Page last updated: 2024-09-02

tryptoline and aphidicolin

tryptoline has been researched along with aphidicolin in 3 studies

Compound Research Comparison

Studies
(tryptoline)
Trials
(tryptoline)
Recent Studies (post-2010)
(tryptoline)
Studies
(aphidicolin)
Trials
(aphidicolin)
Recent Studies (post-2010) (aphidicolin)
2221691,6473136

Protein Interaction Comparison

ProteinTaxonomytryptoline (IC50)aphidicolin (IC50)
DNA polymerase catalytic subunitHuman alphaherpesvirus 1 strain KOS0.438
DNA polymerase catalytic subunitHuman alphaherpesvirus 1 strain 170.5
DNA polymerase catalytic subunitHuman herpesvirus 5 strain AD1690.4435
DNA polymerase catalytic subunitHuman herpesvirus 3 strain Dumas1.6
DNA polymerase alpha catalytic subunitHomo sapiens (human)2.98
DNA polymerase catalytic subunitHuman herpesvirus 6 (strain Uganda-1102)0.4

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Batista-Gonzalez, A; Brunhofer, G; Fallarero, A; Gopi Mohan, C; Karlsson, D; Shinde, P; Vuorela, P1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Fallarero, A; Hanski, L; Isojärvi, J; Karhu, E; Vuorela, P1

Other Studies

3 other study(ies) available for tryptoline and aphidicolin

ArticleYear
Exploration of natural compounds as sources of new bifunctional scaffolds targeting cholinesterases and beta amyloid aggregation: the case of chelerythrine.
    Bioorganic & medicinal chemistry, 2012, Nov-15, Volume: 20, Issue:22

    Topics: Acetylcholinesterase; Amyloid beta-Peptides; Benzophenanthridines; Binding Sites; Butyrylcholinesterase; Catalytic Domain; Cholinesterase Inhibitors; Humans; Isoquinolines; Kinetics; Molecular Docking Simulation; Structure-Activity Relationship

2012
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Identification of Privileged Antichlamydial Natural Products by a Ligand-Based Strategy.
    Journal of natural products, 2017, 10-27, Volume: 80, Issue:10

    Topics: Anti-Bacterial Agents; Azithromycin; Biological Products; Cell Line; Cell Survival; Chlamydophila pneumoniae; Drug Discovery; Humans; Ligands; Microbial Sensitivity Tests; Molecular Structure

2017