tubercidin and adenosine kinase
tubercidin has been researched along with adenosine kinase in 95 studies
Research
Studies (95)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 24 (25.26) | 18.7374 |
1990's | 36 (37.89) | 18.2507 |
2000's | 25 (26.32) | 29.6817 |
2010's | 9 (9.47) | 24.3611 |
2020's | 1 (1.05) | 2.80 |
Authors
Authors | Studies |
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Gupta, RS; Siminovitch, L | 1 |
Townsend, LB; Wotring, LL | 1 |
Berne, RM; Coleman, SD; Ely, SW; Matherne, GP | 1 |
Duley, JA; Montero, C; Simmonds, HA; Smolenski, RT | 1 |
de Jong, JW; Den Boer, PJ; Grootegoed, JA; Mackenbach, P | 1 |
Bontemps, F; van den Berghe, G | 1 |
Kather, H | 1 |
Barankiewicz, J; Gruber, HE; Jimenez, R; Ronlov, G | 1 |
Meghji, P; Middleton, KM; Newby, AC | 1 |
Bhaumik, D; Datta, AK | 1 |
Gupta, RS; Mehta, KD | 5 |
Gupta, RS; Singh, B; Stetsko, DK | 1 |
Fox, IH; Hurley, MC; Lin, B | 1 |
Baird-Lambert, J; Davies, LP; Marwood, JF | 1 |
Allan, PW; Bennett, LL; Brockman, RW; Rose, LM; Shaddix, SC | 1 |
Basuyau, JP; Chedeville, A; Claeyssens, S; Hamet, M; Lavoinne, A | 1 |
Dovey, HF; McKerrow, JH; Wang, CC | 1 |
Berens, RL; LaFon, SW; Marr, JJ; Nelson, DJ | 1 |
Holmquist, CA; Newby, AC | 1 |
Dalke, P; Lyda, TS; Magill, CW; Magill, JM | 1 |
Plagemann, PG; Wohlhueter, RM | 2 |
Lobelle-Rich, PA; Reeves, RE | 1 |
Baird-Lambert, JA; Davies, LP; Jamieson, DD; Kazlauskas, R | 1 |
Cass, CE; Phillips, JR; Selner, M | 1 |
Holmquist, CA; Illingworth, J; Newby, AC; Pearson, JD | 1 |
Hori, M; Inoue, M; Kamada, T; Kitakaze, M; Komamura, K; Minamino, T; Node, K; Takeda, H | 1 |
Corsi, C; Fratti, S; Pazzagli, M; Pedata, F; Pepeu, G | 1 |
Fredholm, BB; Lloyd, HG | 1 |
el Kouni, MH; Iltzsch, MH; Tankersley, KO; Uber, SS | 1 |
Decking, UK; Haas, HL; Pak, MA; Schrader, J | 1 |
Bullough, DA; Montag, A; Mullane, KM; Young, MA; Zhang, C | 1 |
Bollen, M; Massillon, D; Stalmans, W; van de Werve, G | 1 |
Carson, DA; Cottam, HB; Di Pasquale, G; Raychaudhuri, A; Shih, HC; Wasson, DB | 1 |
Phillis, JW; Smith-Barbour, M | 1 |
Bontemps, F; Van den Berghe, G; Vincent, MF | 1 |
Sciotti, VM; Van Wylen, DG | 1 |
Bading, B; Deussen, A; Kelm, M; Schrader, J | 1 |
Flückiger-Isler, RE; Walter, P | 1 |
Geiger, JD; Parkinson, FE | 1 |
Hrnjez, BJ; Matthews, JB; Mun, EC; Smith, JA; Tally, KJ | 1 |
Gupta, RS | 1 |
Golembiowska, K; Sawynok, J; White, TD | 1 |
Cook, AF; Davies, LP | 1 |
Kroll, K; Stepp, DW | 1 |
DaRe, J; Foster, AC; Jelovich, LA; Miller, LP; Ugarkar, B; Yao, L | 1 |
Chopp, M; Jiang, N; Kowaluk, EA; Lee, CH; Mazdiyasni, H | 1 |
Dubey, RK; Gillespie, DG; Jackson, EK; Mi, Z | 1 |
Kalsi, KK; Kochan, Z; Smolenski, RT; Yacoub, MH; Zych, M | 1 |
Manthei, SA; Reiling, CM; Van Wylen, DG | 1 |
Hebb, MO; White, TD | 1 |
Gordon, PB; Grotterød, EM; Kovács, AL; Seglen, PO | 1 |
Jarvis, MF; Kowaluk, EA; Lynch, JJ | 1 |
Deussen, A; Kelm, M; Schäfer, S; Stappert, M | 1 |
Barankiewicz, J; Castellino, AJ; Dumas, DP; Erion, MD; Foster, AC; Gruber, HE; Ugarkar, BG; Wiesner, JB | 1 |
Britton, DR; Jarvis, MF; Kowaluk, EA; Lee, CH; Mikusa, J; Williams, M | 1 |
Dubey, RK; Gillespie, DG; Jackson, EK; Shue, H | 1 |
Brennan, RG; Ealick, SE; Mathews, II; Roos, DS; Schumacher, MA; Scott, DM; Ullman, B | 2 |
Abbracchio, MP; Camurri, A; Ceruti, S; Falzano, L; Fiorentini, C; Frank, C; Giammarioli, AM; Malorni, W; Rufini, S | 1 |
Browne, CE; DaRe, JM; Erion, MD; Kopcho, JJ; Schanzer, JM; Ugarkar, BG; Wiesner, JB | 1 |
Castellino, AJ; DaRe, JM; Erion, MD; Kopcho, JJ; Schanzer, JM; Ugarkar, BG; Wiesner, JB | 1 |
Gołembiowska, K; Zylewska, A | 1 |
Cerniway, RJ; Headrick, JP; Matherne, GP; Peart, J | 1 |
Baldwin, SA; Cass, CE; LaRivière, CG; Parkinson, FE; Powell, AE; Sinclair, CJ; Xiong, W; Young, JD | 1 |
Gray, CC; Kalsi, KK; Kochan, Z; Smolenski, RT; Yacoub, MH; Zych, M | 1 |
Cioroch, M; Makarewicz, W; Skladanowski, AC; Tkacz, K | 1 |
Benton, HP; Kollias-Baker, C; MacDonald, MH; Tesch, AM | 1 |
Kumar, R; Sharma, BK; Singh, P | 1 |
Boison, D; Fritschy, JM; Gouder, N; Scheurer, L | 1 |
Benton, HP; MacDonald, MH; Petrov, R; Tesch, AM | 1 |
Boison, D; Crestani, F; Fedele, DE; Gabernet, L; Gouder, N; Güttinger, M; Rülicke, T; Scheurer, L | 1 |
Boyer, SH; Erion, MD; Gomez-Galeno, JE; Kopcho, J; Matelich, MC; Mendonca, R; Nagahisa, A; Nakane, M; Ollis, K; Solbach, J; Tsuchiya, M; Ugarkar, BG; Wiesner, JB | 1 |
