Page last updated: 2024-08-24

triazoles and zm 241385

triazoles has been researched along with zm 241385 in 347 studies

Research

Studies (347)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's43 (12.39)18.2507
2000's194 (55.91)29.6817
2010's105 (30.26)24.3611
2020's5 (1.44)2.80

Authors

AuthorsStudies
Brooks, R; Collis, MG; Keddie, JR; Poucher, SM; Shaw, GR1
Hourani, SM; Prentice, DJ2
Brooks, R; Keddie, JR; McKillop, D; Poucher, SM; Shaw, GR1
Jacobson, KA; Palmer, TM; Poucher, SM; Stiles, GL1
Poucher, SM2
Dixon, AK; Richardson, PJ; Widdowson, L1
Apasov, S; Huang, S; Kojima, H; Koshiba, M; Sitkovsky, MV1
Constantino, MD; Cunha, RA; Ribeiro, JA2
Hourani, SM; Payne, SL; Prentice, DJ1
McGrath, JC; Moore, FP; Thomson, NC1
Fukamachi, H; Nakahata, T; Suzuki, H; Takei, M1
Conforti, L; Kobayashi, S; Millhorn, DE; Pun, RY1
Coney, AM; Marshall, JM1
Jones, PA; Smith, RA; Stone, TW2
Baraldi, PG; Borea, PA; Cacciari, B; Dionisotti, S; Ongini, E; Varani, K1
Baker, SP; Baraldi, PG; Belardinelli, L; Cacciari, B; Monopoli, A; Ongini, E; Shryock, JC; Snowdy, S; Spalluto, G1
O'Regan, MH; Phillis, JW; Song, D1
Bryan, PT; Marshall, JM1
O'Kane, EM; Stone, TW1
Cutler, BS; Dobson, JG; Fenton, RA; Li, Jm; Peyton, BD; Powell, CC; Wheeler, HB1
Dionisotti, S; Fredholm, BB; Gessi, S; Irenius, E; Ongini, E1
Chung, ES; Dobson, JG; Fenton, RA; Honeyman, TW; Lorbar, M; McGinn, RJ; Meyer, TE; Norton, GR; Woodiwiss, AJ1
Cseppentö, A; Kovács, P; Nagy, E; Szabó, JZ; Szentmiklósi, AJ; Ujfalusi, A1
Huang, L; Linden, J; Macdonald, T; Okusa, MD1
Cunha, RA; Lopes, LV; Ribeiro, JA3
Fredholm, BB; Lindström, K1
Buster, BL; Linden, J; Scheld, WM; Sullivan, GW1
Benovic, JL; Kelly, E; Parent, JL; Willets, JM1
Palmer, TM; Stiles, GL1
Bordoni, F; Corradetti, R; Latini, S; Pedata, F; Pepeu, G1
Enyeart, JJ; Xu, L1
Brunsden, AM; Grundy, D1
Davie, CS; Everitt, DE; Standen, NB1
Fei, Q; Loutzenhiser, R; Parker, M; Tang, L1
Jacobson, KA; Ji, XD1
Harada, N; Katsuragi, T; Okajima, K1
Dashwood, MR; Spyer, KM; St Lambert, JH; Thomas, T1
Costentin, J; El Yacoubi, M; Ledent, C; Parmentier, M; Vaugeois, JM1
Hong, KW; Shin, HK; Shin, YW1
Abebe, W; Arif Hasan, AZ; Mustafa, SJ1
Jabbari-T, J; Oberhauser, V; Rump, LC; von Kügelgen, I1
Cunha, RA; Pereira, MF; Ribeiro, JA1
Clark, KL; Guyton, RA; Nakamura, M; Velez, DV; Vinten-Johansen, J; Zhao, ZQ1
Anderson, R; Ramafi, G; Theron, AJ; Visser, SS1
Olah, ME; Roudabush, FL1
Agostinho, P; Cunha, RA; Melo, J; Oliveira, CR; Rego, AC1
Matsuki, N; Nakazawa, K; Ohno, Y; Sato, K1
Costentin, J; El Yacoubi, M; Ledent, C; Parmentier, M; Vaugeois, J1
Feoktistov, I; Mustafa, SJ; Olanrewaju, HA; Qin, W; Scemama, JL1
Gao, ZG; Ijzerman, AP; Jacobson, KA; Jiang, Q1
Gao, ZG; Ijzerman, AP1
Harada, N; Katsuragi, T; Murakami, K; Ohshima, K; Okajima, K; Sato, C; Usune, S1
Cunha, RA; Hernández, MD; Miras-Portugal, MT; Pereira, MF; Pintor, J; Ribeiro, JA1
Koos, BJ; Maeda, T2
Kaszkin, M; Pfeilschifter, J; Scholz-Pedretti, K1
Hein, TW; Kuo, L; Muthuchamy, M; Wang, W; Zoghi, B1
Alexander, SP; Millns, PJ1
Costentin, J; Daoust, M; El Yacoubi, M; Ledent, C; Parmentier, M; Vaugeois, J1
Linden, J; Macdonald, TL; Rieger, JM; Scheld, WM; Sullivan, GW1
Coyne, EF; Meno, JR; Ngai, AC; West, GA; Winn, HR1
Barringhaus, KG; Bishop, GG; Gimple, LW; Hesselbacher, SE; Linden, J; Macdonald, T; McPherson, JA; Powers, ER; Rieger, JM; Sanders, JM; Sarembock, IJ; Sullivan, G1
Linden, J; Macdonald, TL; Peirce, SM; Rieger, JM; Skalak, TC1
Jan, C; Koos, BJ; Maeda, T1
Baker, SP; Belardinelli, L; Blackburn, B; Elzein, E; Gao, Z; Lasley, RD; Li, Z; Meyer, S; Palle, V; Zablocki, JA1
Bernardi, G; Calabresi, P; Centonze, D; Pisani, A; Saulle, E1
Nikbakht, MR; Stone, TW1
Hamann, M; Richter, A1
Breschi, MC; Calderone, V; Martinotti, E; Nieri, P1
Culmsee, C; Kemp, BE; Mattson, MP; Monnig, J1
Crum, AV; Meno, JR; Winn, HR1
Inoue, H; Kikkawa, K; Mochida, H; Noto, T1
Edmunds, NJ; Marshall, JM1
Harvey, V; Jones, J; Knight, AR; Misra, A; Quirk, K1
Furue, H; Kumamoto, E; Lao, LJ; Luo, C; Yoshimura, M1
Grisshammer, R; Weiss, HM1
Higashi, H; Marwaha, AS; Meno, JR; Winn, HR1
Ellis, KM; Fozard, JR; Mazzoni, L; Tigani, B; Villela Dantas, MF1
Jan, C; Koos, BJ; Lopez, G; Maeda, T1
Cunha, RA; Fredholm, BB; Kull, B; Lopes, LV; Ribeiro, JA1
Belem, PC; Chen, JF; Cronstein, B; Elson, G; Fink, JS; Jacobson, M; Leibovich, SJ; Montesinos, C; Pinhal-Enfield, G; Ramanathan, M; Rosania, A; Schwarzschild, MA1
Gao, ZG; IJzerman, AP; Jacobson, KA; Kim, SG; Melman, N; Soltysiak, KA1
Bril, A; Broadley, KJ; Khandoudi, N; Maddock, HL1
Chicz-DeMet, A; DeMet, EM1
Cunha, RA; Oliveira, CR; Rebola, N1
Daoust, M; Ledent, C; Naassila, M1
Borea, PA; Cattabriga, E; Iannotta, V; Manfredini, R; Pancaldi, C; Portaluppi, F; Uluoglu, C; Varani, K1
Abbracchio, MP; Borea, PA; Camurri, A; Capecchi, PL; Cattabeni, F; Ceccatelli, L; Diciolla, F; Laghi-Pasini, F; Lazzerini, PE; Maccherini, M; Ulouglu, C; Varani, K1
D'Ambrosio, R; Iliff, JJ; Ngai, AC; Winn, HR1
Diniz, C; Gonçalves, J; Leal, S1
Duling, BR; Linden, J; Platts, SH1
Antoniou, K; Ferré, S; Fuxe, K; Goldberg, SR; Justinova, Z; Karcz-Kubicha, M; Müller, CE; Pezzola, A; Popoli, P; Quarta, D; Reggio, R; Solinas, M; Terasmaa, A1
Cunha, RA; Dall'Igna, OP; Dall'lgna, OP; Lara, DR; Porciúncula, LO; Souza, DO1
Adamski, D; Berger, F; Charles, MP; Kholler, B; Pelletier, L; Wion, D1
Boehm, S; Freissmuth, M; Just, H; Klinger, M; Korkhov, VM; Kudlacek, O; Nanoff, C; Pankevych, H; Vartian, N; Yang, Q1
Fredholm, BB; Hellsten, Y; Lynge, J; Nordsborg, N; Schulte, G1
Cunha, RA; de Mendonca, A; Oliveira, CR; Rebola, N; Ribeiro, JA; Sebastião, AM1
O'Regan, MH; Phillis, JW1
Corradetti, R; Latini, S; Pedata, F; Pugliese, AM1
Brodmann, M; Lischnig, U; Lueger, A; Pilger, E; Stark, G1
Addae, JI; Stone, TW; Youssef, FF1
Mustafa, JS; Rekik, M1
Costentin, J; El Yacoubi, M; Vaugeois, JM1
Benwell, K; Cliffe, IA; Dourish, CT; Gillespie, RJ; Knight, AR; Lerpiniere, J; Misra, A; Pratt, RM; Revell, D; Upton, R; Weiss, SM1
Day, YJ; Huang, L; Linden, J; Marshall, MA; McDuffie, MJ; Okusa, MD1
Brooke, RE; Deuchars, J; Deuchars, SA1
Goulart, EC; Kaster, MP; Rodrigues, AL; Rosa, AO; Rosso, MM; Santos, AR1
Furuta, S; Honma, I; Kumagai, M; Miyazaki, S; Onodera, K; Sakurada, S; Sato, T1
Kwok, YN; Yip, L1
Abebe, W; Mozaffari, MS1
Easton, AS; Inglis, VI; Jones, MP; Tse, AD1
Bier, D; Coenen, HH; Holschbach, MH; Olsson, RA; Schulze, A; Sihver, W; Wutz, W1
Galluzzo, M; Grieco, R; Pèzzola, A; Pintor, A; Popoli, P; Reggio, R1
Diógenes, MJ; Fernandes, CC; Ribeiro, JA; Sebastião, AM1
Konishi, S; Rusakov, D; Saitow, F; Satake, S1
Etherington, LA; Frenguelli, BG1
Ho, CM; Ho, ST; Peng, SC; Su, CK; Tsai, SK1
Awadallah, NW; Chan, ES; Cronstein, BN; Montesinos, MC; Rahman, MM; Reiss, AB1
Domenici, MR; Frank, C; Grieco, R; Martire, A; Pepponi, R; Pintor, A; Popoli, P; Potenza, RL; Tebano, MT1
Barbu, DE; Lungu, CL; O'Regan, MH; Phillis, JW1
Dziubina, A; Gołembiowska, K3
Domenici, MR; Martire, A; Pepponi, R; Popoli, P; Potenza, RL; Tebano, MT1
Batista, LC; Prediger, RD; Takahashi, RN1
Bailey, A; Hourani, S; Kelly, M; Kitchen, I; Ledent, C1
Colgan, SP; Eltzschig, HK; Ibla, JC; Morote-Garcia, JC; Resta, R; Thompson, LF; Van De Wiele, CJ1
Bohorquez, F; Kawasaki, Y; Kim, YH; Koos, BJ1
Lappas, CM; Linden, J; Rieger, JM1
Briones, R; Donoso, MV; Huidobro-Toro, JP; López, R; Miranda, R1
Ballard-Croft, C; Keith, BJ; Kristo, G; Lasley, RD; Mentzer, RM; Reid, EA; Yoshimura, Y1
Fuxe, K; Rinken, A; Terasmaa, A; Uustare, A; Vonk, A1
Ackley, MA; Baldwin, SA; King, AE1
Abbracchio, MP; Camurri, A; Capecchi, PL; Diciolla, F; Laghi-Pasini, F; Lazzerini, PE; Maccherini, M; Mazzola, A; Pompella, G1
Prediger, RD; Takahashi, RN1
Hikichi, T; Kawahara, A; Kitaya, N; Mori, F; Takahashi, J; Yoshida, A1
Fernandes, D; Prediger, RD; Takahashi, RN1
Bonan, CD; Cammarota, M; Izquierdo, I; Pereira, GS; Rossato, JI; Sarkis, JJ1
Arun, KH; Kaul, CL; Kumar, S; Sharma, SS1
Herrera, S; Kasza, K; Mendelson, WB; Szafran, MJ; Tung, A1
Amerson, BS; Guyton, RA; Halkos, ME; Headrick, JP; Kerendi, F; Kin, H; Lofye, MT; Vinten-Johansen, J; Zatta, AJ; Zhao, ZQ1
Boeck, CR; Bronzatto, MJ; Kroth, EH; Vendite, D1
Almeida, T; Cunha, RA; Oliveira, CR; Richardson, PJ; Rodrigues, RJ1
Linden, J; Marshall, MA; Murphree, LJ; Sullivan, GW1
Angulo, E; Casadó, V; Chen, JF; Ejarque, A; Franco, R; Lluis, C; Moratalla, R; Saura, J; Schwarzschild, MA; Serratosa, J; Tusell, JM1
Belardinelli, L; Biaggioni, I; Dhalla, AK; Wang, WQ; Wong, MY1
Marshall, JM; Ray, CJ3
Deussen, A; Frøbert, O; Gravholt, CH; Haink, G; Levin, M; Simonsen, U1
Fathollahi, Y; Mirnajafi-Zadeh, J; Namvar, S; Rezvani, ME; Zeraati, M1
Allen-Gipson, DS; Sisson, JH; Spurzem, JR; Wong, J; Wyatt, TA1
Antonioli, L; Blandizzi, C; Colucci, R; Del Tacca, M; Fornai, M; Ghisu, N1
Cheng, JJ; Huang, NK; Lai, WL; Lin, YR; Lu, MK1
Alexander, SP; Beckett, SR; Harper, LK; Marsden, CA; McCreary, AC1
Baghdoyan, HA; Coleman, CG; Lydic, R1
Fang, X; Gao, N; Hu, HZ; Liu, S; Wang, GD; Wang, XY; Wood, JD; Xia, Y1
Ay, I; Tuncer, M1
Csóka, B; Deitch, EA; Haskó, G; Ledent, C; Lu, Q; Németh, ZH; Pacher, P; Spolarics, Z; Wilmanski, J; Xu, D1
Abbracchio, MP; Bates, G; Borea, PA; Camurri, A; Cattaneo, E; Tarditi, A; Varani, K; Woodman, B1
Aceves, J; Erlij, D; Florán, B; Florán, L; Gonzalez, B; Paz, F1
Greengard, P; Higashi, H; Kuroiwa, M; Nishi, A; Shuto, T; Snyder, GL; Sotogaku, N; Tanaka, M; Yabuuchi, K1
O'Leary, DS; Scislo, TJ1
Koos, BJ; Kruger, L; Linden, J; Murray, TF; Yan, X1
Day, YJ; Kern, JA; Li, Y; Linden, J; Liu, L; Oskouian, RJ; Rieger, JM1
Chan, ES; Chen, JF; Cronstein, BN; Delano, DL; Desai, A; Fernandez, P; Friedman, SL; Montesinos, MC; Pillinger, MH; Reiss, AB; Schwarzschild, MA; Yee, H1
Conde, SV; Gonzalez, C; Obeso, A; Rigual, R; Rocher, A; Vicario, I1
Brown, R; Fredholm, BB; Lai, EY; Mrowka, R; Patzak, A; Persson, AE; Persson, PB; Spielmann, N; Steege, A1
Huxley, VH; Wang, J1
Chan, ES; Chen, JF; Cronstein, BN; Desai, A; Fernandez, P; Khoa, DN; Merchant, AA; Montesinos, MC; Pillinger, MH; Reiss, AB; Schwarzschild, MA; Tomic-Canic, M; Trzaska, S; Tung, CF1
Ellman, PI; Kern, JA; Kron, IL; Laurent, JJ; Linden, J; Maxey, TS; Okonkwo, DO; Reece, TB; Tache-Leon, C; Tribble, CG1
Baunez, C; Bernardi, G; Calabresi, P; Centonze, D; De Chiara, V; Gubellini, P; Picconi, B; Prosperetti, C; Rossi, S; Tscherter, A1
Keith, BJ; Kristo, G; Lasley, RD; Mentzer, RM1
Auchampach, JA; Ge, ZD; Gross, GJ; Jacobson, MA; Kreckler, LM; Peart, JN; Wan, TC1
Grden, M; Kocbuch, K; Pawelczyk, T; Podgorska, M; Szutowicz, A1
Gao, C; Gao, N; Hu, HZ; Liu, S; Wood, JD; Xia, Y1
Cunha-Reis, D; Fontinha, BM; Ribeiro, JA; Sebastião, AM1
Hao, I; Leibovich, SJ; Pinhal-Enfield, G; Ramanathan, M1
Beukers, MW; Blad, CC; Brouwer, J; den Dulk, H; Ijzerman, AP; Li, Q; Ye, K1
Bairam, A; Kinkead, R; Montandon, G2
Fatokun, AA; Smith, RA; Stone, TW1
Einav, S; Galun, E; Linden, J; Matot, I; Rivo, J; Zeira, E1
Behan, WM; Stone, TW1
Agnati, L; Filip, M; Franco, R; Fuxe, K; Lluís, C; Marcellino, D; Navarro, G; Roberts, DC1
Biskup, W; Celiński, K; Cichoz-Lach, H; Czechowska, G; Korobowicz, E; Korolczuk, A; Madro, A; Prozorow-Król, B; Słomka, M1
Awad, AS; Huang, L; Li, L; Linden, J; Lobo, PI; McDuffie, M; Okusa, MD; Sevigny, CP1
Albasanz, JL; Castillo, CA; Fernández, M; Martín, M1
Bradding, P; Brightling, CE; Cruse, G; Duffy, SM1
Hurley, DJ; Moore, JN; Murray, TF; Sun, WC; Vandenplas, ML1
Fathollahi, Y; Hosseinmardi, N; Mirnajafi-Zadeh, J; Shahabi, P1
Canas, PM; Cunha, RA; Oliveira, CR; Porciúncula, LO; Silva, CG1
Hofmann, PA; Ledent, C; Morrison, RR; Mustafa, SJ; Tan, XL1
Hamano, R; Iwagaki, H; Kanke, T; Liu, K; Nishibori, M; Sendo, T; Takahashi, HK; Tanaka, N; Yoshino, T1
Fathollahi, Y; Mirnajafi-Zadeh, J; Palizvan, MR; Rezvani, ME1
Baranyi, M; Illes, P; Sperlágh, B; Vizi, ES; Zsilla, G1
Belcastro, V; Borsini, F; Calabresi, P; Centonze, D; Costa, C; Picconi, B; Tantucci, M; Tozzi, A; Tscherter, A1
Cao, Z; Hurley, DJ; Linden, J; Moore, JN; Murray, TF; Sun, WC; Vandenplas, ML1
Armida, M; Chen, JF; Domenici, MR; Grò, C; Martire, A; Pepponi, R; Popoli, P; Potenza, RL; Schwarzschild, MA; Tebano, MT1
Awad, AS; Linden, J; Liu, L; Okusa, MD; Rosin, DL; Rouse, M; Sedor, JR; Vergis, AL1
Albasanz, JL; Barrachina, M; Ferrer, I; Martín, M; Perez, S1
Binfaré, RW; Budni, J; Lobato, KR; Rodrigues, AL; Rosa, AO; Santos, AR1
Coskun, C; Mutlu, D; Savci, V; Suzer, O; Yalcin, M; Yilmaz, MS1
Blackburn, MR; Chan, ES; Chiriboga, L; Cronstein, BN; Fernández, P; Trzaska, S; Wilder, T1
Chen, JF; Kulik, T; Kung, D; Kusano, Y; Miekisiak, G; Winn, HR1
Broadley, KJ; Smith, N1
Casanello, P; Escudero, C; Sobrevia, L1
Cormack, LK; Feinberg, LM; Schallert, K; Schallert, T; Spinetta, MJ; Stroud, C; Woodlee, MT1
Cherezov, V; Chien, EY; Griffith, MT; Hanson, MA; Ijzerman, AP; Jaakola, VP; Lane, JR; Stevens, RC1
Bendor, J; Flajolet, M; Futter, M; Greengard, P; Nairn, AC; Nuangchamnong, N; Shen, W; Surmeier, DJ; Wallach, I; Wang, Z1
Hamilton, JB; Lancaster, DM; Patel, N; Pietersen, AN; Vreugdenhil, M1
Fathollahi, Y; Jahanshahi, A; Javan, M; Mirnajafi-Zadeh, J; Mohammad-Zadeh, M; Motamedi, F; Noorbakhsh, SM1
Ahlawat, R; Chavez-Valdez, R; Cristofalo, EA; Gauda, EB; Nathan, A; Wills-Karp, M1
Carlström, M; Lai, EY; Patzak, A; Persson, AE1
Baghdoyan, HA; Lydic, R; Van Dort, CJ1
Ichinose, TK; O'Leary, DS; Scislo, TJ1
Fernandes, D; Pamplona, FA; Pandolfo, P; Pires, VA; Prediger, RD; Takahashi, RN1
Miriel, VA; Rivers, RJ; Thengchaisri, N1
Church, JE; Coupar, IM; Pouton, CW; Rose'Meyer, RB; Urmaliya, VB; White, PJ1
Jin, M; Koizumi, S; Linden, J; Odashima, M; Ohnishi, H; Otaka, M; Watanabe, S1
Dziubina, A; Gołembiowska, K; Kamińska, K; Kowalska, M1
Autuori, A; Belcastro, V; Borsini, F; Calabresi, P; Costa, C; Di Filippo, M; Luchetti, E; Picconi, B; Siliquini, S; Tantucci, M; Tozzi, A1
Cipriani, S; Galli, A; Gianfriddo, M; Giovannini, MG; Mello, T; Pedata, F; Pugliese, AM; Traini, C1
Bertram, EH; Hargus, NJ; Patel, MK1
Abola, E; Brooks, CL; Dixon, JS; Michino, M; Moult, J; Stevens, RC1
Csóka, B; Haskó, G; Leibovich, SJ; Lukashev, D; Luo, W; Ramanathan, M; Sitkovsky, MV1
Ackerman, Z; Avraham, Y; Berry, EM; Magen, I; Mechoulam, R; Vorobiev, L1
Ferrante, A; Ferretti, R; Martire, A; Pepponi, R; Popoli, P1
Chen, JF; Chiodi, V; Domenici, MR; Ferrante, A; Frank, C; Ledent, C; Martire, A; Pepponi, R; Popoli, P; Tebano, MT1
Borea, PA; Catarzi, D; Colotta, V; Filacchioni, G; Lenzi, O; Morizzo, E; Moro, S; Paoletta, S; Poli, D; Varani, K; Varano, F; Vincenzi, F1
Maass, A; Müller, CE; Schiedel, AC; Sherbiny, FF1
Carroll, MA; Doumad, AB; Falck, JR; Li, J; Liclican, EL; Stier, CT; Wang, J1
Bernstein, SH; Burack, WR; Cochran, MR; Hilchey, SP; Hyrien, O; Kobie, JJ; Mosmann, TR; Quataert, SA; Secor-Socha, S; Wang, JC1
Aronhime, SN; Chen, JF; Echeverry, G; Kulik, TB; Kusano, Y; Miekisiak, G; Winn, HR1
Albasanz, JL; Barrachina, M; Buira, SP; Dentesano, G; Ferrer, I; Martín, M; Moreno, J1
Boeck, CR; Calo', G; de Castro, AA; Dos Santos Casagrande, T; Gavioli, EC; Guerrini, R; Martinello, C; Moretti, M1
Berghaus, LJ; Hurley, DJ; Linden, J; Moore, JN; Sun, WC; Thompson, R; Vandenplas, ML1
Abrol, R; Goddard, WA; Griffith, AR; Kim, SK; Li, Y; Trzaskowski, B1
Chen, SR; Li, DP; Pan, HL1
Arnould, I; Bellamy, JF; Besnard, F; Blouquit-Laye, S; Buenestado, A; Chapelier, A; Devillier, P; Grassin Delyle, S; Naline, E1
Cairo, G; Gammella, E; Tacchini, L1
Ijzerman, AP; Jaakola, VP; Katritch, V; Lane, JR; Lin, JY; Stevens, RC1
Ledent, C; Palmer, TM; Rutherford, C; Safhi, MM; Sands, WA1
Belcher, JD; Geng, JG; Huo, Y; Slungaard, A; Tang, R; Viollet, B; Wang, H; Wang, J; Wu, C; Zhang, C; Zhang, W; Zhu, C1
Pao, AC; Rajagopal, M1
Carlström, M; Welch, WJ; Wilcox, CS1
Ashok, Y; Jaakola, VP; Nanekar, RT; Piirainen, H1
Li, GQ; Lu, HH; Mo, Q; Qian, J; Tang, LM; Wang, F; Wang, XH; Zhu, J; Zhu, JF1
Fredholm, BB; Hao, JX; Li, L; Schulte, G; Wiesenfeld-Hallin, Z; Xu, XJ1
Ledent, C; Pouton, CW; Short, JL; Urmaliya, VB; White, PJ1
Beukers, MW; Guo, D; Ijzerman, AP; Müller, CE; Peeters, MC; van Westen, GJ; Wisse, LE1
Che, PL; Du, J; Ha, B; Wang, Z; Yarema, KJ1
Casadó, V; Cinca, J; Ciruela, F; Fernandes, J; Franco, R; Hove-Madsen, L; Llach, A; Lluís, C; Molina, CE; Prat-Vidal, C1
Alves-Do-Prado, W; Bornia, EC; Correia-de-Sá, P1
Carlini, M; Cesari, D; Da Pozzo, E; Daniele, S; Dell'Osso, L; Golia, F; Martini, C; Panighini, A; Picchetti, M; Trincavelli, ML1
Cherezov, V; Gao, ZG; Han, GW; Jacobson, KA; Katritch, V; Stevens, RC; Wu, H; Xu, F1
Chen, JF; Feng, L; Garcia, GE; Johnson, RJ; Truong, LD1
Choukèr, A; Feuerecker, M; Kaufmann, I; Salam, A; Schelling, G; Thiel, M1
Bennett, K; Edwards, PC; Langmead, CJ; Lebon, G; Leslie, AG; Tate, CG; Warne, T1
Andrews, SP; Congreve, M; Errey, JC; Marshall, FH; Mason, JS; Robertson, N; Tehan, B; Weir, M; Zhukov, A1
Cronstein, BN; Williams, AJ1
Brown, RM; Duncan, JR; Lawrence, AJ; Ledent, C; Stagnitti, MR1
Bennett, K; Congreve, M; Doré, AS; Errey, JC; Hollenstein, K; Hurrell, E; Magnani, F; Marshall, FH; Ng, I; Robertson, N; Tate, CG; Tehan, B; Weir, M1
Ayers, PW; Burger, SK; Liu, Y; Vöhringer-Martinez, E1
Moriya, T; Nakahata, N; Nakata, H; Obara, Y; Suzuki, T1
Akamine, AT; Almeida, VI; Crippa, JA; Dal-Pizzol, F; Ferraz-de-Paula, V; Hallak, JE; Mariano-Souza, DP; Palermo-Neto, J; Pinheiro, ML; Quevedo, J; Quinteiro-Filho, WM; Ribeiro, A; Vitoretti, LB; Zuardi, AW1
Chancellor, MB; de Groat, WC; Kitta, T; Kuno, S; Nonomura, K; Yoshimura, N1
Dell'anno, MT; Fisone, G; Pallottino, S1
Chen, X; Kang, H; Li, X; Liu, X; Liu, Z; Shu, K; Zhu, S1
Blanco, C; Colettis, N; Hartley, RC; Harvey, AL; Jamieson, AG; Jerusalinsky, D; Kornisiuk, E; Snitcofsky, M; Stone, TW; Young, LC1
Chiriboga, L; Cronstein, BN; Perez-Aso, M1
Lochner, A; Moolman, JA; Salie, R1
Cherezov, V; Chubukov, P; Chun, E; Han, GW; Heitman, LH; IJzerman, AP; Katritch, V; Liu, W; Roth, CB; Stevens, RC; Thompson, AA; Xu, F1
Azevedo, MS; Cechinel-Filho, V; Ferreira, VM; Lucena, GM; Matheus, FC; Prediger, RD; Tessele, PB1
Falck, JR; Morisseau, C; Mustafa, SJ; Nayeem, MA; Pradhan, I; Zeldin, DC1
Coppi, E; Galli, A; Maraula, G; Mello, T; Pedata, F; Pugliese, AM; Traini, C1
Martins, DF; Mazzardo-Martins, L; Piovezan, AP; Santos, AR; Soldi, F; Stramosk, J1
Ashok, Y; Jaakola, VP; Nanekar, RT1
Ailawadi, G; Barbery, C; Bhamidipati, CM; Kron, IL; Laubach, VE; Meher, AK; Mehta, GS; Moehle, CW; Owens, GK; Sharma, AK; Su, G; Upchurch, GR; Vigneshwar, NG1
Adams, C; Choi, DS; Hinton, DJ; Kang, NY; Kim, T; Lee, MR; Nam, HW; Oliveros, A; Ruby, CL1
An, JH; Chen, JF; Dai, SS; Li, W; Ning, YL; Wang, H; Yang, N; Zhou, YG; Zhu, PF1
Han, K; Pang, X; Yang, M1
Almerico, AM; Lauria, A; Pantano, L; Tutone, M1
Capuano, B; Jörg, M; Mak, FS; Miller, ND; Scammells, PJ; Shonberg, J; Yuriev, E1
Alam, MN; Hsieh, KC; Kumar, S; McGinty, D; Rai, S; Szymusiak, R1
Agostinho, P; Castro, AA; Cunha, RA; Garção, P; Köfalvi, A; Prediger, RD; Szabó, EC; Tomé, ÂR; Wopereis, S1
Bacilieri, M; Cacciari, B; Ciancetta, A; Cosconati, S; Da Settimo, F; Federico, S; Klotz, KN; Moro, S; Novellino, E; Paoletta, S; Spalluto, G; Taliani, S1
Carrillo-Salinas, FJ; Feliú, A; Guaza, C; Iñigo, PM; Mecha, M; Mestre, L1
Antonia, SJ; Khalil, FK; Luddy, K; Mediavilla-Varela, M; Neuger, AM; Noyes, D; Soliman, H1
Feng, LY; Huang, L; Wu, DD; Zhang, L1
Bencivelli, D; Borea, PA; Casetta, I; Corciulo, C; Gentile, M; Granieri, E; Varani, K; Vincenzi, F1
Bernardo, A; De Nuccio, C; Ferrante, A; Minghetti, L; Pepponi, R; Popoli, P; Visentin, S1
Minic, Z; O'Leary, DS; Scislo, TJ1
Alves-Do-Prado, W; Ambiel, CR; Antônio, MB; Correia-de-Sá, P; de Paula Ramos, E1
Alarcón, M; Badimon, L; Caballero, J; Fuentes, E; Padró, T; Palomo, I; Pérez, P; Vilahur, G1
Frøbert, O; Hedegaard, ER; Mogensen, S; Nielsen, BD; Rembold, CM; Simonsen, U1
Albasanz, JL; Barrachina, M; Blanch, M; Díaz-Sánchez, S; Ferrer, I; Martín, M; Monje, A; Pereira-Veiga, T; Planchat, LM; Villar-Menéndez, I1
Exley, M; Kini, R; Madasu, M; Nowak, M; Ohta, A; Sitkovsky, M; Subramanian, M1
Bruzzese, L; By, Y; Condo, J; Durand-Gorde, JM; Fenouillet, E; Fromonot, J; Guieu, R; Kipson, N; Ruf, J1
Brussee, J; Guo, D; Hazeu, M; Heitman, LH; Ijzerman, AP; Mocking, T; van Veldhoven, JP; Xia, L1
Alarcón, M; Caballero, J; Fuentes, E; Palomo, I; Rojas, A1
Lappas, CM1
Arias-Montaño, JA; Escamilla-Sánchez, J; González-Pantoja, R; Márquez-Gómez, R; Morales-Figueroa, GE1
Liu, W; Manaenko, A; Sun, X; Ye, Z; Zhang, L; Zhang, R1
Dimitrieva, TV; Pliyev, BK; Savchenko, VG1
Åqvist, J; Gutiérrez-de-Terán, H; Keränen, H1
Cataño-Cañizalez, YG; Cortés-Garcia, JD; Cortez-Espinosa, N; Guzman-Flores, JM; Portales-Perez, DP; Rodríguez-Rivera, JG; Vargas-Morales, JM1
Bilos, A; Geraci, S; Gretz, N; Heemskerk, S; Kraenzlin, B; Masereeuw, R; Peters, E; Pickkers, P; Wilmer, MJ1
Chaimovitz, C; Douvdevani, A; Eini, H; Frishman, V; Kachko, L; Lewis, EC; Yulzari, R1
Cortés-Garcia, JD; Cortez-Espinosa, N; García-Hernández, MH; Guzmán-Flores, JM; Layseca-Espinosa, E; López-López, C; Portales-Cervantes, L; Portales-Pérez, DP1
Kimura, E; Matsuno, A; Midorikawa, T; Monoi, N; Murakoshi, M; Nagamori, Y; Nakamura, Y; Nishino, H; Oka, K; Sano, T; Sugafuji, T; Sugiyama, K; Uchiyama, A; Urade, Y1
Cronstein, BN; Levine, J; Low, YC; Mediero, A; Perez-Aso, M1
Guo, D; Hankemeier, T; Hölscher, A; Holzheimer, M; IJzerman, AP; Louvel, J; Massink, A; Spijksma, G1
Cai, L; Luo, HM; Pi, T; Ren, XM; Su, CF; Wu, WT; Zhang, W; Zhou, XW1
Sabio, M; Topiol, S1
Christopoulos, A; Gregory, KJ; May, LT; Tan, CY; Vecchio, EA; White, PJ1
Dror, RO; Guo, D; Heitman, LH; IJzerman, AP; Liu, R; Mocking, T; Pan, AC; Shaw, DE1
Huang, P; Huang, S; Liu, X; Luo, X; Qi, J; Shen, X; Wang, J; Yang, Z; Zhong, Y1
Bortolato, A; Cheng, RK; Cooke, RM; Deflorian, F; Doré, AS; Errey, JC; Guo, D; Heitman, LH; IJzerman, AP; Marshall, FH; Segala, E1
Bethge, P; Blanchet, C; Cunha, RA; Frick, A; Gonçalves, FQ; Gonçalves, N; Gorlewicz, A; Grosjean, N; Haberl, MG; Lemos, C; Malezieux, M; Mulle, C; Nägerl, UV; Viana da Silva, S; Zhang, P1
Kimura, E; Midorikawa, T; Monoi, N; Murakoshi, M; Murata-Matsuno, A; Nakamura, Y; Nishino, H; Oka, K; Sano, T; Sugafuji, T; Sugiyama, K; Uchiyama, A; Urade, Y1
Amin, MN; Chiang, MJ; Cole, PA; Gabrielson, K; Giddens, J; Hsiao, PY; Kalin, JH; Lo, YC; Powell, JD; Sun, IH; Sysa-Shah, P; Wang, LX1
Bonaventura, J; Brugarolas, M; Casadó, V; Cellai, L; Chang, CP; Chern, Y; Cortés, A; Dettori, I; Ferré, S; Guitart, X; Narayanan, M; Orrú, M; Pedata, F; Rea, W1
Adam, RM; Chung, YG; Cristofaro, V; Doyle, C; Lukianov, SN; Sack, BS; Schäfer, M; Sullivan, MP1
Bai, W; Chen, JF; Chen, X; Chen, XY; Li, P; Liu, D; Ning, YL; Peng, Y; Wang, H; Yang, N; Zhao, Y; Zhao, ZA; Zhou, YG1
Colmenero, AV; Gabel, M; Hambrecht-Wiedbusch, VS; Imperial, JP; Liu, LJ; Vanini, G1
Guo, D; IJzerman, AP1
Chen, JF; Li, P; Ning, YL; Peng, Y; Yang, N; Zeng, XJ; Zhao, Y; Zhao, ZA; Zhou, YG1
Ernst, OP; García, AE; Larda, ST; Lyda, B; Neale, C; Pichugin, D; Pomès, R; Prosser, RS; Sljoka, A; Sunahara, RK; Tsuchimura, N; Ye, L1
Bajnok, A; Orbán, C; Sava, F; Toldi, G; Vásárhelyi, Z1
Ávila-Ibarra, LR; de Lourdes Mora-García, M; Del Carmen Fuentes-Castañeda, M; Don-López, CA; García-Rocha, R; Gutiérrez-Serrano, V; Hernández-Montes, J; Monroy-García, A; Torres-Pineda, DB; Weiss-Steider, B1
Cao, J; Dong, Z; Li, W; Lin, H; Shi, Y; Xiao, R; Zhang, X1
Chelvanambi, M; Fabian, KPL; Hong, CS; Lang, S; Ludwig, S; Razzo, BM; Storkus, WJ; Whiteside, TL1
Dziodzio, J; Eldridge, A; Emery, IF; Ichinose, F; Leclerc, A; Lord, C; Lucas, FL; May, T; McCrum, B; Riker, R; Robich, MP; Ryzhov, S; Sawyer, DB; Seder, DB1
Conde, SV; Gonzalez, C; Martins, FO; Melo, BF; Monteiro, EC; Olea, E; Prieto-Lloret, J; Ribeiro, MJ; Sacramento, JF1
Baudry, JY; Green, AT; Hu, X; Humphreys, BM; Parks, JM; Smith, JC; Smith, MD1
Bill, RM; Dafforn, TR; Jamshad, M; Lin, YP; Little, HA; Poyner, DR; Routledge, SJ; Simms, J; Spickett, CM; Thakker, A; Wheatley, M1
Byeon, JJ; Choi, JM; Kim, N; Lee, BI; Lim, JH; Na, YG; Park, MH; Park, MJ; Park, SJ; Park, Y; Shin, SH; Shin, YG1
Buccioni, M; Coelho, JE; Dal Ben, D; Lambertucci, C; Lopes, LV; Marques-Morgado, I; Martí Navia, A; Marucci, G; Spinaci, A; Volpini, R1
Dong, X; Fan, Y; Li, L; Liu, X; Lu, Q; Sun, B; Yang, Y; Zhang, H; Zhao, J; Zhu, J1
Briddon, SJ; Franks, HA; Harwood, CR; Hill, SJ; Kellam, B; Kindon, ND; Otun, O; Patera, F; Stoddart, LA; Veprintsev, DB; Woolard, J1

