u 37883a has been researched along with adamantane in 63 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 40 (63.49) | 18.2507 |
2000's | 17 (26.98) | 29.6817 |
2010's | 6 (9.52) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Graham, BE; Humphrey, SJ; Ludens, JH; Perricone, SC; Skaletzky, LL; Zins, GR | 1 |
Kadowitz, PJ; McMahon, TJ; Minkes, RK; Santiago, JA | 1 |
Choe, E; Ferrara, J; Flint, L; Franklin, E; Grivas, T; Hyman, A; Lippton, H | 1 |
Clark, MA; Humphrey, SJ; Ludens, JH; Smith, MP | 1 |
Clark, MA; Lawson, JA; Ludens, JH | 2 |
Giebisch, G; Klein-Robbenhaar, G; Wang, T; Wang, WH | 1 |
Fosset, M; Humphrey, S; Lazdunski, M; Meisheri, K | 1 |
Humphrey, SJ; Jackson, WF; Smith, MP | 1 |
Graham, BE; Humphrey, SJ; Perricone, SC; Skaletzky, LL; Zandt, RA; Zins, GR | 1 |
De Weille, J; Fosset, M; Guillemare, E; Honore, E; Lazdunski, M; Meisheri, K | 1 |
Khan, SA; Meisheri, KD; Ohrnberger, CE | 1 |
Ferrara, JJ; Flint, LM; Force, SD; Franklin, EW; Hyman, AL; Lippton, HL; Taheri, PA | 1 |
Cipkus-Dubray, LA; Humphrey, SJ; Jones, AW; Khan, SA; Meisheri, KD; Smith, MP | 1 |
Champion, HC; Del Rio, O; Garrison, EA; Kadowitz, PJ; Santiago, JA; Smith, RE | 1 |
Humphrey, SJ | 1 |
Cheng, DY; DeWitt, BJ; Kadowitz, PJ; Neely, CF; Suzuki, F | 1 |
Buchanan, LV; Cimini, MG; Gibson, JK; Humphrey, SJ; Khan, SA; Meisheri, KD; Smith, MP | 1 |
Bivalacqua, TJ; Champion, HC; Coy, DH; Erickson, CC; Kadowitz, PJ; Murphy, WA; Simoneaux, ML | 1 |
Champion, HC; Cheng, DY; DeWitt, BJ; Kandowitz, PJ; Marrone, JR; McMahon, TJ | 1 |
Choe, EU; Cruz, MP; Ferrara, JJ; Flint, LM; Hyman, AL; Lippton, HL; Pigott, JD; Sabates, BL | 1 |
Jasińska, R; Makowski, P; Pikuła, S; Szewczyk, A | 1 |
Champion, HC; Kadowitz, PJ | 1 |
Bivalacqua, TJ; Champion, HC; Czapla, MA; Ilgenfritz, C; Kadowitz, PJ; Santiago, JA | 1 |
Blantz, RC; Osswald, H; Thomson, S; Vallon, V | 1 |
Humphrey, SJ; Ludens, JH | 1 |
Chen, X; Freedman, JE; Lin, YJ | 1 |
Albinus, M; Blach, D; Vallon, V | 1 |
Löffler-Walz, C; Quast, U | 1 |
Albinus, M; Brenner, I; Kirschenmann, D; Osswald, H; Vallon, V | 1 |
Anwar, M; Banister, RE; Feng, CJ; Kadowitz, PJ; Kaye, AD; Nossaman, BD | 1 |
Bivalacqua, TJ; Champion, HC; Friedman, DE; Kadowitz, PJ; Kastin, AJ; Zadina, JE | 1 |
Anwar, M; Banister, R; Banister, RE; Feng, C; Feng, CJ; Kadowitz, P; Kadowitz, PJ; Kaye, A; Kaye, AD; Nossaman, B; Nossaman, BD; Turner, K | 1 |
Huang, DY; Osswald, H; Vallon, V | 2 |
Abassi, RA; Bivalacqua, TJ; Champion, HC; Kadowitz, PJ; Lambert, DG | 1 |
Beech, DJ; Cheong, A; Hough, E; McDonald, RL; McHugh, D; Partridge, C; Sivaprasadarao, A; Surah-Narwal, S; Xu, SZ | 1 |
Barrett-Jolley, R; Everitt, D; Köppel, H; Quayle, JM; Wellman, GC | 1 |
Fujita, T; Hayashi, I; Inamura, N; Kumagai, Y; Majima, M | 2 |
Bivalacqua, TJ; Champion, HC; Kadowitz, PJ; Kastin, AJ; Zadina, JE | 1 |
Anwar, M; De Witt, BJ; Feng, CJ; Kadowitz, PJ; Kaye, AD; Nossaman, BD; Smith, DE | 1 |
Ikeda, S; Kyotani, S; Min, KY; Mori, H; Nagaya, N; Nakanishi, N; Ninomiya, I; Oya, H; Shimouchi, A; Shirai, M | 1 |
Bivalacqua, TJ; Champion, HC; Coy, DH; Kadowitz, PJ; Murphy, WA; Pierce, RL | 1 |
Bivalacqua, TJ; Champion, HC; Kadowitz, PJ; Shah, MK | 1 |
Cha, SH; Endou, H; Fujita, T; Hayashi, I; Higashihara, M; Majima, M; Yamanaka, M | 1 |
