Page last updated: 2024-09-03

tyrosyl-arginyl-phenylalanyl-lysinamide and norbinaltorphimine

tyrosyl-arginyl-phenylalanyl-lysinamide has been researched along with norbinaltorphimine in 2 studies

Compound Research Comparison

Studies
(tyrosyl-arginyl-phenylalanyl-lysinamide)
Trials
(tyrosyl-arginyl-phenylalanyl-lysinamide)
Recent Studies (post-2010)
(tyrosyl-arginyl-phenylalanyl-lysinamide)
Studies
(norbinaltorphimine)
Trials
(norbinaltorphimine)
Recent Studies (post-2010) (norbinaltorphimine)
740179180205

Protein Interaction Comparison

ProteinTaxonomytyrosyl-arginyl-phenylalanyl-lysinamide (IC50)norbinaltorphimine (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.0104
Kappa-type opioid receptorMus musculus (house mouse)0.0029
Mu-type opioid receptorHomo sapiens (human)0.212
Delta-type opioid receptorHomo sapiens (human)0.024
Kappa-type opioid receptorHomo sapiens (human)0.0036

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Maslov, LN; Naryzhnaya, NV; Tam, SW1
Neilan, CL; Nguyen, TM; Pasternak, GW; Schiller, PW1

Other Studies

2 other study(ies) available for tyrosyl-arginyl-phenylalanyl-lysinamide and norbinaltorphimine

ArticleYear
Ligands for opioid and sigma-receptors improve cardiac electrical stability in rat models of post-infarction cardiosclerosis and stress.
    Life sciences, 1999, Volume: 65, Issue:1

    Topics: Animals; Anti-Arrhythmia Agents; beta-Endorphin; Disease Models, Animal; Dynorphins; Enkephalin, Leucine-2-Alanine; Heart; Immobilization; Ligands; Morphine; Myocardial Infarction; Myocardium; Naloxone; Naltrexone; Narcotic Antagonists; Oligopeptides; Piperidines; Pyrrolidines; Rats; Receptors, Opioid; Receptors, Opioid, delta; Stress, Physiological; Ventricular Fibrillation

1999
Pharmacological characterization of the dermorphin analog [Dmt(1)]DALDA, a highly potent and selective mu-opioid peptide.
    European journal of pharmacology, 2001, May-04, Volume: 419, Issue:1

    Topics: Analgesics; Animals; Drug Tolerance; Humans; Mice; Morphine; Naloxone; Naltrexone; Narcotic Antagonists; Oligodeoxyribonucleotides, Antisense; Oligopeptides; Opioid Peptides; Pain Measurement; Receptors, Opioid, mu; Time Factors

2001