Chambers, MG; Mason, RM; Mistry, D | 1 |
Boison, D; Pignataro, G; Simon, RP | 1 |
Allan, PW; Liu, MC; Long, MC; Luo, MZ; Parker, WB; Sartorelli, AC | 1 |
Bhagwat, SS; Cowart, MD; Gomtsyan, A; Jakob, CL; Jarvis, MF; Kowaluk, EA; Lee, CH; Matulenko, MA; Muchmore, SW; Severin, JM; Smith, RA; Stewart, AO; Yu, H | 1 |
Brdar, B; Reich, E | 1 |
Carneiro, FS; Carneiro, ZN; Giachini, FRC; Inscho, EW; Leite, R; Lima, VV; Tostes, RC; Webb, RC | 1 |
Cho, CY; Geierstanger, BH; Ginsberg, MH; Goldfinger, LE; Hong, J; Lee, J; Nam, TG; Orth, AP; Peters, EC; Schultz, PG | 1 |
Boison, D; Dale, N; Etherington, LA; Frenguelli, BG; Irving, AJ; Meechan, L; Patterson, GE | 1 |
Boison, D; Li, T; Shen, HY | 1 |
Fukuda, M; Hino, H; Ishii, E; Kuzume, K; Morimoto, T; Suzuki, Y | 1 |
Bhutoria, S; Ghoshal, N | 1 |
Agarwal, T; Cui, XA; Gupta, RS; Singh, B | 1 |
Birkus, G; Bourderioux, A; Cihlar, T; Dzubák, P; Feng, JY; Hajdúch, M; Hocek, M; Konecný, P; Naus, P; Perlíková, P; Pichová, I; Pohl, R; Ray, AS; Stray, KM; Votruba, I; Wang, T | 1 |
Boison, D; Granja, TF; Köhler, D; Morote-García, JC; Rosenberger, P; Schneider, M; Straub, A; Streienberger, A | 1 |
Boison, D; Ciancetta, A; Jacobson, KA; Osborne, D; Toti, KS | 1 |
Acharya, MM; Allen, BD; Baddour, AA; Baulch, JE; Giedzinski, E; Kawashita, T; Nguyen, TH; Parihar, VK; Syage, AR; Yoon, N; Yu, L | 1 |
Bigej, R; Boison, D; Friedman, JL; Saleumvong, B; Sandau, US; Yahya, M | 1 |
Ashraf, O; Boison, D; Chitravanshi, V; Fedele, DE; Huynh, T; Murugan, M; Purnell, BS | 1 |
Other Studies
95 other study(ies) available for tubercidin and adenosine kinase
Article | Year |
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Genetic and biochemical studies with the adenosine analogs toyocamycin and tubercidin: mutation at the adenosine kinase locus in Chinese hamster cells.
Topics: Adenosine Kinase; Animals; Antibiotics, Antineoplastic; Cell Line; Cricetinae; Cricetulus; Drug Resistance; Female; Mutation; Ovary; Phenotype; Phosphotransferases; Ribonucleosides; Toyocamycin; Tubercidin | 1978 |
Study of the cytotoxicity and metabolism of 4-amino-3-carboxamido-1-(beta-D-ribofuranosyl)pyrazolo[3,4-d]pyrimidine using inhibitors of adenosine kinase and adenosine deaminase.
Topics: Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Cell Survival; Cells, Cultured; Enzyme Inhibitors; Leukemia L1210; Mice; Nucleoside Deaminases; Phosphotransferases; Ribonucleosides; Tubercidin | 1979 |
Inhibition of adenosine metabolism increases myocardial interstitial adenosine concentrations and coronary flow.
Topics: Adenine; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Coronary Circulation; Extracellular Space; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Myocardium; Perfusion; Tubercidin; Vascular Resistance | 1992 |
Effects of adenosine analogues on ATP concentrations in human erythrocytes. Further evidence for a route independent of adenosine kinase.
Topics: Adenine Phosphoribosyltransferase; Adenosine Kinase; Adenosine Triphosphate; Erythrocytes; Humans; Hypoxanthine; Hypoxanthines; Pentostatin; Tubercidin | 1991 |
Effects of glucose and adenosine on the ATP content of hamster spermatids.
Topics: Adenine; Adenosine; Adenosine Kinase; Adenosine Triphosphate; Animals; Cricetinae; Cyclic AMP; Dipyridamole; Dose-Response Relationship, Drug; Fructose; Galactose; Glucose; Hypoxanthine; Hypoxanthines; In Vitro Techniques; Male; Mannose; Spermatids; Tubercidin | 1990 |
Adenine nucleotide catabolism in human erythrocytes: pathways and regulation.
Topics: Adenine Nucleotides; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Adenosine Monophosphate; Erythrocytes; Humans; Hydrolysis; Hypoxanthines; Kinetics; Nucleotidases; Pentostatin; Phosphorylation; Tubercidin | 1990 |
Pathways of purine metabolism in human adipocytes. Further evidence against a role of adenosine as an endogenous regulator of human fat cell function.
Topics: Adenosine; Adenosine Deaminase Inhibitors; Adenosine Diphosphate; Adenosine Kinase; Adenosine Monophosphate; Adenosine Triphosphate; Adipose Tissue; Glycerophosphates; Humans; Hypoxanthine; Hypoxanthines; Inosine; Inosine Monophosphate; Isoproterenol; Lipolysis; Pentostatin; Purines; Tubercidin | 1990 |
Selective adenosine release from human B but not T lymphoid cell line.