Kamishima, T; Kovalev, H; Lodwick, D; Quayle, JM | 1 |
Galun, E; Matot, I; Rivo, J; Zeira, E | 1 |
Aishima, M; Brading, AF; Ito, Y; Takahashi-Yanaga, F; Teramoto, N; Tomoda, T; Yunoki, T; Zhu, HL | 1 |
Cao, K; Hanna, ST; Wang, R | 1 |
Ito, Y; Naito, S; Teramoto, N; Tomoda, T; Yunoki, T | 1 |
Teramoto, N | 1 |
Al Abed, A; Brock, JA; Tan, JH | 1 |
Jiang, B; Wang, R; Wu, L | 1 |
Baber, SR; Bivalacqua, TJ; Champion, HC; Kadowitz, PJ; Nossaman, BD | 1 |
Baun, M; Boni, LJ; Hay-Schmidt, A; Jansen-Olesen, I; Olesen, J; Ploug, KB | 1 |
Hay-Schmidt, A; Jansen-Olesen, I; Klaerke, DA; Olesen, J; Ploug, KB; Sheykhzade, M; Strøbech, L; Sørensen, MA | 1 |
Chan, YL; Clapp, LH; Dyson, A; Orie, NN; Singer, M; Stidwill, RP; Taylor, V | 1 |
Chang, SW; Chen, YZ; Fang, SY; Hsu, CY; Huang, CC; Lam, CF; Liu, YC; Roan, JN; Tsai, YC | 1 |
Inoue, T; Murai, M; Ochiai, T; Ra, C; Suzuki, Y; Suzuki-Karasaki, M | 1 |
Asfar, P; Collin, S; Fremont-Orlowski, S; Ganster, F; Issa, K; Kimmoun, A; Levy, B; Mertes, PM | 1 |
Inai, T; Node, K; Takahara, K; Teramoto, N; Yamamoto, T | 1 |
Busch, CJ; Lasitschka, F; Turzo, M; Vaith, J; Weigand, MA | 1 |
1 review(s) available for u 37883a and adamantane
Article | Year |
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Pharmacological Profile of U-37883A, a Channel Blocker of Smooth Muscle-Type ATP-Sensitive K Channels.
Topics: Adamantane; Animals; Diuretics; Morpholines; Muscle, Smooth, Vascular; Potassium Channel Blockers; Potassium Channels | 2006 |
62 other study(ies) available for u 37883a and adamantane
Article | Year |
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Diuretic activity of N'-disubstituted morpholinoguanidine analogs of U-37883A in rats and dogs.
Topics: Adamantane; Animals; Diuretics; Dogs; Heart Rate; In Vitro Techniques; Morpholines; Myocardial Contraction; Perfusion; Potassium; Rats; Sodium; Species Specificity | 1995 |
Role of K+ATP channels and EDRF in reactive hyperemia in the hindquarters vascular bed of cats.
Topics: Adamantane; Adenosine Triphosphate; Animals; Arginine; Cats; Glyburide; Hindlimb; Hyperemia; Ischemia; Morpholines; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Potassium Channels; Pulmonary Circulation; Regional Blood Flow; Vasodilation; Vasodilator Agents | 1995 |
Femoral vasodilation to cromakalim is blocked by U37883A, a non-sulphonylurea that selectively inhibits KATP channels.
Topics: Adamantane; Analysis of Variance; Animals; Benzopyrans; Cromakalim; Dogs; Drug Interactions; Femur; Injections, Intravenous; Isoproterenol; Morpholines; Nitroglycerin; Potassium Channels; Pyrroles; Regional Blood Flow; Serotonin; Serotonin Receptor Agonists; Vasodilation; Vasodilator Agents | 1995 |
Renal and vascular effects of chemically distinct ATP-sensitive K+ channel blockers in rats.
Topics: Adamantane; Adenosine Triphosphate; Anesthesia; Animals; Blood Glucose; Dose-Response Relationship, Drug; Guanidines; Hemodynamics; Kidney; Male; Morpholines; Natriuresis; Pinacidil; Potassium Channels; Rats; Rats, Sprague-Dawley; Sodium; Vasodilator Agents | 1995 |
Effects of a K+ channel blocker on glomerular filtration rate and electrolyte excretion in conscious rats.
