tyrosyl-arginyl-phenylalanyl-lysinamide has been researched along with u-50488 in 2 studies
Studies (tyrosyl-arginyl-phenylalanyl-lysinamide) | Trials (tyrosyl-arginyl-phenylalanyl-lysinamide) | Recent Studies (post-2010) (tyrosyl-arginyl-phenylalanyl-lysinamide) | Studies (u-50488) | Trials (u-50488) | Recent Studies (post-2010) (u-50488) |
---|---|---|---|---|---|
74 | 0 | 17 | 1,664 | 3 | 209 |
Protein | Taxonomy | tyrosyl-arginyl-phenylalanyl-lysinamide (IC50) | u-50488 (IC50) |
---|---|---|---|
Delta-type opioid receptor | Rattus norvegicus (Norway rat) | 2.15 | |
Kappa-type opioid receptor | Mus musculus (house mouse) | 0.0027 | |
Mu-type opioid receptor | Rattus norvegicus (Norway rat) | 2.15 | |
Kappa-type opioid receptor | Rattus norvegicus (Norway rat) | 0.7171 | |
Kappa-type opioid receptor | Cavia porcellus (domestic guinea pig) | 0.0958 | |
Kappa-type opioid receptor | Homo sapiens (human) | 0.0537 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 1 (50.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Kudernatsch, MB; Schlösser, B; Sutor, B; ten Bruggencate, G | 1 |
Fasolo, J; Soong, Y; Szeto, HH; Wu, D | 1 |
2 other study(ies) available for tyrosyl-arginyl-phenylalanyl-lysinamide and u-50488
Article | Year |
---|---|
Delta, mu and kappa opioid receptor agonists inhibit dopamine overflow in rat neostriatal slices.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Dopamine; Dopamine Uptake Inhibitors; Electric Stimulation; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine-2-Alanine; Enkephalins; In Vitro Techniques; Male; Neostriatum; Nomifensine; Oligopeptides; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu | 1995 |
Resensitization of blood pressure response to mu-opioid peptide agonists after acute desensitization.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Blood Pressure; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Female; Oligopeptides; Opioid Peptides; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Sheep | 2001 |