Page last updated: 2024-08-17

triiodothyronine and kb 2115

triiodothyronine has been researched along with kb 2115 in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (10.00)29.6817
2010's8 (80.00)24.3611
2020's1 (10.00)2.80

Authors

AuthorsStudies
Hashizume, K; Ichikawa, K; Kikuchi, N; Matsuzawa, A; Miyamoto, T; Nagano, R; Nakamura, T; Ohnota, H; Ozawa, T; Shiohara, H1
Asano, Y; Maeda, K; Takahashi, N; Watanabe, N1
Banner, B; Conde-Knape, K; Danzi, S; Dvorozniak, M; Haynes, NE; Huang, KS; Kelly, MJ; Klein, I; Larigan, JD; Mennona, F; Pietranico-Cole, S; Qian, Y; Reynolds, CH; Scott, N; So, SS; Taub, R; Thakkar, K; Tilley, J; Vermeulen, J1
Josseaume, C; Lorcy, Y1
Angelin, B; Baxter, JD; Carlsson, B; Klein, I; Kristensen, JD; Ladenson, PW; Olsson, AG; Ridgway, EC1
Baxter, JD; Gustafsson, JÅ; Hsueh, WA; Lin, JZ; Martagón, AJ; Phillips, KJ; Webb, P1
Boilard, E; Levesque, T; Park, EA; Sharma, P1
Angelin, B; Carlsson, B; Chester Ridgway, E; Eriksson, M; Klein, I; Kristensen, JD; Ladenson, PW; Olsson, AG1
Columbano, A; Ledda-Columbano, GM; Leoni, VP; Mattu, S; Perra, A; Pibiri, M; Puliga, E; Szydlowska, M1
Zucchi, R1

Reviews

1 review(s) available for triiodothyronine and kb 2115

ArticleYear
Thyroid Hormone Analogues: An Update.
    Thyroid : official journal of the American Thyroid Association, 2020, Volume: 30, Issue:8

    Topics: Acetates; Anilides; Animals; Central Nervous System Diseases; Clinical Trials as Topic; Diiodothyronines; Drug Design; Dyslipidemias; Humans; Liver Diseases; Male; Mice; Mutation; Non-alcoholic Fatty Liver Disease; Phenols; Pyridazines; Rats; Signal Transduction; Thyroid Hormone Receptors alpha; Thyroid Hormone Receptors beta; Thyroid Hormones; Thyronines; Triiodothyronine; Uracil

2020

Trials

2 trial(s) available for triiodothyronine and kb 2115

ArticleYear
Use of the thyroid hormone analogue eprotirome in statin-treated dyslipidemia.
    The New England journal of medicine, 2010, Mar-11, Volume: 362, Issue:10

    Topics: Adult; Anilides; Cholesterol, LDL; Double-Blind Method; Drug Therapy, Combination; Dyslipidemias; Female; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Lipoproteins; Male; Middle Aged; Thyroid Hormones; Triglycerides; Triiodothyronine

2010
Reductions in serum levels of LDL cholesterol, apolipoprotein B, triglycerides and lipoprotein(a) in hypercholesterolaemic patients treated with the liver-selective thyroid hormone receptor agonist eprotirome.
    Journal of internal medicine, 2015, Volume: 277, Issue:3

    Topics: Anilides; Anticholesteremic Agents; Apolipoproteins B; Blood Pressure; Bone and Bones; Cholesterol, LDL; Double-Blind Method; Drug Administration Schedule; Female; Heart Rate; Humans; Hypercholesterolemia; Lipoprotein(a); Male; Middle Aged; Thyrotropin; Triglycerides; Triiodothyronine

2015

Other Studies

7 other study(ies) available for triiodothyronine and kb 2115

ArticleYear
Discovery of novel indane derivatives as liver-selective thyroid hormone receptor β (TRβ) agonists for the treatment of dyslipidemia.
    Bioorganic & medicinal chemistry, 2012, Jun-01, Volume: 20, Issue:11

    Topics: Animals; Arginine; Cholesterol; Disease Models, Animal; Drug Design; Drug Evaluation, Preclinical; Dyslipidemias; Humans; Indans; Ligands; Liver; Male; Malonates; Models, Molecular; Molecular Mimicry; Molecular Structure; Rats; Rats, Wistar; Small Molecule Libraries; Structure-Activity Relationship; Thyroid Hormone Receptors beta

2012
Synthesis and pharmacological characterization of 1-benzyl-4-aminoindole-based thyroid hormone receptor β agonists.
    Bioorganic & medicinal chemistry, 2014, Jan-01, Volume: 22, Issue:1

    Topics: Animals; Indoles; Rats; Thyroid Hormone Receptors beta

2014
Discovery of 2-[3,5-dichloro-4-(5-isopropyl-6-oxo-1,6-dihydropyridazin-3-yloxy)phenyl]-3,5-dioxo-2,3,4,5-tetrahydro[1,2,4]triazine-6-carbonitrile (MGL-3196), a Highly Selective Thyroid Hormone Receptor β agonist in clinical trials for the treatment of dys
    Journal of medicinal chemistry, 2014, May-22, Volume: 57, Issue:10

    Topics: Animals; Bone Density; Clinical Trials as Topic; Drug Discovery; Dyslipidemias; Humans; Male; Mice; Mice, Inbred C57BL; Pyridazines; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Thyroid Hormone Receptors beta; Uracil

2014
[Thyroid hormone analogs: an important biological supply and new therapeutic possibilities].
    Annales d'endocrinologie, 2008, Volume: 69 Suppl 1

    Topics: Acetates; Anilides; Anticholesteremic Agents; Humans; Hypolipidemic Agents; Phenols; Phenyl Ethers; Phenylacetates; Receptors, Thyroid Hormone; Signal Transduction; Thyroid Hormones; Triiodothyronine

2008
Thyroid hormone receptor agonists reduce serum cholesterol independent of the LDL receptor.
    Endocrinology, 2012, Volume: 153, Issue:12

    Topics: Acetates; Anilides; Animals; Apolipoproteins B; Cholesterol; Cholesterol 7-alpha-Hydroxylase; Feces; Lipoproteins; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Phenols; Receptors, LDL; Receptors, Thyroid Hormone; Thyroid Hormone Receptors beta; Triglycerides; Triiodothyronine

2012
Thyroid hormone status regulates the expression of secretory phospholipases.
    Biochemical and biophysical research communications, 2014, Jan-31, Volume: 444, Issue:1

    Topics: Anilides; Animals; Gene Expression Regulation, Enzymologic; Group II Phospholipases A2; Hep G2 Cells; Hepatocytes; Humans; Hyperlipidemias; Hyperthyroidism; Hypothyroidism; Inflammation; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Transgenic; Phospholipases A2, Secretory; Rats; Rats, Sprague-Dawley; RNA, Messenger; Thyroid Hormone Receptors beta; Triiodothyronine

2014
The Thyromimetic KB2115 (Eprotirome) Induces Rat Hepatocyte Proliferation.
    Gene expression, 2017, Jul-07, Volume: 17, Issue:3

    Topics: Anilides; Animal Feed; Animals; Apoptosis; Body Weight; Cell Proliferation; Cyclin D1; Heart; Hepatocytes; Liver; Male; Organ Size; Rats; Rats, Inbred F344; Receptors, Thyroid Hormone; Regenerative Medicine; Time Factors; Transaminases; Triiodothyronine

2017