Page last updated: 2024-09-03

tyrosyl-arginyl-phenylalanyl-sarcosine and fentanyl

tyrosyl-arginyl-phenylalanyl-sarcosine has been researched along with fentanyl in 1 studies

Compound Research Comparison

Studies
(tyrosyl-arginyl-phenylalanyl-sarcosine)
Trials
(tyrosyl-arginyl-phenylalanyl-sarcosine)
Recent Studies (post-2010)
(tyrosyl-arginyl-phenylalanyl-sarcosine)
Studies
(fentanyl)
Trials
(fentanyl)
Recent Studies (post-2010) (fentanyl)
150115,2884,3104,483

Protein Interaction Comparison

ProteinTaxonomytyrosyl-arginyl-phenylalanyl-sarcosine (IC50)fentanyl (IC50)
ATP-dependent translocase ABCB1Homo sapiens (human)6.5
Delta-type opioid receptorMus musculus (house mouse)0.6342
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0122
Mu-type opioid receptorRattus norvegicus (Norway rat)0.1888
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.0122
Mu-type opioid receptorHomo sapiens (human)0.0058
Delta-type opioid receptorHomo sapiens (human)0.3092
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)5.893
Kappa-type opioid receptorHomo sapiens (human)1.58
Mu-type opioid receptorCavia porcellus (domestic guinea pig)0.0031
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.8197
Sigma non-opioid intracellular receptor 1Cavia porcellus (domestic guinea pig)4.973
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.354

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lambert, DG; Smart, D1

Other Studies

1 other study(ies) available for tyrosyl-arginyl-phenylalanyl-sarcosine and fentanyl

ArticleYear
Tyr-D-Arg2-Phe-sarcosine4 activates phospholipase C-coupled mu2-opioid receptors in SH-SY5Y cells.
    European journal of pharmacology, 1996, Jun-03, Volume: 305, Issue:1-3

    Topics: Analgesics; Analgesics, Opioid; Cyclic AMP; Fentanyl; Humans; Inositol 1,4,5-Trisphosphate; Neuroblastoma; Oligopeptides; Receptors, Opioid, mu; Second Messenger Systems; Tumor Cells, Cultured; Type C Phospholipases

1996