Reviews

3 review(s) available for triazoles and zm 241385

ArticleYear
Community-wide assessment of GPCR structure modelling and ligand docking: GPCR Dock 2008.
    Nature reviews. Drug discovery, 2009, Volume: 8, Issue:6

    Topics: Animals; Crystallization; Crystallography, X-Ray; Drug Design; Drug Industry; Humans; Ligands; Models, Molecular; Predictive Value of Tests; Protein Binding; Receptor, Adenosine A2A; Receptors, G-Protein-Coupled; Structure-Activity Relationship; Triazines; Triazoles

2009
Structural features of adenosine receptors: from crystal to function.
    Biochimica et biophysica acta, 2011, Volume: 1808, Issue:5

    Topics: Crystallography, X-Ray; Humans; Protein Conformation; Receptors, Purinergic P1; Triazines; Triazoles

2011
Molecular Basis of Ligand Dissociation from G Protein-Coupled Receptors and Predicting Residence Time.
    Methods in molecular biology (Clifton, N.J.), 2018, Volume: 1705

    Topics: Cholinergic Antagonists; Drug Discovery; Humans; Kinetics; Ligands; Models, Molecular; Molecular Conformation; Molecular Docking Simulation; Molecular Dynamics Simulation; Protein Binding; Quantitative Structure-Activity Relationship; Receptors, Cholinergic; Receptors, G-Protein-Coupled; Receptors, Purinergic P1; Tiotropium Bromide; Triazines; Triazoles

2018

Trials

3 trial(s) available for triazoles and zm 241385

ArticleYear
Effects of doxazosin and propranolol on A2A adenosine receptors in essential hypertension.
    Hypertension (Dallas, Tex. : 1979), 2002, Volume: 40, Issue:6

    Topics: Adenosine-5'-(N-ethylcarboxamide); Adult; Antihypertensive Agents; Binding, Competitive; Blood Pressure; Body Mass Index; Cyclic AMP; Diastole; Doxazosin; Female; Humans; Hypertension; Lymphocytes; Male; Middle Aged; Neutrophils; Propranolol; Radioligand Assay; Receptor, Adenosine A2A; Receptors, Purinergic P1; Reference Values; Systole; Treatment Outcome; Triazines; Triazoles

2002
Plasma glutamate-modulated interaction of A2AR and mGluR5 on BMDCs aggravates traumatic brain injury-induced acute lung injury.
    The Journal of experimental medicine, 2013, Apr-08, Volume: 210, Issue:4

    Topics: Acute Lung Injury; Adenosine; Adenosine A2 Receptor Agonists; Adult; Animals; Bone Marrow Cells; Brain Injuries; Disease Models, Animal; Female; Glutamic Acid; Humans; Male; Mice; Mice, Knockout; Middle Aged; Phenethylamines; Protein Kinase C; Receptor, Adenosine A2A; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Signal Transduction; Triazines; Triazoles; Type C Phospholipases

2013
Japanese sake yeast supplementation improves the quality of sleep: a double-blind randomised controlled clinical trial.
    Journal of sleep research, 2016, Volume: 25, Issue:1

    Topics: Adenosine A2 Receptor Antagonists; Adult; Alcoholic Beverages; Cell Extracts; Cross-Over Studies; Double-Blind Method; Electroencephalography; Female; HEK293 Cells; Humans; Male; Powders; Receptor, Adenosine A2A; Saccharomyces cerevisiae; Sleep; Sleep Stages; Triazines; Triazoles

2016

Other Studies

341 other study(ies) available for triazoles and zm 241385

ArticleYear
In vivo characterisation of ZM 241385, a selective adenosine A2A receptor antagonist.
    European journal of pharmacology, 1996, Apr-22, Volume: 301, Issue:1-3

    Topics: Adenosine; Animals; Cardiovascular Agents; Decerebrate State; Dogs; Female; Heart Rate; Hindlimb; In Vitro Techniques; Myocardial Contraction; Purinergic P1 Receptor Antagonists; Rats; Rats, Inbred SHR; Regional Blood Flow; Triazines; Triazoles; Vasodilation

1996
Activation of multiple sites by adenosine analogues in the rat isolated aorta.
    British journal of pharmacology, 1996, Volume: 118, Issue:6

    Topics: Adenosine; Animals; Aorta, Thoracic; Endothelium, Vascular; Enzyme Inhibitors; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Rats; Rats, Wistar; Receptors, Purinergic P1; Sulfonamides; Theophylline; Triazines; Triazoles; Xanthines

1996
Pharmacodynamics of ZM 241385, a potent A2a adenosine receptor antagonist, after enteric administration in rat, cat and dog.
    The Journal of pharmacy and pharmacology, 1996, Volume: 48, Issue:6

    Topics: Administration, Oral; Animals; Cats; Dogs; Drug Interactions; Female; Hemodynamics; Hypertension; Injections, Intravenous; Intubation, Gastrointestinal; Male; Purinergic P1 Receptor Antagonists; Rats; Species Specificity; Theophylline; Triazines; Triazoles; Vasodilation; Vasodilator Agents

1996
125I-4-(2-[7-amino-2-[2-furyl][1,2,4]triazolo[2,3-a][1,3,5] triazin-5-yl-amino]ethyl)phenol, a high affinity antagonist radioligand selective for the A2a adenosine receptor.
    Molecular pharmacology, 1995, Volume: 48, Issue:6

    Topics: Animals; Cattle; CHO Cells; Cricetinae; Iodine Radioisotopes; Purinergic P1 Receptor Antagonists; Radioligand Assay; Receptors, Purinergic P1; Recombinant Proteins; Triazines; Triazoles

1995
The role of the A(2A) adenosine receptor subtype in functional hyperaemia in the hindlimb of anaesthetized cats.
    The Journal of physiology, 1996, Apr-15, Volume: 492 ( Pt 2)

    Topics: Adenosine; Animals; Arteries; Cats; Gases; Hindlimb; Hydrogen-Ion Concentration; Hyperemia; Isometric Contraction; Male; Muscles; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Regional Blood Flow; Theophylline; Triazines; Triazoles

1996
Ischaemic skeletal muscle hyperaemia in the anaesthetized cat: no contribution of A2A adenosine receptors.
    The Journal of physiology, 1997, Apr-01, Volume: 500 ( Pt 1)

    Topics: Anesthesia, General; Animals; Blood Pressure; Cats; Electric Stimulation; Femoral Nerve; Hindlimb; Hyperemia; Ischemia; Isometric Contraction; Male; Muscle Contraction; Muscle, Skeletal; Oxygen Consumption; Purinergic P1 Receptor Antagonists; Receptor, Adenosine A2A; Receptors, Purinergic P1; Regional Blood Flow; Sciatic Nerve; Triazines; Triazoles

1997
Adenosine analogues relax guinea-pig taenia caeci via an adenosine A2B receptor and a xanthine-resistant site.
    European journal of pharmacology, 1997, Mar-26, Volume: 323, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cecum; Dose-Response Relationship, Drug; Guinea Pigs; Male; Muscle Relaxation; Muscle, Smooth; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Theophylline; Triazines; Triazoles; Vasodilator Agents; Xanthines

1997
Desensitisation of the adenosine A1 receptor by the A2A receptor in the rat striatum.
    Journal of neurochemistry, 1997, Volume: 69, Issue:1

    Topics: Adenosine; Animals; Antihypertensive Agents; Corpus Striatum; Enzyme Inhibitors; Isoquinolines; Phenethylamines; Presynaptic Terminals; Protein Kinase C; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Purinergic P1; Sensitivity and Specificity; Sulfonamides; Synaptosomes; Triazines; Triazoles; Tritium; Xanthines

1997
Memory of extracellular adenosine A2A purinergic receptor-mediated signaling in murine T cells.
    The Journal of biological chemistry, 1997, Oct-10, Volume: 272, Issue:41

    Topics: Adenosine; Animals; Cell Division; Exocytosis; Extracellular Matrix; Fas Ligand Protein; fas Receptor; Interleukin-2; Membrane Glycoproteins; Mice; Mice, Inbred DBA; Phenethylamines; Purinergic P1 Receptor Agonists; Receptor, Adenosine A2A; Receptors, Antigen, T-Cell; Receptors, Purinergic P1; Signal Transduction; T-Lymphocytes; Triazines; Triazoles

1997
ZM241385 is an antagonist of the facilitatory responses produced by the A2A adenosine receptor agonists CGS21680 and HENECA in the rat hippocampus.
    British journal of pharmacology, 1997, Volume: 122, Issue:7

    Topics: Acetylcholine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Antihypertensive Agents; Binding Sites; Hippocampus; Ligands; Membranes; Phenethylamines; Platelet Aggregation Inhibitors; Purinergic P1 Receptor Agonists; Rats; Synaptic Transmission; Synaptosomes; Triazines; Triazoles; Visual Cortex

1997
Activation of two sites by adenosine receptor agonists to cause relaxation in rat isolated mesenteric artery.
    British journal of pharmacology, 1997, Volume: 122, Issue:7

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Anti-Arrhythmia Agents; Dinucleoside Phosphates; Dose-Response Relationship, Drug; Male; Mesenteric Arteries; Purinergic P1 Receptor Agonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Theophylline; Triazines; Triazoles; Vasodilation; Vasodilator Agents

1997
Adenosine A1 receptor-mediated activation of AMP-activated protein kinase in bovine bronchial rings.
    Biochemical Society transactions, 1997, Volume: 25, Issue:4

    Topics: Adenosine-5'-(N-ethylcarboxamide); Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Bronchi; Cattle; Enzyme Activation; In Vitro Techniques; Multienzyme Complexes; Phenylisopropyladenosine; Protein Kinases; Protein Serine-Threonine Kinases; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Ribonucleotides; Triazines; Triazoles; Xanthines

1997
Inhibitory effect of adenosine on degranulation of human cultured mast cells upon cross-linking of Fc epsilon RI.
    Biochemical and biophysical research communications, 1998, Jan-26, Volume: 242, Issue:3

    Topics: Adenosine; Antibodies; Chymases; Cross-Linking Reagents; Cyclic AMP; Guanosine; Humans; Immunoglobulin E; Mast Cells; Mitogen-Activated Protein Kinase 1; Phenethylamines; Phosphorylation; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, IgE; RNA, Messenger; Serine Endopeptidases; Thioinosine; Thionucleosides; Triazines; Triazoles; Tryptases

1998
Adenosine modulates hypoxia-induced responses in rat PC12 cells via the A2A receptor.
    The Journal of physiology, 1998, Apr-01, Volume: 508 ( Pt 1)

    Topics: Adenosine; Adenosine Deaminase; Adrenal Gland Neoplasms; Animals; Calcium; Cell Hypoxia; Fluorescent Dyes; Fura-2; Lung; Membrane Potentials; Patch-Clamp Techniques; PC12 Cells; Pheochromocytoma; Purinergic P1 Receptor Antagonists; Rats; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Receptor, Adenosine A3; Receptors, Purinergic P1; RNA, Messenger; Theophylline; Transcription, Genetic; Triazines; Triazoles

1998
Role of adenosine and its receptors in the vasodilatation induced in the cerebral cortex of the rat by systemic hypoxia.
    The Journal of physiology, 1998, Jun-01, Volume: 509 ( Pt 2)

    Topics: Adenosine; Animals; Blood Flow Velocity; Blood-Brain Barrier; Erythrocytes; Hypoxia; Laser-Doppler Flowmetry; Male; Parietal Lobe; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Theophylline; Triazines; Triazoles; Vasodilation

1998
Protection against kainate-induced excitotoxicity by adenosine A2A receptor agonists and antagonists.
    Neuroscience, 1998, Volume: 85, Issue:1

    Topics: Adenosine; Animals; Excitatory Amino Acid Agonists; Hippocampus; Kainic Acid; Male; Neurons; Neuroprotective Agents; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Triazines; Triazoles; Xanthines

1998
Protection against hippocampal kainate excitotoxicity by intracerebral administration of an adenosine A2A receptor antagonist.
    Brain research, 1998, Aug-03, Volume: 800, Issue:2

    Topics: Adenosine; Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Brain Chemistry; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Hippocampus; Kainic Acid; Male; Neurotoxins; Phenethylamines; Rats; Rats, Wistar; Triazines; Triazoles

1998
Binding affinity of adenosine receptor agonists and antagonists at human cloned A3 adenosine receptors.
    Life sciences, 1998, Volume: 63, Issue:5

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Binding, Competitive; Cell Line; Cloning, Molecular; Humans; Kidney; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyrimidines; Quinazolines; Receptor, Adenosine A3; Receptors, Purinergic P1; Transfection; Triazines; Triazoles

1998
A2A-adenosine receptor reserve for coronary vasodilation.
    Circulation, 1998, Aug-18, Volume: 98, Issue:7

    Topics: Adenosine; Animals; Coronary Circulation; Female; Guinea Pigs; Heart; In Vitro Techniques; Kinetics; Male; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyrimidines; Receptor, Adenosine A2A; Receptors, Purinergic P1; Triazines; Triazoles; Vasodilation

1998
The role of adenosine in rat coronary flow regulation during respiratory and metabolic acidosis.
    European journal of pharmacology, 1998, Sep-04, Volume: 356, Issue:2-3

    Topics: Acidosis; Acidosis, Respiratory; Adenosine; Animals; Caffeine; Coronary Circulation; Hypercapnia; Male; Purinergic P1 Receptor Antagonists; Pyrimidines; Rats; Rats, Sprague-Dawley; Theophylline; Triazines; Triazoles

1998
Adenosine receptor subtypes and vasodilatation in rat skeletal muscle during systemic hypoxia: a role for A1 receptors.
    The Journal of physiology, 1999, Jan-01, Volume: 514 ( Pt 1)

    Topics: Adenosine; Animals; Antihypertensive Agents; Blood Gas Analysis; Hydrogen-Ion Concentration; Hypoxia; Male; Muscle, Skeletal; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Regional Blood Flow; Respiration; Triazines; Triazoles; Vasodilation; Vasodilator Agents; Xanthines

1999
Interaction between adenosine A1 and A2 receptor-mediated responses in the rat hippocampus in vitro.
    European journal of pharmacology, 1998, Nov-27, Volume: 362, Issue:1

    Topics: Adenosine; Animals; Excitatory Postsynaptic Potentials; Hippocampus; Male; Organ Culture Techniques; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyrazines; Rats; Rats, Wistar; Receptors, Purinergic P1; Triazines; Triazoles

1998
Adenosine A2a receptors increase arterial endothelial cell nitric oxide.
    The Journal of surgical research, 1998, Volume: 80, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Carotid Arteries; Cells, Cultured; Endothelium, Vascular; Humans; Iliac Artery; Nitric Oxide; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Quinazolines; Receptor, Adenosine A2A; Receptors, Purinergic P1; Swine; Triazines; Triazoles; Xanthines

1998
Comparison of CGS 15943, ZM 241385 and SCH 58261 as antagonists at human adenosine receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:1

    Topics: Animals; Cell Line; CHO Cells; Cricetinae; Cyclic AMP; Humans; Purinergic P1 Receptor Antagonists; Pyrimidines; Quinazolines; Rats; Transfection; Triazines; Triazoles; Xanthines

1999
Adenosine A1 receptor-mediated antiadrenergic effects are modulated by A2a receptor activation in rat heart.
    The American journal of physiology, 1999, Volume: 276, Issue:2

    Topics: Adenosine; Adrenergic alpha-Antagonists; Animals; Calcium; Drug Synergism; Heart; In Vitro Techniques; Intracellular Membranes; Male; Myocardium; Osmolar Concentration; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Triazines; Triazoles

1999
Sensitization by chronic diazepam treatment of A2A adenosine receptor-mediated relaxation in rat pulmonary artery.
    Life sciences, 1999, Volume: 64, Issue:2

    Topics: Adenosine; Animals; Carrier Proteins; Diazepam; Dinucleoside Phosphates; Dipyridamole; Dose-Response Relationship, Drug; Female; Heart; Heart Atria; Muscle Relaxation; Phenethylamines; Pulmonary Artery; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Purinergic P1; Thioinosine; Triazines; Triazoles; Verapamil

1999
G protein coupling of CGS 21680 binding sites in the rat hippocampus and cortex is different from that of adenosine A1 and striatal A2A receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:4

    Topics: Adenosine; Animals; Binding Sites; Binding, Competitive; Brain; Cerebral Cortex; Cholera Toxin; Corpus Striatum; Ethylmaleimide; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Hippocampus; Male; Membranes; Pertussis Toxin; Phenethylamines; Purinergic P1 Receptor Agonists; Pyrimidines; Rats; Rats, Wistar; Receptors, Purinergic P1; Triazines; Triazoles; Tritium; Virulence Factors, Bordetella

1999
Selective A2A adenosine receptor activation reduces ischemia-reperfusion injury in rat kidney.
    The American journal of physiology, 1999, Volume: 277, Issue:3

    Topics: Animals; Humans; Kidney; Male; Necrosis; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Reperfusion Injury; Triazines; Triazoles

1999
Increase in the number, G protein coupling, and efficiency of facilitatory adenosine A2A receptors in the limbic cortex, but not striatum, of aged rats.
    Journal of neurochemistry, 1999, Volume: 73, Issue:4

    Topics: Adenosine; Aging; Animals; Cell Membrane; Cerebral Cortex; Corpus Striatum; Cyclic AMP; Dentate Gyrus; GTP-Binding Proteins; Kinetics; Limbic System; Male; Organ Specificity; Phenethylamines; Purinergic P1 Receptor Agonists; Radioligand Assay; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Purinergic P1; Triazines; Triazoles; Tritium

1999
Autoradiographic comparison of the potency of several structurally unrelated adenosine receptor antagonists at adenosine A1 and A(2A) receptors.
    European journal of pharmacology, 1999, Sep-10, Volume: 380, Issue:2-3

    Topics: Adenosine; Animals; Autoradiography; Binding, Competitive; Brain; Caffeine; In Vitro Techniques; Male; Phenethylamines; Purinergic P1 Receptor Antagonists; Pyrazines; Quinazolines; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Receptors, Purinergic P1; Theophylline; Triazines; Triazoles; Tritium; Xanthines