Topics: Adenosine; Adenosine Kinase; Adenosine Triphosphate; Animals; B-Lymphocytes; Cell Line; Deoxyglucose; Hypoxanthine; Hypoxanthines; Inosine; Kinetics; Models, Biological; Pentostatin; Rats; T-Lymphocytes; Tubercidin | 1990 |
Absolute rates of adenosine formation during ischaemia in rat and pigeon hearts.
Topics: 5'-Nucleotidase; Adenine; Adenosine; Adenosine Deaminase; Adenosine Kinase; Adult; AMP Deaminase; Animals; Columbidae; Coronary Disease; Female; Heart; Histocytochemistry; Humans; Male; Middle Aged; Myocardium; Nucleotidases; Nucleotides; Phosphoric Monoester Hydrolases; Rats; Rats, Inbred Strains; Species Specificity; Tubercidin | 1988 |
Reaction kinetics and inhibition of adenosine kinase from Leishmania donovani.
Topics: Adenosine; Adenosine Diphosphate; Adenosine Kinase; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Kinetics; Leishmania donovani; Methylthioinosine; Phosphotransferases; Substrate Specificity; Tubercidin | 1988 |
Involvement of adenosine kinase in the phosphorylation of formycin B in CHO cells.
Topics: Adenosine; Adenosine Kinase; Amides; Animals; Antibiotics, Antineoplastic; Cell Line; Cricetinae; Drug Resistance; Female; Formycins; Methylthioinosine; Mutation; Ovary; Phosphorylation; Phosphotransferases; Pyrazoles; Ribonucleosides; Ribose; Toyocamycin; Tubercidin | 1985 |
Inhibition of metabolic cooperation by phorbol esters in a cell culture system based on adenosine kinase deficient mutants of V79 cells.
Topics: Adenosine; Adenosine Kinase; Animals; Cell Communication; Cell Count; Cell Line; Cricetinae; Cricetulus; Diphtheria Toxin; Dose-Response Relationship, Drug; Drug Resistance; Mutation; Peptide Elongation Factor 2; Peptide Elongation Factors; Phorbol Esters; Phorbols; Phosphorylation; Phosphotransferases; Tetradecanoylphorbol Acetate; Tubercidin | 1985 |
Regulation of deoxyadenosine and nucleoside analog phosphorylation by human placental adenosine kinase.
Topics: Adenosine Diphosphate; Adenosine Kinase; Adenosine Monophosphate; Adenosine Triphosphate; Deoxyadenosines; Female; Humans; Hydrogen-Ion Concentration; Kinetics; Methylthioinosine; Nucleosides; Nucleotides; Phosphorylation; Phosphotransferases; Placenta; Potassium Chloride; Pregnancy; Tubercidin; Vidarabine | 1985 |
Novel mutants of CHO cells resistant to adenosine analogs and containing biochemically altered form of adenosine kinase in cell extracts.
Topics: Adenosine; Adenosine Kinase; Animals; Antibiotics, Antineoplastic; Cell Line; Cricetinae; Cricetulus; Drug Resistance; Formycins; Genetic Markers; Hybrid Cells; Mutation; Phenotype; Phosphorylation; Phosphotransferases; Tubercidin | 1986 |
Immunological studies with different classes of mutants affected at the adenosine kinase locus in CHO cells.
Topics: Adenosine Kinase; Amides; Animals; Antibody Specificity; Cell Line; Cricetinae; Cricetulus; Cross Reactions; Drug Resistance; Female; Formycins; Immunosorbent Techniques; Methylthioinosine; Mutation; Ovary; Phosphotransferases; Pyrazoles; Ribonucleosides; Ribose; Toyocamycin; Tubercidin | 1986 |
Studies on several pyrrolo[2,3-d]pyrimidine analogues of adenosine which lack significant agonist activity at A1 and A2 receptors but have potent pharmacological activity in vivo.
Topics: Adenosine; Adenosine Deaminase; Adenosine Kinase; Adenosine-5'-(N-ethylcarboxamide); Animals; Blood Pressure; Brain; Cyclic AMP; Guanosine; Guinea Pigs; Heart Rate; Male; Mice; Muscle Relaxation; Phenylisopropyladenosine; Receptors, Cell Surface; Receptors, Purinergic; Tubercidin | 1986 |
Genetic and biochemical characteristics of three different types of mutants of mammalian cells affected in adenosine kinase.
Topics: Adenosine; Adenosine Kinase; Animals; Binding, Competitive; Biological Transport; Cell Line; Cricetinae; Cross Reactions; Drug Resistance; Formycins; Mutation; Phosphotransferases; Purine Nucleosides; Structure-Activity Relationship; Tubercidin | 1986 |
Alterations in nucleotide pools induced by 3-deazaadenosine and related compounds. Role of adenylate deaminase.
Topics: Adenine; Adenosine Kinase; Alanine; Aminoglycosides; AMP Deaminase; Animals; Anti-Bacterial Agents; Cell Survival; Coformycin; Hypoxanthine; Hypoxanthines; Mice; Nucleotide Deaminases; Nucleotides; Time Factors; Tubercidin | 1988 |
Influence of 2-chloroadenosine on the nucleotide content of isolated rat hepatocytes.
Topics: 2-Chloroadenosine; Adenosine; Adenosine Diphosphate; Adenosine Kinase; Adenosine Triphosphate; Animals; Chromatography, High Pressure Liquid; Kinetics; Liver; Male; Nucleotides; Phosphorylation; Piperazines; Rats; Rats, Inbred Strains; Spectrophotometry; Tubercidin | 1988 |
Action of tubercidin and other adenosine analogs on Schistosoma mansoni schistosomules.
Topics: Adenosine; Adenosine Kinase; Adenosine Monophosphate; Animals; Antibiotics, Antineoplastic; Formycins; Movement; Nucleotides; Purine-Nucleoside Phosphorylase; Ribonucleosides; Schistosoma mansoni; Substrate Specificity; Tubercidin; Vidarabine | 1985 |
Inosine analogs. Their metabolism in mouse L cells and in Leishmania donovani.
Topics: Adenosine Kinase; Adenosine Triphosphate; Animals; Cell Line; Chromatography, High Pressure Liquid; Enzyme Inhibitors; Fibroblasts; Guanosine Triphosphate; Inosine; Inosine Triphosphate; Leishmania; Mice; Tubercidin | 1985 |
Adenosine production inside rat polymorphonuclear leucocytes.