Topics: Adamantane; Animals; Diuretics; Dose-Response Relationship, Drug; Electrolytes; Glomerular Filtration Rate; Male; Morpholines; Natriuresis; Osmolar Concentration; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Water | 1995 |
Effects of a novel KATP channel blocker on renal tubule function and K channel activity.
Topics: Adamantane; Animals; Diuretics; Kidney Tubules; Loop of Henle; Male; Morpholines; Natriuresis; Perfusion; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley | 1995 |
Receptor binding characterization in kidney membrane of [3H]U-37883, a novel ATP-sensitive K+ channel blocker with diuretic/natriuretic properties.
Topics: Adamantane; Adenosine Triphosphate; Animals; Binding, Competitive; Diuretics; Endopeptidases; Kidney; Kinetics; Morpholines; Natriuresis; Potassium Channels; Sensitivity and Specificity; Swine; Tritium | 1995 |
Selective in vivo antagonism of pinacidil-induced hypotension by the guanidine U37883A in anesthetized rats.
Topics: Adamantane; Anesthesia; Animals; Blood Pressure; Diuretics; Dose-Response Relationship, Drug; Female; Guanidines; Heart; Heart Rate; Hypotension; Morpholines; Pinacidil; Potassium Channels; Rats; Rats, Sprague-Dawley; Tachycardia; Vasodilator Agents | 1994 |
Synthesis and diuretic activity of alkyl- and arylguanidine analogs of N,N'-dicyclohexyl-4-morpholinecarboxamidine in rats and dogs.
Topics: Adamantane; Administration, Oral; Animals; Blood Pressure; Diuretics; Dogs; Drug Interactions; Female; Heart Rate; Male; Minoxidil; Morpholines; Potassium Channels; Rats; Rats, Sprague-Dawley | 1994 |
Functional receptors in Xenopus oocytes for U-37883A, a novel ATP-sensitive K+ channel blocker: comparison with rat insulinoma cells.
Topics: Adamantane; Adenosine Triphosphate; Animals; Binding Sites; Female; Glyburide; Insulinoma; Morpholines; Oocytes; Potassium Channels; Rats; Tumor Cells, Cultured; Xenopus laevis | 1994 |
Synergistic effects of glyburide and U-37883A, two structurally different vascular ATP-sensitive potassium channel antagonists.
Topics: Adamantane; Adenosine Triphosphate; Animals; Benzopyrans; Cromakalim; Drug Synergism; Gallopamil; Glyburide; In Vitro Techniques; Ion Channel Gating; Male; Mesenteric Arteries; Minoxidil; Morpholines; Potassium Channels; Pyrroles; Rabbits; Vasodilation | 1993 |
Analysis of regional hemodynamic regulation in response to scald injury.
Topics: Adamantane; Animals; Arginine; Atropine; Blood Pressure; Burns; Diphenhydramine; Dogs; Femoral Artery; Hemodynamics; Hindlimb; Histamine; Isoproterenol; Meclofenamic Acid; Methoxamine; Methysergide; Morpholines; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitroglycerin; Pulmonary Circulation; Ranitidine; Regional Blood Flow; Ritanserin; Serotonin; Serotonin Receptor Agonists; Time Factors; Triazines; Ultrasonography; Vascular Resistance; Vasodilation; Verapamil; Xanthines | 1994 |
4-morpholinecarboximidine-N-1-adamantyl-N'-cyclohexylhydrochloride (U-37883A): pharmacological characterization of a novel antagonist of vascular ATP-sensitive K+ channel openers.
Topics: Adamantane; Adenosine Triphosphate; Animals; Benzopyrans; Blood Pressure; Cats; Cromakalim; Dogs; Female; In Vitro Techniques; Male; Mesenteric Arteries; Minoxidil; Morpholines; Potassium; Potassium Channels; Pyrroles; Rabbits; Rats; Rats, Sprague-Dawley; Vasodilation | 1993 |
Analysis of responses to kallidin, DABK, and DAK in feline hindlimb vascular bed.
Topics: Adamantane; Animals; Arginine; Atropine; Blood Vessels; Bradykinin; Bradykinin Receptor Antagonists; Cats; Female; Hindlimb; Kallidin; Male; Meclofenamic Acid; Morpholines; Muscarinic Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Potassium Channels | 1995 |
Effects of K-ATP blocking guanidine diuretics during experimental kaliuresis in rats and dogs.
