Page last updated: 2024-08-26

u 69593 and cyclazocine

u 69593 has been researched along with cyclazocine in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19905 (55.56)18.7374
1990's3 (33.33)18.2507
2000's1 (11.11)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bettaney, J; Dray, A; James, IF; Ketchum, SB; Perkins, MN1
Magnan, J; Tiberi, M1
Cicero, TJ; Giordano, AL; Nock, B; O'Connor, LH1
Bykov, V; De Costa, BR; France, CP; Jacobson, AE; Rice, KC; Rothman, RB; Woods, JH1
Cicero, TJ; Nock, B; O'Connor, LH; Rajpara, A2
Magnan, J; Mongeau, R; Payette, P; Tiberi, M1
Berzetei, IP; Duckles, SP; Fong, A; Yamamura, HI1
Bidlack, JM; Cioffi, CL; Cohen, DJ; Colasurdo, AM; Duan, W; Wentland, MP; Xu, G; Ye, Y1

Other Studies

9 other study(ies) available for u 69593 and cyclazocine

ArticleYear
Opioid receptor ligands in the neonatal rat spinal cord: binding and in vitro depression of the nociceptive responses.
    British journal of pharmacology, 1990, Volume: 99, Issue:3

    Topics: Animals; Animals, Newborn; Benzeneacetamides; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; In Vitro Techniques; Kinetics; Ligands; Morphine; Muscle, Smooth, Vascular; Naloxone; Narcotics; Nociceptors; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Spinal Cord

1990
Demonstration of the heterogeneity of the kappa-opioid receptors in guinea-pig cerebellum using selective and nonselective drugs.
    European journal of pharmacology, 1990, Jun-12, Volume: 188, Issue:6

    Topics: Animals; Benzeneacetamides; Benzomorphans; Binding, Competitive; Cerebellum; Computers; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Ethylketocyclazocine; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Membranes; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1990
Affinity of drugs and peptides for U-69,593-sensitive and -insensitive kappa opiate binding sites: the U-69,593-insensitive site appears to be the beta endorphin-specific epsilon receptor.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:2

    Topics: Analgesics; Animals; Benzeneacetamides; Binding, Competitive; Brain; Culture Techniques; Cyclazocine; Ethylketocyclazocine; Narcotics; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa

1990
Pharmacological activities of optically pure enantiomers of the kappa opioid agonist, U50,488, and its cis diastereomer: evidence for three kappa receptor subtypes.
    European journal of pharmacology, 1989, Aug-29, Volume: 167, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Behavior, Animal; Benzeneacetamides; Benzodiazepines; Benzomorphans; Binding, Competitive; Brain Chemistry; Cyclazocine; Discrimination, Psychological; Ethylketocyclazocine; Female; Guinea Pigs; Macaca mulatta; Male; Membranes; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Stereoisomerism

1989
[3H]U-69593 labels a subtype of kappa opiate receptor with characteristics different from that labeled by [3H]ethylketocyclazocine.
    Life sciences, 1988, Volume: 42, Issue:23

    Topics: Animals; Benzeneacetamides; Binding, Competitive; Brain; Cell Membrane; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Ethylketocyclazocine; Male; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Sodium Chloride; Temperature; Tritium

1988
Autoradiography of [3H]U-69593 binding sites in rat brain: evidence for kappa opioid receptor subtypes.
    European journal of pharmacology, 1988, Sep-01, Volume: 154, Issue:1

    Topics: Analgesics; Animals; Autoradiography; Benzeneacetamides; Benzomorphans; Binding Sites; Brain Chemistry; Cyclazocine; Ethylketocyclazocine; Male; Pyrrolidines; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, kappa; Temperature

1988
[3H]U69,593 binding in guinea-pig brain: comparison with [3H]ethylketazocine binding at the kappa-opioid sites.
    Canadian journal of physiology and pharmacology, 1988, Volume: 66, Issue:11

    Topics: Benzeneacetamides; Brain; Cyclazocine; Ethylketocyclazocine; Kinetics; Pyrrolidines; Radioligand Assay; Receptors, Opioid

1988
Characterization of kappa opioid receptors in the rabbit ear artery.
    European journal of pharmacology, 1988, Jul-14, Volume: 151, Issue:3

    Topics: Animals; Benzeneacetamides; Benzomorphans; Cyclazocine; Dynorphins; Ethylketocyclazocine; In Vitro Techniques; Male; Mice; Muscle, Smooth, Vascular; Narcotic Antagonists; Peptide Fragments; Pyrrolidines; Rabbits; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1988
8-Aminocyclazocine analogues: synthesis and structure-activity relationships.
    Bioorganic & medicinal chemistry letters, 2000, Jan-17, Volume: 10, Issue:2

    Topics: Analgesics; Animals; Benzeneacetamides; Binding, Competitive; Brain; Cyclazocine; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Guinea Pigs; Molecular Structure; Naltrexone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid; Stereoisomerism; Structure-Activity Relationship

2000