Topics: 5'-Nucleotidase; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Chromatography, High Pressure Liquid; Coformycin; Neutrophils; Nucleotidases; Pentostatin; Rats; Tubercidin | 1981 |
Adenosine kinase-deficient mutant of Neurospora crassa.
Topics: Adenosine; Adenosine Kinase; Kinetics; Mutation; Neurospora; Neurospora crassa; Phosphotransferases; Purine Nucleosides; Purine Nucleotides; Tubercidin | 1982 |
Adenosine metabolism in wild-type and enzyme-deficient variants of Chinese hamster ovary and Novikoff rat hepatoma cells.
Topics: 2-Aminopurine; Adenine Nucleotides; Adenosine; Adenosine Kinase; Animals; Cell Division; Cell Line; Cell-Free System; Coformycin; Cricetinae; Female; Kinetics; Liver Neoplasms, Experimental; Ovary; Pentostatin; Phosphorylation; Phosphotransferases; Purine-Nucleoside Phosphorylase; Rats; Tubercidin | 1983 |
Formycin B-resistant mutants of Chinese hamster ovary cells: novel genetic and biochemical phenotype affecting adenosine kinase.
Topics: Adenosine; Adenosine Kinase; Animals; Antibiotics, Antineoplastic; Biological Transport; Cell Line; Cells, Cultured; Cricetinae; Drug Resistance; Formycins; Mutation; Phosphotransferases; Toyocamycin; Tubercidin | 1983 |
The partial purification and characterization of adenosine kinase from Entamoeba histolytica.
Topics: Adenosine; Adenosine Kinase; Adenosine Triphosphate; Animals; Chromatography, Affinity; Entamoeba histolytica; Glycerol; Kinetics; Phosphotransferases; Substrate Specificity; Tubercidin; Vidarabine | 1983 |
Halogenated pyrrolopyrimidine analogues of adenosine from marine organisms: pharmacological activities and potent inhibition of adenosine kinase.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenine; Adenosine; Adenosine Kinase; Adenylyl Cyclases; Animals; Brain; Bronchodilator Agents; Cardiovascular System; Central Nervous System; Guinea Pigs; In Vitro Techniques; Male; Marine Biology; Mice; Phosphotransferases; Rats; Ribonucleosides; Theophylline; Tubercidin | 1984 |
Resistance to 9-beta-D-arabinofuranosyladenine in cultured leukemia L 1210 cells.
Topics: Adenosine Kinase; Animals; Cell Division; Coformycin; DNA Replication; Drug Resistance; Leukemia L1210; Mice; Pentostatin; Tubercidin; Vidarabine | 1983 |
The control of adenosine concentration in polymorphonuclear leucocytes, cultured heart cells and isolated perfused heart from the rat.
Topics: Adenosine; Adenosine Kinase; Animals; Cells, Cultured; Coformycin; Heart; In Vitro Techniques; Male; Myocardium; Neutrophils; Pentostatin; Perfusion; Rats; Rats, Inbred Strains; Tubercidin | 1983 |
Adenosine and tubercidin binding and transport in Chinese hamster ovary and Novikoff rat hepatoma cells.
Topics: Adenosine; Adenosine Kinase; Animals; Biological Transport; Cell Line; Cricetinae; Female; Kinetics; Liver Neoplasms, Experimental; Ovary; Phosphorylation; Rats; Ribonucleosides; Thymidine; Tubercidin; Uridine | 1983 |
Activation of protein kinase C increases adenosine production in the hypoxic canine coronary artery through the extracellular pathway.
Topics: 5'-Nucleotidase; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Arteries; Coronary Vessels; Dogs; Enzyme Activation; Hypoxia; In Vitro Techniques; Pentostatin; Protein Kinase C; Tubercidin | 1995 |
Regulation of extracellular adenosine levels in the striatum of aging rats.
Topics: 2-Amino-5-phosphonovalerate; Adenine; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Aging; Amino Acids; Animals; Corpus Striatum; Enzyme Inhibitors; Extracellular Space; Male; Microdialysis; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Tubercidin | 1995 |
Involvement of adenosine deaminase and adenosine kinase in regulating extracellular adenosine concentration in rat hippocampal slices.
Topics: Adenine; Adenosine; Adenosine Deaminase; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Basal Metabolism; Electric Stimulation; Hippocampus; In Vitro Techniques; Male; Purines; Rats; Tubercidin | 1995 |
Structure-activity relationship for the binding of nucleoside ligands to adenosine kinase from Toxoplasma gondii.
Topics: Adenosine; Adenosine Kinase; Animals; Antiprotozoal Agents; Drug Design; Ligands; Purine Nucleosides; Structure-Activity Relationship; Toxoplasma; Tubercidin | 1995 |
Inhibition of adenosine kinase increases endogenous adenosine and depresses neuronal activity in hippocampal slices.
Topics: Adenosine; Adenosine Kinase; Animals; Hippocampus; In Vitro Techniques; Inosine; Kinetics; Membrane Potentials; Neurons; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Tubercidin; Xanthines | 1994 |
Adenosine-mediated inhibition of platelet aggregation by acadesine. A novel antithrombotic mechanism in vitro and in vivo.
Topics: Adenosine; Adenosine Deaminase; Adenosine Kinase; Aminoimidazole Carboxamide; Animals; Aspirin; Blood Physiological Phenomena; Coronary Thrombosis; Coronary Vessels; Dipyridamole; Disease Models, Animal; Dogs; Erythrocytes; Humans; Male; Plasma; Platelet Aggregation; Purinergic P1 Receptor Antagonists; Regional Blood Flow; Ribonucleosides; Theophylline; Tubercidin | 1994 |
Identification of the glycogenic compound 5-iodotubercidin as a general protein kinase inhibitor.
Topics: Adenosine Kinase; Animals; Glucagon; Glycogen Synthase; Liver; Male; Peptides; Phosphorylase Kinase; Phosphorylation; Protein Kinase Inhibitors; Rats; Rats, Wistar; Tubercidin; Vasopressins | 1994 |
New adenosine kinase inhibitors with oral antiinflammatory activity: synthesis and biological evaluation.
