Page last updated: 2024-09-03

tyrosyl-prolyl-leucyl-glycinamide and spiperone

tyrosyl-prolyl-leucyl-glycinamide has been researched along with spiperone in 2 studies

Compound Research Comparison

Studies
(tyrosyl-prolyl-leucyl-glycinamide)
Trials
(tyrosyl-prolyl-leucyl-glycinamide)
Recent Studies (post-2010)
(tyrosyl-prolyl-leucyl-glycinamide)
Studies
(spiperone)
Trials
(spiperone)
Recent Studies (post-2010) (spiperone)
109002,9441385

Protein Interaction Comparison

ProteinTaxonomytyrosyl-prolyl-leucyl-glycinamide (IC50)spiperone (IC50)
Bile salt export pumpHomo sapiens (human)10
D(2) dopamine receptorHomo sapiens (human)0.0008
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)0.097
D(4) dopamine receptorHomo sapiens (human)0.0005
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)0.097
Histamine H1 receptorCavia porcellus (domestic guinea pig)0.097
D(3) dopamine receptorHomo sapiens (human)0.0635
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)0.097
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0001
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.955

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Krowicki, ZK1
Kastin, AJ; Kostrzewa, RM1

Other Studies

2 other study(ies) available for tyrosyl-prolyl-leucyl-glycinamide and spiperone

ArticleYear
Dopamine receptor antagonists block the effect of Tyr-MIF-1 (Tyr-Pro-Leu-Gly-NH2) on the opiate form of footshock-induced analgesia.
    Neuropeptides, 1991, Volume: 19, Issue:4

    Topics: Amino Acid Sequence; Animals; Benzazepines; Dopamine Antagonists; Drug Synergism; Foot; Haloperidol; Hot Temperature; Male; Molecular Sequence Data; MSH Release-Inhibiting Hormone; Naloxone; Pain; Rats; Rats, Inbred Strains; Receptors, Dopamine; Spiperone; Transcutaneous Electric Nerve Stimulation

1991
Tyr-MIF-1 attenuates development of tolerance to spiperone-induced catalepsy in rats.
    Brain research bulletin, 1993, Volume: 31, Issue:6

    Topics: Amino Acid Sequence; Animals; Benzazepines; Catalepsy; Drug Administration Schedule; Drug Tolerance; Male; Molecular Sequence Data; Motor Activity; MSH Release-Inhibiting Hormone; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Spiperone; Stereotyped Behavior

1993