1999
Neutrophil A2A adenosine receptor inhibits inflammation in a rat model of meningitis: synergy with the type IV phosphodiesterase inhibitor, rolipram.
    The Journal of infectious diseases, 1999, Volume: 180, Issue:5

    Topics: Adenosine; Animals; Blood-Brain Barrier; Cell Adhesion; Cyclic AMP; Disease Models, Animal; Drug Synergism; Humans; Leukocytosis; Meningitis, Bacterial; Neutrophil Activation; Neutrophils; Phosphodiesterase Inhibitors; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Purinergic P1; Respiratory Burst; Rolipram; Superoxides; Triazines; Triazoles; Tumor Necrosis Factor-alpha

1999
Selective reduction in A2 adenosine receptor desensitization following antisense-induced suppression of G protein-coupled receptor kinase 2 expression.
    Journal of neurochemistry, 1999, Volume: 73, Issue:5

    Topics: Animals; beta-Adrenergic Receptor Kinases; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; DNA, Antisense; G-Protein-Coupled Receptor Kinase 2; G-Protein-Coupled Receptor Kinase 3; Gene Expression; Glioma; Homeostasis; Hybrid Cells; Mice; Neuroblastoma; Phosphorylation; Rats; Receptors, Purinergic P1; Transfection; Triazines; Triazoles; Tumor Cells, Cultured

1999
Stimulation of A(2A) adenosine receptor phosphorylation by protein kinase C activation: evidence for regulation by multiple protein kinase C isoforms.
    Biochemistry, 1999, Nov-09, Volume: 38, Issue:45

    Topics: Acetophenones; Animals; Benzopyrans; Carbazoles; CHO Cells; Consensus Sequence; Cricetinae; Cyclic AMP; Dogs; Endothelin-1; Enzyme Activation; Enzyme Inhibitors; Glioma; Indoles; Isoenzymes; Maleimides; Mutagenesis, Site-Directed; Phosphorylation; Protein Kinase C; Rats; Receptor, Adenosine A2A; Receptors, Purinergic P1; Signal Transduction; Tetradecanoylphorbol Acetate; Triazines; Triazoles; Tumor Cells, Cultured

1999
Effect of A2A adenosine receptor stimulation and antagonism on synaptic depression induced by in vitro ischaemia in rat hippocampal slices.
    British journal of pharmacology, 1999, Volume: 128, Issue:5

    Topics: Adenosine; Animals; Excitatory Postsynaptic Potentials; Hippocampus; Hypoxia-Ischemia, Brain; In Vitro Techniques; Male; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyrimidines; Rats; Rats, Wistar; Receptor, Adenosine A2A; Synapses; Synaptic Transmission; Triazines; Triazoles; Xanthines

1999
Adenosine inhibits a non-inactivating K+ current in bovine adrenal cortical cells by activation of multiple P1 receptors.
    The Journal of physiology, 1999, Nov-15, Volume: 521 Pt 1

    Topics: Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Cattle; GTP-Binding Proteins; In Vitro Techniques; Male; Membrane Potentials; Patch-Clamp Techniques; Potassium; Potassium Channel Blockers; Potassium Channels; Receptors, Purinergic P1; Signal Transduction; Triazines; Triazoles; Xanthines; Zona Fasciculata

1999
Sensitization of visceral afferents to bradykinin in rat jejunum in vitro.
    The Journal of physiology, 1999, Dec-01, Volume: 521 Pt 2

    Topics: Adenosine; Animals; Bradykinin; Bucladesine; Cyclooxygenase Inhibitors; Dinoprostone; Histamine; Histamine Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Jejunum; Male; Membrane Potentials; Naproxen; Neurons, Afferent; Piperidines; Ranitidine; Rats; Rats, Inbred Strains; Serotonin; Stimulation, Chemical; Triazines; Triazoles; Xanthines

1999
Increase in the vasorelaxant potency of K(ATP) channel opening drugs by adenosine A(1) and A(2) receptors in the pig coronary artery.
    European journal of pharmacology, 1999, Oct-27, Volume: 383, Issue:2

    Topics: Adenosine; Animals; ATP-Binding Cassette Transporters; Coronary Vessels; Cromakalim; Dose-Response Relationship, Drug; Drug Interactions; In Vitro Techniques; KATP Channels; Nicorandil; Phenethylamines; Pinacidil; Potassium Channels; Potassium Channels, Inwardly Rectifying; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Swine; Triazines; Triazoles; Vasodilator Agents; Xanthines

1999
ZM 241385, an adenosine A(2A) receptor antagonist, inhibits hippocampal A(1) receptor responses.
    European journal of pharmacology, 1999, Nov-03, Volume: 383, Issue:3

    Topics: Animals; Dinucleoside Phosphates; Enzyme Inhibitors; Hippocampus; Male; Phenylisopropyladenosine; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Purinergic P1; Triazines; Triazoles

1999
Afferent arteriolar adenosine A2a receptors are coupled to KATP in in vitro perfused hydronephrotic rat kidney.
    The American journal of physiology, 1999, Volume: 277, Issue:6

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Arterioles; Blood Pressure; Enzyme Inhibitors; Hydronephrosis; Kidney; Perfusion; Potassium Channels; Potassium Chloride; Rats; Receptor, Adenosine A2A; Receptors, Purinergic P1; Renal Artery; Renal Circulation; Triazines; Triazoles; Vasoconstriction; Vasodilation; Vasodilator Agents; Xanthines

1999
Cross talk between A(1) and A(2A) adenosine receptors in the hippocampus and cortex of young adult and old rats.
    Journal of neurophysiology, 1999, Volume: 82, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Aging; Animals; Binding, Competitive; Cerebral Cortex; Electrophysiology; Hippocampus; In Vitro Techniques; Male; Phenethylamines; Protein Kinase C; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor Cross-Talk; Receptor, Adenosine A2A; Receptors, Purinergic P1; Synaptic Membranes; Triazines; Triazoles; Xanthines

1999
Use of the triazolotriazine [3H]ZM 241385 as a radioligand at recombinant human A2B adenosine receptors.
    Drug design and discovery, 1999, Volume: 16, Issue:3

    Topics: Animals; Cell Line; CHO Cells; Cricetinae; Humans; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Radioligand Assay; Receptor, Adenosine A2B; Receptors, Purinergic P1; Recombinant Proteins; Triazines; Triazoles; Tritium

1999
[Adenosine reduces ischemia/reperfusion-induced liver injury by inhibiting leukocyte activation].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1999, Volume: 114 Suppl 1

    Topics: Adenosine; Alkynes; Animals; Humans; In Vitro Techniques; Leukocyte Elastase; Liver; Male; Monocytes; N-Formylmethionine Leucyl-Phenylalanine; Neutrophil Activation; Neutrophils; Rats; Rats, Wistar; Receptors, Purinergic P1; Reperfusion Injury; Transaminases; Triazines; Triazoles; Tumor Necrosis Factor-alpha

1999
Localization and action of adenosine A2a receptors in regions of the brainstem important in cardiovascular control.
    Neuroscience, 2000, Volume: 95, Issue:2

    Topics: Adenosine; Animals; Aorta; Autoradiography; Blood Pressure; Brain Stem; Image Processing, Computer-Assisted; Iodine Radioisotopes; Phrenic Nerve; Pressoreceptors; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Reflex; Stimulation, Chemical; Triazines; Triazoles

2000
The anxiogenic-like effect of caffeine in two experimental procedures measuring anxiety in the mouse is not shared by selective A(2A) adenosine receptor antagonists.
    Psychopharmacology, 2000, Volume: 148, Issue:2

    Topics: Adenosine; Administration, Oral; Animals; Anxiety; Behavior, Animal; Caffeine; Darkness; Drug Administration Schedule; Injections, Intraperitoneal; Light; Male; Maze Learning; Mice; Mice, Knockout; Neuroprotective Agents; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyrimidines; Reaction Time; Receptor, Adenosine A2A; Triazines; Triazoles; Xanthines

2000
Role of adenosine A(2B) receptors in vasodilation of rat pial artery and cerebral blood flow autoregulation.
    American journal of physiology. Heart and circulatory physiology, 2000, Volume: 278, Issue:2

    Topics: Animals; Arteries; Cerebrovascular Circulation; Cyclic AMP; Cyclic GMP; Enzyme Inhibitors; Flavins; Homeostasis; Male; NG-Nitroarginine Methyl Ester; Nitrates; Nitrites; Pia Mater; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2B; Receptors, Purinergic P1; Thionucleotides; Triazines; Triazoles; Vasodilation

2000
Antagonism of coronary artery relaxation by adenosine A2A-receptor antagonist ZM241385.
    Journal of cardiovascular pharmacology, 2000, Volume: 35, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Antihypertensive Agents; Coronary Vessels; Dinoprost; Dose-Response Relationship, Drug; Drug Interactions; Endothelium, Vascular; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Phenethylamines; Purinergic P1 Receptor Antagonists; Pyrimidines; Receptors, Purinergic P1; Swine; Triazines; Triazoles; Vasodilator Agents

2000
Adenosine mediates nitric-oxide-independent renal vasodilation by activation of A2A receptors.
    Journal of hypertension, 1999, Volume: 17, Issue:12 Pt 2

    Topics: Adenosine; Animals; Endothelium, Vascular; Female; In Vitro Techniques; Male; Nitric Oxide; Phenethylamines; Potassium; Potassium Channels; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rabbits; Receptors, Purinergic; Renal Artery; Triazines; Triazoles; Vasodilation; Vasodilator Agents

1999
Tonic adenosine neuromodulation is preserved in motor nerve endings of aged rats.
    Neurochemistry international, 2000, Volume: 36, Issue:7

    Topics: Acetylcholine; Adenosine; Aging; Animals; Electric Stimulation; Male; Motor Neurons; Nerve Endings; Neurotransmitter Agents; Phrenic Nerve; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Triazines; Triazoles; Xanthines

2000
A novel adenosine analog, AMP579, inhibits neutrophil activation, adherence and neutrophil-mediated injury to coronary vascular endothelium.
    European journal of pharmacology, 2000, May-26, Volume: 397, Issue:1

    Topics: Animals; Cell Adhesion; Cell Degranulation; Coronary Vessels; Dogs; Dose-Response Relationship, Drug; Endothelium, Vascular; Female; Imidazoles; In Vitro Techniques; Male; Neutrophil Activation; Neutrophils; Pyridines; Quinazolines; Superoxides; Triazines; Triazoles; Vasodilation; Xanthines

2000
Accelerated resequestration of cytosolic calcium and suppression of the pro-inflammatory activities of human neutrophils by CGS 21680 in vitro.
    British journal of pharmacology, 2000, Volume: 130, Issue:4

    Topics: Adenosine; Calcium; Calcium Radioisotopes; Cyclic AMP; Cytosol; Dose-Response Relationship, Drug; Fura-2; Humans; Inflammation; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Pancreatic Elastase; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P2 Receptor Antagonists; Superoxides; Thapsigargin; Triazines; Triazoles

2000
Down-regulation of vascular endothelial growth factor expression after A(2A) adenosine receptor activation in PC12 pheochromocytoma cells.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 293, Issue:3

    Topics: Adenosine; Animals; Down-Regulation; Endothelial Growth Factors; Gene Expression Regulation; Lymphokines; PC12 Cells; Phenethylamines; Rats; Receptors, Purinergic P1; RNA, Messenger; Signal Transduction; Triazines; Triazoles; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors

2000
Adenosine A2A receptors regulate the extracellular accumulation of excitatory amino acids upon metabolic dysfunction in chick cultured retinal cells.
    Experimental eye research, 2000, Volume: 70, Issue:5

    Topics: Adenosine; Analysis of Variance; Animals; Aspartic Acid; Bicuculline; Cells, Cultured; Chick Embryo; Chromatography, High Pressure Liquid; Excitatory Amino Acids; Extracellular Space; GABA-A Receptor Antagonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Glycolysis; Humans; Ischemia; Organophosphorus Compounds; Purinergic P1 Receptor Antagonists; Pyrimidines; Receptor, Adenosine A2A; Receptors, Purinergic P1; Retina; Triazines; Triazoles; Xanthines

2000
Extracellular ATP reduces optically monitored electrical signals in hippocampal slices through metabolism to adenosine.
    European journal of pharmacology, 2000, Jul-07, Volume: 399, Issue:2-3

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Dose-Response Relationship, Drug; Electric Stimulation; Electrophysiology; Hippocampus; Organ Culture Techniques; Rats; Rats, Wistar; Signal Transduction; Triazines; Triazoles; Uridine Diphosphate; Xanthines

2000
SCH 58261 and ZM 241385 differentially prevent the motor effects of CGS 21680 in mice: evidence for a functional 'atypical' adenosine A(2A) receptor.
    European journal of pharmacology, 2000, Jul-28, Volume: 401, Issue:1

    Topics: Adenosine; Animals; Dose-Response Relationship, Drug; Drug Interactions; Exploratory Behavior; Injections, Intraventricular; Male; Maze Learning; Mice; Mice, Knockout; Motor Activity; Neuroprotective Agents; Phenethylamines; Pyrimidines; Receptor, Adenosine A2A; Receptors, Purinergic P1; Time Factors; Triazines; Triazoles

2000
Adenosine A(2A) and A(2B) receptors in cultured human and porcine coronary artery endothelial cells.
    American journal of physiology. Heart and circulatory physiology, 2000, Volume: 279, Issue:2

    Topics: 2-Chloroadenosine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Affinity Labels; Animals; Binding, Competitive; Cells, Cultured; Coronary Vessels; Cyclic AMP; Endothelium, Vascular; Gene Expression Regulation; Humans; Iodine Radioisotopes; Iodobenzenes; Kinetics; Phenethylamines; Purinergic P1 Receptor Antagonists; Radioligand Assay; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Receptors, Purinergic P1; Reverse Transcriptase Polymerase Chain Reaction; Swine; Transcription, Genetic; Triazines; Triazoles

2000
Site-directed mutagenesis studies of human A(2A) adenosine receptors: involvement of glu(13) and his(278) in ligand binding and sodium modulation.
    Biochemical pharmacology, 2000, Sep-01, Volume: 60, Issue:5

    Topics: Animals; Binding, Competitive; Drug Interactions; Glutamic Acid; Guanosine Triphosphate; Histidine; Humans; In Vitro Techniques; Kinetics; Models, Molecular; Mutagenesis, Site-Directed; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Radioligand Assay; Receptor, Adenosine A2A; Receptors, Purinergic P1; Sodium; Triazines; Triazoles; Tritium

2000
Allosteric modulation of A(2A) adenosine receptors by amiloride analogues and sodium ions.
    Biochemical pharmacology, 2000, Sep-01, Volume: 60, Issue:5

    Topics: Allosteric Regulation; Amiloride; Animals; Binding, Competitive; Cell Membrane; Corpus Striatum; Diuretics; Dose-Response Relationship, Drug; Drug Interactions; In Vitro Techniques; Purinergic P1 Receptor Antagonists; Radiopharmaceuticals; Rats; Receptor, Adenosine A2A; Receptors, Purinergic P1; Sodium; Sodium Chloride; Time Factors; Triazines; Triazoles; Tritium

2000
Adenosine and selective A(2A) receptor agonists reduce ischemia/reperfusion injury of rat liver mainly by inhibiting leukocyte activation.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 294, Issue:3

    Topics: Adenosine; Alkynes; Animals; Calcium; Cells, Cultured; Chemokine CXCL1; Chemokines, CXC; Chemotactic Factors; Growth Substances; Humans; Intercellular Signaling Peptides and Proteins; Ischemia; Leukocyte Elastase; Lipopolysaccharides; Liver; Male; Monocytes; Neutrophil Activation; Peroxidase; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A2A; Reperfusion Injury; Triazines; Triazoles; Tumor Necrosis Factor-alpha

2000
Diadenosine polyphosphates facilitate the evoked release of acetylcholine from rat hippocampal nerve terminals.
    Brain research, 2000, Oct-06, Volume: 879, Issue:1-2

    Topics: Acetylcholine; Animals; Dinucleoside Phosphates; Hippocampus; Male; Presynaptic Terminals; Pyridoxal Phosphate; Rats; Rats, Wistar; Receptors, Purinergic P1; Suramin; Synaptosomes; Triazines; Triazoles; Tritium; Xanthines

2000
Adenosine A(2A) receptors mediate cardiovascular responses to hypoxia in fetal sheep.
    American journal of physiology. Heart and circulatory physiology, 2001, Volume: 280, Issue:1

    Topics: Adenosine; Animals; Blood Gas Analysis; Blood Pressure; Female; Fetal Hypoxia; Heart Rate; Hydrogen-Ion Concentration; Phenethylamines; Pregnancy; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptor, Adenosine A2A; Receptors, Purinergic P1; Sheep; Triazines; Triazoles; Xanthines

2001
Potentiation of cytokine induction of group IIA phospholipase A(2) in rat mesangial cells by ATP and adenosine via the A2A adenosine receptor.
    British journal of pharmacology, 2001, Volume: 132, Issue:1

    Topics: 5'-Nucleotidase; Adenosine; Adenosine Deaminase; Adenosine Triphosphate; Animals; Blotting, Northern; Cells, Cultured; Enzyme Induction; Enzyme Inhibitors; Glomerular Mesangium; Group II Phospholipases A2; Interleukin-1; Phospholipases A; Purinergic P2 Receptor Antagonists; Rats; Receptor, Adenosine A2A; Receptors, Purinergic P1; RNA, Messenger; Signal Transduction; Suramin; Triazines; Triazoles; Uridine Triphosphate; Vasodilator Agents

2001
Functional and molecular characterization of receptor subtypes mediating coronary microvascular dilation to adenosine.
    Journal of molecular and cellular cardiology, 2001, Volume: 33, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Animals; Antihypertensive Agents; Blotting, Western; Colforsin; Coronary Vessels; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Female; Glyburide; Heart; Hypoglycemic Agents; In Situ Hybridization; Male; Microcirculation; Myocardium; Peptides; Phenethylamines; Potassium Channel Blockers; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Reverse Transcriptase Polymerase Chain Reaction; Stress, Physiological; Swine; Thionucleotides; Tissue Distribution; Triazines; Triazoles

2001
[(3)H]ZM241385--an antagonist radioligand for adenosine A(2A) receptors in rat brain.
    European journal of pharmacology, 2001, Jan-12, Volume: 411, Issue:3

    Topics: Animals; Autoradiography; Binding, Competitive; Brain Chemistry; Female; Half-Life; In Vitro Techniques; Male; Membranes; Purinergic P1 Receptor Antagonists; Radioligand Assay; Rats; Rats, Wistar; Receptor, Adenosine A2A; Thermodynamics; Triazines; Triazoles

2001
Absence of the adenosine A(2A) receptor or its chronic blockade decrease ethanol withdrawal-induced seizures in mice.
    Neuropharmacology, 2001, Volume: 40, Issue:3

    Topics: Administration, Oral; Alcohol Withdrawal Seizures; Animals; Beverages; Cacao; Disease Models, Animal; Drug Administration Schedule; Eating; Ethanol; Female; Flavoring Agents; Injections, Intraperitoneal; Male; Mice; Mice, Knockout; Purinergic P1 Receptor Antagonists; Receptor, Adenosine A2A; Receptors, Purinergic P1; Triazines; Triazoles

2001
Cyclic AMP-dependent inhibition of human neutrophil oxidative activity by substituted 2-propynylcyclohexyl adenosine A(2A) receptor agonists.
    British journal of pharmacology, 2001, Volume: 132, Issue:5

    Topics: Adenosine; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Humans; Neutrophils; Receptor, Adenosine A2A; Receptors, Purinergic P1; Respiratory Burst; Triazines; Triazoles

2001
Receptor subtypes mediating adenosine-induced dilation of cerebral arterioles.
    American journal of physiology. Heart and circulatory physiology, 2001, Volume: 280, Issue:5

    Topics: Adenosine; Adenosine Triphosphate; Animals; Antihypertensive Agents; Arterioles; Cerebrovascular Circulation; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Phenethylamines; Quinazolines; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Triazines; Triazoles; Vasodilation

2001
Adenosine A(2A) receptor stimulation reduces inflammation and neointimal growth in a murine carotid ligation model.
    Arteriosclerosis, thrombosis, and vascular biology, 2001, Volume: 21, Issue:5

    Topics: Animals; Arteriosclerosis; Carotid Artery Injuries; Cell Adhesion Molecules; Female; Inflammation; Leukocyte Count; Macrophages; Mice; Mice, Inbred C57BL; Neutrophils; Purinergic P1 Receptor Antagonists; Receptor, Adenosine A2A; Receptors, Purinergic P1; Triazines; Triazoles

2001
Selective A(2A) adenosine receptor activation reduces skin pressure ulcer formation and inflammation.
    American journal of physiology. Heart and circulatory physiology, 2001, Volume: 281, Issue:1

    Topics: Animals; Cell Line; Cyclohexanecarboxylic Acids; Dermatitis; Drug Combinations; Humans; Ischemia; Leukocytes; Male; Necrosis; Pressure Ulcer; Purines; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Receptors, Purinergic P1; Reference Values; Regional Blood Flow; Reperfusion Injury; Skin; Triazines; Triazoles

2001
Adenosine A(1) and A(2A) receptors modulate sleep state and breathing in fetal sheep.
    Journal of applied physiology (Bethesda, Md. : 1985), 2001, Volume: 91, Issue:1

    Topics: Adenosine; Animals; Fetus; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Respiratory Physiological Phenomena; Sheep; Sleep Stages; Triazines; Triazoles; Xanthines

2001
Novel short-acting A2A adenosine receptor agonists for coronary vasodilation: inverse relationship between affinity and duration of action of A2A agonists.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 298, Issue:1

    Topics: Adenosine; Animals; Antihypertensive Agents; Coronary Vessels; Corpus Striatum; Cyclic AMP; Dose-Response Relationship, Drug; Female; Humans; Male; PC12 Cells; Phenethylamines; Purinergic P1 Receptor Agonists; Purines; Pyrazoles; Rats; Receptor, Adenosine A2A; Receptors, Purinergic P1; Swine; Triazines; Triazoles; Vasodilation; Vasodilator Agents

2001
Adenosine-mediated inhibition of striatal GABAergic synaptic transmission during in vitro ischaemia.
    Brain : a journal of neurology, 2001, Volume: 124, Issue:Pt 9

    Topics: Adenosine; Adenosine Triphosphate; Animals; Brain Ischemia; Corpus Striatum; gamma-Aminobutyric Acid; Male; Membrane Potentials; Neural Inhibition; Organ Culture Techniques; Patch-Clamp Techniques; Potassium Channels; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Synaptic Transmission; Triazines; Triazoles; Xanthines

2001
Suppression of presynaptic responses to adenosine by activation of NMDA receptors.
    European journal of pharmacology, 2001, Sep-07, Volume: 427, Issue:1

    Topics: Action Potentials; Adenosine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Baclofen; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; GABA Agonists; Glycine; Hippocampus; In Vitro Techniques; Kainic Acid; Long-Term Potentiation; Male; N-Methylaspartate; Phenethylamines; Presynaptic Terminals; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, N-Methyl-D-Aspartate; Time Factors; Triazines; Triazoles

2001
Effects of adenosine receptor agonists and antagonists in a genetic animal model of primary paroxysmal dystonia.
    British journal of pharmacology, 2001, Volume: 134, Issue:2

    Topics: Adenosine; Animals; Caffeine; Cricetinae; Disease Models, Animal; Dose-Response Relationship, Drug; Dystonia; Female; Male; Mesocricetus; Muscle Contraction; Mutation; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Quinazolines; Theobromine; Theophylline; Triazines; Triazoles; Xanthines

2001
Adenosine-mediated hypotension in in vivo guinea-pig: receptors involved and role of NO.
    British journal of pharmacology, 2001, Volume: 134, Issue:4

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Blood Pressure; Diphenhydramine; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guinea Pigs; Heart Rate; Hypotension; Male; Methylene Blue; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Theophylline; Triazines; Triazoles; Vasodilator Agents; Xanthines

2001
AMP-activated protein kinase is highly expressed in neurons in the developing rat brain and promotes neuronal survival following glucose deprivation.
    Journal of molecular neuroscience : MN, 2001, Volume: 17, Issue:1

    Topics: Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Apoptosis; Brain; Cell Survival; Cells, Cultured; Glucose; Hypoglycemic Agents; Immunohistochemistry; Male; Multienzyme Complexes; Neurons; Neuroprotective Agents; Oligonucleotides, Antisense; Protein Serine-Threonine Kinases; Protein Subunits; Rats; Rats, Sprague-Dawley; Ribonucleotides; Triazines; Triazoles; Xanthines

2001
Effect of adenosine receptor blockade on pial arteriolar dilation during sciatic nerve stimulation.
    American journal of physiology. Heart and circulatory physiology, 2001, Volume: 281, Issue:5

    Topics: Adenine; Administration, Topical; Animals; Electric Stimulation; Enzyme Inhibitors; Evoked Potentials, Somatosensory; Injections, Intraperitoneal; Male; Pia Mater; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Sciatic Nerve; Theophylline; Triazines; Triazoles; Vasodilation; Vasodilator Agents; Xanthines

2001
Role of adenosine and P2 receptors in the penile tumescence in anesthetized dogs.
    European journal of pharmacology, 2001, Aug-03, Volume: 425, Issue:1

    Topics: Adenosine; Adenosine Diphosphate; Adenosine Triphosphate; Anesthesia; Animals; Dogs; Dose-Response Relationship, Drug; Enzyme Inhibitors; Injections, Intravenous; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Penile Erection; Penis; Purinergic P2 Receptor Agonists; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Theophylline; Thionucleotides; Triazines; Triazoles

2001
Oxygen delivery and oxygen consumption in rat hindlimb during systemic hypoxia: role of adenosine.
    The Journal of physiology, 2001, Nov-01, Volume: 536, Issue:Pt 3

    Topics: Adenosine; Animals; Hemodynamics; Hindlimb; Hypoxia; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Nitroprusside; Oxygen Consumption; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Purinergic P1; Triazines; Triazoles; Vital Capacity; Xanthines

2001
Solubilisation and immunoprecipitation of rat striatal adenosine A(2A) receptors.
    European journal of pharmacology, 2001, Nov-16, Volume: 431, Issue:2

    Topics: Adenosine; Animals; Cholic Acids; Corpus Striatum; Detergents; Phenethylamines; Precipitin Tests; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Radioligand Assay; Rats; Receptor, Adenosine A2A; Receptors, Purinergic P1; Solubility; Triazines; Triazoles

2001
Adenosine inhibits excitatory transmission to substantia gelatinosa neurons of the adult rat spinal cord through the activation of presynaptic A(1) adenosine receptor.
    Pain, 2001, Volume: 94, Issue:3

    Topics: Adenosine; Age Factors; Analgesics; Animals; Antihypertensive Agents; Excitatory Postsynaptic Potentials; In Vitro Techniques; Male; Neural Inhibition; Neurons; Patch-Clamp Techniques; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Substantia Gelatinosa; Triazines; Triazoles; Xanthines

2001
Purification and characterization of the human adenosine A(2a) receptor functionally expressed in Escherichia coli.
    European journal of biochemistry, 2002, Volume: 269, Issue:1

    Topics: Escherichia coli; Humans; Receptors, Purinergic P1; Recombinant Fusion Proteins; Solubility; Triazines; Triazoles

2002
Hippocampal injury and neurobehavioral deficits following hyperglycemic cerebral ischemia: effect of theophylline and ZM 241385.
    Journal of neurosurgery, 2002, Volume: 96, Issue:1

    Topics: Adenosine; Animals; Blood Glucose; Cell Death; Cerebral Infarction; Escape Reaction; Hippocampus; Injections, Intraperitoneal; Male; Maze Learning; Neurons; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Theophylline; Triazines; Triazoles

2002
Effects of CGS 21680, a selective adenosine A2A receptor agonist, on allergic airways inflammation in the rat.
    European journal of pharmacology, 2002, Mar-08, Volume: 438, Issue:3

    Topics: Adenosine; Allergens; Animals; Anti-Inflammatory Agents; Asthma; Blood Pressure; Budesonide; Dose-Response Relationship, Drug; Inflammation; Lung; Male; Ovalbumin; Phenethylamines; Purinergic P1 Receptor Agonists; Rats; Rats, Inbred BN; Receptor, Adenosine A2A; Triazines; Triazoles; Vascular Resistance

2002
Adenosine A(2A) receptors mediate hypoxic inhibition of fetal breathing in sheep.
    American journal of obstetrics and gynecology, 2002, Volume: 186, Issue:4

