Page last updated: 2024-08-16

trifluoperazine and bepridil

trifluoperazine has been researched along with bepridil in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19906 (33.33)18.7374
1990's4 (22.22)18.2507
2000's4 (22.22)29.6817
2010's4 (22.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Benz, RD; Contrera, JF; Kruhlak, NL; Matthews, EJ; Weaver, JL1
Cai, W; Hao, Y; Hu, P; Ma, D; Pan, H; Xie, X; Yu, AD; Yu, J; Yuan, J; Zhang, L; Zhu, H1
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Herzig, JW; Quast, U1
Ovaska, M; Taskinen, J1
Lugnier, C; Schaeffer, P; Stoclet, JC1
Monteforte, PB; Silver, PJ1
Hofmann, F; Zimmer, M1
Barron, E; Marshall, RJ; Martorana, M; Winslow, E1
Agre, P; Bennett, V; Virshup, D1
Pollak, PT1
Choi, D; Kleerekoper, Q; Liu, W; Putkey, JA1
Kobayashi, S; Kumagai, M; Makioka, A; Takeuchi, T1
Berek, JS; Chung, YM; Hu, MC; Ma, J; Park, SH; Yang, Q1
Belevych, N; Biesiadecki, BJ; Cuesta, A; Davis, JP; Hwang, PM; Li, MX; Price, M; Reiser, PJ; Tikunova, SB1

Reviews

1 review(s) available for trifluoperazine and bepridil

ArticleYear
A systematic review and critical comparison of internal standards for the routine liquid chromatographic assay of amiodarone and desethylamiodarone.
    Therapeutic drug monitoring, 1996, Volume: 18, Issue:2

    Topics: Amiodarone; Anti-Arrhythmia Agents; Bepridil; Chromatography, High Pressure Liquid; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Monitoring; Estrogen Antagonists; Tamoxifen; Trifluoperazine

1996

Other Studies

17 other study(ies) available for trifluoperazine and bepridil

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Assessment of the health effects of chemicals in humans: II. Construction of an adverse effects database for QSAR modeling.
    Current drug discovery technologies, 2004, Volume: 1, Issue:4

    Topics: Adverse Drug Reaction Reporting Systems; Artificial Intelligence; Computers; Databases, Factual; Drug Prescriptions; Drug-Related Side Effects and Adverse Reactions; Endpoint Determination; Models, Molecular; Quantitative Structure-Activity Relationship; Software; United States; United States Food and Drug Administration

2004
Small molecule regulators of autophagy identified by an image-based high-throughput screen.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Nov-27, Volume: 104, Issue:48

    Topics: Autophagy; Calcium Channel Blockers; Cell Line, Tumor; Drug Evaluation, Preclinical; Fluspirilene; Glioblastoma; Green Fluorescent Proteins; Humans; Intracellular Membranes; Loperamide; Microtubule-Associated Proteins; Mycotoxins; Peptides; Phagosomes; Phosphatidylinositol Phosphates; Pimozide; Protein Kinases; Recombinant Fusion Proteins; Sirolimus; Small Molecule Libraries; TOR Serine-Threonine Kinases; Trifluoperazine; Zinc Fingers

2007
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
On the role of Ca++ binding proteins as possible targets for Ca++ sensitizing agents.
    Zeitschrift fur Kardiologie, 1992, Volume: 81 Suppl 4

    Topics: Amrinone; Animals; Bepridil; Calcium; Calcium-Binding Proteins; Calmodulin; Cardiotonic Agents; Dose-Response Relationship, Drug; Milrinone; Models, Cardiovascular; Myocardial Contraction; Piperazines; Pyridones; Swine; Trifluoperazine; Troponin; Troponin C

1992
A model for human cardiac troponin C and for modulation of its Ca2+ affinity by drugs.
    Proteins, 1991, Volume: 11, Issue:2

    Topics: Amino Acid Sequence; Asparagine; Bepridil; Binding Sites; Calcium; Calmodulin; Glycine; Humans; Models, Molecular; Molecular Sequence Data; Myocardium; Protein Conformation; Pyridazines; Trifluoperazine; Troponin; Troponin C; Vasodilator Agents

1991
Interaction of calmodulin and calcium antagonists with [3H]diltiazem and [3H]nitrendipine binding sites.
    Journal of cardiovascular pharmacology, 1988, Volume: 12 Suppl 4

