Page last updated: 2024-09-03

tyrosyl-arginyl-phenylalanyl-lysinamide and u-50488

tyrosyl-arginyl-phenylalanyl-lysinamide has been researched along with u-50488 in 2 studies

Compound Research Comparison

Studies
(tyrosyl-arginyl-phenylalanyl-lysinamide)
Trials
(tyrosyl-arginyl-phenylalanyl-lysinamide)
Recent Studies (post-2010)
(tyrosyl-arginyl-phenylalanyl-lysinamide)
Studies
(u-50488)
Trials
(u-50488)
Recent Studies (post-2010) (u-50488)
740171,6643209

Protein Interaction Comparison

ProteinTaxonomytyrosyl-arginyl-phenylalanyl-lysinamide (IC50)u-50488 (IC50)
Delta-type opioid receptorRattus norvegicus (Norway rat)2.15
Kappa-type opioid receptorMus musculus (house mouse)0.0027
Mu-type opioid receptorRattus norvegicus (Norway rat)2.15
Kappa-type opioid receptorRattus norvegicus (Norway rat)0.7171
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)0.0958
Kappa-type opioid receptorHomo sapiens (human)0.0537

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kudernatsch, MB; Schlösser, B; Sutor, B; ten Bruggencate, G1
Fasolo, J; Soong, Y; Szeto, HH; Wu, D1

Other Studies

2 other study(ies) available for tyrosyl-arginyl-phenylalanyl-lysinamide and u-50488

ArticleYear
Delta, mu and kappa opioid receptor agonists inhibit dopamine overflow in rat neostriatal slices.
    Neuroscience letters, 1995, May-19, Volume: 191, Issue:1-2

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Dopamine; Dopamine Uptake Inhibitors; Electric Stimulation; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; In Vitro Techniques; Male; Neostriatum; Nomifensine; Oligopeptides; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu

1995
Resensitization of blood pressure response to mu-opioid peptide agonists after acute desensitization.
    Anesthesia and analgesia, 2001, Volume: 93, Issue:3

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Blood Pressure; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Female; Oligopeptides; Opioid Peptides; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sheep

2001