Topics: Adamantane; Animals; Creatinine; Diuretics; Dogs; Female; Guanidines; Male; Morpholines; Potassium; Potassium Chloride; Rats; Rats, Sprague-Dawley; Sodium; Sodium Chloride | 1995 |
Adenosine A1 and A2 receptors mediate tone-dependent responses in feline pulmonary vascular bed.
Topics: Adamantane; Adenosine; Adenosine Triphosphate; Animals; Arginine; Cats; Female; Male; Methylene Blue; Morpholines; Muscle Tonus; Muscle, Smooth, Vascular; Prostaglandin-Endoperoxide Synthases; Pulmonary Circulation; Purinergic P1 Receptor Agonists; Receptors, Purinergic P1; Xanthines | 1996 |
Cardiovascular effects of the K-ATP channel blocker U-37883A and structurally related morpholinoguanidines.
Topics: Adamantane; Adenosine Triphosphate; Administration, Oral; Analysis of Variance; Animal Welfare; Animals; Blood Pressure; Diuretics; Dogs; Electrophysiology; Female; Guanidines; Heart Rate; Injections, Intravenous; Male; Mesenteric Arteries; Morpholines; Myocardial Contraction; Papillary Muscles; Pinacidil; Potassium Channels; Rabbits; Rats; Rats, Sprague-Dawley; Species Specificity; Stroke Volume; Structure-Activity Relationship; Vascular Resistance; Vasodilator Agents; Ventricular Function, Left | 1996 |
Proadrenomedullin NH2-terminal 20 peptide has cAMP-mediated vasodilator activity in the mesenteric vascular bed of the cat.
Topics: Adamantane; Adrenomedullin; Animals; Cats; Cyclic AMP; Denervation; Enzyme Inhibitors; Female; Male; Mesenteric Artery, Superior; Morpholines; NG-Nitroarginine Methyl Ester; Peptide Fragments; Peptides; Phentolamine; Proteins; Purinones; Pyrrolidinones; Reserpine; Rolipram; Sympathetic Nervous System; Sympatholytics; Vasodilation | 1996 |
Effects of U-37883A, a vascular selective KATP+ channel antagonist, in the pulmonary and hindlimb circulation.
Topics: Adamantane; Animals; Blood Vessels; Cats; Extremities; Female; Glyburide; Male; Morpholines; Potassium Channel Blockers; Pulmonary Circulation; Vasodilation | 1996 |
Adrenomedullin mediates coronary vasodilation through adenosine receptors and KATP channels.
Topics: Adamantane; Adenosine Triphosphate; Adrenomedullin; Animals; Calcitonin Gene-Related Peptide; Calcitonin Gene-Related Peptide Receptor Antagonists; Coronary Circulation; Coronary Vessels; Dogs; Morpholines; Peptide Fragments; Peptides; Potassium Channels; Receptors, Purinergic P1; Vascular Resistance; Vasodilation; Xanthines | 1997 |
An antagonist of ATP-regulated potassium channels, the guanidine derivative U-37883A, stimulates the synthesis of phosphatidylserine in rat liver endoplasmic reticulum membranes.
Topics: Adamantane; Adenosine Triphosphate; Animals; Calcium; Endoplasmic Reticulum; Kinetics; Male; Microsomes, Liver; Morpholines; Phosphatidylserines; Phospholipids; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Serine | 1997 |
NO release and the opening of K+ATP channels mediate vasodilator responses to histamine in the cat.
Topics: Adamantane; Adenosine Triphosphate; Animals; Cats; Cyclic AMP; Cyclic GMP; Enzyme Inhibitors; Female; Histamine; Histamine Agonists; Histamine Antagonists; Male; Morpholines; NG-Nitroarginine Methyl Ester; Nitric Oxide; Potassium Channels; Prostaglandins; Tetraethylammonium; Tetraethylammonium Compounds; Vasodilation; Vasodilator Agents | 1997 |
Comparison of responses to T-kinin and bradykinin in the mesenteric vascular bed of the cat.
Topics: Adamantane; Analysis of Variance; Animals; Bradykinin; Bradykinin Receptor Antagonists; Cats; Cimetidine; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Female; Histamine Antagonists; Male; Meclofenamic Acid; Mesentery; Morpholines; NG-Nitroarginine Methyl Ester; Piperidines; Potassium Channels; Pyrilamine | 1997 |
Potential role of luminal potassium in tubuloglomerular feedback.
Topics: Adamantane; Animals; Carrier Proteins; Cell Polarity; Feedback; Glomerular Filtration Rate; Ion Transport; Kidney Tubules, Distal; Kidney Tubules, Proximal; Male; Morpholines; Natriuresis; Perfusion; Potassium; Potassium Channels; Rats; Rats, Inbred Strains; Sodium Chloride; Sodium-Potassium-Chloride Symporters | 1997 |
The natriuretic activity of the K+ channel blocker U-37883A displays an ADH-dependence.