    Topics: Animals; Carbon Dioxide; Electroencephalography; Electrooculography; Eye Movements; Female; Fetal Blood; Fetal Hypoxia; Fetal Movement; Fetus; Hydrogen-Ion Concentration; Oxygen; Pregnancy; Purinergic P1 Receptor Antagonists; Receptor, Adenosine A2A; Receptors, Purinergic P1; Respiration; Sheep; Triazines; Triazoles; Xanthines

2002
Adenosine A(2A) receptor facilitation of hippocampal synaptic transmission is dependent on tonic A(1) receptor inhibition.
    Neuroscience, 2002, Volume: 112, Issue:2

    Topics: Adenosine; Animals; Binding, Competitive; CHO Cells; Cricetinae; Cyclic AMP; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; GABA Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Humans; In Vitro Techniques; Ligands; Male; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Purinergic P1; Signal Transduction; Synaptic Transmission; Transfection; Triazines; Triazoles; Xanthines

2002
Synergistic up-regulation of vascular endothelial growth factor expression in murine macrophages by adenosine A(2A) receptor agonists and endotoxin.
    The American journal of pathology, 2002, Volume: 160, Issue:6

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Blotting, Western; Cells, Cultured; Drosophila Proteins; Endothelial Growth Factors; Female; Interferon-gamma; Lipopolysaccharides; Lymphokines; Macrophages, Peritoneal; Male; Membrane Glycoproteins; Mice; Mice, Inbred C3H; Mice, Inbred C57BL; Mice, Knockout; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Phenethylamines; Protein Kinase Inhibitors; Purinergic P1 Receptor Agonists; Receptor, Adenosine A2A; Receptors, Cell Surface; Receptors, Purinergic P1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Theobromine; Toll-Like Receptor 4; Toll-Like Receptors; Triazines; Triazoles; Up-Regulation; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors; Xanthines

2002
Selective allosteric enhancement of agonist binding and function at human A3 adenosine receptors by a series of imidazoquinoline derivatives.
    Molecular pharmacology, 2002, Volume: 62, Issue:1

    Topics: Adenosine; Allosteric Regulation; Animals; Binding, Competitive; CHO Cells; Cricetinae; Dose-Response Relationship, Drug; Imidazoles; Iodine Radioisotopes; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Quinolines; Radioligand Assay; Rats; Receptor, Adenosine A2A; Receptor, Adenosine A3; Receptors, Purinergic P1; Triazines; Triazoles; Tritium; Xanthines

2002
Effects of adenosine receptor agonists on guinea-pig isolated working hearts and the role of endothelium and NO.
    The Journal of pharmacy and pharmacology, 2002, Volume: 54, Issue:6

    Topics: Adenosine; Animals; Cyclooxygenase Inhibitors; Endothelium, Vascular; Guinea Pigs; Heart; Hemodynamics; In Vitro Techniques; Indomethacin; Male; Nitric Oxide; Nitric Oxide Synthase; Phenethylamines; Prostaglandins; Purinergic P1 Receptor Agonists; Triazines; Triazoles

2002
Localization of adenosine A2A-receptors in rat brain with [3H]ZM-241385.
    Naunyn-Schmiedeberg's archives of pharmacology, 2002, Volume: 366, Issue:5

    Topics: Animals; Brain; Male; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Receptors, Purinergic P1; Triazines; Triazoles; Tritium

2002
Transducing system operated by adenosine A(2A) receptors to facilitate acetylcholine release in the rat hippocampus.
    European journal of pharmacology, 2002, Nov-01, Volume: 454, Issue:1

    Topics: Acetylcholine; Adenylyl Cyclases; Animals; Blotting, Western; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Activation; Hippocampus; In Vitro Techniques; Male; Nerve Endings; Protein Kinase C; Purinergic P1 Receptor Antagonists; Pyrimidines; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Purinergic P1; Signal Transduction; Synaptosomes; Triazines; Triazoles; Xanthines

2002
Low ethanol sensitivity and increased ethanol consumption in mice lacking adenosine A2A receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Dec-01, Volume: 22, Issue:23

    Topics: Administration, Oral; Alcohol Drinking; Animals; Behavior, Animal; Body Temperature; Choice Behavior; Dose-Response Relationship, Drug; Drug Resistance; Drug Tolerance; Ethanol; Female; Hypothermia; Injections, Intraperitoneal; Male; Mice; Mice, Knockout; Purinergic P1 Receptor Antagonists; Quinine; Receptor, Adenosine A2A; Receptors, Purinergic P1; Reflex; Sex Factors; Sucrose; Triazines; Triazoles

2002
Changes of peripheral A2A adenosine receptors in chronic heart failure and cardiac transplantation.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2003, Volume: 17, Issue:2

    Topics: Binding, Competitive; Female; Heart Failure; Heart Transplantation; Humans; Kinetics; Lymphocytes; Male; Myocardium; Neutrophils; Receptor, Adenosine A2A; Receptors, Purinergic P1; Triazines; Triazoles; Tritium

2003
Adenosine receptors mediate glutamate-evoked arteriolar dilation in the rat cerebral cortex.
    American journal of physiology. Heart and circulatory physiology, 2003, Volume: 284, Issue:5

    Topics: Animals; Arterioles; Blood Pressure; Cerebrovascular Circulation; Excitatory Amino Acid Agonists; Glutamic Acid; Male; N-Methylaspartate; Pia Mater; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Triazines; Triazoles; Vasodilation

2003
Regional differences in the adenosine A(2) receptor-mediated modulation of contractions in rat vas deferens.
    European journal of pharmacology, 2003, Jan-24, Volume: 460, Issue:2-3

    Topics: Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Epididymis; Immunohistochemistry; In Vitro Techniques; Male; Muscle Contraction; Norepinephrine; Phenethylamines; Prostate; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Purinergic P1; Theobromine; Triazines; Triazoles; Vas Deferens; Xanthines

2003
Rapid modification of the glycocalyx caused by ischemia-reperfusion is inhibited by adenosine A2A receptor activation.
    American journal of physiology. Heart and circulatory physiology, 2003, Volume: 284, Issue:6

    Topics: Animals; Arterioles; Biotransformation; Capillaries; Cyclohexanecarboxylic Acids; Erythrocytes; Glycocalyx; Male; Mice; Mice, Inbred C57BL; Muscle, Skeletal; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Receptor, Adenosine A2A; Reperfusion Injury; Triazines; Triazoles

2003
Involvement of adenosine A1 and A2A receptors in the motor effects of caffeine after its acute and chronic administration.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2003, Volume: 28, Issue:7

    Topics: Adenosine; Amphetamine; Animals; Behavior, Animal; Caffeine; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Male; Motor Activity; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Receptors, Purinergic P1; Theophylline; Time Factors; Triazines; Triazoles; Tritium; Xanthines

2003
Neuroprotection by caffeine and adenosine A2A receptor blockade of beta-amyloid neurotoxicity.
    British journal of pharmacology, 2003, Volume: 138, Issue:7

    Topics: Adenosine A2 Receptor Antagonists; Alzheimer Disease; Amyloid beta-Peptides; Animals; Brain; Caffeine; Cells, Cultured; Central Nervous System Diseases; Cerebellum; Neurons; Neuroprotective Agents; Peptide Fragments; Rats; Rats, Wistar; Receptor, Adenosine A2A; Theophylline; Triazines; Triazoles

2003
Induction of neurite outgrowth in PC12 cells by the bacterial nucleoside N6-methyldeoxyadenosine is mediated through adenosine A2a receptors and via cAMP and MAPK signaling pathways.
    Biochemical and biophysical research communications, 2003, May-16, Volume: 304, Issue:4

    Topics: Adenosine; Animals; CDC2 Protein Kinase; CDC2-CDC28 Kinases; Cyclic AMP; Cyclin-Dependent Kinase 2; Cyclin-Dependent Kinases; Deoxyadenosines; DNA-Binding Proteins; Enzyme Inhibitors; ets-Domain Protein Elk-1; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Neurites; PC12 Cells; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Rats; Receptor, Adenosine A2A; Receptors, Purinergic P1; Second Messenger Systems; Transcription Factors; Triazines; Triazoles

2003
The human D2 dopamine receptor synergizes with the A2A adenosine receptor to stimulate adenylyl cyclase in PC12 cells.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2003, Volume: 28, Issue:7

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenine; Adenosine; Adenosine Deaminase; Adenosine Diphosphate; Adenylyl Cyclases; Animals; Benzamides; Binding, Competitive; Cell Cycle; Cell Membrane; Cofilin 1; Colforsin; Cyclic AMP; Cytoskeletal Proteins; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Enzyme Activation; Gene Expression; Glutamic Acid; Humans; Membrane Potentials; Patch-Clamp Techniques; PC12 Cells; Pertussis Toxin; Phenethylamines; Phosphodiesterase Inhibitors; Phosphoproteins; Propionates; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyrrolidines; Quinpirole; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, Purinergic P1; Thionucleotides; Transfection; Triazines; Triazoles; Xenopus Proteins

2003
Adenosine A 2B receptors modulate cAMP levels and induce CREB but not ERK1/2 and p38 phosphorylation in rat skeletal muscle cells.
    Biochemical and biophysical research communications, 2003, Jul-18, Volume: 307, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cells, Cultured; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Muscle, Skeletal; p38 Mitogen-Activated Protein Kinases; Pertussis Toxin; Phenethylamines; Phosphorylation; Rats; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Receptors, Purinergic P1; RNA; Triazines; Triazoles

2003
Enhanced adenosine A2A receptor facilitation of synaptic transmission in the hippocampus of aged rats.
    Journal of neurophysiology, 2003, Volume: 90, Issue:2

    Topics: Adenosine; Adrenergic beta-Agonists; Aging; Animals; Blotting, Western; Cyclic AMP; Electrophysiology; Excitatory Postsynaptic Potentials; Hippocampus; Isoproterenol; Male; Neurons; Phenethylamines; Presynaptic Terminals; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Purinergic P1; Synaptic Transmission; Triazines; Triazoles; Xanthines

2003
Effects of adenosine receptor antagonists on pial arteriolar dilation during carbon dioxide inhalation.
    European journal of pharmacology, 2003, Aug-29, Volume: 476, Issue:3

    Topics: Adenosine; Administration, Inhalation; Animals; Caffeine; Carbon Dioxide; Cerebral Cortex; Cerebral Veins; Cerebrovascular Circulation; Drug Interactions; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Purinergic P1 Receptor Antagonists; Quinazolines; Rats; Rats, Sprague-Dawley; Triazines; Triazoles; Vasodilation; Vasodilator Agents; Xanthines

2003
Brief, repeated, oxygen-glucose deprivation episodes protect neurotransmission from a longer ischemic episode in the in vitro hippocampus: role of adenosine receptors.
    British journal of pharmacology, 2003, Volume: 140, Issue:2

    Topics: Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Antagonists; Animals; Brain Ischemia; Electric Stimulation; Excitatory Postsynaptic Potentials; Glucose; Hippocampus; Hypoxia; In Vitro Techniques; Ischemic Preconditioning; Male; Oxygen; Purinergic P1 Receptor Antagonists; Pyridines; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptor, Adenosine A2A; Receptor, Adenosine A3; Receptors, Purinergic P1; Synaptic Transmission; Time Factors; Triazines; Triazoles; Xanthines

2003
The effect of caffeine on peripheral vascular resistance in isolated perfused guinea pig hind limbs.
    Journal of cardiovascular pharmacology, 2003, Volume: 42, Issue:4

    Topics: Adenosine; Animals; Caffeine; Dose-Response Relationship, Drug; Female; Flavins; Guinea Pigs; Hindlimb; Hypoxia; Iliac Artery; Iloprost; Male; Nitrogen; Norepinephrine; Perfusion; Triazines; Triazoles; Vascular Resistance; Vasoconstriction; Vasodilation

2003
LTP-induced depression of response to hypoxia in hippocampus: effects of adenosine receptor activation.
    Neuroreport, 2003, Oct-06, Volume: 14, Issue:14

    Topics: Adenosine; Animals; Electric Stimulation; Hippocampus; Hypoxia; In Vitro Techniques; Long-Term Potentiation; Male; Membrane Potentials; Purinergic P1 Receptor Agonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Triazines; Triazoles

2003
Modulation of A2A adenosine receptors and associated Galphas proteins by ZM 241385 treatment of porcine coronary artery.
    Journal of cardiovascular pharmacology, 2003, Volume: 42, Issue:6

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Coronary Vessels; Cyclic AMP; Male; Muscle, Smooth, Vascular; Swine; Triazines; Triazoles; Up-Regulation; Vasodilation

2003
Adenosine A2A receptors and depression.
    Neurology, 2003, Dec-09, Volume: 61, Issue:11 Suppl 6

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Animals; Antidepressive Agents; Behavior, Animal; Caffeine; Depression; Disease Models, Animal; Dopamine Antagonists; Drug Interactions; Haloperidol; Mice; Mice, Knockout; Motor Activity; Neurotransmitter Agents; Parkinsonian Disorders; Purines; Pyrimidines; Receptor, Adenosine A2A; Triazines; Triazoles

2003
Discovery of nonxanthine adenosine A2A receptor antagonists for the treatment of Parkinson's disease.
    Neurology, 2003, Dec-09, Volume: 61, Issue:11 Suppl 6

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Animals; Antiparkinson Agents; Binding, Competitive; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Design; Drug Evaluation, Preclinical; Humans; Ligands; Mefloquine; Mice; Motor Activity; Neuroprotective Agents; Parkinsonian Disorders; Phenethylamines; Purines; Pyrimidines; Radioligand Assay; Rats; Triazines; Triazoles

2003
Protection from ischemic liver injury by activation of A2A adenosine receptors during reperfusion: inhibition of chemokine induction.
    American journal of physiology. Gastrointestinal and liver physiology, 2004, Volume: 286, Issue:2

    Topics: Adenosine A2 Receptor Agonists; Animals; Blood Cells; Chemokines; Cyclohexanecarboxylic Acids; Cytokines; Drug Administration Schedule; Edema; Gene Deletion; Ischemia; Leukocytes; Liver; Liver Circulation; Liver Diseases; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Purines; Radioligand Assay; Receptor, Adenosine A2A; Reperfusion Injury; RNA, Messenger; Triazines; Triazoles

2004
Input-specific modulation of neurotransmitter release in the lateral horn of the spinal cord via adenosine receptors.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Jan-07, Volume: 24, Issue:1

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Cells, Cultured; Excitatory Postsynaptic Potentials; Immunohistochemistry; Interneurons; Male; Neural Inhibition; Neurons; Neurotransmitter Agents; Patch-Clamp Techniques; Phenethylamines; Presynaptic Terminals; Rats; Receptor, Adenosine A1; Receptor, Adenosine A2A; Spinal Cord; Triazines; Triazoles

2004
Adenosine administration produces an antidepressant-like effect in mice: evidence for the involvement of A1 and A2A receptors.
    Neuroscience letters, 2004, Jan-23, Volume: 355, Issue:1-2

    Topics: Adenosine; Animals; Antidepressive Agents; Caffeine; Depressive Disorder; Disease Models, Animal; Female; Male; Mice; Motor Activity; Receptor, Adenosine A1; Receptor, Adenosine A2A; Stress, Psychological; Triazines; Triazoles; Xanthines

2004
Involvement of adenosine A1 receptors in forced walking stress-induced analgesia in mice.
    Methods and findings in experimental and clinical pharmacology, 2003, Volume: 25, Issue:10

    Topics: Adenosine A1 Receptor Antagonists; Analgesia; Animals; Behavior, Animal; Formaldehyde; Male; Mice; Mice, Inbred Strains; Pain; Receptor, Adenosine A1; Stress, Psychological; Theophylline; Triazines; Triazoles; Walking; Xanthines

2003
Role of adenosine A2A receptor in the regulation of gastric somatostatin release.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 309, Issue:2

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Gastric Mucosa; Male; Phenethylamines; Rats; Rats, Wistar; Receptor, Adenosine A2A; Somatostatin; Stomach; Tissue Distribution; Triazines; Triazoles; Xanthines

2004
Effect of taurine deficiency on adenosine receptor-mediated relaxation of the rat aorta.
    Vascular pharmacology, 2003, Volume: 40, Issue:4

    Topics: 2-Chloroadenosine; Acetylcholine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Aorta, Thoracic; beta-Alanine; Endothelium, Vascular; Enzyme Inhibitors; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Phenylephrine; Rats; Rats, Inbred WKY; Receptors, Purinergic P1; Taurine; Triazines; Triazoles; Vasoconstrictor Agents; Vasodilator Agents

2003
Neutrophils both reduce and increase permeability in a cell culture model of the blood-brain barrier.
    Brain research, 2004, Feb-20, Volume: 998, Issue:2

    Topics: Adenosine; Adenosine Deaminase; Animals; Aprotinin; Blood-Brain Barrier; Capillary Permeability; Catalase; Cell Culture Techniques; Cell Movement; Cells, Cultured; Egtazic Acid; Electric Impedance; Endothelial Cells; Free Radicals; Humans; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Superoxide Dismutase; Triazines; Triazoles

2004
Binding of tritiated and radioiodinated ZM241,385 to brain A2A adenosine receptors.
    Nuclear medicine and biology, 2004, Volume: 31, Issue:2

    Topics: Animals; Brain; Iodine Radioisotopes; Isotope Labeling; Metabolic Clearance Rate; Organ Specificity; Protein Binding; Radionuclide Imaging; Radiopharmaceuticals; Rats; Receptor, Adenosine A2A; Tissue Distribution; Triazines; Triazoles; Tritium

2004
Adenosine A 2A receptor antagonists prevent the increase in striatal glutamate levels induced by glutamate uptake inhibitors.
    Journal of neurochemistry, 2004, Volume: 89, Issue:1

    Topics: Adenosine A2 Receptor Antagonists; Animals; Corpus Striatum; Dicarboxylic Acids; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Excitatory Amino Acid Transporter 2; Glutamic Acid; Kainic Acid; Male; Microdialysis; Neuroprotective Agents; Neurotransmitter Uptake Inhibitors; Pyrimidines; Pyrrolidines; Rats; Rats, Wistar; Receptor, Adenosine A2A; Triazines; Triazoles

2004
Activation of adenosine A2A receptor facilitates brain-derived neurotrophic factor modulation of synaptic transmission in hippocampal slices.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Mar-24, Volume: 24, Issue:12

    Topics: Adenosine; Adenosine Kinase; Animals; Brain-Derived Neurotrophic Factor; Bucladesine; Carbazoles; Electric Stimulation; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Indole Alkaloids; Long-Term Potentiation; Male; Patch-Clamp Techniques; Phenethylamines; Potassium; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptor, trkB; Synaptic Transmission; Triazines; Triazoles

2004
AMPA receptor-mediated presynaptic inhibition at cerebellar GABAergic synapses: a characterization of molecular mechanisms.
    The European journal of neuroscience, 2004, Volume: 19, Issue:9

    Topics: Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Benzoxazines; Calcium; Calcium Channel Blockers; Cerebellum; Chelating Agents; Colforsin; Cyclopropanes; Drug Interactions; Egtazic Acid; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Morpholines; Naphthalenes; Neural Inhibition; Neurons; Piperidines; Presynaptic Terminals; Pyrazoles; Rats; Rats, Wistar; Receptors, AMPA; Ryanodine; Synapses; Triazines; Triazoles

2004
Endogenous adenosine modulates epileptiform activity in rat hippocampus in a receptor subtype-dependent manner.
    The European journal of neuroscience, 2004, Volume: 19, Issue:9

    Topics: Adenosine; Animals; Animals, Newborn; Dihydropyridines; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Indoles; Maleimides; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Seizures; Theophylline; Time Factors; Triazines; Triazoles

2004
The role of intraspinal adenosine A1 receptors in sympathetic regulation.
    European journal of pharmacology, 2004, May-10, Volume: 492, Issue:1

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Agonists; Adenosine A3 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Dihydropyridines; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Spinal Cord; Splanchnic Nerves; Sympathetic Nervous System; Synaptic Transmission; Theobromine; Theophylline; Triazines; Triazoles

2004
Adenosine A2A receptor occupancy stimulates expression of proteins involved in reverse cholesterol transport and inhibits foam cell formation in macrophages.
    Journal of leukocyte biology, 2004, Volume: 76, Issue:3

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Arteriosclerosis; ATP Binding Cassette Transporter 1; ATP-Binding Cassette Transporters; Carrier Proteins; Cell Differentiation; Cholestanetriol 26-Monooxygenase; Cholesterol; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Down-Regulation; Foam Cells; Gene Expression Regulation, Enzymologic; Humans; Macrophages; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Phenethylamines; Receptor, Adenosine A2A; RNA, Messenger; Steroid Hydroxylases; Triazines; Triazoles; Up-Regulation

2004
Adenosine A2A receptor blockade differentially influences excitotoxic mechanisms at pre- and postsynaptic sites in the rat striatum.
    Journal of neuroscience research, 2004, Jul-01, Volume: 77, Issue:1

    Topics: 4-Aminopyridine; Adenosine; Adenosine A2 Receptor Antagonists; Animals; Calcium; Corpus Striatum; Dose-Response Relationship, Drug; Glutamic Acid; In Vitro Techniques; L-Lactate Dehydrogenase; Male; Models, Biological; N-Methylaspartate; Neurodegenerative Diseases; Neurons; Neuroprotective Agents; Neurotoxins; Phenethylamines; Pyrimidines; Quinolinic Acid; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, N-Methyl-D-Aspartate; Synaptic Membranes; Synaptic Transmission; Triazines; Triazoles

2004
Adenosine's role in hypercapnia-evoked cerebral vasodilation in the rat.
    Neuroscience letters, 2004, Jul-15, Volume: 365, Issue:1

    Topics: Adenosine; Animals; Carbon Dioxide; Cerebrovascular Circulation; Hypercapnia; Male; Microscopy, Video; Nitric Oxide; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Triazines; Triazoles; Vasodilation

2004
Striatal adenosine A(2A) receptor blockade increases extracellular dopamine release following l-DOPA administration in intact and dopamine-denervated rats.
    Neuropharmacology, 2004, Volume: 47, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adenosine A2 Receptor Antagonists; Analysis of Variance; Animals; Area Under Curve; Brain Chemistry; Chromatography, High Pressure Liquid; Corpus Striatum; Denervation; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Drug Interactions; Extracellular Space; Homovanillic Acid; Hydroxyindoleacetic Acid; Levodopa; Male; Malonates; Methyltyrosines; Rats; Rats, Wistar; Receptor, Adenosine A2A; Reserpine; Serotonin; Substantia Nigra; Time Factors; Triazines; Triazoles; Xanthines

2004
Permissive role of adenosine A2A receptors on metabotropic glutamate receptor 5 (mGluR5)-mediated effects in the striatum.
    Journal of neurochemistry, 2004, Volume: 90, Issue:5

    Topics: Adenosine; Animals; Carbazoles; Cells, Cultured; Corpus Striatum; Dose-Response Relationship, Drug; Drug Interactions; Electrophysiology; Embryo, Mammalian; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; Glycine; In Vitro Techniques; Indoles; Male; Membrane Potentials; N-Methylaspartate; Phenethylamines; Phenylacetates; Pregnancy; Purinergic P1 Receptor Agonists; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Adenosine A2; Receptors, Metabotropic Glutamate; Triazines; Triazoles

2004
Adenosine A1 receptors modulate the anxiolytic-like effect of ethanol in the elevated plus-maze in mice.
    European journal of pharmacology, 2004, Sep-19, Volume: 499, Issue:1-2

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Analysis of Variance; Animals; Anti-Anxiety Agents; Anxiety; Caffeine; Dose-Response Relationship, Drug; Drug Synergism; Ethanol; Male; Maze Learning; Mice; Receptor, Adenosine A1; Triazines; Triazoles; Xanthines

2004
Characterization of [3H]ZM 241385 binding in wild-type and adenosine A2A receptor knockout mice.
    European journal of pharmacology, 2004, Nov-03, Volume: 504, Issue:1-2

    Topics: Animals; Binding Sites; Brain; Dose-Response Relationship, Drug; Male; Mice; Mice, Knockout; Protein Binding; Receptor, Adenosine A2A; Triazines; Triazoles; Tritium

2004
Crucial role for ecto-5'-nucleotidase (CD73) in vascular leakage during hypoxia.
    The Journal of experimental medicine, 2004, Dec-06, Volume: 200, Issue:11

    Topics: 5'-Nucleotidase; Adenosine; Animals; Capillary Permeability; Hypoxia; Lung; Mice; Triazines; Triazoles

2004
Adenosine A2A-receptor blockade abolishes the roll-off respiratory response to hypoxia in awake lambs.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2005, Volume: 288, Issue:5

    Topics: Adenosine A2 Receptor Antagonists; Animals; Animals, Newborn; Blood Pressure; Body Temperature; Carbon Dioxide; Heart Rate; Hydrogen-Ion Concentration; Hypoxia; Oxygen; Receptor, Adenosine A2A; Respiration; Sheep; Tidal Volume; Time Factors; Triazines; Triazoles; Xanthines

2005
A2A adenosine receptor induction inhibits IFN-gamma production in murine CD4+ T cells.
    Journal of immunology (Baltimore, Md. : 1950), 2005, Jan-15, Volume: 174, Issue:2

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; CD4-Positive T-Lymphocytes; Cell Line; Cyclic AMP; Cyclohexanecarboxylic Acids; Gene Dosage; Humans; Interferon-gamma; Lymphocyte Activation; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Purines; Receptor, Adenosine A2A; Receptors, Antigen, T-Cell; RNA, Messenger; Rolipram; Triazines; Triazoles

2005
A2B adenosine receptor mediates human chorionic vasoconstriction and signals through arachidonic acid cascade.
    American journal of physiology. Heart and circulatory physiology, 2005, Volume: 288, Issue:5

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Arachidonic Acid; Chorion; Endothelium, Vascular; Female; Humans; In Vitro Techniques; Placenta; Pregnancy; Receptor, Adenosine A2B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Triazines; Triazoles; Vasoconstriction; Vasodilator Agents; Xanthines

2005
In vivo adenosine receptor preconditioning reduces myocardial infarct size via subcellular ERK signaling.
    American journal of physiology. Heart and circulatory physiology, 2005, Volume: 288, Issue:5

    Topics: Animals; Butadienes; Enzyme Inhibitors; Imidazoles; Ischemic Preconditioning, Myocardial; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Myocardial Infarction; Nitriles; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Reperfusion Injury; Subcellular Fractions; Triazines; Triazoles; Xanthines

2005
Kinetic and functional properties of [3H]ZM241385, a high affinity antagonist for adenosine A2A receptors.
    Life sciences, 2005, Feb-11, Volume: 76, Issue:13

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Algorithms; Animals; Binding, Competitive; Cell Membrane; CHO Cells; Cricetinae; Cyclic AMP; GTP-Binding Proteins; Kinetics; Ligands; Neostriatum; Phenethylamines; Radioligand Assay; Triazines; Triazoles

2005
Adenosine contributes to mu-opioid synaptic inhibition in rat substantia gelatinosa in vitro.
    Neuroscience letters, 2005, Mar-11, Volume: 376, Issue:2

    Topics: Adenosine; Analgesics, Opioid; Animals; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Excitatory Postsynaptic Potentials; Neural Inhibition; Neurons; Organ Culture Techniques; Patch-Clamp Techniques; Rats; Receptors, Opioid, mu; Receptors, Purinergic P1; Substantia Gelatinosa; Synapses; Triazines; Triazoles; Xanthines

2005
Upregulation of A2A adenosine receptor expression by TNF-alpha in PBMC of patients with CHF: a regulatory mechanism of inflammation.
    Journal of cardiac failure, 2005, Volume: 11, Issue:1

    Topics: Adenosine; Blotting, Western; Female; Heart Failure; Humans; Lipopolysaccharides; Male; Middle Aged; Neutrophils; Phenethylamines; Receptor, Adenosine A2A; Receptors, Purinergic P1; Reverse Transcriptase Polymerase Chain Reaction; Triazines; Triazoles; Tumor Necrosis Factor-alpha; Up-Regulation

2005
Modulation of short-term social memory in rats by adenosine A1 and A(2A) receptors.
    Neuroscience letters, 2005, Mar-16, Volume: 376, Issue:3

    Topics: Adenosine; Animals; Behavior, Animal; Brain; Caffeine; Dose-Response Relationship, Drug; Drug Administration Schedule; Injections, Intraperitoneal; Male; Memory, Short-Term; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptor, Adenosine A2A; Social Behavior; Triazines; Triazoles; Xanthines

