tripitramine has been researched along with pirenzepine in 7 studies
Studies (tripitramine) | Trials (tripitramine) | Recent Studies (post-2010) (tripitramine) | Studies (pirenzepine) | Trials (pirenzepine) | Recent Studies (post-2010) (pirenzepine) |
---|---|---|---|---|---|
17 | 0 | 0 | 3,812 | 587 | 140 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 6 (85.71) | 18.2507 |
2000's | 1 (14.29) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bolognesi, ML; Budriesi, R; Canossa, M; Chiarini, A; Melchiorre, C; Minarini, A; Spampinato, S | 1 |
Bolognesi, ML; Chiarini, A; Melchiorre, C; Minarini, A; Spampinato, S | 1 |
Bellucci, C; Bolognesi, ML; Giorgi, G; Marucci, G; Matera, R; Melchiorre, C; Minarini, A; Rosini, M; Tumiatti, V | 1 |
Angeli, P; Bianchi, S; Imeri, L; Mancia, M | 1 |
Potter, LT; Purkerson, SL | 1 |
Brown, DA; Caulfield, MP; Fernandez-Fernandez, JM; Halley, P; Wanaverbecq, N | 1 |
Budriesi, R; Chiarini, A; Melchiorre, C; Minarini, A; Spampinato, S; Tumiatti, V | 1 |
7 other study(ies) available for tripitramine and pirenzepine
Article | Year |
---|---|
Design, synthesis, and biological activity of methoctramine-related tetraamines bearing an 11-acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4] benzodiazepin-6-one moiety: structural requirements for optimum occupancy of muscarinic receptor subtypes as revealed b
Topics: Animals; Atrial Function; Benzodiazepines; Cells, Cultured; Cerebral Cortex; Drug Design; Female; Guinea Pigs; Heart Atria; Ileum; Male; Molecular Structure; Muscarinic Antagonists; Muscle Contraction; Myocardial Contraction; Myocardium; Polyamines; Rats; Receptors, Muscarinic; Structure-Activity Relationship; Submandibular Gland | 1994 |
Synthesis and biological activity of some methoctramine-related tetraamines bearing a 11-acetyl-5,11-dihydro-6H-pyrido[2,3-b][1,4]-benzodiazepin-6-one moiety as antimuscarinics: a second generation of highly selective M2 muscarinic receptor antagonists.
Topics: Animals; Benzodiazepines; Diamines; Guinea Pigs; Molecular Structure; Muscarinic Antagonists; Rats; Receptors, Muscarinic; Structure-Activity Relationship | 1993 |
Design, synthesis, and biological evaluation of pirenzepine analogs bearing a 1,2-cyclohexanediamine and perhydroquinoxaline units in exchange for the piperazine ring as antimuscarinics.
Topics: Animals; CHO Cells; Cricetinae; Cricetulus; Cyclohexylamines; Gene Expression Regulation; Guinea Pigs; Heart Atria; Humans; Male; Models, Molecular; Molecular Structure; Muscarinic Antagonists; Muscle, Skeletal; Pirenzepine; Protein Binding; Quinoxalines; Rabbits; Receptors, Muscarinic; Structure-Activity Relationship; Vas Deferens | 2008 |
Muscarinic receptor subtypes in the medial preoptic area and sleep-wake cycles.
Topics: Animals; Benzodiazepines; Body Temperature Regulation; Male; Microinjections; Muscarinic Antagonists; Piperidines; Pirenzepine; Preoptic Area; Rats; Receptors, Muscarinic; Sleep; Sleep, REM; Wakefulness | 1996 |
Use of antimuscarinic toxins to facilitate studies of striatal m4 muscarinic receptors.
Topics: Alkaloids; Animals; Benzodiazepines; Binding, Competitive; Cats; CHO Cells; Corpus Striatum; Cricetinae; Elapid Venoms; Furans; Gallamine Triethiodide; Humans; Male; Muscarinic Antagonists; N-Methylscopolamine; Naphthalenes; Neurotoxins; Piperidines; Pirenzepine; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Receptor, Muscarinic M4; Receptors, Muscarinic; Recombinant Proteins | 1998 |
Selective activation of heterologously expressed G protein-gated K+ channels by M2 muscarinic receptors in rat sympathetic neurones.
Topics: Animals; Barium; Benzodiazepines; Biolistics; Calcium Channels; Carbachol; Cells, Cultured; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Green Fluorescent Proteins; GTP-Binding Proteins; Luminescent Proteins; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Pirenzepine; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic; Recombinant Proteins; Superior Cervical Ganglion; Transfection | 1999 |
The design of novel methoctramine-related tetraamines as muscarinic receptor subtype selective antagonists.
Topics: Animals; Atrial Function; Benzodiazepines; Benzodiazepinones; Diamines; Drug Design; Guinea Pigs; Heart Atria; Ileum; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Piperidines; Pirenzepine; Rats; Receptors, Muscarinic; Structure-Activity Relationship; Submandibular Gland; Trachea | 1995 |