triazoles has been researched along with vx680 in 2 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 2 (100.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Barr, AJ; Elkins, JM; Knapp, S; Salah, E; Ugochukwu, E; von Delft, F | 1 |
Bossemeyer, D; de Oliveira, TM; Engh, RA; Pflug, A | 1 |
2 other study(ies) available for triazoles and vx680
Article | Year |
---|---|
Crystal structures of ABL-related gene (ABL2) in complex with imatinib, tozasertib (VX-680), and a type I inhibitor of the triazole carbothioamide class.
Topics: Amino Acid Motifs; Benzamides; Crystallography, X-Ray; Humans; Imatinib Mesylate; Models, Molecular; Piperazines; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Protein-Tyrosine Kinases; Pyrimidines; Triazoles | 2011 |
Mutants of protein kinase A that mimic the ATP-binding site of Aurora kinase.
Topics: Adenosine Triphosphate; Amino Acid Sequence; Amino Acid Substitution; Aurora Kinases; Binding Sites; Crystallography, X-Ray; Cyclic AMP-Dependent Protein Kinases; Cyclin-Dependent Kinases; Enzyme Inhibitors; Humans; Kinetics; Molecular Sequence Data; Piperazines; Protein Serine-Threonine Kinases; Recombinant Fusion Proteins; Sequence Alignment; Triazoles | 2011 |