Topics: Adamantane; Animals; Blood Pressure; Diuretics; Furosemide; Glomerular Filtration Rate; Heart Rate; Male; Morpholines; Natriuresis; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Sodium Chloride; Vasopressins; Water | 1998 |
K-ATP-blocking diuretic PNU-37883A reduces plasma renin activity in dogs.
Topics: Adamantane; Animals; Diuretics; Dogs; Drug Interactions; Female; Furosemide; Infusions, Intra-Arterial; Infusions, Intravenous; Male; Morpholines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Renal Artery; Renin | 1998 |
U-37883A potently inhibits dopamine-modulated K+ channels on rat striatal neurons.
Topics: Adamantane; Animals; Corpus Striatum; Dopamine; Morpholines; Neurons; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Rats | 1998 |
Effect of KATP channel blocker U37883A on renal function in experimental diabetes mellitus in rats.
Topics: Adamantane; Adenosine Triphosphate; Animals; Diabetes Mellitus, Experimental; Glomerular Filtration Rate; Kidney; Male; Morpholines; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Renal Circulation; Renin; Streptozocin | 1998 |
Interaction of the diuretics torasemide and U-37883A with the K(ATP) channel in rat isolated aorta.
Topics: Adamantane; Adenosine Triphosphate; Animals; Aorta; Binding, Competitive; Diuretics; Dose-Response Relationship, Drug; Furosemide; In Vitro Techniques; Isometric Contraction; Male; Morpholines; Potassium Channels; Protein Binding; Rats; Rats, Sprague-Dawley; Rubidium; Rubidium Radioisotopes; Sulfonamides; Torsemide | 1998 |
Potassium diet as a determinant for the renal response to systemic potassium channel modulation in anesthetized rats.
Topics: Adamantane; Animals; Blood Pressure; Body Fluids; Diuretics; Dose-Response Relationship, Drug; Glomerular Filtration Rate; Guanidines; Heart Rate; Juxtaglomerular Apparatus; Kidney; Male; Morpholines; Potassium; Potassium Channels; Potassium, Dietary; Pyridines; Rats; Rats, Sprague-Dawley; Renin; Sodium; Vasodilator Agents | 1998 |
Pulmonary vasodilation by ketamine is mediated in part by L-type calcium channels.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adamantane; Anesthetics, Dissociative; Animals; Arachidonic Acid; Arginine; Blood Pressure; Calcium Channel Blockers; Calcium Channels; Cromakalim; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Ketamine; Lung; Male; Meclofenamic Acid; Morpholines; Potassium Channels; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Vasodilation; Verapamil | 1998 |
Nitric oxide release mediates vasodilator responses to endomorphin 1 but not nociceptin/OFQ in the hindquarters vascular bed of the rat.
Topics: Adamantane; Animals; Blood Vessels; Endorphins; Endothelium, Vascular; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Meclofenamic Acid; Morpholines; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nociceptin; Oligopeptides; Opioid Peptides; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Regional Blood Flow; Vasodilation; Vasodilator Agents | 1998 |
Responses to propofol in the pulmonary vascular bed of the rat.
Topics: Acetylcholine; Adamantane; Adenosine Triphosphate; Adrenergic beta-Agonists; Anesthetics, Intravenous; Animals; Arachidonic Acid; Arginine; Blood Pressure; Chelating Agents; Cyclooxygenase Inhibitors; Dimethyl Sulfoxide; Diuretics; Dose-Response Relationship, Drug; Edetic Acid; Enzyme Inhibitors; Isoproterenol; Lung; Male; Meclofenamic Acid; Morpholines; Nitric Oxide Synthase; Nitroglycerin; Potassium Channel Blockers; Propofol; Pulmonary Circulation; Rats; Rats, Sprague-Dawley; Solvents; Vasodilator Agents | 1999 |
Eukaliuric diuresis and natriuresis in response to the KATP channel blocker U37883A: micropuncture studies on the tubular site of action.
Topics: Adamantane; Animals; Diuresis; Diuretics; Furosemide; Glomerular Filtration Rate; Glyburide; Hypoglycemic Agents; Kidney Tubules, Distal; Kidney Tubules, Proximal; Loop of Henle; Morpholines; Natriuresis; Potassium Channels; Punctures; Rats | 1999 |
Analysis of vasoconstrictor responses to histamine in the hindlimb vascular bed of the rabbit.
