tyrosyl-prolyl-tryptophyl-glycinamide has been researched along with endomorphin 1 in 5 studies
| Studies (tyrosyl-prolyl-tryptophyl-glycinamide) | Trials (tyrosyl-prolyl-tryptophyl-glycinamide) | Recent Studies (post-2010) (tyrosyl-prolyl-tryptophyl-glycinamide) | Studies (endomorphin 1) | Trials (endomorphin 1) | Recent Studies (post-2010) (endomorphin 1) |
|---|---|---|---|---|---|
| 25 | 0 | 0 | 448 | 2 | 109 |
| Protein | Taxonomy | tyrosyl-prolyl-tryptophyl-glycinamide (IC50) | endomorphin 1 (IC50) |
|---|---|---|---|
| Delta-type opioid receptor | Mus musculus (house mouse) | 0.026 | |
| Mu-type opioid receptor | Rattus norvegicus (Norway rat) | 0.0005 | |
| Mu-type opioid receptor | Homo sapiens (human) | 0.0275 | |
| Mu-type opioid receptor | Mus musculus (house mouse) | 0.0363 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 2 (40.00) | 18.2507 |
| 2000's | 3 (60.00) | 29.6817 |
| 2010's | 0 (0.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Ge, LJ; Hackler, L; Kastin, AJ; Zadina, JE | 1 |
| Harrison, LM; Kastin, AJ; Zadina, JE | 1 |
| Fasold, MB; Horner, KA; Kastin, AJ; Smith, RR; Zadina, JE | 1 |
| Fujimura, T; Ito, K; Mizoguchi, H; Nakayama, D; Sakurada, S; Sakurada, T; Sakurada, W; Sato, T; Sawai, T; Watanabe, H | 1 |
| Mizoguchi, H; Nakayama, D; Sakurada, S; Sakurada, T; Watanabe, C; Watanabe, H | 1 |
5 other study(ies) available for tyrosyl-prolyl-tryptophyl-glycinamide and endomorphin 1
| Article | Year |
|---|---|
A potent and selective endogenous agonist for the mu-opiate receptor.
Topics: Amino Acid Sequence; Analgesics, Opioid; Animals; Brain Chemistry; Cattle; Endorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Mice; MSH Release-Inhibiting Hormone; Oligopeptides; Radioimmunoassay; Receptors, Opioid, mu | 1997 |
Differential effects of endomorphin-1, endomorphin-2, and Tyr-W-MIF-1 on activation of G-proteins in SH-SY5Y human neuroblastoma membranes.
Topics: Cell Membrane; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; MSH Release-Inhibiting Hormone; Narcotic Antagonists; Neuroblastoma; Oligopeptides; Receptors, Opioid; Tumor Cells, Cultured | 1998 |
Saturable brain-to-blood transport of endomorphins.
Topics: Animals; Binding, Competitive; Blood-Brain Barrier; Brain; Calcitonin Gene-Related Peptide; Carrier Proteins; Iodine Radioisotopes; Ligation; Male; Membrane Transport Proteins; Mice; Mice, Inbred ICR; MSH Release-Inhibiting Hormone; Oligopeptides; Pain; Radioligand Assay; Receptors, Opioid, mu; Sciatic Nerve | 2001 |
Involvement of spinal mu1-opioid receptors on the Tyr-d-Arg-Phe-sarcosine-induced antinociception.
Topics: Analgesics; Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Hot Temperature; Hyperalgesia; Injections, Spinal; Male; Mice; MSH Release-Inhibiting Hormone; Oligopeptides; Pain Measurement; Protein Isoforms; Receptors, Opioid, mu; Spinal Cord | 2006 |
A Tyr-W-MIF-1 analog containing D-Pro2 discriminates among antinociception in mice mediated by different classes of mu-opioid receptors.
Topics: Analgesics, Opioid; Animals; Brain; Disease Models, Animal; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Hot Temperature; Injections, Intraventricular; Male; Mice; MSH Release-Inhibiting Hormone; Naloxone; Narcotic Antagonists; Oligopeptides; Pain; Pain Measurement; Pain Threshold; Reaction Time; Receptors, Opioid, mu; Somatostatin; Time Factors | 2007 |