Topics: Adenosine Kinase; Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Cells, Cultured; Drug Evaluation, Preclinical; Humans; Kinetics; Lymphocytes; Pleurisy; Pyrazoles; Pyridines; Rats; Rats, Sprague-Dawley; Tubercidin | 1993 |
The adenosine kinase inhibitor, 5-iodotubercidin, is not protective against cerebral ischemic injury in the gerbil.
Topics: Adenosine Kinase; Animals; Body Temperature; Brain Ischemia; Gerbillinae; Hippocampus; Male; Motor Activity; Tubercidin | 1993 |
Mechanisms of elevation of adenosine levels in anoxic hepatocytes.
Topics: 5'-Nucleotidase; Adenine Nucleotides; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Amobarbital; Animals; Carbon Dioxide; Cell Membrane; Liver; Male; Nitrogen; Oxygen; Pentostatin; Phosphoric Monoester Hydrolases; Potassium Cyanide; Rats; Rats, Wistar; Tubercidin | 1993 |
Increases in interstitial adenosine and cerebral blood flow with inhibition of adenosine kinase and adenosine deaminase.
Topics: Adenine; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Brain; Cerebrovascular Circulation; Dialysis Solutions; Dose-Response Relationship, Drug; Extracellular Space; Hypoxanthine; Hypoxanthines; Inosine; Male; Rats; Rats, Wistar; Tubercidin | 1993 |
Formation and salvage of adenosine by macrovascular endothelial cells.
Topics: 5'-Nucleotidase; Adenine Nucleotides; Adenosine; Adenosine Deaminase; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Calcimycin; Cells, Cultured; Chromatography, High Pressure Liquid; Endothelium, Vascular; Firefly Luciferin; Kinetics; Luciferases; Microspheres; Phosphorylation; Swine; Tubercidin | 1993 |
Stimulation of rat liver glycogen synthesis by the adenosine kinase inhibitor 5-iodotubercidin.
Topics: 2-Chloroadenosine; Adenosine; Adenosine Kinase; Adenosine Triphosphate; Amino Acids; Animals; Cells, Cultured; Liver; Liver Glycogen; Male; Rats; Rats, Wistar; Tubercidin | 1993 |
Effects of iodotubercidin on adenosine kinase activity and nucleoside transport in DDT1 MF-2 smooth muscle cells.
Topics: Adenosine Kinase; Animals; Cricetinae; Dose-Response Relationship, Drug; Kinetics; Muscle, Smooth; Nucleosides; Radioligand Assay; Tubercidin | 1996 |
Adenosine scavenging: a novel mechanism of chloride secretory control in intestinal epithelial cells.
Topics: Adenosine; Adenosine Kinase; Adenosine Triphosphate; Biological Transport; Buffers; Cells, Cultured; Chlorides; Chromatography, High Pressure Liquid; Cyclic AMP; Dipyridamole; Enzyme Inhibitors; Humans; Intestinal Mucosa; Membrane Proteins; Nucleosides; Phosphodiesterase Inhibitors; Phosphorylation; Tubercidin; Vasodilator Agents | 1996 |
Adenosine-AMP exchange activity is an integral part of the mammalian adenosine kinase.
Topics: Adenosine; Adenosine Kinase; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Arsenates; Cattle; CHO Cells; Cricetinae; Enzyme Inhibitors; Enzyme Stability; Kinetics; Liver; Magnesium; Mutation; Phosphates; Temperature; Toyocamycin; Tubercidin | 1996 |
Adenosine kinase inhibitors augment release of adenosine from spinal cord slices.
Topics: Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Deoxyadenosines; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Male; Pentostatin; Rats; Rats, Sprague-Dawley; Spinal Cord; Tubercidin | 1996 |
Inhibition of adenosine kinase and adenosine uptake in guinea-pig CNS tissue by halogenated tubercidin analogues.
Topics: Adenosine; Adenosine Kinase; Animals; Cerebral Cortex; Enzyme Inhibitors; Guinea Pigs; In Vitro Techniques; Tubercidin | 1995 |
Adenosine kinetics in canine coronary circulation.
Topics: Adenosine; Adenosine Kinase; Animals; Biological Transport; Capillaries; Computer Simulation; Coronary Circulation; Dipyridamole; Dogs; Endothelium, Vascular; Female; Hemodynamics; In Vitro Techniques; Indicator Dilution Techniques; Kinetics; Male; Models, Cardiovascular; Nitroglycerin; Tubercidin; Veins | 1996 |
Pre- and peristroke treatment with the adenosine kinase inhibitor, 5'-deoxyiodotubercidin, significantly reduces infarct volume after temporary occlusion of the middle cerebral artery in rats.
Topics: Adenosine Kinase; Animals; Cerebral Arteries; Cerebral Infarction; Cerebrovascular Disorders; Constriction, Pathologic; Male; Rats; Tubercidin | 1996 |
Adenosine kinase inhibition protects brain against transient focal ischemia in rats.
Topics: Adenosine Kinase; Animals; Arterial Occlusive Diseases; Body Temperature; Body Weight; Brain; Cerebral Infarction; Enzyme Inhibitors; Ischemic Attack, Transient; Male; Neuroprotective Agents; Rats; Rats, Wistar; Tubercidin | 1997 |
Exogenous and endogenous adenosine inhibits fetal calf serum-induced growth of rat cardiac fibroblasts: role of A2B receptors.
Topics: Adenine; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Adenosine-5'-(N-ethylcarboxamide); Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Cattle; Cell Division; Culture Media; Dipyridamole; DNA Replication; Enzyme Inhibitors; Fibroblasts; Heart; Male; Myocardium; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Tubercidin; Xanthines | 1997 |
Adenine/ribose supply increases adenosine production and protects ATP pool in adenosine kinase-inhibited cardiac cells.
Topics: Adenine; Adenosine; Adenosine Kinase; Adenosine Triphosphate; Animals; Cells, Cultured; Endothelium, Vascular; Enzyme Inhibitors; Heart; In Vitro Techniques; Kinetics; Male; Myocardium; Purines; Rats; Rats, Sprague-Dawley; Ribose; Tubercidin; Uridine | 1998 |
Dual cardiac microdialysis to assess drug-induced changes in interstitial purine metabolites: adenosine deaminase inhibition versus adenosine kinase inhibition.
