Page last updated: 2024-08-24

triazoles and vx680

triazoles has been researched along with vx680 in 2 studies

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Barr, AJ; Elkins, JM; Knapp, S; Salah, E; Ugochukwu, E; von Delft, F1
Bossemeyer, D; de Oliveira, TM; Engh, RA; Pflug, A1

Other Studies

2 other study(ies) available for triazoles and vx680

ArticleYear
Crystal structures of ABL-related gene (ABL2) in complex with imatinib, tozasertib (VX-680), and a type I inhibitor of the triazole carbothioamide class.
    Journal of medicinal chemistry, 2011, Apr-14, Volume: 54, Issue:7

    Topics: Amino Acid Motifs; Benzamides; Crystallography, X-Ray; Humans; Imatinib Mesylate; Models, Molecular; Piperazines; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Protein-Tyrosine Kinases; Pyrimidines; Triazoles

2011
Mutants of protein kinase A that mimic the ATP-binding site of Aurora kinase.
    The Biochemical journal, 2011, Nov-15, Volume: 440, Issue:1

    Topics: Adenosine Triphosphate; Amino Acid Sequence; Amino Acid Substitution; Aurora Kinases; Binding Sites; Crystallography, X-Ray; Cyclic AMP-Dependent Protein Kinases; Cyclin-Dependent Kinases; Enzyme Inhibitors; Humans; Kinetics; Molecular Sequence Data; Piperazines; Protein Serine-Threonine Kinases; Recombinant Fusion Proteins; Sequence Alignment; Triazoles

2011