    Topics: Animals; Bepridil; Calcium Channel Blockers; Calcium Channels; Calmodulin; Diltiazem; Imidazoles; Phosphodiesterase Inhibitors; Pyrrolidines; Rats; Receptors, Nicotinic; Sulfonamides; Trifluoperazine

1988
Differential effects of pharmacological modulators of cardiac myofibrillar ATPase activity in normal and myopathic (BIO 14.6) hamsters.
    European journal of pharmacology, 1988, Mar-15, Volume: 147, Issue:3

    Topics: Adenosine Triphosphatases; Animals; Anti-Arrhythmia Agents; Bepridil; Calcium; Calcium Channel Blockers; Cricetinae; Disease Models, Animal; Electrophoresis, Polyacrylamide Gel; Heart Failure; Imidazoles; Male; Myocardium; Myofibrils; Perhexiline; Pyrrolidines; Trifluoperazine

1988
Differentiation of the drug-binding sites of calmodulin.
    European journal of biochemistry, 1987, Apr-15, Volume: 164, Issue:2

    Topics: 2',3'-Cyclic-Nucleotide Phosphodiesterases; Animals; Bepridil; Binding Sites; Calmodulin; In Vitro Techniques; Kinetics; Myosin-Light-Chain Kinase; Nimodipine; Pyrrolidines; Trifluoperazine

1987
Comparative antiarrhythmic and electrophysiological effects of drugs known to inhibit calmodulin (TFP, W7 and bepridil).
    British journal of pharmacology, 1986, Volume: 89, Issue:3

    Topics: Action Potentials; Animals; Anti-Arrhythmia Agents; Bepridil; Calmodulin; Coronary Vessels; Guinea Pigs; Heart; Hemodynamics; In Vitro Techniques; Ligation; Male; Phentolamine; Phenylephrine; Pyrrolidines; Rats; Rats, Inbred Strains; Sulfonamides; Trifluoperazine

1986
Bepridil and cetiedil. Vasodilators which inhibit Ca2+-dependent calmodulin interactions with erythrocyte membranes.
    The Journal of clinical investigation, 1984, Volume: 74, Issue:3

    Topics: Adult; Azepines; Bepridil; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Calmodulin; Calmodulin-Binding Proteins; Erythrocyte Membrane; Humans; Kinetics; Phosphoprotein Phosphatases; Pyrrolidines; Trifluoperazine; Vasodilator Agents

1984
Identification of binding sites for bepridil and trifluoperazine on cardiac troponin C.
    The Journal of biological chemistry, 1998, Apr-03, Volume: 273, Issue:14

    Topics: Animals; Bepridil; Binding Sites; Calcium; Humans; Myocardium; Protein Binding; Protein Conformation; Trifluoperazine; Troponin C

1998
Possible role of calcium ions, calcium channels and calmodulin in excystation and metacystic development of Entamoeba invadens.
    Parasitology research, 2002, Volume: 88, Issue:9

    Topics: Animals; Bepridil; Calcium; Calcium Channel Blockers; Calcium Channels; Calmodulin; Chelating Agents; Culture Media; Entamoeba; Entamoebiasis; Gallic Acid; Trifluoperazine

2002
Pharmacological activation of FOXO3 suppresses triple-negative breast cancer in vitro and in vivo.
    Oncotarget, 2016, Jul-05, Volume: 7, Issue:27

    Topics: Animals; Apoptosis; Bepridil; Breast Neoplasms; Cell Nucleus; Dopamine; Female; Forkhead Box Protein O3; Gene Expression Regulation, Neoplastic; Gene Silencing; Humans; Kruppel-Like Transcription Factors; MCF-7 Cells; Mice; Mice, Nude; Neoplastic Stem Cells; Phosphorylation; Proto-Oncogene Proteins c-myc; Receptors, Dopamine D2; RNA, Small Interfering; Trifluoperazine; Triple Negative Breast Neoplasms

2016
3-Chlorodiphenylamine activates cardiac troponin by a mechanism distinct from bepridil or TFP.
    The Journal of general physiology, 2019, 01-07, Volume: 151, Issue:1

    Topics: Animals; Bepridil; Calcium; Diphenylamine; Female; Heart; Humans; Myocardium; Rats; Rats, Wistar; Trifluoperazine; Troponin C; Troponin I

2019