tripitramine has been researched along with carbachol in 3 studies
Studies (tripitramine) | Trials (tripitramine) | Recent Studies (post-2010) (tripitramine) | Studies (carbachol) | Trials (carbachol) | Recent Studies (post-2010) (carbachol) |
---|---|---|---|---|---|
17 | 0 | 0 | 13,918 | 81 | 968 |
Protein | Taxonomy | tripitramine (IC50) | carbachol (IC50) |
---|---|---|---|
Muscarinic acetylcholine receptor M2 | Homo sapiens (human) | 0.7849 | |
Muscarinic acetylcholine receptor M4 | Homo sapiens (human) | 2.0626 | |
Muscarinic acetylcholine receptor M1 | Rattus norvegicus (Norway rat) | 3.4134 | |
Muscarinic acetylcholine receptor M3 | Rattus norvegicus (Norway rat) | 2.9961 | |
Muscarinic acetylcholine receptor M4 | Rattus norvegicus (Norway rat) | 2.535 | |
Muscarinic acetylcholine receptor M5 | Rattus norvegicus (Norway rat) | 2.9961 | |
Muscarinic acetylcholine receptor M2 | Rattus norvegicus (Norway rat) | 2.6638 | |
Muscarinic acetylcholine receptor M1 | Homo sapiens (human) | 4.849 | |
Muscarinic acetylcholine receptor M3 | Homo sapiens (human) | 4.99 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 3 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bolognesi, ML; Budriesi, R; Chiarini, A; Melchiorre, C; Minarini, A | 1 |
Brown, DA; Caulfield, MP; Fernandez-Fernandez, JM; Halley, P; Wanaverbecq, N | 1 |
Akici, A; El-Fakahany, EE; Karaalp, A; Oktay, S; Skender, E | 1 |
3 other study(ies) available for tripitramine and carbachol
Article | Year |
---|---|
In vitro characterization of tripitramine, a polymethylene tetraamine displaying high selectivity and affinity for muscarinic M2 receptors.
Topics: Animals; Benzodiazepines; Carbachol; Diamines; Dose-Response Relationship, Drug; Duodenum; Guinea Pigs; Heart Atria; Ileum; In Vitro Techniques; Lung; Male; Muscarinic Antagonists; Rats; Receptors, Muscarinic; Trachea; Vas Deferens | 1995 |
Selective activation of heterologously expressed G protein-gated K+ channels by M2 muscarinic receptors in rat sympathetic neurones.
Topics: Animals; Barium; Benzodiazepines; Biolistics; Calcium Channels; Carbachol; Cells, Cultured; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Green Fluorescent Proteins; GTP-Binding Proteins; Luminescent Proteins; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Pirenzepine; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic; Recombinant Proteins; Superior Cervical Ganglion; Transfection | 1999 |
Muscarinic M(2) receptors are not primarily involved in the contraction of guinea-pig gallbladder smooth muscle.
Topics: Alkaloids; Animals; Benzodiazepines; Carbachol; Cevanes; Female; Gallamine Triethiodide; Gallbladder; Guinea Pigs; In Vitro Techniques; Male; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Receptor, Muscarinic M2; Receptors, Muscarinic | 1999 |