2005
Adenosine agonist regulation of outward active transport of fluorescein across retinal pigment epithelium in rabbits.
    Experimental eye research, 2005, Volume: 80, Issue:4

    Topics: Adenosine; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Biological Transport, Active; Dihydropyridines; Fluorescein; Fluoresceins; Fluorophotometry; Injections, Intravenous; Male; Pigment Epithelium of Eye; Purinergic P1 Receptor Antagonists; Rabbits; Retinal Detachment; Triazines; Triazoles; Xanthines

2005
Blockade of adenosine A2A receptors reverses short-term social memory impairments in spontaneously hypertensive rats.
    Behavioural brain research, 2005, Apr-30, Volume: 159, Issue:2

    Topics: Adenosine A2 Receptor Antagonists; Analysis of Variance; Animals; Caffeine; Discrimination Learning; Habituation, Psychophysiologic; Male; Memory Disorders; Memory, Short-Term; Rats; Rats, Inbred SHR; Rats, Wistar; Receptor, Adenosine A2A; Recognition, Psychology; Smell; Social Behavior; Social Environment; Species Specificity; Triazines; Triazoles; Xanthines

2005
Activation of adenosine receptors in the posterior cingulate cortex impairs memory retrieval in the rat.
    Neurobiology of learning and memory, 2005, Volume: 83, Issue:3

    Topics: Adenosine; Animals; Avoidance Learning; Cerebral Cortex; Exploratory Behavior; Gyrus Cinguli; Male; Memory; Microinjections; Phenethylamines; Purinergic Agonists; Purinergic Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptor, Adenosine A2A; Triazines; Triazoles; Xanthines

2005
Effects of adenosine and adenosine A2A receptor agonist on motor nerve conduction velocity and nerve blood flow in experimental diabetic neuropathy.
    Neurological research, 2005, Volume: 27, Issue:1

    Topics: Adenosine; Animals; Blood Glucose; Body Weight; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Drug Interactions; Neural Conduction; Phenethylamines; Purinergic P2 Receptor Agonists; Rats; Regional Blood Flow; Sciatic Nerve; Staining and Labeling; Streptozocin; Theophylline; Time Factors; Triazines; Triazoles

2005
Effect of sleep deprivation on righting reflex in the rat is partially reversed by administration of adenosine A1 and A2 receptor antagonists.
    Anesthesiology, 2005, Volume: 102, Issue:6

    Topics: Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Animals; Drug Combinations; Male; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptors, Adenosine A2; Reflex; Sleep Deprivation; Theophylline; Triazines; Triazoles

2005
Postconditioning reduces infarct size via adenosine receptor activation by endogenous adenosine.
    Cardiovascular research, 2005, Jul-01, Volume: 67, Issue:1

    Topics: Adenosine; Animals; Male; Myocardial Infarction; Myocardial Reperfusion; Myocardium; Perfusion; Purinergic P1 Receptor Antagonists; Random Allocation; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Theophylline; Triazines; Triazoles; Xanthines

2005
Adenosine receptors co-operate with NMDA preconditioning to protect cerebellar granule cells against glutamate neurotoxicity.
    Neuropharmacology, 2005, Volume: 49, Issue:1

    Topics: Adenosine Diphosphate; Adenosine Triphosphatases; Animals; Animals, Newborn; Cell Death; Cells, Cultured; Cerebellum; Cyclic AMP; Drug Antagonism; Excitatory Amino Acid Agonists; Glutamic Acid; Hydrolysis; N-Methylaspartate; Neurons; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Purinergic P1; Theophylline; Triazines; Triazoles

2005
Dual presynaptic control by ATP of glutamate release via facilitatory P2X1, P2X2/3, and P2X3 and inhibitory P2Y1, P2Y2, and/or P2Y4 receptors in the rat hippocampus.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Jul-06, Volume: 25, Issue:27

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Adenylyl Imidodiphosphate; Animals; Astrocytoma; Calcium; Cell Line; Cell Line, Tumor; Glutamic Acid; Hippocampus; Kidney; Male; Potassium; Pyramidal Cells; Pyridoxal Phosphate; Rats; Rats, Wistar; Receptors, Presynaptic; Receptors, Purinergic P2; Receptors, Purinergic P2X; Receptors, Purinergic P2X2; Receptors, Purinergic P2X3; Receptors, Purinergic P2Y1; Receptors, Purinergic P2Y2; Recombinant Fusion Proteins; RNA, Messenger; Subcellular Fractions; Suramin; Synaptosomes; Transfection; Triazines; Triazoles; Xanthines

2005
Lipopolysaccharide rapidly modifies adenosine receptor transcripts in murine and human macrophages: role of NF-kappaB in A(2A) adenosine receptor induction.
    The Biochemical journal, 2005, Nov-01, Volume: 391, Issue:Pt 3

    Topics: Animals; Cells, Cultured; Cyclohexanecarboxylic Acids; Gene Expression Regulation; Humans; Lipopolysaccharides; Macrophages; Mice; NF-kappa B; Nitriles; Protein Binding; Purines; Receptor, Adenosine A2A; RNA, Messenger; Sulfones; Transcription, Genetic; Triazines; Triazoles; Tumor Necrosis Factor-alpha

2005
Adenosine A2A receptor stimulation potentiates nitric oxide release by activated microglia.
    Journal of neurochemistry, 2005, Volume: 95, Issue:4

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Analysis of Variance; Animals; Animals, Newborn; Blotting, Western; Cell Proliferation; Cells, Cultured; Cerebral Cortex; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Immunohistochemistry; Indoles; Lipopolysaccharides; Maleimides; Mice; Mice, Inbred C57BL; Microglia; Nitric Oxide; Nitrites; Phenethylamines; Protein Binding; Radioligand Assay; Receptor, Adenosine A2A; Time Factors; Triazines; Triazoles; Tritium; Tumor Necrosis Factor-alpha

2005
Tachycardia caused by A2A adenosine receptor agonists is mediated by direct sympathoexcitation in awake rats.
    The Journal of pharmacology and experimental therapeutics, 2006, Volume: 316, Issue:2

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Male; Norepinephrine; Purines; Pyrazoles; Rats; Rats, Sprague-Dawley; Sympathetic Nervous System; Tachycardia; Time Factors; Triazines; Triazoles

2006
The cellular mechanisms by which adenosine evokes release of nitric oxide from rat aortic endothelium.
    The Journal of physiology, 2006, Jan-01, Volume: 570, Issue:Pt 1

    Topics: Adenosine; Animals; Aorta, Thoracic; Apamin; Arachidonic Acids; Calcium; Endothelium, Vascular; In Vitro Techniques; Large-Conductance Calcium-Activated Potassium Channels; Male; Nitric Oxide; Peptides; Phospholipases A; Phospholipases A2; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptors, Adenosine A2; Second Messenger Systems; Small-Conductance Calcium-Activated Potassium Channels; Triazines; Triazoles; Vasodilator Agents; Xanthines

2006
Adenosine concentration in the porcine coronary artery wall and A2A receptor involvement in hypoxia-induced vasodilatation.
    The Journal of physiology, 2006, Jan-15, Volume: 570, Issue:Pt 2

    Topics: Acetamides; Adenosine; Adenosine A2 Receptor Antagonists; Adenosine Deaminase; Adenosine Deaminase Inhibitors; Adenosine Kinase; Animals; Coronary Vessels; Dose-Response Relationship, Drug; Glucose; Hypoxia; In Vitro Techniques; Lactates; Purines; Pyruvic Acid; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Swine; Triazines; Triazoles; Vasodilation

2006
Adenosine A1 and A2A receptors of hippocampal CA1 region have opposite effects on piriform cortex kindled seizures in rats.
    Seizure, 2006, Volume: 15, Issue:1

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Cerebral Cortex; Electric Stimulation; Hippocampus; Kindling, Neurologic; Male; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptor, Adenosine A2A; Receptors, Purinergic P2; Seizures; Triazines; Triazoles; Xanthines

2006
Adenosine A2A receptors promote adenosine-stimulated wound healing in bronchial epithelial cells.
    American journal of physiology. Lung cellular and molecular physiology, 2006, Volume: 290, Issue:5

    Topics: Adenosine; Bronchi; Cell Division; Cell Line; Cell Movement; Humans; Kinetics; Receptor, Adenosine A2A; Respiratory Mucosa; Transcription, Genetic; Triazines; Triazoles; Wound Healing; Wounds and Injuries

2006
A2a receptors mediate inhibitory effects of adenosine on colonic motility in the presence of experimental colitis.
    Inflammatory bowel diseases, 2006, Volume: 12, Issue:2

    Topics: Adenosine; Animals; Colitis; Disease Models, Animal; Gastrointestinal Motility; Intestinal Mucosa; Male; Muscle Contraction; Muscle, Smooth; Nitric Oxide; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Reverse Transcriptase Polymerase Chain Reaction; Sensitivity and Specificity; Tissue Culture Techniques; Triazines; Triazoles

2006
Adenosine as an active component of Antrodia cinnamomea that prevents rat PC12 cells from serum deprivation-induced apoptosis through the activation of adenosine A(2A) receptors.
    Life sciences, 2006, Jun-13, Volume: 79, Issue:3

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Aminohydrolases; Animals; Apoptosis; Culture Media, Serum-Free; Inosine; PC12 Cells; Polyporales; Rats; Triazines; Triazoles

2006
Effects of the A 2A adenosine receptor antagonist KW6002 in the nucleus accumbens in vitro and in vivo.
    Pharmacology, biochemistry, and behavior, 2006, Volume: 83, Issue:1

    Topics: Animals; Binding, Competitive; Conditioning, Operant; Dopamine; Dose-Response Relationship, Drug; Extracellular Space; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Microdialysis; Motor Activity; Nucleus Accumbens; Purines; Rats; Receptor, Adenosine A2A; Triazines; Triazoles; Xanthines

2006
Dialysis delivery of an adenosine A2A agonist into the pontine reticular formation of C57BL/6J mouse increases pontine acetylcholine release and sleep.
    Journal of neurochemistry, 2006, Volume: 96, Issue:6

    Topics: Acetylcholine; Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Dose-Response Relationship, Drug; Extracellular Fluid; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred C57BL; Microdialysis; Neural Inhibition; Neural Pathways; Phenethylamines; Pons; Receptor, Adenosine A2A; Reticular Formation; Sleep; Sleep, REM; Synaptic Transmission; Triazines; Triazoles; Up-Regulation; Wakefulness

2006
Neurogenic secretion mediated by the purinergic P2Y1 receptor in guinea-pig small intestine.
    European journal of pharmacology, 2006, Apr-24, Volume: 536, Issue:1-2

    Topics: Adenosine Diphosphate; Adenosine Triphosphate; Animals; Bumetanide; Chlorides; Dose-Response Relationship, Drug; Electric Stimulation; Electrolytes; Gene Expression; Guinea Pigs; In Vitro Techniques; Intestine, Small; Male; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2; Receptors, Purinergic P2Y1; Receptors, Vasoactive Intestinal Polypeptide, Type I; Signal Transduction; Sodium Potassium Chloride Symporter Inhibitors; Tetrodotoxin; Theophylline; Triazines; Triazoles; Vasoactive Intestinal Peptide

2006
Both endothelium and afferent nerve endings play a role in acetylcholine-induced renal vasodilation.
    Life sciences, 2006, Jul-24, Volume: 79, Issue:9

    Topics: Acetylcholine; Animals; Calcitonin Gene-Related Peptide; Capsaicin; Cyclic AMP-Dependent Protein Kinases; Cyclooxygenase Inhibitors; Endothelium, Vascular; Enzyme Inhibitors; Female; Glycyrrhetinic Acid; Indomethacin; Male; Nerve Endings; Neurons, Afferent; Nitric Oxide; Nitric Oxide Synthase Type III; Nitroarginine; Octoxynol; Rats; Rats, Wistar; Renal Circulation; Second Messenger Systems; Triazines; Triazoles; Vasodilator Agents

2006
Adenosine A2A receptor inactivation increases survival in polymicrobial sepsis.
    Journal of immunology (Baltimore, Md. : 1950), 2006, May-01, Volume: 176, Issue:9

    Topics: Adenosine A2 Receptor Antagonists; Animals; Apoptosis; Bacteremia; Biomarkers; Cytokines; Gene Expression Profiling; Male; Mice; Mice, Knockout; Oligonucleotide Array Sequence Analysis; Receptor, Adenosine A2A; Spleen; Survival Rate; Triazines; Triazoles

2006
Early and transient alteration of adenosine A2A receptor signaling in a mouse model of Huntington disease.
    Neurobiology of disease, 2006, Volume: 23, Issue:1

    Topics: Adenylyl Cyclases; Animals; Basal Ganglia; Cyclic AMP; Disease Models, Animal; Huntington Disease; Mice; Mice, Transgenic; Receptors, Adenosine A2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Triazines; Triazoles

2006
Adenosine A2A receptor stimulation decreases GAT-1-mediated GABA uptake in the globus pallidus of the rat.
    Neuropharmacology, 2006, Volume: 51, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenosine A2 Receptor Agonists; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Data Interpretation, Statistical; Enzyme Inhibitors; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Globus Pallidus; In Vitro Techniques; Isoquinolines; Male; Okadaic Acid; Phenethylamines; Rats; Rats, Wistar; Sulfonamides; Synapses; Triazines; Triazoles

2006
Role of adenosine A1 receptors in the modulation of dopamine D1 and adenosine A2A receptor signaling in the neostriatum.
    Neuroscience, 2006, Aug-11, Volume: 141, Issue:1

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Animals; Benzazepines; Dopamine and cAMP-Regulated Phosphoprotein 32; Dopamine Antagonists; Drug Interactions; Gene Expression; In Vitro Techniques; Mice; Mice, Inbred C57BL; Neostriatum; Phenethylamines; Raclopride; Receptor, Adenosine A1; Receptor, Adenosine A2A; Receptors, Dopamine D1; Signal Transduction; Threonine; Triazines; Triazoles; Xanthines

2006
Adenosine receptors located in the NTS contribute to renal sympathoinhibition during hypotensive phase of severe hemorrhage in anesthetized rats.
    American journal of physiology. Heart and circulatory physiology, 2006, Volume: 291, Issue:5

    Topics: Anesthesia; Animals; Blood Pressure; Heart Rate; Hemorrhage; Kidney; Male; Microinjections; Neural Inhibition; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, Purinergic P1; Solitary Nucleus; Sympathetic Nervous System; Theophylline; Triazines; Triazoles

2006
Characterization of [125I]ZM 241385 binding to adenosine A2A receptors in the pineal of sheep brain.
    Brain research, 2006, Jun-22, Volume: 1096, Issue:1

    Topics: Adenosine; Algorithms; Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Brain Chemistry; Data Interpretation, Statistical; Diencephalon; Female; In Vitro Techniques; Iodine Radioisotopes; Membranes; Pineal Gland; Pregnancy; Receptor, Adenosine A2A; Receptors, G-Protein-Coupled; Sheep; Thalamic Nuclei; Triazines; Triazoles

2006
Mouse spinal cord compression injury is reduced by either activation of the adenosine A2A receptor on bone marrow-derived cells or deletion of the A2A receptor on non-bone marrow-derived cells.
    Neuroscience, 2006, Sep-15, Volume: 141, Issue:4

    Topics: Adenosine A2 Receptor Agonists; Analysis of Variance; Animals; Bone Marrow Cells; Bone Marrow Transplantation; Disease Models, Animal; Dose-Response Relationship, Drug; Enzyme Activation; Female; Mice; Mice, Knockout; Motor Activity; Myelin Sheath; Piperidines; Radioligand Assay; Receptor, Adenosine A2A; Spinal Cord Compression; Time Factors; Triazines; Triazoles

2006
Adenosine A(2A) receptors play a role in the pathogenesis of hepatic cirrhosis.
    British journal of pharmacology, 2006, Volume: 148, Issue:8

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Animals; Blotting, Western; Caffeine; Carbon Tetrachloride; Cell Line; Chromatography, High Pressure Liquid; Ethanol; Hepatocytes; Humans; Liver Cirrhosis; Matrix Metalloproteinases, Membrane-Associated; Methotrexate; Mice; Mice, Inbred C57BL; Rats; Receptor, Adenosine A2A; Reverse Transcriptase Polymerase Chain Reaction; Thioacetamide; Triazines; Triazoles

2006
Caffeine inhibition of rat carotid body chemoreceptors is mediated by A2A and A2B adenosine receptors.
    Journal of neurochemistry, 2006, Volume: 98, Issue:2

    Topics: Adenosine; Animals; Caffeine; Carotid Body; Catecholamines; Central Nervous System Stimulants; Chemoreceptor Cells; Dose-Response Relationship, Drug; Female; Hypoxia; Immunohistochemistry; Male; Potassium; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Receptors, Presynaptic; Respiratory Mechanics; Triazines; Triazoles; Xanthines

2006
Contribution of adenosine receptors in the control of arteriolar tone and adenosine-angiotensin II interaction.
    Kidney international, 2006, Volume: 70, Issue:4

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Angiotensin II; Animals; Arterioles; Feedback; Female; Kidney Glomerulus; Kidney Tubules; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Phenethylamines; Purines; Receptor, Adenosine A1; Receptors, Adenosine A2; Theophylline; Triazines; Triazoles; Vasoconstriction; Vasodilation

2006
Adenosine A2A receptor modulation of juvenile female rat skeletal muscle microvessel permeability.
    American journal of physiology. Heart and circulatory physiology, 2006, Volume: 291, Issue:6

    Topics: Adenine; Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Aging; Animals; Arterioles; Cell Membrane Permeability; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Gene Expression Regulation; Muscle, Skeletal; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptor, Adenosine A2A; Receptor, Adenosine A2B; RNA, Messenger; Serum Albumin; Triazines; Triazoles; Vasodilator Agents; Venules

2006
Adenosine A2A receptors in diffuse dermal fibrosis: pathogenic role in human dermal fibroblasts and in a murine model of scleroderma.
    Arthritis and rheumatism, 2006, Volume: 54, Issue:8

    Topics: Animals; Cells, Cultured; Collagen; Dermis; Disease Models, Animal; Enzyme Inhibitors; Fibroblasts; Fibrosis; Gene Expression; Humans; Hydroxyproline; Male; MAP Kinase Kinase 1; Mice; Mice, Inbred C57BL; Mice, Knockout; Receptor, Adenosine A2A; RNA, Messenger; Scleroderma, Diffuse; Triazines; Triazoles

2006
Functional and cytoarchitectural spinal cord protection by ATL-146e after ischemia/reperfusion is mediated by adenosine receptor agonism.
    Journal of vascular surgery, 2006, Volume: 44, Issue:2

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Cell Survival; Cyclohexanecarboxylic Acids; Disease Models, Animal; Microtubule-Associated Proteins; Neurons; Neuroprotective Agents; Paraplegia; Purines; Rabbits; Receptor, Adenosine A2A; Reperfusion Injury; Spinal Cord; Spinal Cord Ischemia; Time Factors; Triazines; Triazoles

2006
Deficits of glutamate transmission in the striatum of experimental hemiballism.
    Neuroscience, 2006, Nov-17, Volume: 143, Issue:1

    Topics: Anesthetics, Local; Animals; Corpus Striatum; Disease Models, Animal; Dopamine Antagonists; Dyskinesias; Electric Stimulation; Excitatory Postsynaptic Potentials; Glutamic Acid; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Sulpiride; Synaptic Transmission; Tetrodotoxin; Triazines; Triazoles

2006
The A2a/A2b receptor antagonist ZM-241385 blocks the cardioprotective effect of adenosine agonist pretreatment in in vivo rat myocardium.
    American journal of physiology. Heart and circulatory physiology, 2007, Volume: 292, Issue:1

    Topics: Adenosine A2 Receptor Antagonists; Animals; Cardiotonic Agents; Drug Combinations; Male; Myocardial Ischemia; Premedication; Purinergic P1 Receptor Agonists; Rats; Rats, Sprague-Dawley; Treatment Outcome; Triazines; Triazoles

2007
Cl-IB-MECA [2-chloro-N6-(3-iodobenzyl)adenosine-5'-N-methylcarboxamide] reduces ischemia/reperfusion injury in mice by activating the A3 adenosine receptor.
    The Journal of pharmacology and experimental therapeutics, 2006, Volume: 319, Issue:3

    Topics: Adenosine; Adenosine A3 Receptor Agonists; Animals; Blood Pressure; Cardiotonic Agents; Cell Degranulation; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Histamine; In Vitro Techniques; Male; Mice; Mice, Knockout; Myocardial Infarction; Myocardial Reperfusion Injury; Myocardium; p-Methoxy-N-methylphenethylamine; Pyridines; Radioligand Assay; Receptor, Adenosine A3; Triazines; Triazoles

2006
Expression of adenosine receptors in cardiac fibroblasts as a function of insulin and glucose level.
    Archives of biochemistry and biophysics, 2006, Nov-01, Volume: 455, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclases; Animals; Blotting, Western; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Fibroblasts; Gene Expression; Glucose; Heart Ventricles; Insulin; Male; Phenethylamines; Protein Isoforms; Rats; Rats, Wistar; Receptors, Purinergic P1; RNA, Messenger; Triazines; Triazoles

2006
Stimulation of adenosine A1 and A2A receptors by AMP in the submucosal plexus of guinea pig small intestine.
    American journal of physiology. Gastrointestinal and liver physiology, 2007, Volume: 292, Issue:2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Action Potentials; Adenosine; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Adenosine Diphosphate; Adenosine Monophosphate; Animals; Boron Compounds; Enzyme Inhibitors; Estrenes; Excitatory Postsynaptic Potentials; Guinea Pigs; Ileum; Indoles; Male; Maleimides; Norepinephrine; Phenethylamines; Pyrrolidinones; Quinazolines; Receptor, Adenosine A1; Receptor, Adenosine A2A; Signal Transduction; Submucous Plexus; Synaptic Transmission; Tetrodotoxin; Theophylline; Triazines; Triazoles

2007
Tonic adenosine A1 and A2A receptor activation is required for the excitatory action of VIP on synaptic transmission in the CA1 area of the hippocampus.
    Neuropharmacology, 2007, Volume: 52, Issue:2

    Topics: Adenosine; Adenosine Deaminase; Analysis of Variance; Animals; Drug Interactions; Electric Stimulation; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Male; Membrane Potentials; Neuroprotective Agents; Patch-Clamp Techniques; Pyrimidines; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptor, Adenosine A2A; Synaptic Transmission; Triazines; Triazoles; Vasoactive Intestinal Peptide; Xanthines

2007
Synergistic up-regulation of vascular endothelial growth factor (VEGF) expression in macrophages by adenosine A2A receptor agonists and endotoxin involves transcriptional regulation via the hypoxia response element in the VEGF promoter.
    Molecular biology of the cell, 2007, Volume: 18, Issue:1

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Cell Hypoxia; DNA; Exons; Female; Hypoxia-Inducible Factor 1, alpha Subunit; Lipopolysaccharides; Macrophages; Mice; NF-kappa B; Response Elements; RNA, Messenger; Sequence Deletion; Toll-Like Receptor 4; Transcription, Genetic; Triazines; Triazoles; Tumor Necrosis Factor-alpha; Up-Regulation; Vascular Endothelial Growth Factor A

2007
ZM241385, DPCPX, MRS1706 are inverse agonists with different relative intrinsic efficacies on constitutively active mutants of the human adenosine A2B receptor.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 320, Issue:2

    Topics: Adenosine A2 Receptor Agonists; Humans; Mutation; Purines; Saccharomyces cerevisiae; Triazines; Triazoles; Xanthines

2007
Disruption of adenosinergic modulation of ventilation at rest and during hypercapnia by neonatal caffeine in young rats: role of adenosine A(1) and A(2A) receptors.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2007, Volume: 292, Issue:4

    Topics: Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Animals; Caffeine; Central Nervous System Stimulants; Hypercapnia; Injections, Intraperitoneal; Male; Plethysmography; Pulmonary Ventilation; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptor, Adenosine A2A; Rest; Time Factors; Triazines; Triazoles; Xanthines

2007
Cell death in rat cerebellar granule neurons induced by hydrogen peroxide in vitro: mechanisms and protection by adenosine receptor ligands.
    Brain research, 2007, Feb-09, Volume: 1132, Issue:1

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Animals, Newborn; Apoptosis; Brain Diseases; Catalase; Cell Death; Cell Survival; Cells, Cultured; Cerebellar Cortex; Dose-Response Relationship, Drug; Enzyme Inhibitors; Hydrogen Peroxide; Necrosis; Neurons; Oxidative Stress; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptors, Adenosine A2; Receptors, Purinergic P1; Time Factors; Triazines; Triazoles

2007
Attenuation of reperfusion lung injury and apoptosis by A2A adenosine receptor activation is associated with modulation of Bcl-2 and Bax expression and activation of extracellular signal-regulated kinases.
    Shock (Augusta, Ga.), 2007, Volume: 27, Issue:3

    Topics: Adenosine A2 Receptor Agonists; Animals; Apoptosis; bcl-2-Associated X Protein; Cats; Extracellular Signal-Regulated MAP Kinases; Lung; Lung Injury; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Piperidines; Proto-Oncogene Proteins c-bcl-2; Pulmonary Alveoli; Receptor, Adenosine A2A; Reperfusion Injury; Triazines; Triazoles; Wounds and Injuries

2007
Interleukin-1beta but not tumor necrosis factor-alpha potentiates neuronal damage by quinolinic acid: protection by an adenosine A2A receptor antagonist.
    Journal of neuroscience research, 2007, Volume: 85, Issue:5

    Topics: Adenosine A2 Receptor Antagonists; Animals; Brain Injuries; Brain Ischemia; Cytoprotection; Drug Synergism; Hippocampus; Interleukin-1beta; Male; Nerve Degeneration; Neuroprotective Agents; Neurotoxins; Pyramidal Cells; Quinolinic Acid; Rats; Rats, Wistar; Receptor, Adenosine A2A; Triazines; Triazoles; Tumor Necrosis Factor-alpha

2007
Increase in A2A receptors in the nucleus accumbens after extended cocaine self-administration and its disappearance after cocaine withdrawal.
    Brain research, 2007, Apr-27, Volume: 1143

    Topics: Animals; Behavior, Animal; Binding, Competitive; Cocaine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Male; Nucleus Accumbens; Raclopride; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Reinforcement Schedule; Self Administration; Substance Withdrawal Syndrome; Time Factors; Triazines; Triazoles; Tritium

2007
The role of adenosine A2a receptors in experimental acute pancreatitis.
    Advances in medical sciences, 2006, Volume: 51

    Topics: Acute Disease; Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Amylases; Animals; Disease Models, Animal; Immunohistochemistry; Lipase; Male; Pancreas; Pancreatitis; Phenethylamines; Rats; Rats, Wistar; Receptor, Adenosine A2A; Taurocholic Acid; Triazines; Triazoles

2006
Activation of adenosine 2A receptors attenuates allograft rejection and alloantigen recognition.
    Journal of immunology (Baltimore, Md. : 1950), 2007, Apr-01, Volume: 178, Issue:7

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Antibodies, Monoclonal; Antigen-Presenting Cells; Antigens, CD; Antigens, Differentiation; CD3 Complex; CD40 Ligand; CTLA-4 Antigen; Cytokines; Graft Rejection; Interferon-gamma; Interleukin-2 Receptor alpha Subunit; Isoantigens; Lymphocyte Activation; Mice; Mice, Knockout; Piperidines; Programmed Cell Death 1 Receptor; Receptor, Adenosine A2A; Reperfusion Injury; Skin Transplantation; T-Lymphocytes; Triazines; Triazoles; ZAP-70 Protein-Tyrosine Kinase

2007
Endogenous expression of adenosine A1, A2 and A3 receptors in rat C6 glioma cells.
    Neurochemical research, 2007, Volume: 32, Issue:6

    Topics: Adenylyl Cyclases; Animals; Blotting, Western; Brain Neoplasms; Cell Line, Tumor; Cell Membrane; Fluorescent Antibody Technique; Glioma; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Molecular Sequence Data; Nerve Tissue Proteins; Protein Binding; Rats; Receptor, Adenosine A1; Receptor, Adenosine A3; Receptors, Adenosine A2; Reverse Transcriptase Polymerase Chain Reaction; Triazines; Triazoles; Xanthines

