Page last updated: 2024-09-03

tyrosyl-arginyl-phenylalanyl-sarcosine and naloxone

tyrosyl-arginyl-phenylalanyl-sarcosine has been researched along with naloxone in 6 studies

Compound Research Comparison

Studies
(tyrosyl-arginyl-phenylalanyl-sarcosine)
Trials
(tyrosyl-arginyl-phenylalanyl-sarcosine)
Recent Studies (post-2010)
(tyrosyl-arginyl-phenylalanyl-sarcosine)
Studies
(naloxone)
Trials
(naloxone)
Recent Studies (post-2010) (naloxone)
150120,1341,2573,321

Protein Interaction Comparison

ProteinTaxonomytyrosyl-arginyl-phenylalanyl-sarcosine (IC50)naloxone (IC50)
Cytochrome P450 2D6Homo sapiens (human)2
Delta-type opioid receptorMus musculus (house mouse)0.043
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0219
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0019
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0019
Mu-type opioid receptorHomo sapiens (human)0.0397
Delta-type opioid receptorHomo sapiens (human)0.1896
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.05
Kappa-type opioid receptorHomo sapiens (human)0.0795
Mu-type opioid receptorMus musculus (house mouse)0.0154
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0089
Beta-2 adrenergic receptorCavia porcellus (domestic guinea pig)0.0055

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (50.00)18.2507
2000's3 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Feuerstein, G; Paakkari, I; Paakkari, P1
Búzás, B; Cox, BM; Izenwasser, S1
Feuerstein, G; Paakkari, I; Paakkari, P; Sirén, AL; Vonhof, S1
Cheong, YP; Cho, KP; Kim, CJ; Kim, JK; Kim, KW; Kwun, J; Woo, RS1
Barone, FC; Feuerstein, GZ; Millison, JH; Paakkari, P; Price, WJ; Sirén, AK; Vonhof, S1
Gudka, BD; Sirén, AL; Vonhof, S1

Other Studies

6 other study(ies) available for tyrosyl-arginyl-phenylalanyl-sarcosine and naloxone

ArticleYear
Dermorphin tetrapeptide analog induces naloxonazine-reversible respiratory stimulation.
    Progress in clinical and biological research, 1990, Volume: 328

    Topics: Analgesics; Animals; Naloxone; Oligopeptides; Rats; Rats, Inbred Strains; Receptors, Opioid; Receptors, Opioid, mu; Respiration; Tidal Volume

1990
Differential regulation of adenylyl cyclase activity by mu and delta opioids in rat caudate putamen and nucleus accumbens.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 267, Issue:1

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Benzeneacetamides; Caudate Nucleus; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalins; Male; Molecular Sequence Data; Naloxone; Naltrexone; Nucleus Accumbens; Oligopeptides; Putamen; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, delta; Receptors, Opioid, mu; Signal Transduction; Somatostatin

1993
Dermorphin analog Tyr-D-Arg2-Phe-sarcosine-induced opioid analgesia and respiratory stimulation: the role of mu 1-receptors?
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:2

    Topics: Amino Acid Sequence; Analgesics; Animals; Catalepsy; Dose-Response Relationship, Drug; Male; Molecular Sequence Data; Naloxone; Oligopeptides; Opioid Peptides; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Respiration

1993
Receptor selectivity of Met-enkephalin-Arg6-Phe7, an endogenous opioid peptide, in cerebral cortex of human and rat.
    Life sciences, 2000, May-26, Volume: 67, Issue:1

    Topics: Adult; Animals; Benzeneacetamides; Benzomorphans; Binding Sites; Cerebral Cortex; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Methionine; Ethylketocyclazocine; Female; Humans; Male; Naloxone; Naltrexone; Norepinephrine; Oligopeptides; Peptide Fragments; Peptides; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Somatostatin

2000
Receptor binding and biological activity of the dermorphin analog Tyr-D-Arg(2)-Phe-Sar (TAPS).
    European journal of pharmacology, 2001, Mar-23, Volume: 416, Issue:1-2

    Topics: Analgesics; Animals; Binding, Competitive; Catalepsy; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Injections, Spinal; Male; Muscle Contraction; Naloxone; Nociceptors; Oligopeptides; Opioid Peptides; Pulmonary Ventilation; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Time Factors

2001
Tolerance and dependence following chronic intracerebroventricular infusions of Tyr-D-Arg2-Phe-Sar4 (TAPS).
    European journal of pharmacology, 2003, Jan-10, Volume: 459, Issue:1

    Topics: Analgesics, Opioid; Animals; Dose-Response Relationship, Drug; Drug Tolerance; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; In Vitro Techniques; Infusion Pumps; Injections, Intraventricular; Male; Morphine; Naloxone; Oligopeptides; Pain; Rats; Rats, Sprague-Dawley; Substance Withdrawal Syndrome; Substance-Related Disorders; Time Factors

2003