Page last updated: 2024-09-03

tyrosyl-prolyl-tryptophyl-glycinamide and naloxonazine

tyrosyl-prolyl-tryptophyl-glycinamide has been researched along with naloxonazine in 2 studies

Compound Research Comparison

Studies
(tyrosyl-prolyl-tryptophyl-glycinamide)
Trials
(tyrosyl-prolyl-tryptophyl-glycinamide)
Recent Studies (post-2010)
(tyrosyl-prolyl-tryptophyl-glycinamide)
Studies
(naloxonazine)
Trials
(naloxonazine)
Recent Studies (post-2010) (naloxonazine)
2500200030

Protein Interaction Comparison

ProteinTaxonomytyrosyl-prolyl-tryptophyl-glycinamide (IC50)naloxonazine (IC50)
Mu-type opioid receptorHomo sapiens (human)0.0072
Delta-type opioid receptorHomo sapiens (human)0.136
Kappa-type opioid receptorHomo sapiens (human)0.085

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fujimura, T; Ito, K; Kawamura, S; Mizoguchi, H; Murayama, K; Nakayama, D; Sakurada, C; Sakurada, S; Sakurada, T; Sato, T; Watanabe, C; Watanabe, H1
Mizoguchi, H; Nakayama, D; Sakurada, S; Sakurada, T; Watanabe, C; Watanabe, H1

Other Studies

2 other study(ies) available for tyrosyl-prolyl-tryptophyl-glycinamide and naloxonazine

ArticleYear
A Tyr-W-MIF-1 analog containing D-Pro2 acts as a selective mu2-opioid receptor antagonist in the mouse.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 312, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Male; Mice; MSH Release-Inhibiting Hormone; Naloxone; Naltrexone; Narcotic Antagonists; Oligopeptides; Receptors, Opioid, mu

2005
A Tyr-W-MIF-1 analog containing D-Pro2 discriminates among antinociception in mice mediated by different classes of mu-opioid receptors.
    European journal of pharmacology, 2007, Jun-01, Volume: 563, Issue:1-3

    Topics: Analgesics, Opioid; Animals; Brain; Disease Models, Animal; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Hot Temperature; Injections, Intraventricular; Male; Mice; MSH Release-Inhibiting Hormone; Naloxone; Narcotic Antagonists; Oligopeptides; Pain; Pain Measurement; Pain Threshold; Reaction Time; Receptors, Opioid, mu; Somatostatin; Time Factors

2007