Topics: Adamantane; Adrenergic alpha-Antagonists; Angiotensin Receptor Antagonists; Animals; Benzimidazoles; Biphenyl Compounds; Blood Vessels; Cyclooxygenase Inhibitors; Enzyme Inhibitors; Hindlimb; Histamine; Injections, Intravenous; Male; Meclofenamic Acid; Morpholines; NG-Nitroarginine Methyl Ester; Phentolamine; Rabbits; Receptor, Angiotensin, Type 1; Receptor, Angiotensin, Type 2; Receptors, Histamine; Tetrazoles; Vasoconstriction; Vasoconstrictor Agents | 1999 |
Block of human aorta Kir6.1 by the vascular KATP channel inhibitor U37883A.
Topics: Adamantane; Animals; Aorta; Cricetinae; Humans; Membrane Potentials; Mice; Morpholines; Potassium Channel Blockers; Potassium Channels, Inwardly Rectifying; Rats; Xenopus laevis | 1999 |
Inhibition of vascular K(ATP) channels by U-37883A: a comparison with cardiac and skeletal muscle.
Topics: Adamantane; Adenosine Triphosphate; Animals; Cromakalim; In Vitro Techniques; Male; Mesenteric Arteries; Morpholines; Muscle Relaxation; Muscle, Skeletal; Myocardium; Potassium Channel Blockers; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar | 1999 |
Early increases in renal kallikrein secretion on administration of potassium or ATP-sensitive potassium channel blockers in rats.
Topics: Adamantane; Adenosine Triphosphate; Animals; Chlorides; Dose-Response Relationship, Drug; Gluconates; Glyburide; In Vitro Techniques; Kallikreins; Kidney; Male; Morpholines; Perfusion; Polyethylene Glycols; Potassium; Potassium Channel Blockers; Potassium Chloride; Rats; Rats, Sprague-Dawley; Sodium; Time Factors; Urination | 1999 |
K+ loading, but not Na+ loading, and blockade of ATP-sensitive K+ channels augment renal kallikrein secretion.
Topics: Adamantane; Animals; ATP-Binding Cassette Transporters; Glyburide; Kallikreins; KATP Channels; Kidney; Male; Morpholines; Potassium; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Sprague-Dawley; Sodium | 1999 |
Vasodilator responses to the endomorphin peptides, but not nociceptin/OFQ, are mediated by nitric oxide release.
Topics: Adamantane; Analgesics, Opioid; Animals; Diuretics; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Hindlimb; Meclofenamic Acid; Morpholines; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nociceptin; Oligopeptides; Opioid Peptides; Rats; Rats, Sprague-Dawley; Vasodilation; Vasodilator Agents | 1999 |
Sodium reabsorption in thick ascending limb of Henle's loop: effect of potassium channel blockade in vivo.
Topics: Adamantane; Animals; Barium; Cesium; Charybdotoxin; Dose-Response Relationship, Drug; Glyburide; Loop of Henle; Male; Models, Biological; Morpholines; Potassium; Potassium Channel Blockers; Potassium Channels; Quinine; Rats; Rats, Wistar; Sodium; Verapamil | 2000 |
Analysis of responses of garlic derivatives in the pulmonary vascular bed of the rat.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adamantane; Allyl Compounds; Animals; Antihypertensive Agents; Antioxidants; Bronchodilator Agents; Cromakalim; Cyclooxygenase Inhibitors; Disulfides; Diuretics; Enzyme Inhibitors; Garlic; Hypertension, Pulmonary; Lung Diseases, Obstructive; Male; Meclofenamic Acid; Morpholines; NG-Nitroarginine Methyl Ester; Plants, Medicinal; Pulmonary Circulation; Rats; Rats, Sprague-Dawley; Respiration; Sulfhydryl Compounds; Sulfinic Acids; Vasoconstrictor Agents | 2000 |
K(ATP) channels predominantly regulate conduit vessel tone in normoxic cat pulmonary arteries in vivo.
Topics: Adamantane; Adenosine Triphosphate; Animals; Blood Pressure; Cats; Cromakalim; Dose-Response Relationship, Drug; Glyburide; Morpholines; Potassium Channels; Pulmonary Artery; Vasoconstriction; Vasodilator Agents | 2001 |
Analysis of responses to hAmylin, hCGRP, and hADM in isolated resistance arteries from the mesenteric vascular bed of the rat.
Topics: Acetylcholine; Adamantane; Adrenomedullin; Amyloid; Animals; Arginine; Calcitonin Gene-Related Peptide; Cromakalim; Dose-Response Relationship, Drug; Endothelium, Vascular; Enzyme Inhibitors; Humans; In Vitro Techniques; Islet Amyloid Polypeptide; Mesenteric Arteries; Morpholines; Nitric Oxide Synthase; Oxadiazoles; Peptide Fragments; Peptides; Perfusion; Potassium Channel Blockers; Quinoxalines; Rats; Receptors, Calcitonin Gene-Related Peptide; Receptors, Islet Amyloid Polypeptide; Receptors, Peptide; Vascular Resistance; Vasodilator Agents | 2001 |
Differential responses to ATPgammaS in the mesenteric and hindlimb vascular bed of the cat.