2007
Adenosine closes the K+ channel KCa3.1 in human lung mast cells and inhibits their migration via the adenosine A2A receptor.
    European journal of immunology, 2007, Volume: 37, Issue:6

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Benzimidazoles; Calcium Channel Agonists; Cations; Cell Movement; Culture Media, Conditioned; Electric Stimulation; Electrophysiology; Histamine; Humans; Immunoglobulin E; Intermediate-Conductance Calcium-Activated Potassium Channels; Lung; Mast Cells; Phenethylamines; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Triazines; Triazoles

2007
Effects of stimulation of adenosine A2A receptors on lipopolysaccharide-induced production of reactive oxygen species by equine neutrophils.
    American journal of veterinary research, 2007, Volume: 68, Issue:6

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Cyclic AMP; Dose-Response Relationship, Drug; Horses; Lipopolysaccharides; Neutrophils; Reactive Oxygen Species; Receptor, Adenosine A2A; Rolipram; Triazines; Triazoles

2007
The role of adenosine A1 and A2A receptors of entorhinal cortex on piriform cortex kindled seizures in rats.
    Pharmacological research, 2007, Volume: 56, Issue:2

    Topics: Adenosine; Animals; Anticonvulsants; Convulsants; Disease Models, Animal; Electric Stimulation; Electrodes, Implanted; Entorhinal Cortex; Kindling, Neurologic; Male; Microinjections; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptor, Adenosine A2A; Seizures; Triazines; Triazoles; Xanthines

2007
Blockade of adenosine A(2A) receptors prevents staurosporine-induced apoptosis of rat hippocampal neurons.
    Neurobiology of disease, 2007, Volume: 27, Issue:2

    Topics: Adenosine A2 Receptor Antagonists; Animals; Apoptosis; Blotting, Western; Cells, Cultured; Enzyme Inhibitors; Hippocampus; Immunohistochemistry; Male; Mitochondria; Neurons; Phosphoprotein Phosphatases; Rats; Rats, Wistar; Staurosporine; Synaptophysin; Triazines; Triazoles

2007
Targeted deletion of A2A adenosine receptors attenuates the protective effects of myocardial postconditioning.
    American journal of physiology. Heart and circulatory physiology, 2007, Volume: 293, Issue:4

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Animals; Disease Models, Animal; Mice; Mice, Knockout; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Myocardial Reperfusion Injury; Myocardium; Phosphorylation; Proto-Oncogene Proteins c-akt; Receptor, Adenosine A2A; Research Design; Signal Transduction; Time Factors; Triazines; Triazoles; Troponin I; Ventricular Function, Left; Ventricular Pressure

2007
Stimulation of adenosine A2A receptor inhibits LPS-induced expression of intercellular adhesion molecule 1 and production of TNF-alpha in human peripheral blood mononuclear cells.
    Shock (Augusta, Ga.), 2008, Volume: 29, Issue:2

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Agonists; Adenosine A3 Receptor Antagonists; CD40 Antigens; Cells, Cultured; Cyclic AMP; Enzyme-Linked Immunosorbent Assay; Flavins; Flow Cytometry; Humans; Intercellular Adhesion Molecule-1; Leukocytes, Mononuclear; Lipopolysaccharide Receptors; Lipopolysaccharides; Receptor, Adenosine A2A; Triazines; Triazoles; Tumor Necrosis Factor-alpha; Xanthines

2008
Anticonvulsant effect of A1 but not A2A adenosine receptors of piriform cortex in amygdala-kindled rats.
    Canadian journal of physiology and pharmacology, 2007, Volume: 85, Issue:6

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Amygdala; Analysis of Variance; Animals; Anticonvulsants; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; Kindling, Neurologic; Male; Microinjections; Models, Anatomic; Phenethylamines; Rats; Rats, Sprague-Dawley; Theophylline; Triazines; Triazoles

2007
Purinergic modulation of glutamate release under ischemic-like conditions in the hippocampus.
    Neuroscience, 2007, Oct-12, Volume: 149, Issue:1

    Topics: Adenosine; Adenosine Triphosphate; Analgesics; Animals; Dose-Response Relationship, Drug; Glucose; Glutamic Acid; Hippocampus; Hypoxia; In Vitro Techniques; Ischemia; Male; Phenethylamines; Purinergic Agonists; Purinergic Antagonists; Pyrimidines; Rats; Rats, Wistar; Receptors, Purinergic; Sodium Channel Blockers; Tetrodotoxin; Triazines; Triazoles; Xanthines

2007
Interaction of A2A adenosine and D2 dopamine receptors modulates corticostriatal glutamatergic transmission.
    Neuropharmacology, 2007, Volume: 53, Issue:6

    Topics: Adenine; Adenosine; Animals; Cerebral Cortex; Corpus Striatum; Dopamine Agonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Male; Neurons; Organ Culture Techniques; Patch-Clamp Techniques; Phenethylamines; Quinpirole; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Dopamine D2; Synaptic Transmission; Triazines; Triazoles

2007
Adenosine A2A receptor agonists inhibit lipopolysaccharide-induced production of tumor necrosis factor-alpha by equine monocytes.
    Veterinary immunology and immunopathology, 2008, Jan-15, Volume: 121, Issue:1-2

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding, Competitive; Cyclic AMP; Horses; Immunoenzyme Techniques; Lipopolysaccharides; Monocytes; Phenethylamines; Piperidines; Receptor, Adenosine A2A; Regression Analysis; Triazines; Triazoles; Tumor Necrosis Factor-alpha

2008
Adenosine A(2A) receptors are required for normal BDNF levels and BDNF-induced potentiation of synaptic transmission in the mouse hippocampus.
    Journal of neurochemistry, 2008, Volume: 104, Issue:1

    Topics: Adenosine A2 Receptor Antagonists; Animals; Brain-Derived Neurotrophic Factor; Dose-Response Relationship, Drug; Drug Interactions; Enzyme-Linked Immunosorbent Assay; Excitatory Postsynaptic Potentials; Gene Expression Regulation; Hippocampus; In Vitro Techniques; Mice; Mice, Knockout; Patch-Clamp Techniques; Receptor, Adenosine A2A; Synaptic Transmission; Triazines; Triazoles

2008
Activation of adenosine 2A receptors preserves structure and function of podocytes.
    Journal of the American Society of Nephrology : JASN, 2008, Volume: 19, Issue:1

    Topics: Adenosine A2 Receptor Agonists; Albuminuria; Animals; Diabetic Nephropathies; Mice; Mice, Inbred C57BL; Piperidines; Podocytes; Proteinuria; Purine Nucleosides; Receptors, Adenosine A2; Triazines; Triazoles

2008
Up-regulation of adenosine receptors in the frontal cortex in Alzheimer's disease.
    Brain pathology (Zurich, Switzerland), 2008, Volume: 18, Issue:2

    Topics: Adenylyl Cyclases; Aged; Aged, 80 and over; Alzheimer Disease; Analysis of Variance; Cell Membrane; Colforsin; Cyclic AMP; Female; Frontal Lobe; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Male; Middle Aged; Protein Binding; Receptors, Purinergic P1; Triazines; Triazoles; Tritium; Up-Regulation; Xanthines

2008
Involvement of the adenosine A1 and A2A receptors in the antidepressant-like effect of zinc in the forced swimming test.
    Progress in neuro-psychopharmacology & biological psychiatry, 2008, May-15, Volume: 32, Issue:4

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A2 Receptor Agonists; Aniline Compounds; Animals; Antidepressive Agents; Caffeine; Central Nervous System Stimulants; Dipyridamole; Female; Male; Mice; Motor Activity; Nucleoside Transport Proteins; Receptor, Adenosine A1; Receptor, Adenosine A2A; Swimming; Triazines; Triazoles; Xanthines; Zinc

2008
Hypotensive effects of intravenously administered uridine and cytidine in conscious rats: involvement of adenosine receptors.
    European journal of pharmacology, 2008, Apr-14, Volume: 584, Issue:1

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A2 Receptor Agonists; Animals; Antihypertensive Agents; Blood Pressure; Caffeine; Carotid Arteries; Consciousness; Cytidine; Dose-Response Relationship, Drug; Heart Rate; Hypotension; Injections, Intravenous; Injections, Intraventricular; Male; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptor, Adenosine A2A; Theobromine; Theophylline; Time Factors; Triazines; Triazoles; Uridine; Ventricular Function, Left; Ventricular Pressure; Xanthines

2008
Pharmacological blockade of A2A receptors prevents dermal fibrosis in a model of elevated tissue adenosine.
    The American journal of pathology, 2008, Volume: 172, Issue:6

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Animals; Collagen; Fibrosis; Interleukin-13; Mice; Receptor, Adenosine A2A; Skin; Transforming Growth Factor beta1; Triazines; Triazoles

2008
Cerebral blood flow response in adenosine 2a receptor knockout mice during transient hypoxic hypoxia.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2008, Volume: 28, Issue:10

    Topics: Adrenergic alpha-2 Receptor Antagonists; Aminophylline; Animals; Blood Pressure; Cardiotonic Agents; Cerebrovascular Circulation; Female; Hyperemia; Hypoxia, Brain; Ischemic Attack, Transient; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Receptors, Adrenergic, alpha-2; Triazines; Triazoles

2008
Neonatal caffeine induces sex-specific developmental plasticity of the hypoxic respiratory chemoreflex in adult rats.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2008, Volume: 295, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Anesthesia; Animals; Animals, Newborn; Caffeine; Carotid Body; Central Nervous System Stimulants; Female; Gene Expression; Hypoxia; Male; Neural Inhibition; Phrenic Nerve; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Dopamine D2; Reflex; Respiration; RNA, Messenger; Sex Characteristics; Triazines; Triazoles; Tyrosine 3-Monooxygenase

2008
Adenosine receptor subtypes in the airways responses to 5'-adenosine monophosphate inhalation of sensitized guinea-pigs.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 2008, Volume: 38, Issue:9

    Topics: Adenosine Monophosphate; Administration, Inhalation; Animals; Anti-Inflammatory Agents; Asthma; Bronchial Hyperreactivity; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Bronchodilator Agents; Dexamethasone; Dose-Response Relationship, Drug; Guinea Pigs; Immunization; Purinergic P1 Receptor Antagonists; Purines; Quinazolines; Receptors, Purinergic P1; Triazines; Triazoles; Xanthines

2008
Human equilibrative nucleoside transporters 1 and 2 may be differentially modulated by A2B adenosine receptors in placenta microvascular endothelial cells from pre-eclampsia.
    Placenta, 2008, Volume: 29, Issue:9

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adult; Endothelial Cells; Equilibrative Nucleoside Transporter 1; Equilibrative-Nucleoside Transporter 2; Female; Gene Expression Regulation; Humans; Phenethylamines; Placenta; Pre-Eclampsia; Pregnancy; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Triazines; Triazoles

2008
Alcohol-induced retrograde memory impairment in rats: prevention by caffeine.
    Psychopharmacology, 2008, Volume: 201, Issue:3

    Topics: Adenosine A2 Receptor Antagonists; Amnesia, Retrograde; Animals; Caffeine; Central Nervous System Depressants; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Drug Therapy, Combination; Ethanol; Exploratory Behavior; Habituation, Psychophysiologic; Injections, Intraperitoneal; Male; Odorants; Pentylenetetrazole; Phosphodiesterase 5 Inhibitors; Purinones; Rats; Rats, Long-Evans; Rats, Sprague-Dawley; Recognition, Psychology; Seizures; Smell; Time Factors; Triazines; Triazoles; Wood

2008
The 2.6 angstrom crystal structure of a human A2A adenosine receptor bound to an antagonist.
    Science (New York, N.Y.), 2008, Nov-21, Volume: 322, Issue:5905

    Topics: Adenosine A2 Receptor Antagonists; Animals; Binding Sites; Crystallography, X-Ray; Humans; Ligands; Protein Binding; Protein Conformation; Receptor, Adenosine A2A; Structure-Activity Relationship; Triazines; Triazoles; Tryptophan; Turkeys

2008
FGF acts as a co-transmitter through adenosine A(2A) receptor to regulate synaptic plasticity.
    Nature neuroscience, 2008, Volume: 11, Issue:12

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Animals; Cell Differentiation; Cells, Cultured; Chlorocebus aethiops; Cyclic AMP; Embryo, Mammalian; Fibroblast Growth Factors; Hippocampus; Immunoprecipitation; In Vitro Techniques; Long-Term Potentiation; Mitogen-Activated Protein Kinase Kinases; Neurites; Neurons; Patch-Clamp Techniques; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptor Protein-Tyrosine Kinases; Receptor, Adenosine A2A; Receptors, Fibroblast Growth Factor; Synapses; Transfection; Triazines; Triazoles; Two-Hybrid System Techniques

2008
Modulation of gamma oscillations by endogenous adenosine through A1 and A2A receptors in the mouse hippocampus.
    Neuropharmacology, 2009, Volume: 56, Issue:2

    Topics: Adenosine; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Analysis of Variance; Animals; Biological Clocks; Dose-Response Relationship, Drug; Evoked Potentials; Excitatory Amino Acid Agonists; Fourier Analysis; Hippocampus; Hypoxia; In Vitro Techniques; Kainic Acid; Male; Mice; Mice, Inbred C57BL; Phenethylamines; Receptor, Adenosine A1; Receptor, Adenosine A2A; Theophylline; Thioinosine; Time Factors; Triazines; Triazoles

2009
The role of adenosine A(1) receptors in mediating the inhibitory effects of low frequency stimulation of perforant path on kindling acquisition in rats.
    Neuroscience, 2009, Feb-18, Volume: 158, Issue:4

    Topics: Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Analysis of Variance; Animals; Biophysics; Cyclic AMP; Electric Stimulation; Excitatory Postsynaptic Potentials; Hippocampus; Kindling, Neurologic; Male; Neural Inhibition; Perforant Pathway; Rats; Rats, Wistar; Receptor, Adenosine A1; Seizures; Time Factors; Triazines; Triazoles; Xanthines

2009
Caffeine modulates TNF-alpha production by cord blood monocytes: the role of adenosine receptors.
    Pediatric research, 2009, Volume: 65, Issue:2

    Topics: Acetamides; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Antagonists; Adult; Blotting, Western; Caffeine; Cells, Cultured; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme-Linked Immunosorbent Assay; Fetal Blood; Humans; Infant, Newborn; Interleukins; Lipopolysaccharides; Middle Aged; Monocytes; Purines; Quinazolines; Receptor, Adenosine A1; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Receptor, Adenosine A3; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors; Triazines; Triazoles; Tumor Necrosis Factor-alpha; Xanthines

2009
Adenosine A1 and A2a receptors modulate insulinemia, glycemia, and lactatemia in fetal sheep.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2009, Volume: 296, Issue:3

    Topics: Adenosine; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Animals; Blood Gas Analysis; Blood Glucose; Female; Fetus; Hydrogen-Ion Concentration; Hypoxia; Insulin; Lactates; Pregnancy; Receptor, Adenosine A1; Receptor, Adenosine A2A; Sheep; Triazines; Triazoles; Xanthines

2009
Angiotensin II enhances the afferent arteriolar response to adenosine through increases in cytosolic calcium.
    Acta physiologica (Oxford, England), 2009, Volume: 196, Issue:4

    Topics: Adenosine; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Animals; Arterioles; Calcium; Cytosol; Kidney; Male; Mice; Mice, Inbred C57BL; Muscle, Smooth, Vascular; Naphthyridines; Purines; Receptor, Adenosine A1; Receptor, Angiotensin, Type 1; Receptors, Adenosine A2; Triazines; Triazoles; Vasoconstriction

2009
Adenosine A(1) and A(2A) receptors in mouse prefrontal cortex modulate acetylcholine release and behavioral arousal.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2009, Jan-21, Volume: 29, Issue:3

    Topics: Acetylcholine; Adenosine; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Analysis of Variance; Animals; Arousal; Behavior, Animal; Caffeine; Chromatography, High Pressure Liquid; Electroencephalography; Electromyography; Male; Mice; Microdialysis; Phenethylamines; Phosphodiesterase Inhibitors; Prefrontal Cortex; Receptor, Adenosine A1; Receptors, Adenosine A2; Spectrum Analysis; Triazines; Triazoles; Xanthines

2009
Activation of NTS A2a adenosine receptors differentially resets baroreflex control of renal vs. adrenal sympathetic nerve activity.
    American journal of physiology. Heart and circulatory physiology, 2009, Volume: 296, Issue:4

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adrenal Glands; Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Heart Rate; Kidney; Male; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptor, Adenosine A2A; Solitary Nucleus; Sympathetic Nervous System; Theophylline; Triazines; Triazoles

2009
Nitric oxide (NO) does not contribute to the generation or action of adenosine during exercise hyperaemia in rat hindlimb.
    The Journal of physiology, 2009, Apr-01, Volume: 587, Issue:Pt 7

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Animals; Cyclic GMP; Electric Stimulation; Enzyme Inhibitors; Femoral Artery; Hindlimb; Hyperemia; Isometric Contraction; Male; Muscle, Skeletal; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Donors; Nitric Oxide Synthase; Oxygen Consumption; Physical Exertion; Rats; Rats, Wistar; Receptor, Adenosine A2A; Regional Blood Flow; S-Nitroso-N-Acetylpenicillamine; Sciatic Nerve; Time Factors; Triazines; Triazoles; Vasodilation

2009
Elucidation in the rat of the role of adenosine and A2A-receptors in the hyperaemia of twitch and tetanic contractions.
    The Journal of physiology, 2009, Apr-01, Volume: 587, Issue:Pt 7

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Animals; Blood Pressure; Carbon Dioxide; Electric Stimulation; Femoral Artery; Hydrogen-Ion Concentration; Hyperemia; Isometric Contraction; Male; Muscle, Skeletal; Muscle, Smooth, Vascular; Oxygen; Rats; Rats, Wistar; Receptor, Adenosine A2A; Regional Blood Flow; Sciatic Nerve; Theophylline; Time Factors; Triazines; Triazoles; Vasodilation

2009
Adenosine receptor antagonists improve short-term object-recognition ability of spontaneously hypertensive rats: a rodent model of attention-deficit hyperactivity disorder.
    Behavioural pharmacology, 2009, Volume: 20, Issue:2

    Topics: Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Animals; Attention Deficit Disorder with Hyperactivity; Blood Pressure; Caffeine; Disease Models, Animal; Female; Male; Memory, Short-Term; Methylphenidate; Rats; Rats, Inbred SHR; Rats, Wistar; Receptor, Adenosine A1; Receptors, Adenosine A2; Recognition, Psychology; Triazines; Triazoles; Xanthines

2009
Multiple receptor subtypes and multiple mechanisms of dilation are involved in vascular network dilation caused by adenosine.
    Microvascular research, 2009, Volume: 77, Issue:3

    Topics: Adenosine; Animals; Arterioles; Cricetinae; Drug Antagonism; Endothelium, Vascular; Flavins; Mesocricetus; Methacholine Chloride; Nitroprusside; Purinergic P1 Receptor Antagonists; Quinazolines; Receptors, Purinergic P1; Triazines; Triazoles; Vasodilation; Vasodilator Agents

2009
Cardioprotection induced by adenosine A1 receptor agonists in a cardiac cell ischemia model involves cooperative activation of adenosine A2A and A2B receptors by endogenous adenosine.
    Journal of cardiovascular pharmacology, 2009, Volume: 53, Issue:5

    Topics: Acetamides; Adenosine; Adenosine A1 Receptor Agonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Agonists; Adenosine A3 Receptor Antagonists; Aminopyridines; Animals; Apoptosis; Cardiotonic Agents; Cell Line; Cell Survival; Dihydropyridines; Imidazoles; Myocardial Ischemia; Phenethylamines; Purines; Rats; Triazines; Triazoles; Xanthines

2009
Attenuation of gastric mucosal inflammation induced by indomethacin through activation of the A2A adenosine receptor in rats.
    Journal of gastroenterology, 2009, Volume: 44, Issue:5

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Anti-Inflammatory Agents, Non-Steroidal; Chemokine CXCL1; Dinoprostone; Gastric Mucosa; Indomethacin; Inflammation; Interleukin-1beta; Male; Peroxidase; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Stomach Ulcer; Triazines; Triazoles; Tumor Necrosis Factor-alpha

2009
Effect of adenosine A(2A) receptor antagonists on L-DOPA-induced hydroxyl radical formation in rat striatum.
    Neurotoxicity research, 2009, Volume: 15, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adenosine A2 Receptor Antagonists; Animals; Area Under Curve; Benserazide; Catalepsy; Corpus Striatum; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Drug Interactions; Haloperidol; Homovanillic Acid; Hydroxyl Radical; Levodopa; Male; Microdialysis; Rats; Rats, Wistar; Time Factors; Triazines; Triazoles; Xanthines

2009
A2A adenosine receptor antagonists protect the striatum against rotenone-induced neurotoxicity.
    Experimental neurology, 2009, Volume: 217, Issue:1

    Topics: Action Potentials; Adenine; Adenosine A2 Receptor Antagonists; Animals; Cerebral Cortex; Corpus Striatum; Dose-Response Relationship, Drug; In Vitro Techniques; Insecticides; Male; Neurons; Rats; Rats, Wistar; Rotenone; Time Factors; Triazines; Triazoles

2009
The adenosine A2A receptor antagonist ZM241385 enhances neuronal survival after oxygen-glucose deprivation in rat CA1 hippocampal slices.
    British journal of pharmacology, 2009, Volume: 157, Issue:5

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Animals; Astrocytes; Blotting, Western; Brain Ischemia; Cell Hypoxia; Cell Survival; Coloring Agents; Excitatory Postsynaptic Potentials; Glial Fibrillary Acidic Protein; Glucose; Hippocampus; Immunohistochemistry; In Vitro Techniques; Male; Neurons; Neuroprotective Agents; Oxygen; Phenethylamines; Propidium; Pyrazoles; Pyrimidines; Rats; Rats, Wistar; Receptor, Adenosine A2A; Staining and Labeling; Time Factors; Triazines; Triazoles

2009
Adenosine A1 receptors presynaptically modulate excitatory synaptic input onto subiculum neurons.
    Brain research, 2009, Jul-14, Volume: 1280

    Topics: Action Potentials; Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Central Nervous System Agents; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Membrane Potentials; Neurons; Presynaptic Terminals; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptors, Adenosine A2; Synapses; Synaptic Transmission; Triazines; Triazoles; Xanthines

2009
Differential regulation of HIF-1alpha isoforms in murine macrophages by TLR4 and adenosine A(2A) receptor agonists.
    Journal of leukocyte biology, 2009, Volume: 86, Issue:3

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Cells, Cultured; Drug Combinations; Female; Gene Expression Regulation; Genes, Reporter; Hypoxia-Inducible Factor 1, alpha Subunit; Lipopolysaccharides; Luciferases, Renilla; Macrophages, Peritoneal; Mice; Mice, Congenic; Mice, Inbred C57BL; NF-kappa B; Nitriles; Phenethylamines; Protein Isoforms; Purinergic P1 Receptor Agonists; RNA, Messenger; Sulfones; Toll-Like Receptor 4; Transfection; Triazines; Triazoles; Vascular Endothelial Growth Factor A

2009
Cannabidiol ameliorates cognitive and motor impairments in mice with bile duct ligation.
    Journal of hepatology, 2009, Volume: 51, Issue:3

    Topics: Adenosine A2 Receptor Antagonists; Animals; Bile Ducts; Brain-Derived Neurotrophic Factor; Cannabidiol; Chronic Disease; Cognition; Cognition Disorders; Cyclooxygenase 2; Disease Models, Animal; Female; Gait Disorders, Neurologic; Hepatic Encephalopathy; Ligation; Liver Diseases; Mice; Mice, Inbred Strains; Motor Activity; Receptor, Adenosine A2A; Receptors, Tumor Necrosis Factor, Type I; RNA, Messenger; Treatment Outcome; Triazines; Triazoles

2009
Region-specific neuroprotective effect of ZM 241385 towards glutamate uptake inhibition in cultured neurons.
    European journal of pharmacology, 2009, Sep-01, Volume: 617, Issue:1-3

    Topics: Adenosine A2 Receptor Antagonists; Animals; Binding, Competitive; Biological Transport; Biomimetics; Blotting, Western; Cells, Cultured; Cerebral Cortex; Dicarboxylic Acids; Female; Gene Expression Regulation; Glutamic Acid; Neostriatum; Neurons; Neuroprotective Agents; Organ Specificity; Pregnancy; Pyrrolidines; Rats; Receptor, Adenosine A2A; Substrate Specificity; Triazines; Triazoles

2009
Adenosine A2A receptors enable the synaptic effects of cannabinoid CB1 receptors in the rodent striatum.
    Journal of neurochemistry, 2009, Volume: 110, Issue:6

    Topics: Action Potentials; Animals; Benzoxazines; Biophysics; Calcium; Calcium Channel Blockers; Cerebral Cortex; Corpus Striatum; Electric Stimulation; Embryo, Mammalian; Excitatory Amino Acid Agonists; Female; Glycine; In Vitro Techniques; L-Lactate Dehydrogenase; Male; Mice; Mice, Knockout; Morpholines; N-Methylaspartate; Naphthalenes; Neurons; Phenylacetates; Piperidines; Pregnancy; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptors, Adenosine A2; Synapses; Triazines; Triazoles

2009
2-Phenylpyrazolo[4,3-d]pyrimidin-7-one as a new scaffold to obtain potent and selective human A3 adenosine receptor antagonists: new insights into the receptor-antagonist recognition.
    Journal of medicinal chemistry, 2009, Dec-10, Volume: 52, Issue:23

    Topics: Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Antagonists; Amino Acid Sequence; Animals; CHO Cells; Cricetinae; Cricetulus; Humans; Models, Molecular; Molecular Conformation; Molecular Sequence Data; Protein Binding; Pyrazoles; Pyrimidines; Pyrimidinones; Receptor, Adenosine A2A; Receptor, Adenosine A3; Substrate Specificity; Triazines; Triazoles

2009
Homology modelling of the human adenosine A2B receptor based on X-ray structures of bovine rhodopsin, the beta2-adrenergic receptor and the human adenosine A2A receptor.
    Journal of computer-aided molecular design, 2009, Volume: 23, Issue:11

    Topics: Animals; Cattle; Humans; Models, Molecular; Molecular Structure; Mutagenesis, Site-Directed; Protein Binding; Protein Conformation; Receptor, Adenosine A2B; Receptors, Adrenergic, beta-2; Rhodopsin; Triazines; Triazoles; X-Rays

2009
Inhibition of the adenosine2A receptor-epoxyeicosatrienoic acid pathway renders Dahl salt-resistant rats hypertensive.
    Hypertension (Dallas, Tex. : 1979), 2009, Volume: 54, Issue:6

    Topics: Adrenergic alpha-2 Receptor Antagonists; Amides; Animals; Blood Pressure; Drinking; Eicosanoids; Hydroxyeicosatetraenoic Acids; Hypertension, Renal; Male; Natriuresis; Oxidoreductases; Rats; Rats, Inbred Dahl; Receptors, Adrenergic, alpha-2; Sodium Chloride, Dietary; Triazines; Triazoles

2009
Human follicular lymphoma CD39+-infiltrating T cells contribute to adenosine-mediated T cell hyporesponsiveness.
    Journal of immunology (Baltimore, Md. : 1950), 2009, Nov-15, Volume: 183, Issue:10

    Topics: Adenosine; Adenosine Triphosphate; Antigens, CD; Apyrase; CD8-Positive T-Lymphocytes; Clonal Anergy; Humans; Interferon-gamma; Interleukin-2; Lymphocytes, Tumor-Infiltrating; Lymphoma, Follicular; Neuroprotective Agents; Pyrimidines; Receptors, Purinergic P1; T-Lymphocytes, Regulatory; Triazines; Triazoles

2009
Role of adenosine A2 receptors in regulation of cerebral blood flow during induced hypotension.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 2010, Volume: 30, Issue:4

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Cerebrovascular Circulation; Dipyridamole; Hypotension; Male; Mice; Mice, Knockout; Phenethylamines; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Triazines; Triazoles; Vasodilation; Vasodilator Agents

2010
DNA methylation regulates adenosine A(2A) receptor cell surface expression levels.
    Journal of neurochemistry, 2010, Volume: 112, Issue:5

    Topics: Azacitidine; Cell Line; Chromatin Immunoprecipitation; DNA Methylation; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gene Expression Regulation; HeLa Cells; Humans; Immunoprecipitation; Methyl-CpG-Binding Protein 2; Neuroblastoma; Protein Binding; Radioligand Assay; Receptor, Adenosine A2A; Receptors, Cell Surface; RNA, Messenger; S-Adenosylmethionine; Time Factors; Triazines; Triazoles; Tritium

