tryptoline has been researched along with triazoles in 5 studies
Studies (tryptoline) | Trials (tryptoline) | Recent Studies (post-2010) (tryptoline) | Studies (triazoles) | Trials (triazoles) | Recent Studies (post-2010) (triazoles) |
---|---|---|---|---|---|
222 | 1 | 69 | 25,808 | 2,252 | 13,501 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 4 (80.00) | 24.3611 |
2020's | 1 (20.00) | 2.80 |
Authors | Studies |
---|---|
Boonyarat, C; Fokin, VV; Jiaranaikulwanitch, J; Vajragupta, O | 1 |
Fokin, VV; Govitrapong, P; Jiaranaikulwanitch, J; Vajragupta, O | 1 |
Fokin, VV; Govitrapong, P; Jiaranaikulwanitch, J; Tadtong, S; Vajragupta, O | 1 |
Goyal, B; Goyal, D; Narang, SS | 2 |
5 other study(ies) available for tryptoline and triazoles
Article | Year |
---|---|
Triazolyl tryptoline derivatives as β-secretase inhibitors.
Topics: Amyloid Precursor Protein Secretases; Carbolines; Enzyme Inhibitors; Triazoles | 2010 |
From BACE1 inhibitor to multifunctionality of tryptoline and tryptamine triazole derivatives for Alzheimer's disease.
Topics: Alzheimer Disease; Amyloid beta-Peptides; Aspartic Acid Endopeptidases; Binding Sites; Biological Assay; Carbolines; Chelating Agents; Humans; Models, Molecular; Protease Inhibitors; Protective Agents; Triazoles; Tryptamines | 2012 |
Neuritogenic activity of bi-functional bis-tryptoline triazole.
Topics: Amyloid Precursor Protein Secretases; Animals; Aspartic Acid Endopeptidases; Carbolines; Cell Line; Cell Survival; Dose-Response Relationship, Drug; Enzyme Inhibitors; Humans; Mice; Molecular Structure; Neurites; Neuroprotective Agents; Structure-Activity Relationship; Triazoles | 2017 |
Inhibition of Alzheimer's amyloid-β
Topics: Alzheimer Disease; Amyloid beta-Peptides; Amyloid Precursor Protein Secretases; Aspartic Acid Endopeptidases; Carbolines; Humans; Molecular Docking Simulation; Molecular Dynamics Simulation; Neurodegenerative Diseases; Peptide Fragments; Triazoles | 2020 |
Molecular insights into the inhibitory mechanism of bi-functional bis-tryptoline triazole against β-secretase (BACE1) enzyme.
Topics: Amyloid Precursor Protein Secretases; Aspartic Acid Endopeptidases; Binding Sites; Carbolines; Catalytic Domain; Humans; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Models, Molecular; Molecular Docking Simulation; Molecular Dynamics Simulation; Protease Inhibitors; Protein Binding; Protein Folding; Triazoles | 2019 |