Topics: Adenine; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Chromatography, High Pressure Liquid; Extracellular Space; Hypoxanthine; Inosine; Male; Microdialysis; Myocardial Ischemia; Myocardial Reperfusion; Myocardium; Rabbits; Tubercidin | 1998 |
Co-administration of adenosine kinase and deaminase inhibitors produces supra-additive potentiation of N-methyl-D-aspartate-evoked adenosine formation in cortex.
Topics: Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Cerebral Cortex; Deoxyadenosines; Drug Synergism; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Male; N-Methylaspartate; Pentostatin; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Tubercidin | 1998 |
Inhibition of hepatocytic autophagy by adenosine, adenosine analogs and AMP.
Topics: Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Adenosine Monophosphate; Animals; Autophagy; Cells, Cultured; Enzyme Inhibitors; Liver; Male; Pentostatin; Phosphorylation; Rats; Rats, Wistar; Tubercidin | 1998 |
An adenosine kinase inhibitor attenuates tactile allodynia in a rat model of diabetic neuropathic pain.
Topics: Adenosine Kinase; Animals; Anti-Bacterial Agents; Blood Glucose; Body Weight; Diabetes Mellitus, Experimental; Diabetic Neuropathies; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Inhibitors; Male; Morphine; Narcotics; Pain; Pain Threshold; Rats; Rats, Sprague-Dawley; Streptozocin; Theophylline; Tubercidin | 1999 |
Quantification of extracellular and intracellular adenosine production: understanding the transmembranous concentration gradient.
Topics: Adenine; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Biological Transport; Bradykinin; Coronary Circulation; Cytosol; Depression, Chemical; Dipyridamole; Drug Synergism; Enzyme Inhibitors; Extracellular Space; Guinea Pigs; Heart; Models, Biological; Myocardium; Osmolar Concentration; Oxygen; Oxygen Consumption; Piperazines; Thioinosine; Tubercidin | 1999 |
Adenosine kinase inhibitors as a novel approach to anticonvulsant therapy.
Topics: Adenosine; Adenosine Kinase; Animals; Anticonvulsants; Cattle; Cells, Cultured; Deoxyadenosines; Electroshock; Endothelium, Vascular; Enzyme Inhibitors; Male; Microcirculation; Motor Activity; Neocortex; Pyrimidines; Radioligand Assay; Rats; Rats, Inbred Strains; Recombinant Proteins; Seizures; Structure-Activity Relationship; Tubercidin | 1999 |
Site and event specific increase of striatal adenosine release by adenosine kinase inhibition in rats.
Topics: Adenosine; Adenosine Kinase; Animals; Corpus Striatum; Enzyme Inhibitors; Kainic Acid; Male; Microdialysis; Rats; Rats, Sprague-Dawley; Tubercidin | 1999 |
A(2B) receptors mediate antimitogenesis in vascular smooth muscle cells.
Topics: 2-Chloroadenosine; Adenine; Adenosine; Adenosine Kinase; Adenosine-5'-(N-ethylcarboxamide); Animals; Anticoagulants; Antihypertensive Agents; Aorta, Abdominal; Becaplermin; Cell Division; Dinucleoside Phosphates; Enzyme Inhibitors; Hyperplasia; Male; MAP Kinase Signaling System; Muscle, Smooth, Vascular; Oligonucleotides, Antisense; Phenethylamines; Platelet-Derived Growth Factor; Proto-Oncogene Proteins c-sis; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-2; Thymidine; Tritium; Tubercidin; Vasodilator Agents; Xanthines | 2000 |
Crystal structures of Toxoplasma gondii adenosine kinase reveal a novel catalytic mechanism and prodrug binding.
Topics: Adenosine; Adenosine Kinase; Adenosine Triphosphate; Amino Acid Sequence; Animals; Anions; Antiprotozoal Agents; Apoenzymes; Base Sequence; Binding Sites; Catalysis; Conserved Sequence; Crystallography, X-Ray; Humans; Hydrogen Bonding; Magnesium; Models, Molecular; Molecular Sequence Data; Prodrugs; Protein Structure, Secondary; Protein Structure, Tertiary; Toxoplasma; Tubercidin; Water | 2000 |
Crystal structures of Toxoplasma gondii adenosine kinase reveal a novel catalytic mechanism and prodrug binding.
Topics: Adenosine; Adenosine Kinase; Adenosine Triphosphate; Amino Acid Sequence; Animals; Anions; Antiprotozoal Agents; Apoenzymes; Binding Sites; Catalysis; Conserved Sequence; Crystallography, X-Ray; Humans; Hydrogen Bonding; Magnesium; Models, Molecular; Molecular Sequence Data; Prodrugs; Protein Structure, Secondary; Protein Structure, Tertiary; Structure-Activity Relationship; Substrate Specificity; Toxoplasma; Tubercidin; Water | 2000 |
Adenosine- and 2-chloro-adenosine-induced cytopathic effects on myoblastic cells and myotubes: involvement of different intracellular mechanisms.
Topics: 2-Chloroadenosine; Acetylcysteine; Actin Cytoskeleton; Adenosine; Adenosine Kinase; Animals; Apoptosis; Cell Adhesion; Cell Line; Cytoskeleton; Dose-Response Relationship, Drug; Enzyme Inhibitors; Free Radical Scavengers; Homocysteine; Intracellular Fluid; Mice; Microscopy, Electron, Scanning; Muscle, Skeletal; Purinergic P1 Receptor Antagonists; Reactive Oxygen Species; Thioinosine; Tubercidin | 2000 |
Adenosine kinase inhibitors. 1. Synthesis, enzyme inhibition, and antiseizure activity of 5-iodotubercidin analogues.
Topics: Adenosine Kinase; Animals; Anticonvulsants; Electroshock; Enzyme Inhibitors; Humans; Male; Rats; Recombinant Proteins; Seizures; Structure-Activity Relationship; Tubercidin | 2000 |
Adenosine kinase inhibitors. 2. Synthesis, enzyme inhibition, and antiseizure activity of diaryltubercidin analogues.