Topics: Adamantane; Adenosine Triphosphate; Animals; Cats; Female; Hindlimb; Male; Meclofenamic Acid; Mesentery; Morpholines; NG-Nitroarginine Methyl Ester; Phentolamine; Purinergic Agonists; Purinergic Antagonists; Pyridoxal Phosphate; Vascular Resistance | 2001 |
Potassium-induced increase in renal kallikrein secretion is attenuated in dissected renal connecting tubules of young spontaneously hypertensive rats.
Topics: Adamantane; Animals; Dose-Response Relationship, Drug; Hypertension; In Vitro Techniques; Kallikrein-Kinin System; Kallikreins; Kidney Tubules; Male; Morpholines; Potassium Channel Blockers; Potassium Chloride; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Rats, Sprague-Dawley | 2002 |
Molecular analysis of the subtype-selective inhibition of cloned KATP channels by PNU-37883A.
Topics: Adamantane; Adenosine Triphosphate; Animals; Cloning, Molecular; Dose-Response Relationship, Drug; Female; Membrane Proteins; Morpholines; Potassium Channel Blockers; Potassium Channels; Rats; Xenopus laevis | 2004 |
Activation of A3 adenosine receptors attenuates lung injury after in vivo reperfusion.
Topics: Adamantane; Adenosine; Adenosine A3 Receptor Agonists; Adenosine A3 Receptor Antagonists; Animals; ATP-Binding Cassette Transporters; Cats; Dihydropyridines; Enzyme Inhibitors; Hemodynamics; Histamine; In Vitro Techniques; KATP Channels; Lung; Morpholines; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitroarginine; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pulmonary Artery; Reperfusion Injury | 2004 |
Effects of U-37883A on intracellular Ca2+ -activated large-conductance K+ channels in pig proximal urethral myocytes.
Topics: Adamantane; Animals; Calcium; Cells, Cultured; Kinetics; Membrane Potentials; Morpholines; Myocytes, Smooth Muscle; Potassium Channels, Calcium-Activated; Swine; Time Factors; Urethra | 2004 |
Interaction of acetylcholine with Kir6.1 channels heterologously expressed in human embryonic kidney cells.
Topics: Acetylcholine; Adamantane; Adenosine Triphosphate; ATP-Binding Cassette Transporters; Atropine; Barium; Bungarotoxins; Cell Line; Dihydro-beta-Erythroidine; Dimethylphenylpiperazinium Iodide; Dose-Response Relationship, Drug; Gene Expression; Humans; KATP Channels; Mecamylamine; Membrane Potentials; Morpholines; Muscarinic Antagonists; Nicotinic Antagonists; Patch-Clamp Techniques; Potassium Channels, Inwardly Rectifying; Receptors, Nicotinic; Transfection | 2005 |
Multiple actions of U-37883A, an ATP-sensitive K+ channel blocker, on membrane currents in pig urethra.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adamantane; Adenosine Triphosphate; Analysis of Variance; Animals; Barium; Calcium Channel Agonists; Cromakalim; Dose-Response Relationship, Drug; Female; Glyburide; In Vitro Techniques; Membrane Potentials; Morpholines; Muscle Cells; Nitroprusside; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels, Inwardly Rectifying; Swine; Time Factors; Urethra; Vasodilator Agents | 2005 |
Inhibition of KATP channels in the rat tail artery by neurally released noradrenaline acting on postjunctional alpha2-adrenoceptors.
Topics: Adamantane; Adenosine Triphosphate; Animals; Arteries; Calcitonin Gene-Related Peptide; Cromakalim; Dose-Response Relationship, Drug; Electric Impedance; Excitatory Postsynaptic Potentials; Female; Glyburide; In Vitro Techniques; Ion Channel Gating; Morpholines; Muscle, Smooth, Vascular; Norepinephrine; Pinacidil; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Sympathetic Nervous System; Tail; Time Factors | 2007 |
Sulphonylureas induced vasorelaxation of mouse arteries.
Topics: Adamantane; Animals; Arteries; Endothelium, Vascular; Glyburide; In Vitro Techniques; KATP Channels; Male; Mesenteric Arteries; Mice; Mice, Inbred C57BL; Morpholines; Muscle Relaxation; Muscle, Smooth, Vascular; Oxadiazoles; Phenylephrine; Potassium Channel Blockers; Quinoxalines; Sulfonylurea Compounds; Vascular Resistance; Vasoconstrictor Agents | 2007 |
Analysis of vasodilator responses to peroxynitrite in the hindlimb vascular bed of the cat.
