Page last updated: 2024-09-04

tripitramine and carbachol

tripitramine has been researched along with carbachol in 3 studies

Compound Research Comparison

Studies
(tripitramine)
Trials
(tripitramine)
Recent Studies (post-2010)
(tripitramine)
Studies
(carbachol)
Trials
(carbachol)
Recent Studies (post-2010) (carbachol)
170013,91881968

Protein Interaction Comparison

ProteinTaxonomytripitramine (IC50)carbachol (IC50)
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.7849
Muscarinic acetylcholine receptor M4Homo sapiens (human)2.0626
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)3.4134
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)2.535
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)2.9961
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)2.6638
Muscarinic acetylcholine receptor M1Homo sapiens (human)4.849
Muscarinic acetylcholine receptor M3Homo sapiens (human)4.99

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bolognesi, ML; Budriesi, R; Chiarini, A; Melchiorre, C; Minarini, A1
Brown, DA; Caulfield, MP; Fernandez-Fernandez, JM; Halley, P; Wanaverbecq, N1
Akici, A; El-Fakahany, EE; Karaalp, A; Oktay, S; Skender, E1

Other Studies

3 other study(ies) available for tripitramine and carbachol

ArticleYear
In vitro characterization of tripitramine, a polymethylene tetraamine displaying high selectivity and affinity for muscarinic M2 receptors.
    British journal of pharmacology, 1995, Volume: 114, Issue:7

    Topics: Animals; Benzodiazepines; Carbachol; Diamines; Dose-Response Relationship, Drug; Duodenum; Guinea Pigs; Heart Atria; Ileum; In Vitro Techniques; Lung; Male; Muscarinic Antagonists; Rats; Receptors, Muscarinic; Trachea; Vas Deferens

1995
Selective activation of heterologously expressed G protein-gated K+ channels by M2 muscarinic receptors in rat sympathetic neurones.
    The Journal of physiology, 1999, Mar-15, Volume: 515 ( Pt 3)

    Topics: Animals; Barium; Benzodiazepines; Biolistics; Calcium Channels; Carbachol; Cells, Cultured; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Green Fluorescent Proteins; GTP-Binding Proteins; Luminescent Proteins; Male; Membrane Potentials; Neurons; Patch-Clamp Techniques; Pirenzepine; Potassium Channels; Potassium Channels, Inwardly Rectifying; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M2; Receptor, Muscarinic M4; Receptors, Muscarinic; Recombinant Proteins; Superior Cervical Ganglion; Transfection

1999
Muscarinic M(2) receptors are not primarily involved in the contraction of guinea-pig gallbladder smooth muscle.
    Pharmacological research, 1999, Volume: 40, Issue:5

    Topics: Alkaloids; Animals; Benzodiazepines; Carbachol; Cevanes; Female; Gallamine Triethiodide; Gallbladder; Guinea Pigs; In Vitro Techniques; Male; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Receptor, Muscarinic M2; Receptors, Muscarinic

1999