tyrosyl-prolyl-tryptophyl-glycinamide has been researched along with beta-funaltrexamine in 2 studies
Studies (tyrosyl-prolyl-tryptophyl-glycinamide) | Trials (tyrosyl-prolyl-tryptophyl-glycinamide) | Recent Studies (post-2010) (tyrosyl-prolyl-tryptophyl-glycinamide) | Studies (beta-funaltrexamine) | Trials (beta-funaltrexamine) | Recent Studies (post-2010) (beta-funaltrexamine) |
---|---|---|---|---|---|
25 | 0 | 0 | 542 | 1 | 54 |
Protein | Taxonomy | tyrosyl-prolyl-tryptophyl-glycinamide (IC50) | beta-funaltrexamine (IC50) |
---|---|---|---|
Muscarinic acetylcholine receptor M2 | Rattus norvegicus (Norway rat) | 0.082 | |
Prostaglandin G/H synthase 1 | Homo sapiens (human) | 0.082 | |
Delta-type opioid receptor | Mus musculus (house mouse) | 0.082 | |
Kappa-type opioid receptor | Mus musculus (house mouse) | 0.082 | |
Mu-type opioid receptor | Mus musculus (house mouse) | 0.082 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (50.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Gergen, KA; Kastin, AJ; Paul, D; Zadina, JE | 1 |
Fujimura, T; Ito, K; Kawamura, S; Mizoguchi, H; Murayama, K; Nakayama, D; Sakurada, C; Sakurada, S; Sakurada, T; Sato, T; Watanabe, C; Watanabe, H | 1 |
2 other study(ies) available for tyrosyl-prolyl-tryptophyl-glycinamide and beta-funaltrexamine
Article | Year |
---|---|
Intrathecal Tyr-W-MIF-1 produces potent, naloxone-reversible analgesia modulated by alpha 2-adrenoceptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic Uptake Inhibitors; Amino Acid Sequence; Animals; Desipramine; Dose-Response Relationship, Drug; Injections, Spinal; Male; Mice; Molecular Sequence Data; MSH Release-Inhibiting Hormone; Naloxone; Naltrexone; Narcotic Antagonists; Norepinephrine; Receptors, Adrenergic, alpha-2; Yohimbine | 1996 |
A Tyr-W-MIF-1 analog containing D-Pro2 acts as a selective mu2-opioid receptor antagonist in the mouse.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics, Opioid; Animals; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Male; Mice; MSH Release-Inhibiting Hormone; Naloxone; Naltrexone; Narcotic Antagonists; Oligopeptides; Receptors, Opioid, mu | 2005 |