Topics: 3',5'-Cyclic-GMP Phosphodiesterases; Adamantane; Animals; Cats; Female; Hindlimb; Male; Meclofenamic Acid; Morpholines; NG-Nitroarginine Methyl Ester; Nitrates; Nitric Oxide Donors; Perfusion; Peroxynitrous Acid; Phosphodiesterase Inhibitors; Potassium Channel Blockers; Purinones; Regional Blood Flow; Rolipram; Sodium Nitrite; Splanchnic Circulation; Vascular Resistance; Vasoconstrictor Agents; Vasodilator Agents | 2007 |
K(ATP) channel expression and pharmacological in vivo and in vitro studies of the K(ATP) channel blocker PNU-37883A in rat middle meningeal arteries.
Topics: Adamantane; Animals; ATP-Binding Cassette Transporters; Blotting, Western; Cromakalim; Data Interpretation, Statistical; Diuretics; Guanidines; In Vitro Techniques; KATP Channels; Male; Meningeal Arteries; Microscopy, Video; Morpholines; Multidrug Resistance-Associated Proteins; Pinacidil; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Drug; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sulfonylurea Receptors; Vasodilator Agents | 2008 |
K ATP channels in pig and human intracranial arteries.
Topics: Adamantane; Animals; ATP-Binding Cassette Transporters; Cerebral Arteries; Gene Expression; Humans; KATP Channels; Male; Meningeal Arteries; Middle Aged; Morpholines; Potassium Channel Blockers; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Species Specificity; Sulfonylurea Receptors; Swine | 2008 |
Inhibition of vascular adenosine triphosphate-sensitive potassium channels by sympathetic tone during sepsis.
Topics: Adamantane; Animals; Aorta; Blood Vessels; Ganglionic Blockers; Gene Expression; Male; Mesenteric Arteries; Morpholines; Norepinephrine; Pentolinium Tartrate; Rats; Rats, Wistar; Sepsis; Sodium-Potassium-Exchanging ATPase; Vasodilation | 2012 |
Cardiovascular protection of activating KATP channel during ischemia-reperfusion acidosis.
Topics: Acidosis; Adamantane; Animals; Aorta, Abdominal; Calcium; Dose-Response Relationship, Drug; Glyburide; Hemodynamics; KATP Channels; Morpholines; Muscle, Smooth, Vascular; Rats; Rats, Sprague-Dawley; Reperfusion Injury; Tissue Culture Techniques; Vasodilation | 2012 |
Depolarization potentiates TRAIL-induced apoptosis in human melanoma cells: role for ATP-sensitive K+ channels and endoplasmic reticulum stress.
Topics: Adamantane; Antineoplastic Agents; Apoptosis; Caspase 12; Caspase 3; Caspase 7; Endoplasmic Reticulum Stress; Enzyme Activation; Glyburide; Humans; KATP Channels; Melanocytes; Melanoma; Membrane Potential, Mitochondrial; Membrane Potentials; Morpholines; Potassium; Potassium Channel Blockers; TNF-Related Apoptosis-Inducing Ligand; Tumor Cells, Cultured | 2012 |
Compared effects of inhibition and exogenous administration of hydrogen sulphide in ischaemia-reperfusion injury.
Topics: Acidosis, Lactic; Adamantane; Adenosine Triphosphate; Alkynes; Animals; Cytokines; Disease Models, Animal; Gasotransmitters; Glycine; Hemodynamics; Hydrogen Sulfide; KATP Channels; Male; Mitogen-Activated Protein Kinase 8; Mitogen-Activated Protein Kinase 9; Morpholines; Nitric Oxide Synthase Type II; Nitric Oxide Synthase Type III; Norepinephrine; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Rats, Wistar; Reperfusion Injury; Shock, Hemorrhagic; Sulfides; Up-Regulation; Vasoconstrictor Agents | 2013 |
Molecular analysis of ATP-sensitive K(+) channel subunits expressed in mouse portal vein.
Topics: Adamantane; Animals; Glyburide; Imidazoles; KATP Channels; Male; Mice; Mice, Inbred BALB C; Morpholines; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Patch-Clamp Techniques; Pinacidil; Portal Vein; Real-Time Polymerase Chain Reaction; Sulfonylurea Receptors; Thioamides | 2015 |
Role of ATP-sensitive potassium channels on hypoxic pulmonary vasoconstriction in endotoxemia.
Topics: Adamantane; Animals; Endotoxemia; Hypoxia; KATP Channels; Lung; Male; Mice; Mice, Inbred C57BL; Morpholines; Organ Culture Techniques; Vasoconstriction | 2018 |