Topics: Adenosine Kinase; Animals; Anticonvulsants; Enzyme Inhibitors; Humans; Magnetic Resonance Spectroscopy; Rats; Recombinant Proteins; Seizures; Spectrophotometry, Ultraviolet; Structure-Activity Relationship; Tubercidin | 2000 |
Effect of adenosine kinase, adenosine deaminase and transport inhibitors on striatal dopamine and stereotypy after methamphetamine administration.
Topics: Adenosine Deaminase; Adenosine Kinase; Animals; Corpus Striatum; Dilazep; Dopamine; Dopamine Uptake Inhibitors; Enzyme Inhibitors; Male; Methamphetamine; Pentostatin; Purinergic P1 Receptor Agonists; Rats; Rats, Wistar; Tubercidin | 2000 |
Cardioprotection with adenosine metabolism inhibitors in ischemic-reperfused mouse heart.
Topics: Adenine; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Enzyme Inhibitors; Female; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Myocardial Contraction; Myocardial Reperfusion Injury; Myocardium; Perfusion; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Theophylline; Tubercidin | 2001 |
Nucleoside transporter subtype expression: effects on potency of adenosine kinase inhibitors.
Topics: Adenine Nucleotides; Adenosine; Adenosine Kinase; Animals; Carrier Proteins; Deoxyadenosines; Dose-Response Relationship, Drug; Enzyme Inhibitors; Equilibrative Nucleoside Transport Proteins; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Gene Expression; Membrane Proteins; Membrane Transport Proteins; Nucleoside Transport Proteins; Thioinosine; Tritium; Tubercidin; Tumor Cells, Cultured | 2001 |
The effect of adenosine metabolism inhibition and nucleotide precursor supply on adenosine production in human heart endothelial cells.
Topics: Adenine; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Adenosine Triphosphate; Cells, Cultured; Coronary Vessels; Endothelium, Vascular; Enzyme Inhibitors; Humans; Nucleotides; Pentostatin; Phosphates; Ribose; Tubercidin | 2000 |
The cytotoxic effect of purine riboside on COS-7 cells.
Topics: 5'-Nucleotidase; Adenosine Kinase; Animals; Anti-Bacterial Agents; Antineoplastic Agents; Cell Survival; Chlorocebus aethiops; COS Cells; Enzyme Inhibitors; Humans; Kinetics; Purine Nucleosides; Ribonucleosides; Tubercidin | 2000 |
Effects of an adenosine kinase inhibitor and an adenosine deaminase inhibitor on accumulation of extracellular adenosine by equine articular chondrocytes.
Topics: Adenine; Adenosine; Adenosine Deaminase; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Cartilage, Articular; Chondrocytes; Enzyme Inhibitors; Horses; Lipopolysaccharides; Nitric Oxide; Nitrites; Tubercidin | 2002 |
Quantitative structure-activity relationship study of 5-iodo- and diaryl-analogues of tubercidin: inhibitors of adenosine kinase.
Topics: Adenosine Kinase; Drug Design; Iodine; Molecular Structure; Quantitative Structure-Activity Relationship; Tubercidin | 2003 |
Overexpression of adenosine kinase in epileptic hippocampus contributes to epileptogenesis.
Topics: Action Potentials; Adenosine A1 Receptor Antagonists; Adenosine Kinase; Animals; Anticonvulsants; Astrocytes; Brain; Disease Models, Animal; Disease Progression; Electroencephalography; Enzyme Inhibitors; Epilepsy, Temporal Lobe; Glial Fibrillary Acidic Protein; Hippocampus; Immunohistochemistry; Kainic Acid; Mice; Neurons; Tubercidin; Xanthines | 2004 |
Inhibition of adenosine kinase attenuates interleukin-1- and lipopolysaccharide-induced alterations in articular cartilage metabolism.
Topics: Adenosine; Adenosine Kinase; Animals; Cartilage, Articular; Culture Media, Conditioned; Dinoprostone; Enzyme Inhibitors; Glycosaminoglycans; Horses; Interleukin-1; Lipopolysaccharides; Matrix Metalloproteinase 3; Nitric Oxide; Tissue Culture Techniques; Tubercidin | 2005 |
Astrogliosis in epilepsy leads to overexpression of adenosine kinase, resulting in seizure aggravation.
Topics: Adenosine Kinase; Animals; Astrocytes; Behavior, Animal; Brain; Cerebral Cortex; Disease Models, Animal; Electroencephalography; Enzyme Inhibitors; Epilepsy, Temporal Lobe; Gliosis; Hippocampus; Kainic Acid; Locomotion; Male; Mice; Mice, Transgenic; Neurons; Transgenes; Tubercidin; Up-Regulation | 2005 |
Adenosine kinase inhibitors. 5. Synthesis, enzyme inhibition, and analgesic activity of diaryl-erythro-furanosyltubercidin analogues.
Topics: Adenosine; Adenosine Kinase; Administration, Oral; Analgesics; Animals; Area Under Curve; Biological Availability; Callithrix; Dogs; Humans; Male; Rats; Rats, Sprague-Dawley; Stereoisomerism; Structure-Activity Relationship; Tubercidin | 2005 |
The role of adenosine in chondrocyte death in murine osteoarthritis and in a murine chondrocyte cell line.
Topics: 5'-Nucleotidase; Adenine; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Apoptosis; Cartilage, Articular; Cell Death; Cell Line; Chondrocytes; DNA Fragmentation; Enzyme Inhibitors; Homocysteine; Male; Mice; Mice, Inbred Strains; Osteoarthritis; Receptors, Purinergic P1; Reverse Transcriptase Polymerase Chain Reaction; Tubercidin | 2006 |
Transgenic overexpression of adenosine kinase aggravates cell death in ischemia.
Topics: Adenosine; Adenosine Kinase; Animals; Brain Ischemia; Cell Death; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Functional Laterality; Hippocampus; Infarction, Middle Cerebral Artery; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Neuroprotective Agents; Promoter Regions, Genetic; Pyramidal Cells; Receptor, Adenosine A1; Tubercidin; Ubiquitin | 2007 |
Evaluation of 3-deaza-adenosine analogues as ligands for adenosine kinase and inhibitors of Mycobacterium tuberculosis growth.
Topics: Adenosine Kinase; Antitubercular Agents; Humans; Ligands; Mycobacterium tuberculosis; Structure-Activity Relationship; Substrate Specificity; Tubercidin | 2007 |
Crystal structures of human adenosine kinase inhibitor complexes reveal two distinct binding modes.
