mice, Inbred C57BL; Microelectrodes; Naltrexone; Narcotic Antagonists; Neural Pathways; Optogenetics; Prefrontal Cortex; Pyrrolidines; Random Allocation; Rats, Long-Evans; Receptors, Opioid, kappa | 2015 |
Age-dependent regulation of GABA transmission by kappa opioid receptors in the basolateral amygdala of Sprague-Dawley rats.
Topics: Aging; Animals; Basolateral Nuclear Complex; Benzeneacetamides; gamma-Aminobutyric Acid; Glutamic Acid; Inhibitory Postsynaptic Potentials; Male; Naltrexone; Pyrrolidines; Rats; Receptors, Opioid, kappa; Synaptic Transmission | 2017 |