2010
Blockade of adenosine A2A receptor counteracts neuropeptide-S-induced hyperlocomotion in mice.
    Naunyn-Schmiedeberg's archives of pharmacology, 2010, Volume: 381, Issue:2

    Topics: Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Animals; Caffeine; Humans; Male; Mice; Mice, Inbred Strains; Motor Activity; Neuropeptides; Triazines; Triazoles

2010
Lipopolysaccharide and TNF-alpha modify adenosine A(2A) receptor expression and function in equine monocytes.
    Veterinary immunology and immunopathology, 2010, Jun-15, Volume: 135, Issue:3-4

    Topics: Adenosine A2 Receptor Agonists; Animals; Animals, Newborn; Base Sequence; DNA Primers; Horse Diseases; Horses; Humans; In Vitro Techniques; Lipopolysaccharides; Mice; Monocytes; Piperidines; Radioligand Assay; Receptor, Adenosine A2A; Recombinant Proteins; RNA, Messenger; Systemic Inflammatory Response Syndrome; Triazines; Triazoles; Tumor Necrosis Factor-alpha

2010
Predicted 3D structures for adenosine receptors bound to ligands: comparison to the crystal structure.
    Journal of structural biology, 2010, Volume: 170, Issue:1

    Topics: Binding Sites; Crystallization; Humans; Models, Molecular; Molecular Structure; Monte Carlo Method; Protein Conformation; Receptor, Adenosine A2A; Triazines; Triazoles

2010
Adenosine inhibits paraventricular pre-sympathetic neurons through ATP-dependent potassium channels.
    Journal of neurochemistry, 2010, Volume: 113, Issue:2

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Adenosine; Analgesics; Animals; Bicuculline; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; GABA Antagonists; Glyburide; Guanosine Diphosphate; In Vitro Techniques; KATP Channels; Male; Membrane Potentials; Neurons; Paraventricular Hypothalamic Nucleus; Patch-Clamp Techniques; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Sodium Channel Blockers; Tetrodotoxin; Thionucleotides; Tolbutamide; Triazines; Triazoles; Xanthines

2010
The role of adenosine receptors in regulating production of tumour necrosis factor-alpha and chemokines by human lung macrophages.
    British journal of pharmacology, 2010, Volume: 159, Issue:6

    Topics: Acetamides; Cells, Cultured; Chemokines; Female; Humans; Lipopolysaccharides; Lung; Macrophages, Alveolar; Male; Middle Aged; Protein Subunits; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Quinazolines; Receptors, Purinergic P1; Reverse Transcriptase Polymerase Chain Reaction; Triazines; Triazoles; Tumor Necrosis Factor-alpha

2010
Adenosine A(2)A receptor but not HIF-1 mediates Tyrosine hydroxylase induction in hypoxic PC12 cells.
    Journal of neuroscience research, 2010, Volume: 88, Issue:9

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Aryl Hydrocarbon Receptor Nuclear Translocator; Cell Hypoxia; Cyclic AMP Response Element-Binding Protein; DNA; Hypoxia-Inducible Factor 1; Hypoxia-Inducible Factor 1, alpha Subunit; Mutation; PC12 Cells; Phenethylamines; Promoter Regions, Genetic; Rats; Receptor, Adenosine A2A; RNA, Messenger; Signal Transduction; Transcription, Genetic; Transfection; Triazines; Triazoles; Tyrosine 3-Monooxygenase

2010
Ligand binding and subtype selectivity of the human A(2A) adenosine receptor: identification and characterization of essential amino acid residues.
    The Journal of biological chemistry, 2010, Apr-23, Volume: 285, Issue:17

    Topics: Adenosine A2 Receptor Antagonists; Amino Acid Substitution; Binding Sites; Cell Line; Humans; Ligands; Models, Molecular; Mutagenesis; Mutation, Missense; Protein Binding; Receptor, Adenosine A2A; Triazines; Triazoles

2010
Priming of signal transducer and activator of transcription proteins for cytokine-triggered polyubiquitylation and degradation by the A 2A adenosine receptor.
    Molecular pharmacology, 2010, Volume: 77, Issue:6

    Topics: Animals; Blotting, Western; Cells, Cultured; Cytokines; Down-Regulation; Humans; Hydrolysis; Immunoprecipitation; Mice; Mice, Knockout; Phosphorylation; Receptors, Adenosine A2; STAT Transcription Factors; Triazines; Triazoles; Ubiquitination

2010
Acadesine inhibits tissue factor induction and thrombus formation by activating the phosphoinositide 3-kinase/Akt signaling pathway.
    Arteriosclerosis, thrombosis, and vascular biology, 2010, Volume: 30, Issue:5

    Topics: Adenosine A2 Receptor Antagonists; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Apolipoproteins E; Atherosclerosis; Blood Coagulation; Cells, Cultured; Disease Models, Animal; Dose-Response Relationship, Drug; Endothelial Cells; Enzyme Activation; Fibrinolytic Agents; Humans; Lipopolysaccharides; Macrophages; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Monocytes; NF-kappa B; Phosphatidylinositol 3-Kinases; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Pyrazoles; Pyrimidines; Receptor, Adenosine A2A; Ribonucleosides; RNA, Messenger; Sepsis; Signal Transduction; Thromboplastin; Transcription Factor AP-1; Triazines; Triazoles; Up-Regulation; Venous Thrombosis

2010
Adenosine activates a2b receptors and enhances chloride secretion in kidney inner medullary collecting duct cells.
    Hypertension (Dallas, Tex. : 1979), 2010, Volume: 55, Issue:5

    Topics: Adenosine; Animals; Cell Line; Chlorides; Cystic Fibrosis Transmembrane Conductance Regulator; Kidney Medulla; Kidney Tubules, Collecting; Pyrazoles; Pyrimidines; Rats; Receptor, Adenosine A2B; Triazines; Triazoles; Xanthines

2010
Adenosine A(2) receptors modulate tubuloglomerular feedback.
    American journal of physiology. Renal physiology, 2010, Volume: 299, Issue:2

    Topics: Adenosine; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Animals; Arterioles; Blood Pressure; Feedback, Physiological; Kidney Glomerulus; Kidney Tubules; Male; Microcirculation; Perfusion; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A1; Receptor, Adenosine A2A; Renal Circulation; Triazines; Triazoles; Vasoconstriction; Vasodilation; Xanthines

2010
Activation of adenosine A2A receptor attenuates inflammatory response in a rat model of small-for-size liver transplantation.
    Transplantation proceedings, 2010, Volume: 42, Issue:5

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Alanine Transaminase; Animals; Chemokine CXCL2; Cytokines; Enzyme-Linked Immunosorbent Assay; Inflammation; Intercellular Adhesion Molecule-1; Liver; Liver Transplantation; Male; NF-kappa B; Organ Size; Peroxidase; Phenethylamines; Phosphorylation; Rats; Rats, Inbred Lew; Receptor, Adenosine A2A; Triazines; Triazoles; Tumor Necrosis Factor-alpha

2010
Peripheral adenosine A2A receptors are involved in carrageenan-induced mechanical hyperalgesia in mice.
    Neuroscience, 2010, Oct-27, Volume: 170, Issue:3

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Carrageenan; Female; Ganglia, Spinal; Hyperalgesia; Inflammation; Injections, Intraperitoneal; Injections, Subcutaneous; Male; Mice; Mice, Knockout; Pain; Pain Threshold; Phenethylamines; Receptor, Adenosine A2A; Sex Characteristics; Triazines; Triazoles

2010
Cooperative cardioprotection through adenosine A1 and A2A receptor agonism in ischemia-reperfused isolated mouse heart.
    Journal of cardiovascular pharmacology, 2010, Volume: 56, Issue:4

    Topics: Acetamides; Adenosine; Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Blood Pressure; Cardiotonic Agents; Drug Synergism; In Vitro Techniques; Male; Mice; Mice, Knockout; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Myocardial Contraction; Myocardial Reperfusion Injury; Phosphorylation; Purines; Receptor, Adenosine A2A; Triazines; Triazoles; Xanthines

2010
GPCR structure and activation: an essential role for the first extracellular loop in activating the adenosine A2B receptor.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2011, Volume: 25, Issue:2

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Amino Acid Sequence; Aminopyridines; Gene Expression Regulation; Humans; Models, Molecular; Molecular Structure; Mutagenesis, Site-Directed; Protein Conformation; Receptor, Adenosine A2B; Saccharomyces cerevisiae; Triazines; Triazoles

2011
Static magnetic field exposure reproduces cellular effects of the Parkinson's disease drug candidate ZM241385.
    PloS one, 2010, Nov-08, Volume: 5, Issue:11

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine Triphosphate; Analysis of Variance; Animals; Blotting, Western; Calcium; Cell Proliferation; Cyclic AMP; Iron; Magnetic Field Therapy; Magnetics; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Neurites; Parkinson Disease; PC12 Cells; Phenethylamines; Phosphorylation; Rats; Receptor, Adenosine A2A; Triazines; Triazoles

2010
Abnormal calcium handling in atrial fibrillation is linked to up-regulation of adenosine A2A receptors.
    European heart journal, 2011, Volume: 32, Issue:6

    Topics: Adenosine A2 Receptor Antagonists; Aged; Atrial Fibrillation; Blotting, Western; Calcium; Calcium Channels, L-Type; Calcium Signaling; Female; Humans; Male; Middle Aged; Myocytes, Cardiac; Real-Time Polymerase Chain Reaction; Receptor, Adenosine A2A; RNA, Messenger; Sarcoplasmic Reticulum; Triazines; Triazoles; Up-Regulation

2011
Presynaptic facilitatory adenosine A2A receptors mediate fade induced by neuromuscular relaxants that exhibit anticholinesterase activity.
    Clinical and experimental pharmacology & physiology, 2011, Volume: 38, Issue:3

    Topics: Acetylcholine; Animals; Atracurium; Cholinesterase Inhibitors; Diaphragm; Electric Stimulation; Hexamethonium; Male; Muscle Contraction; Neuromuscular Agents; Neuromuscular Junction; Pancuronium; Phrenic Nerve; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptor, Muscarinic M2; Receptors, Nicotinic; Receptors, Presynaptic; Synaptic Transmission; Triazines; Triazoles; Tubocurarine; Vecuronium Bromide

2011
A(2A) adenosine receptor binding parameters in platelets from patients affected by pathological gambling.
    Neuropsychobiology, 2011, Volume: 63, Issue:3

    Topics: Adult; Blood Platelets; Case-Control Studies; Female; Gambling; Humans; Kinetics; Male; Radioligand Assay; Radionuclide Imaging; Receptor, Adenosine A2A; Triazines; Triazoles; Tritium

2011
Structure of an agonist-bound human A2A adenosine receptor.
    Science (New York, N.Y.), 2011, Apr-15, Volume: 332, Issue:6027

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Binding Sites; Crystallography, X-Ray; Humans; Hydrogen Bonding; Ligands; Models, Molecular; Opsins; Protein Conformation; Protein Structure, Secondary; Receptor, Adenosine A2A; Rhodopsin; Triazines; Triazoles

2011
Adenosine A(2A) receptor activation prevents progressive kidney fibrosis in a model of immune-associated chronic inflammation.
    Kidney international, 2011, Volume: 80, Issue:4

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Anti-Inflammatory Agents; Autoantibodies; Disease Models, Animal; Extracellular Matrix Proteins; Fibrosis; Glomerulonephritis; Inflammation Mediators; Kidney; Macrophages; Male; Phenethylamines; Rats; Rats, Inbred WKY; Receptor, Adenosine A2A; Severity of Illness Index; Time Factors; Triazines; Triazoles

2011
Adenosine A2(A) receptor modulates the oxidative stress response of primed polymorphonuclear leukocytes after parabolic flight.
    Human immunology, 2011, Volume: 72, Issue:7

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Adult; Gene Expression Regulation; Gravity, Altered; Humans; Hydrogen Peroxide; Immunologic Factors; Male; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Oxidative Stress; Receptors, Adenosine A2; RNA, Messenger; Triazines; Triazoles; Tumor Necrosis Factor-alpha; Vasodilator Agents

2011
Agonist-bound adenosine A2A receptor structures reveal common features of GPCR activation.
    Nature, 2011, May-18, Volume: 474, Issue:7352

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Binding Sites; CHO Cells; Cricetinae; Cricetulus; Crystallography, X-Ray; Drug Inverse Agonism; Humans; Ligands; Models, Molecular; Molecular Conformation; Receptor, Adenosine A2A; Triazines; Triazoles

2011
Biophysical mapping of the adenosine A2A receptor.
    Journal of medicinal chemistry, 2011, Jul-14, Volume: 54, Issue:13

    Topics: Adenosine A2 Receptor Antagonists; Binding Sites; Drug Design; Ligands; Models, Molecular; Mutation; Pyrimidines; Receptor, Adenosine A2A; Small Molecule Libraries; Triazines; Triazoles; Xanthines

2011
The effect of A(2A) adenosine receptor activation on C-C chemokine receptor 7 expression in human THP1 macrophages during inflammation.
    Inflammation, 2012, Volume: 35, Issue:2

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Cell Line; Cell Movement; Chemokine CCL21; Humans; Inflammation; Macrophages; Phenethylamines; Receptors, Adenosine A2; Receptors, CCR7; RNA, Messenger; Triazines; Triazoles

2012
mGlu5 and adenosine A2A receptor interactions regulate the conditioned effects of cocaine.
    The international journal of neuropsychopharmacology, 2012, Volume: 15, Issue:7

    Topics: Analysis of Variance; Animals; Autoradiography; Brain; Cocaine; Conditioning, Operant; Dopamine Uptake Inhibitors; Drug Interactions; Excitatory Amino Acid Antagonists; Iodine Isotopes; Locomotion; Male; Mice; Mice, Knockout; Protein Binding; Pyridines; Radionuclide Imaging; Receptor, Adenosine A2A; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Thiazoles; Time Factors; Triazines; Triazoles

2012
Effect of adenosine A(2A) receptor antagonists and L-DOPA on hydroxyl radical, glutamate and dopamine in the striatum of 6-OHDA-treated rats.
    Neurotoxicity research, 2012, Volume: 21, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adenosine A2 Receptor Antagonists; Animals; Benserazide; Caffeine; Dopamine; Glutamic Acid; Hydroxyl Radical; Levodopa; Male; Microdialysis; Neostriatum; Oxidopamine; Parkinsonian Disorders; Rats; Rats, Wistar; Receptor, Adenosine A2A; Triazines; Triazoles

2012
Structure of the adenosine A(2A) receptor in complex with ZM241385 and the xanthines XAC and caffeine.
    Structure (London, England : 1993), 2011, Sep-07, Volume: 19, Issue:9

    Topics: Adenosine A2 Receptor Agonists; Amino Acid Motifs; Amino Acid Sequence; Amino Acid Substitution; Binding Sites; Caffeine; Crystallography, X-Ray; HEK293 Cells; Humans; Hydrogen Bonding; Models, Molecular; Molecular Sequence Data; Mutagenesis, Site-Directed; Protein Binding; Protein Stability; Protein Structure, Tertiary; Receptor, Adenosine A2A; Surface Properties; Triazines; Triazoles; Xanthines

2011
Computational study of the binding modes of caffeine to the adenosine A2A receptor.
    The journal of physical chemistry. B, 2011, Dec-01, Volume: 115, Issue:47

    Topics: Amino Acid Substitution; Caffeine; Entropy; Humans; Lipid Bilayers; Molecular Dynamics Simulation; Mutagenesis, Site-Directed; Protein Binding; Protein Structure, Tertiary; Receptor, Adenosine A2A; Triazines; Triazoles

2011
Functional interaction between purinergic receptors: effect of ligands for A2A and P2Y12 receptors on P2Y1 receptor function.
    FEBS letters, 2011, Dec-15, Volume: 585, Issue:24

    Topics: Adenosine A2 Receptor Antagonists; Calcium Signaling; Cell Line, Tumor; Gene Expression Regulation; HEK293 Cells; Humans; Intracellular Space; Ligands; Protein Binding; Purinergic P2Y Receptor Agonists; Purinergic P2Y Receptor Antagonists; Receptor, Adenosine A2A; Receptors, Purinergic P2Y1; Receptors, Purinergic P2Y12; Triazines; Triazoles

2011
Cannabidiol, a non-psychotropic plant-derived cannabinoid, decreases inflammation in a murine model of acute lung injury: role for the adenosine A(2A) receptor.
    European journal of pharmacology, 2012, Mar-05, Volume: 678, Issue:1-3

    Topics: Acute Lung Injury; Adenosine A2 Receptor Antagonists; Animals; Anti-Inflammatory Agents; Bone Marrow Cells; Bronchoalveolar Lavage Fluid; Cannabidiol; Cannabinoids; Capillary Permeability; Chemokines; Cytokines; Disease Models, Animal; Drug Evaluation, Preclinical; Leukocytes; Male; Mice; Mice, Inbred C57BL; Peroxidase; Receptor, Adenosine A2A; Triazines; Triazoles

2012
The effect of adenosine A(2A) receptor antagonists on hydroxyl radical, dopamine, and glutamate in the striatum of rats with altered function of VMAT2.
    Neurotoxicity research, 2012, Volume: 22, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adenosine A2 Receptor Antagonists; Adrenergic Uptake Inhibitors; Animals; Caffeine; Corpus Striatum; Dopamine; Dopamine Agents; Extracellular Space; Glutamic Acid; Homovanillic Acid; Hydroxyl Radical; Levodopa; Male; Microdialysis; Oxidative Stress; Rats; Rats, Wistar; Reserpine; Triazines; Triazoles; Vesicular Monoamine Transport Proteins

2012
Suppression of bladder overactivity by adenosine A2A receptor antagonist in a rat model of Parkinson disease.
    The Journal of urology, 2012, Volume: 187, Issue:5

    Topics: Adenosine A2 Receptor Antagonists; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Female; Parkinson Disease; Rats; Rats, Sprague-Dawley; Triazines; Triazoles; Urinary Bladder, Overactive; Urination

2012
mGlu5R promotes glutamate AMPA receptor phosphorylation via activation of PKA/DARPP-32 signaling in striatopallidal medium spiny neurons.
    Neuropharmacology, 2013, Volume: 66

    Topics: Animals; Corpus Striatum; Cyclic AMP-Dependent Protein Kinases; Dopamine and cAMP-Regulated Phosphoprotein 32; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Phosphorylation; Purinergic P1 Receptor Antagonists; Pyridines; Receptor, Adenosine A2A; Receptor, Metabotropic Glutamate 5; Receptors, AMPA; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Metabotropic Glutamate; Resorcinols; Signal Transduction; Triazines; Triazoles

2013
Effect of adenosine A2A receptor antagonist ZM241385 on amygdala-kindled seizures and progression of amygdala kindling.
    Journal of Huazhong University of Science and Technology. Medical sciences = Hua zhong ke ji da xue xue bao. Yi xue Ying De wen ban = Huazhong keji daxue xuebao. Yixue Yingdewen ban, 2012, Volume: 32, Issue:2

    Topics: Adenosine A2 Receptor Antagonists; Amygdala; Animals; Dose-Response Relationship, Drug; Male; Rats; Rats, Wistar; Receptor, Adenosine A2A; Seizures; Treatment Outcome; Triazines; Triazoles

2012
A novel dihydro-pyrazolo(3,4d)(1,2,4)triazolo(1,5a)pyrimidin-4-one (AJ23) is an antagonist at adenosine A(1) receptors and enhances consolidation of step-down avoidance.
    Behavioural brain research, 2012, Oct-01, Volume: 234, Issue:2

    Topics: Adenosine; Analysis of Variance; Animals; Avoidance Learning; CA1 Region, Hippocampal; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Electric Stimulation; Excitatory Postsynaptic Potentials; HEK293 Cells; Heterocyclic Compounds, 3-Ring; Humans; In Vitro Techniques; Inhibition, Psychological; Male; Protein Binding; Purinergic P1 Receptor Antagonists; Pyrimidines; Rats; Rats, Wistar; Reaction Time; Retention, Psychology; Structure-Activity Relationship; Triazines; Triazoles; Tritium; Xanthines

2012
Pharmacological blockade of adenosine A2A receptors diminishes scarring.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2012, Volume: 26, Issue:10

    Topics: Adenosine A2 Receptor Antagonists; Animals; Blotting, Western; Cicatrix; Collagen; Immunohistochemistry; Male; Mice; Mice, Inbred C57BL; Receptor, Adenosine A2A; Reverse Transcriptase Polymerase Chain Reaction; Triazines; Triazoles; Wound Healing

2012
The mechanism of beta-adrenergic preconditioning: roles for adenosine and ROS during triggering and mediation.
    Basic research in cardiology, 2012, Volume: 107, Issue:5

    Topics: Adenosine; Animals; Ethanolamines; Extracellular Signal-Regulated MAP Kinases; Formoterol Fumarate; Ischemic Preconditioning, Myocardial; Isoproterenol; Myocardial Infarction; Phosphatidylinositol 3-Kinases; Potassium Channels; Protein Kinase C; Proto-Oncogene Proteins c-akt; Rats; Reactive Oxygen Species; Receptors, Adrenergic, beta; Receptors, Purinergic P1; Triazines; Triazoles

2012
Structural basis for allosteric regulation of GPCRs by sodium ions.
    Science (New York, N.Y.), 2012, Jul-13, Volume: 337, Issue:6091

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Allosteric Regulation; Cholesterol; Crystallography, X-Ray; Cytochrome b Group; Escherichia coli Proteins; HEK293 Cells; Humans; Hydrogen Bonding; Ligands; Lipid Bilayers; Lipids; Models, Molecular; Protein Conformation; Protein Engineering; Protein Structure, Secondary; Receptor, Adenosine A2A; Recombinant Fusion Proteins; Sodium; Triazines; Triazoles; Water

2012
Effects of ethanolic extract and naphthoquinones obtained from the bulbs of Cipura paludosa on short-term and long-term memory: involvement of adenosine A₁ and A₂A receptors.
    Basic & clinical pharmacology & toxicology, 2013, Volume: 112, Issue:4

    Topics: Animals; Avoidance Learning; Brazil; Caffeine; Ethanol; Furans; Iridaceae; Male; Memory, Long-Term; Memory, Short-Term; Mice; Naphthoquinones; Plant Extracts; Plant Roots; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A1; Receptors, Adenosine A2; Triazines; Triazoles; Xanthines

2013
Adenosine A2A receptor modulates vascular response in soluble epoxide hydrolase-null mice through CYP-epoxygenases and PPARγ.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2013, Jan-01, Volume: 304, Issue:1

    Topics: 8,11,14-Eicosatrienoic Acid; Adamantane; Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Benzamides; Benzoates; Butyrates; Enzyme Inhibitors; Epoxide Hydrolases; Female; Gene Silencing; Lauric Acids; Male; Mice; NG-Nitroarginine Methyl Ester; Oxygenases; Phenethylamines; Phenylurea Compounds; PPAR gamma; Pyridines; Pyrimidines; Receptor, Adenosine A2A; Triazines; Triazoles; Urea; Vasodilation; Vasodilator Agents

2013
Effects of oxygen and glucose deprivation on synaptic transmission in rat dentate gyrus: role of A2A adenosine receptors.
    Neuropharmacology, 2013, Volume: 67

    Topics: Animals; Cell Proliferation; Dentate Gyrus; Doublecortin Protein; Excitatory Postsynaptic Potentials; Glucose; Male; Organ Culture Techniques; Oxygen; Rats; Rats, Wistar; Receptor, Adenosine A2A; Synaptic Transmission; Triazines; Triazoles

2013
High-intensity swimming exercise reduces neuropathic pain in an animal model of complex regional pain syndrome type I: evidence for a role of the adenosinergic system.
    Neuroscience, 2013, Mar-27, Volume: 234

    Topics: Adenine; Adenosine; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Adenosine Deaminase Inhibitors; Animals; Caffeine; Exercise Therapy; Hyperalgesia; Male; Mice; Naloxone; Narcotic Antagonists; Neuralgia; Neurons; Reflex Sympathetic Dystrophy; Swimming; Triazines; Triazoles; Xanthines

2013
Crystallogenesis of adenosine A(2A) receptor-T4 lysozyme fusion protein: a practical route for the structure.
    Methods in enzymology, 2013, Volume: 520

    Topics: Adenosine A2 Receptor Antagonists; Animals; Humans; Models, Biological; Muramidase; Protein Binding; Protein Conformation; Receptor, Adenosine A2A; Receptors, G-Protein-Coupled; Recombinant Fusion Proteins; Triazines; Triazoles

2013
Adenosine 2A receptor modulates inflammation and phenotype in experimental abdominal aortic aneurysms.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2013, Volume: 27, Issue:6

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Aortic Aneurysm, Abdominal; CD4-Positive T-Lymphocytes; Cytokines; Humans; Inflammation; Male; Matrix Metalloproteinase 9; Mice; Mice, Inbred C57BL; Mice, Knockout; Pancreatic Elastase; Phenethylamines; Phenotype; Receptors, Adenosine A2; Triazines; Triazoles

2013
Adenosine transporter ENT1 regulates the acquisition of goal-directed behavior and ethanol drinking through A2A receptor in the dorsomedial striatum.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Mar-06, Volume: 33, Issue:10

    Topics: Alcohol Drinking; Analysis of Variance; Animals; beta-Galactosidase; Choice Behavior; Conditioning, Operant; Corpus Striatum; CREB-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Equilibrative Nucleoside Transporter 1; Gene Expression Regulation; Goals; Green Fluorescent Proteins; Mice; Mice, Inbred C57BL; Mice, Transgenic; Receptor, Adenosine A2A; Reinforcement Schedule; Signal Transduction; Sucrose; Sweetening Agents; Triazines; Triazoles

2013
Antagonist binding and induced conformational dynamics of GPCR A2A adenosine receptor.
    Proteins, 2013, Volume: 81, Issue:8

    Topics: Adenosine A2 Receptor Antagonists; Animals; Humans; Molecular Docking Simulation; Molecular Dynamics Simulation; Protein Conformation; Purines; Rats; Receptor, Adenosine A2A; Thermodynamics; Triazines; Triazoles

2013
A3 adenosine receptor: homology modeling and 3D-QSAR studies.
    Journal of molecular graphics & modelling, 2013, Volume: 42

    Topics: Adenosine A3 Receptor Antagonists; Amino Acid Sequence; Binding Sites; Drug Discovery; Humans; Intracellular Signaling Peptides and Proteins; Models, Molecular; Molecular Dynamics Simulation; Protein Binding; Quantitative Structure-Activity Relationship; Receptor, Adenosine A2A; Receptor, Adenosine A3; Triazines; Triazoles

2013
Novel adenosine A(2A) receptor ligands: a synthetic, functional and computational investigation of selected literature adenosine A(2A) receptor antagonists for extending into extracellular space.
    Bioorganic & medicinal chemistry letters, 2013, Jun-01, Volume: 23, Issue:11

    Topics: Adenosine A2 Receptor Antagonists; Binding Sites; Humans; Hydrogen Bonding; Ligands; Molecular Docking Simulation; Protein Binding; Protein Structure, Tertiary; Receptor, Adenosine A2A; Triazines; Triazoles

2013
Adenosine A(2A) receptors regulate the activity of sleep regulatory GABAergic neurons in the preoptic hypothalamus.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2013, Jul-01, Volume: 305, Issue:1

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; GABAergic Neurons; Hypothalamus; Infusions, Intraventricular; Male; Microinjections; Models, Animal; Phenethylamines; Preoptic Area; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Sleep; Triazines; Triazoles

2013
Functional interaction between pre-synaptic α6β2-containing nicotinic and adenosine A2A receptors in the control of dopamine release in the rat striatum.
    British journal of pharmacology, 2013, Volume: 169, Issue:7

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Corpus Striatum; Dopamine; Gene Expression Regulation; Male; Motor Skills; Nicotine; Phenethylamines; Presynaptic Terminals; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Nicotinic; Synaptosomes; Triazines; Triazoles

2013
Revisiting a receptor-based pharmacophore hypothesis for human A(2A) adenosine receptor antagonists.
    Journal of chemical information and modeling, 2013, Jul-22, Volume: 53, Issue:7

    Topics: Adenosine A2 Receptor Antagonists; Drug Design; Humans; Molecular Docking Simulation; Protein Conformation; Quantitative Structure-Activity Relationship; Receptor, Adenosine A2A; Static Electricity; Triazines; Triazoles