Topics: Adenosine Kinase; Animals; Binding Sites; Crystallography, X-Ray; Enzyme Inhibitors; Humans; Models, Molecular; Molecular Structure; Morpholines; Protein Binding; Protein Conformation; Pyrimidines; Toxoplasma; Tubercidin | 2006 |
Biochemical and biological properties of 5-bromotubercidin: differential effects on cellular DNA-directed and viral RNA-directed RNA synthesis.
Topics: Acids; Adenosine Kinase; Animals; Antiviral Agents; Cell Line; Cell Proliferation; DNA; Hydrogen-Ion Concentration; Kinetics; Liver; Mice; Molecular Structure; Protein Kinase Inhibitors; Rabbits; RNA, Viral; Solubility; Structure-Activity Relationship; Tubercidin | 2008 |
Adenosine actions are preserved in corpus cavernosum from obese and type II diabetic db/db mouse.
Topics: Acetylcholine; Adenosine; Adenosine Kinase; Animals; Diabetes Mellitus, Type 2; Dipyridamole; Disease Models, Animal; Electric Stimulation; Enzyme Inhibitors; Male; Mice; Mice, Mutant Strains; Mice, Obese; Muscle Contraction; Muscle, Smooth; Nitroprusside; Penis; Phenylephrine; Phosphodiesterase Inhibitors; Tubercidin; Vasoconstrictor Agents; Vasodilator Agents | 2008 |
A small molecule inhibitor of alpha4 integrin-dependent cell migration.
Topics: Actinin; Adenosine Kinase; Aniline Compounds; Animals; Cell Line, Tumor; Cell Movement; CHO Cells; Cricetinae; Cricetulus; Humans; Integrin alpha4; Jurkat Cells; RNA Interference; Signal Transduction; Small Molecule Libraries; Tubercidin | 2009 |
Astrocytic adenosine kinase regulates basal synaptic adenosine levels and seizure activity but not activity-dependent adenosine release in the hippocampus.
Topics: Adenosine; Adenosine Kinase; Animals; Animals, Newborn; Astrocytes; Electric Stimulation; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Glial Fibrillary Acidic Protein; Hippocampus; In Vitro Techniques; Rats; Rats, Sprague-Dawley; Seizures; Synapses; Theophylline; Time Factors; Tubercidin | 2009 |
A novel mouse model for sudden unexpected death in epilepsy (SUDEP): role of impaired adenosine clearance.
Topics: Adenine; Adenosine; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Caffeine; Cause of Death; Death, Sudden; Disease Models, Animal; Enzyme Inhibitors; Epilepsy; Kainic Acid; Mice; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Risk Factors; Seizures; Survival Analysis; Tubercidin | 2010 |
Adenosine A1 receptor blockage mediates theophylline-associated seizures.
Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine Kinase; Animals; Behavior, Animal; Body Temperature; Brain; Disease Models, Animal; Dose-Response Relationship, Drug; Electroencephalography; Enzyme Inhibitors; Hyperthermia, Induced; Injections, Intraperitoneal; Male; Rats; Rats, Inbred Lew; Seizures; Theophylline; Tubercidin | 2010 |
Deciphering ligand dependent degree of binding site closure and its implication in inhibitor design: A modeling study on human adenosine kinase.
Topics: Adenosine Kinase; Binding Sites; Cluster Analysis; Drug Design; Drug Evaluation, Preclinical; Enzyme Inhibitors; Humans; Ligands; Models, Molecular; Protein Conformation; Structural Homology, Protein; Structure-Activity Relationship; Tubercidin; User-Computer Interface | 2010 |
Molecular characterization of Chinese hamster cells mutants affected in adenosine kinase and showing novel genetic and biochemical characteristics.
Topics: Adenosine Kinase; Amino Acid Sequence; Animals; Base Sequence; Cell Line; Cricetinae; Cricetulus; Exons; Formycins; Gene Expression Regulation; Humans; Mice; Molecular Sequence Data; Mutation; Promoter Regions, Genetic; Protein Isoforms; Protein Structure, Tertiary; Rats; Tubercidin | 2011 |
Synthesis and significant cytostatic activity of 7-hetaryl-7-deazaadenosines.
Topics: Adenosine Kinase; Animals; Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cytostatic Agents; Humans; Mice; RNA Polymerase II; Tubercidin | 2011 |
Inhibition of Adenosine Kinase Attenuates Acute Lung Injury.
Topics: Acute Lung Injury; Adenosine Kinase; Animals; B-Lymphocytes; Bronchoalveolar Lavage Fluid; Cell Line; Cytokines; Lipopolysaccharides; Lung; Mice; Pneumonia; Prospective Studies; Tubercidin | 2016 |
South (S)- and North (N)-Methanocarba-7-Deazaadenosine Analogues as Inhibitors of Human Adenosine Kinase.
Topics: Adenosine Kinase; Crystallography, X-Ray; Dose-Response Relationship, Drug; Humans; Models, Molecular; Molecular Conformation; Protein Kinase Inhibitors; Structure-Activity Relationship; Tubercidin | 2016 |
Epigenetic determinants of space radiation-induced cognitive dysfunction.
Topics: 5-Methylcytosine; Adenosine Kinase; Animals; Behavior, Animal; Brain; Dioxygenases; DNA (Cytosine-5-)-Methyltransferases; DNA Methylation; DNA Methyltransferase 3A; DNA-Binding Proteins; Epigenomics; Hippocampus; Male; Mice; Mice, Inbred C57BL; Proto-Oncogene Proteins; Tubercidin; Whole-Body Irradiation | 2017 |
Transient use of a systemic adenosine kinase inhibitor attenuates epilepsy development in mice.
Topics: Adenosine Kinase; Animals; Anticonvulsants; Brain; Enzyme Inhibitors; Epilepsy; Male; Mice; Mice, Inbred C57BL; Tubercidin | 2019 |
Suppression of phrenic nerve activity as a potential predictor of imminent sudden unexpected death in epilepsy (SUDEP).
Topics: Adenosine Kinase; Animals; Kainic Acid; Male; Phrenic Nerve; Predictive Value of Tests; Rats; Rats, Wistar; Seizures; Sudden Unexpected Death in Epilepsy; Tubercidin | 2021 |