2013
Cannabidiol provides long-lasting protection against the deleterious effects of inflammation in a viral model of multiple sclerosis: a role for A2A receptors.
    Neurobiology of disease, 2013, Volume: 59

    Topics: Animals; Brain; Cannabidiol; Cardiovirus Infections; Cell Adhesion; Cells, Cultured; Chemokine CCL2; Chemokine CCL5; Disease Models, Animal; Endothelial Cells; Inflammation; Interleukin-1beta; Mice; Motor Activity; Multiple Sclerosis; Receptor, Adenosine A2A; Triazines; Triazoles; Vascular Cell Adhesion Molecule-1

2013
Antagonism of adenosine A2A receptor expressed by lung adenocarcinoma tumor cells and cancer associated fibroblasts inhibits their growth.
    Cancer biology & therapy, 2013, Volume: 14, Issue:9

    Topics: Adenocarcinoma; Adenocarcinoma of Lung; Adenosine A2 Receptor Antagonists; Animals; Apoptosis; Cell Line, Tumor; Cell Proliferation; Fibroblasts; Heterografts; Humans; Lung Neoplasms; Mice, Nude; Pyrimidines; Receptor, Adenosine A2A; Triazines; Triazoles

2013
Modulation of A₂a receptor antagonist on D₂ receptor internalization and ERK phosphorylation.
    Acta pharmacologica Sinica, 2013, Volume: 34, Issue:10

    Topics: Adenosine A2 Receptor Antagonists; Animals; Arrestins; beta-Arrestins; Bioluminescence Resonance Energy Transfer Techniques; Cells, Cultured; Corpus Striatum; Extracellular Signal-Regulated MAP Kinases; HEK293 Cells; Humans; Neurons; Phosphorylation; Protein Multimerization; Quinpirole; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Receptors, Dopamine D2; src-Family Kinases; Triazines; Triazoles

2013
A(2A) adenosine receptors and Parkinson's disease severity.
    Acta neurologica Scandinavica, 2014, Volume: 129, Issue:4

    Topics: Adenosine A2 Receptor Agonists; Aged; Disease Progression; Dose-Response Relationship, Drug; Dyskinesias; Female; Humans; Lymphocytes; Male; Middle Aged; Parkinson Disease; Protein Binding; Receptor, Adenosine A2A; Statistics, Nonparametric; Triazines; Triazoles; Tritium

2014
The stimulation of adenosine A2A receptors ameliorates the pathological phenotype of fibroblasts from Niemann-Pick type C patients.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Sep-25, Volume: 33, Issue:39

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Calcium; Case-Control Studies; Cell Line; Cholesterol; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electron Transport Complex IV; Extracellular Signal-Regulated MAP Kinases; Female; Fibroblasts; Humans; Lysosomes; Male; Membrane Potential, Mitochondrial; Mitochondria; Niemann-Pick Disease, Type C; Phenethylamines; Phenotype; Receptor, Adenosine A2A; Triazines; Triazoles

2013
Nucleus tractus solitarii A(2a) adenosine receptors inhibit cardiopulmonary chemoreflex control of sympathetic outputs.
    Autonomic neuroscience : basic & clinical, 2014, Volume: 180

    Topics: Adenosine; Adrenal Glands; Animals; Biguanides; Blood Pressure; Chemoreceptor Cells; Heart Atria; Heart Conduction System; Heart Rate; Hypotension; Kidney; Lumbosacral Region; Male; Microinjections; Models, Neurological; Phenethylamines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Reflex; Serotonin 5-HT3 Receptor Agonists; Solitary Nucleus; Sympathetic Nervous System; Triazines; Triazoles

2014
Paradoxical neostigmine-induced TOFfade: on the role of presynaptic cholinergic and adenosine receptors.
    European journal of pharmacology, 2014, Jan-15, Volume: 723

    Topics: Animals; Atropine; Cholinesterase Inhibitors; Diamines; Diaphragm; In Vitro Techniques; Male; Muscarinic Antagonists; Neostigmine; Phrenic Nerve; Pirenzepine; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptors, Cholinergic; Receptors, Presynaptic; Receptors, Purinergic P1; Synaptic Transmission; Triazines; Triazoles

2014
Protective mechanisms of adenosine 5'-monophosphate in platelet activation and thrombus formation.
    Thrombosis and haemostasis, 2014, Mar-03, Volume: 111, Issue:3

    Topics: Adenosine A2 Receptor Agonists; Adenosine Monophosphate; Animals; Blood Platelets; CD40 Ligand; Cells, Cultured; Crotalid Venoms; Cyclic Nucleotide Phosphodiesterases, Type 3; Disease Models, Animal; Humans; Lasers; Lectins, C-Type; Mesenteric Veins; Mice; Molecular Targeted Therapy; P-Selectin; Peptide Fragments; Photochemical Processes; Platelet Activation; Platelet Glycoprotein GPIIb-IIIa Complex; Receptor, Adenosine A2A; Rose Bengal; Stereoisomerism; Thrombosis; Triazines; Triazoles

2014
Mechanisms involved in increased sensitivity to adenosine A(2A) receptor activation and hypoxia-induced vasodilatation in porcine coronary arteries.
    European journal of pharmacology, 2014, Jan-15, Volume: 723

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Coronary Vessels; Cyclic AMP; Dinoprost; HSP20 Heat-Shock Proteins; Hypoxia; In Vitro Techniques; Oxygen; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Swine; Triazines; Triazoles; Vasodilation

2014
Reduced striatal adenosine A2A receptor levels define a molecular subgroup in schizophrenia.
    Journal of psychiatric research, 2014, Volume: 51

    Topics: Actins; Adenosine A1 Receptor Antagonists; Adult; Aged; Aged, 80 and over; Alzheimer Disease; Cell Membrane; DNA Methylation; Female; Humans; Lewy Body Disease; Male; Middle Aged; Positron-Emission Tomography; Postmortem Changes; Psychiatric Status Rating Scales; Putamen; Receptor, Adenosine A2A; Schizophrenia; Triazines; Triazoles; Tritium; Xanthines

2014
Extracellular adenosine controls NKT-cell-dependent hepatitis induction.
    European journal of immunology, 2014, Volume: 44, Issue:4

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Cells, Cultured; Concanavalin A; Flow Cytometry; Galactosylceramides; Hepatitis, Animal; Interferon-gamma; Liver; Mice; Mice, Inbred C57BL; Mice, Knockout; Natural Killer T-Cells; Phenethylamines; Receptor, Adenosine A2A; Triazines; Triazoles; Tumor Necrosis Factor-alpha

2014
NF-κB enhances hypoxia-driven T-cell immunosuppression via upregulation of adenosine A(2A) receptors.
    Cellular signalling, 2014, Volume: 26, Issue:5

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Cell Hypoxia; Cell Survival; Cells, Cultured; Cobalt; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Humans; Hypoxia-Inducible Factor 1, alpha Subunit; Immunosuppression Therapy; Isoquinolines; NF-kappa B; Receptor, Adenosine A2A; Signal Transduction; Sulfites; Sulfonamides; T-Lymphocytes; Triazines; Triazoles; Up-Regulation

2014
Binding kinetics of ZM241385 derivatives at the human adenosine A2A receptor.
    ChemMedChem, 2014, Volume: 9, Issue:4

    Topics: Adenosine A2 Receptor Antagonists; Binding Sites; Dose-Response Relationship, Drug; Humans; Kinetics; Molecular Structure; Receptor, Adenosine A2A; Structure-Activity Relationship; Triazines; Triazoles

2014
Chlorogenic acid inhibits human platelet activation and thrombus formation.
    PloS one, 2014, Volume: 9, Issue:3

    Topics: Adenine; Adenosine Triphosphate; Animals; Binding Sites; Bleeding Time; Cell Communication; Cell Line; Cell Survival; Chlorogenic Acid; Collagen; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Hemorheology; Humans; Inflammation Mediators; Leukocytes; Mice; Models, Molecular; P-Selectin; Platelet Activation; Platelet Adhesiveness; Platelet Aggregation; Platelet Glycoprotein GPIIb-IIIa Complex; Receptor, Adenosine A2A; Thrombosis; Triazines; Triazoles

2014
The plant hormone zeatin riboside inhibits T lymphocyte activity via adenosine A2A receptor activation.
    Cellular & molecular immunology, 2015, Volume: 12, Issue:1

    Topics: Animals; Antigens, CD; CD4-Positive T-Lymphocytes; CD8-Positive T-Lymphocytes; Cells, Cultured; Cyclic AMP; Cytokines; Female; Immunomodulation; Isopentenyladenosine; Leukocytosis; Mice; Mice, Inbred C57BL; Plant Growth Regulators; Receptor, Adenosine A2A; Triazines; Triazoles

2015
Histamine H3 receptor activation counteracts adenosine A2A receptor-mediated enhancement of depolarization-evoked [3H]-GABA release from rat globus pallidus synaptosomes.
    ACS chemical neuroscience, 2014, Aug-20, Volume: 5, Issue:8

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Biphenyl Compounds; gamma-Aminobutyric Acid; Globus Pallidus; Histamine Agonists; Histamine H3 Antagonists; Imidazoles; Male; Membrane Potentials; Nitriles; Phenethylamines; Piperidines; Potassium; Pyrrolidines; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Histamine H3; Synaptosomes; Thiourea; Triazines; Triazoles; Tritium

2014
Helium preconditioning protects mouse liver against ischemia and reperfusion injury through the PI3K/Akt pathway.
    Journal of hepatology, 2014, Volume: 61, Issue:5

    Topics: Adenosine A2 Receptor Antagonists; Animals; Apoptosis; Disease Models, Animal; Helium; Ischemic Preconditioning; Liver; Liver Transplantation; Male; Mice; Mice, Inbred BALB C; NF-kappa B; Phosphatidylinositol 3-Kinases; Phosphorylation; Proto-Oncogene Proteins c-akt; PTEN Phosphohydrolase; Reperfusion Injury; Signal Transduction; Transplantation Conditioning; Triazines; Triazoles; Warm Ischemia

2014
Diadenosine diphosphate (Ap₂A) delays neutrophil apoptosis via the adenosine A2A receptor and cAMP/PKA pathway.
    Biochemistry and cell biology = Biochimie et biologie cellulaire, 2014, Volume: 92, Issue:5

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine A2 Receptor Antagonists; Apoptosis; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dideoxyadenosine; Dinucleoside Phosphates; Humans; Neutrophils; Pyrazoles; Pyrimidines; Receptor, Adenosine A2A; Thionucleotides; Triazines; Triazoles

2014
Structural and energetic effects of A2A adenosine receptor mutations on agonist and antagonist binding.
    PloS one, 2014, Volume: 9, Issue:10

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Binding Sites; Humans; Ligands; Mutant Proteins; Mutation; Receptor, Adenosine A2A; Thermodynamics; Triazines; Triazoles

2014
Expression of CD73 and A2A receptors in cells from subjects with obesity and type 2 diabetes mellitus.
    Immunobiology, 2015, Volume: 220, Issue:8

    Topics: 5'-Nucleotidase; Adenosine; Adult; Antigens, CD; Apoptosis; Apyrase; Body Mass Index; CD8-Positive T-Lymphocytes; Diabetes Mellitus, Type 2; Gene Expression Regulation; GPI-Linked Proteins; Humans; Inflammation; Lymphocyte Subsets; Lymphocytes; Obesity; Phenethylamines; Receptor, Adenosine A2A; Triazines; Triazoles

2015
Alkaline phosphatase protects against renal inflammation through dephosphorylation of lipopolysaccharide and adenosine triphosphate.
    British journal of pharmacology, 2015, Volume: 172, Issue:20

    Topics: Acute Kidney Injury; Adrenergic alpha-2 Receptor Antagonists; Alkaline Phosphatase; Animals; Cells, Cultured; Cytokines; Epithelial Cells; Fluoresceins; Gene Expression Regulation; Humans; Inflammation; Kidney; Lipopolysaccharides; Male; Oligosaccharides; Protective Agents; Purines; Rats, Sprague-Dawley; Recombinant Proteins; Triazines; Triazoles

2015
Caffeine promotes anti-tumor immune response during tumor initiation: Involvement of the adenosine A2A receptor.
    Biochemical pharmacology, 2015, Nov-01, Volume: 98, Issue:1

    Topics: Adenosine A2 Receptor Antagonists; Animals; Caffeine; Cell Line, Tumor; Cyclopentanes; Fibrosarcoma; Mice; Mice, Knockout; Neoplasms, Experimental; Receptor, Adenosine A2A; Triazines; Triazoles

2015
Evaluation of the expression and function of the P2X7 receptor and ART1 in human regulatory T-cell subsets.
    Immunobiology, 2016, Volume: 221, Issue:1

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine Triphosphate; Adolescent; ADP Ribose Transferases; Adult; Antigens, CD; Apyrase; Cell Death; Cell Proliferation; Female; Gene Expression Regulation; GPI-Linked Proteins; Humans; Immunophenotyping; L-Selectin; Male; NAD; Phenethylamines; Primary Cell Culture; Receptors, Adenosine A2; Receptors, Purinergic P2X7; Signal Transduction; T-Lymphocyte Subsets; Triazines; Triazoles

2016
Adenosine A2A receptor plays an important role in radiation-induced dermal injury.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2016, Volume: 30, Issue:1

    Topics: Adenosine A2 Receptor Antagonists; Animals; Collagen; Keratinocytes; Mice; Mice, Inbred C57BL; Myofibroblasts; Radiodermatitis; Receptor, Adenosine A2A; Triazines; Triazoles

2016
Mass spectrometry-based ligand binding assays on adenosine A1 and A2A receptors.
    Purinergic signalling, 2015, Volume: 11, Issue:4

    Topics: Animals; Cell Membrane; CHO Cells; Cricetinae; Cricetulus; Deuterium; Humans; Isotope Labeling; Ligands; Mass Spectrometry; Radioligand Assay; Receptor, Adenosine A1; Receptor, Adenosine A2A; Receptors, G-Protein-Coupled; Reference Standards; Reproducibility of Results; Triazines; Triazoles; Xanthines

2015
PI3K/Akt signaling pathway is involved in the neurotrophic effect of senegenin.
    Molecular medicine reports, 2016, Volume: 13, Issue:2

    Topics: Animals; Cell Survival; Chromones; Drugs, Chinese Herbal; Humans; Morpholines; Neurites; Neurodegenerative Diseases; Neurons; Phosphatidylinositol 3-Kinases; Polygala; Primary Cell Culture; Proto-Oncogene Proteins c-akt; Rats; Signal Transduction; Triazines; Triazoles

2016
7TM X-ray structures for class C GPCRs as new drug-discovery tools. 1. mGluR5.
    Bioorganic & medicinal chemistry letters, 2016, Jan-15, Volume: 26, Issue:2

    Topics: Benzamides; Binding Sites; Crystallography, X-Ray; Drug Discovery; Indoles; Ligands; Models, Molecular; Molecular Docking Simulation; Molecular Structure; Protein Domains; Pyrazoles; Pyridines; Pyrimidines; Receptor, Metabotropic Glutamate 5; Thiazoles; Triazines; Triazoles

2016
Ligand-Independent Adenosine A2B Receptor Constitutive Activity as a Promoter of Prostate Cancer Cell Proliferation.
    The Journal of pharmacology and experimental therapeutics, 2016, Volume: 357, Issue:1

    Topics: Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine Deaminase; Animals; Cell Line, Tumor; Cell Proliferation; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Drug Design; Humans; Inositol Phosphates; Ligands; Male; MAP Kinase Signaling System; Prostatic Neoplasms; Receptor, Adenosine A2B; Signal Transduction; Sulfonamides; Triazines; Triazoles; Xanthines

2016
Molecular Basis of Ligand Dissociation from the Adenosine A2A Receptor.
    Molecular pharmacology, 2016, Volume: 89, Issue:5

    Topics: Adenosine A2 Receptor Antagonists; Amino Acid Substitution; Binding Sites; Cell Membrane; Databases, Protein; HEK293 Cells; Humans; Hydrogen Bonding; Hydrophobic and Hydrophilic Interactions; Kinetics; Ligands; Models, Molecular; Molecular Conformation; Molecular Dynamics Simulation; Mutation; Radioligand Assay; Receptor, Adenosine A2A; Recombinant Proteins; Solubility; Triazines; Triazoles

2016
The Effect of A2A Receptor Antagonist on Microglial Activation in Experimental Glaucoma.
    Investigative ophthalmology & visual science, 2016, Volume: 57, Issue:3

    Topics: Adenosine A2 Receptor Antagonists; Animals; Blotting, Western; Cell Count; Cells, Cultured; Chronic Disease; Cytokines; Disease Models, Animal; Enzyme-Linked Immunosorbent Assay; Flow Cytometry; Glaucoma; Immunohistochemistry; Intravitreal Injections; Male; Microglia; Ocular Hypertension; Rats; Rats, Sprague-Dawley; Real-Time Polymerase Chain Reaction; Retinal Ganglion Cells; RNA; Triazines; Triazoles

2016
Controlling the Dissociation of Ligands from the Adenosine A2A Receptor through Modulation of Salt Bridge Strength.
    Journal of medicinal chemistry, 2016, 07-14, Volume: 59, Issue:13

    Topics: Cells, Cultured; Crystallography, X-Ray; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Ligands; Models, Molecular; Molecular Structure; Protein Engineering; Receptor, Adenosine A2A; Structure-Activity Relationship; Triazines; Triazoles

2016
Early synaptic deficits in the APP/PS1 mouse model of Alzheimer's disease involve neuronal adenosine A2A receptors.
    Nature communications, 2016, 06-17, Volume: 7

    Topics: Adenosine A2 Receptor Antagonists; Alzheimer Disease; Amyloid beta-Protein Precursor; Animals; CA3 Region, Hippocampal; Dendritic Spines; Disease Models, Animal; Gene Expression Regulation; Humans; Long-Term Potentiation; Memory, Episodic; Mice; Mice, Transgenic; Neuroprotective Agents; Presenilin-1; Pyrimidines; Receptor, Adenosine A2A; Receptors, N-Methyl-D-Aspartate; RNA, Small Interfering; Signal Transduction; Synapses; Triazines; Triazoles

2016
Oral administration of Japanese sake yeast (Saccharomyces cerevisiae sake) promotes non-rapid eye movement sleep in mice via adenosine A
    Journal of sleep research, 2016, Volume: 25, Issue:6

    Topics: Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Administration, Oral; Alcoholic Beverages; Animals; Electroencephalography; Electromyography; Eye Movements; Japan; Locomotion; Male; Mice; Mice, Inbred C57BL; Receptor, Adenosine A2A; Saccharomyces cerevisiae; Sleep; Sleep, REM; Theophylline; Time Factors; Triazines; Triazoles

2016
An Fc-Small Molecule Conjugate for Targeted Inhibition of the Adenosine 2A Receptor.
    Chembiochem : a European journal of chemical biology, 2016, 10-17, Volume: 17, Issue:20

    Topics: Adenosine A2 Receptor Antagonists; Animals; Female; Humans; Immunoglobulin Fab Fragments; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Models, Molecular; Molecular Structure; Receptor, Adenosine A2A; Respiratory Tract Infections; Triazines; Triazoles; Vaccinia virus

2016
Equilibrative nucleoside transporter ENT1 as a biomarker of Huntington disease.
    Neurobiology of disease, 2016, Volume: 96

    Topics: Adenosine; Adenosine A2 Receptor Antagonists; Animals; Biomarkers; Corpus Striatum; Disease Models, Animal; Gene Expression Regulation; Humans; Huntingtin Protein; Huntington Disease; Locomotion; Nucleoside Transport Proteins; Prefrontal Cortex; Psychomotor Disorders; Purines; Rats; Rats, Transgenic; Receptor, Adenosine A2A; Triazines; Triazoles; Trinucleotide Repeat Expansion; Tritium

2016
Inosine attenuates spontaneous activity in the rat neurogenic bladder through an A
    Scientific reports, 2017, 03-15, Volume: 7

    Topics: Adenosine A2 Receptor Antagonists; Animals; Disease Models, Animal; Humans; Inosine; Potassium Channels; Rats; Receptor, Adenosine A2A; Spinal Cord Injuries; Sulfonamides; Triazines; Triazoles; Urinary Bladder, Neurogenic; Urinary Bladder, Overactive; Xanthines

2017
Adenosine A
    Translational psychiatry, 2017, 05-09, Volume: 7, Issue:5

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adult; Aged; Animals; Brain Injuries, Traumatic; Cognitive Dysfunction; Disease Models, Animal; Female; Glycogen Synthase Kinase 3 beta; Glycogen Synthase Kinases; Hippocampus; Humans; Indoles; Isoquinolines; Male; Maleimides; Mice; Mice, Knockout; Middle Aged; Neurons; Phenethylamines; Phosphorylation; Protein Kinase Inhibitors; Receptor, Adenosine A2A; Signal Transduction; Sulfonamides; tau Proteins; Triazines; Triazoles

2017
Preemptive Caffeine Administration Blocks the Increase in Postoperative Pain Caused by Previous Sleep Loss in the Rat: A Potential Role for Preoptic Adenosine A2A Receptors in Sleep-Pain Interactions.
    Sleep, 2017, 09-01, Volume: 40, Issue:9

    Topics: Adenosine A2 Receptor Antagonists; Animals; Caffeine; Female; Hyperalgesia; Male; Pain, Postoperative; Preoptic Area; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Sex Characteristics; Sleep; Sleep Deprivation; Triazines; Triazoles

2017
Impaired autophagic flux is associated with the severity of trauma and the role of A
    Cell death & disease, 2018, 02-14, Volume: 9, Issue:2

    Topics: Adenosine A2 Receptor Antagonists; Animals; Autophagosomes; Autophagy; Autophagy-Related Protein 12; Autophagy-Related Protein 5; Beclin-1; Brain Injuries, Traumatic; Cerebral Cortex; Chloroquine; Disease Models, Animal; Female; Gene Expression Regulation; Humans; Mice; Mice, Inbred C57BL; Mice, Knockout; Microtubule-Associated Proteins; Neurons; Neuroprotective Agents; Receptor, Adenosine A2A; Sequestosome-1 Protein; Signal Transduction; Trauma Severity Indices; Triazines; Triazoles

2018
Mechanistic insights into allosteric regulation of the A
    Nature communications, 2018, 04-10, Volume: 9, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Allosteric Regulation; Amino Acid Sequence; Animals; Binding Sites; Calcium; Cations, Divalent; Crystallography, X-Ray; Gene Expression; Humans; Kinetics; Magnesium; Models, Molecular; Molecular Dynamics Simulation; Protein Binding; Protein Conformation, alpha-Helical; Protein Conformation, beta-Strand; Protein Interaction Domains and Motifs; Receptor, Adenosine A2A; Recombinant Proteins; Sf9 Cells; Spodoptera; Thermodynamics; Triazines; Triazoles

2018
Effects of caffeine and phosphodiesterase inhibitors on activation of neonatal T lymphocytes.
    Immunobiology, 2018, Volume: 223, Issue:11

    Topics: Adenosine A2 Receptor Antagonists; Adult; Aging; Caffeine; Calcium Signaling; Cells, Cultured; Cyclic AMP; Cytokines; Female; Humans; Infant, Newborn; Leukocytes, Mononuclear; Lymphocyte Activation; Male; Milrinone; Phosphodiesterase Inhibitors; Reactive Oxygen Species; Sildenafil Citrate; T-Lymphocytes; Triazines; Triazoles

2018
Cervical cancer cells produce TGF-β1 through the CD73-adenosine pathway and maintain CD73 expression through the autocrine activity of TGF-β1.
    Cytokine, 2019, Volume: 118

    Topics: 5'-Nucleotidase; Acetamides; Adenosine; Adenosine A2 Receptor Antagonists; Autocrine Communication; Cell Line, Tumor; Female; GPI-Linked Proteins; HeLa Cells; Humans; Immunosuppression Therapy; Purines; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Transforming Growth Factor beta1; Triazines; Triazoles; Tumor Microenvironment; Uterine Cervical Neoplasms

2019
Ischemia postconditioning protects dermal microvascular endothelial cells of rabbit epigastric skin flaps against apoptosis via adenosine A2a receptors.
    Journal of plastic surgery and hand surgery, 2019, Volume: 53, Issue:2

    Topics: Abdomen; Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Apoptosis; Dermis; Endothelial Cells; Ischemic Postconditioning; Models, Animal; Phenethylamines; Rabbits; Surgical Flaps; Triazines; Triazoles

2019
Impact of combination immunochemotherapies on progression of 4NQO-induced murine oral squamous cell carcinoma.
    Cancer immunology, immunotherapy : CII, 2019, Volume: 68, Issue:7

    Topics: 4-Nitroquinoline-1-oxide; Animals; Antineoplastic Combined Chemotherapy Protocols; Cancer Vaccines; Cisplatin; Combined Modality Therapy; Female; Immunotherapy; Mice; Mice, Inbred C57BL; Mouth Neoplasms; Neoplasms, Experimental; Squamous Cell Carcinoma of Head and Neck; Treatment Outcome; Triazines; Triazoles; Vaccines, Subunit

2019
Number of Circulating CD 73-Expressing Lymphocytes Correlates With Survival After Cardiac Arrest.
    Journal of the American Heart Association, 2019, 07-02, Volume: 8, Issue:13

    Topics: 5'-Nucleotidase; Adenosine A2 Receptor Antagonists; Adenosine Diphosphate; Adenosine Monophosphate; Aged; Antigens, CD; Apyrase; Cardiopulmonary Resuscitation; Case-Control Studies; Enzyme Inhibitors; Female; Heart Arrest; Humans; In Vitro Techniques; Leukocyte Count; Lymphocytes; Male; Middle Aged; Myeloid Cells; Prognosis; Reactive Oxygen Species; Triazines; Triazoles; Tumor Necrosis Factor-alpha; Vascular Endothelial Growth Factor A

2019
Contribution of adenosine and ATP to the carotid body chemosensory activity in ageing.
    The Journal of physiology, 2019, Volume: 597, Issue:19

    Topics: Adenosine; Adenosine Triphosphate; Aging; Animals; Antinematodal Agents; Carotid Body; Chemoreceptor Cells; Female; Gene Expression Regulation; Male; Rats; Rats, Wistar; Suramin; Triazines; Triazoles

2019
Ligand-Dependent Sodium Ion Dynamics within the A
    The journal of physical chemistry. B, 2019, 09-26, Volume: 123, Issue:38

    Topics: Binding Sites; Humans; Ions; Ligands; Molecular Dynamics Simulation; Receptor, Adenosine A2A; Sodium; Triazines; Triazoles

2019
Ligand-induced conformational changes in a SMALP-encapsulated GPCR.
    Biochimica et biophysica acta. Biomembranes, 2020, 06-01, Volume: 1862, Issue:6

    Topics: Hydrophobic and Hydrophilic Interactions; Ligands; Lipids; Maleates; Pichia; Protein Conformation; Receptor, Adenosine A2A; Spectrometry, Fluorescence; Styrene; Triazines; Triazoles; Tryptophan

2020
In Vitro, In Silico, and In Vivo Assessments of Pharmacokinetic Properties of ZM241385.
    Molecules (Basel, Switzerland), 2020, Mar-02, Volume: 25, Issue:5

    Topics: Adenosine A2 Receptor Antagonists; Animals; Computer Simulation; Male; Parkinson Disease; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Triazines; Triazoles

2020
Adenosine Receptors as Neuroinflammation Modulators: Role of A
    Cells, 2020, 07-21, Volume: 9, Issue:7

    Topics: Adenosine; Adenosine A1 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Cells, Cultured; Inflammation; Male; Neuroglia; Neurons; Rats, Wistar; Receptors, Purinergic P1; Triazines; Triazoles

2020
Suppression of adenosine A
    Biochemical pharmacology, 2021, Volume: 183

    Topics: Adenosine A2 Receptor Antagonists; Animals; Antineoplastic Agents, Alkylating; Cyclophosphamide; Cystitis; Female; Hyperalgesia; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Triazines; Triazoles; TRPV Cation Channels; Urinary Bladder; Urinary Bladder, Overactive

2021
Ligand-directed covalent labelling of a GPCR with a fluorescent tag in live cells.
    Communications biology, 2020, 11-27, Volume: 3, Issue:1

    Topics: Affinity Labels; Drug Design; Fluorescent Dyes; HEK293 Cells; Humans; Ligands; Receptor, Adenosine A2A; Receptors, G-Protein-Coupled; Triazines; Triazoles

2020