Page last updated: 2024-08-24

triazoles and vx680

triazoles has been researched along with vx680 in 2 studies

Research

Studies (2)

Timeframe	Studies, this research(%)	All Research%
pre-1990	0 (0.00)	18.7374
1990's	0 (0.00)	18.2507
2000's	0 (0.00)	29.6817
2010's	2 (100.00)	24.3611
2020's	0 (0.00)	2.80

Authors

Authors	Studies
Barr, AJ; Elkins, JM; Knapp, S; Salah, E; Ugochukwu, E; von Delft, F	1
Bossemeyer, D; de Oliveira, TM; Engh, RA; Pflug, A	1

Other Studies

2 other study(ies) available for triazoles and vx680

Article	Year
Crystal structures of ABL-related gene (ABL2) in complex with imatinib, tozasertib (VX-680), and a type I inhibitor of the triazole carbothioamide class. Journal of medicinal chemistry, 2011, Apr-14, Volume: 54, Issue:7 Topics: Amino Acid Motifs; Benzamides; Crystallography, X-Ray; Humans; Imatinib Mesylate; Models, Molecular; Piperazines; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Protein-Tyrosine Kinases; Pyrimidines; Triazoles	2011
Mutants of protein kinase A that mimic the ATP-binding site of Aurora kinase. The Biochemical journal, 2011, Nov-15, Volume: 440, Issue:1 Topics: Adenosine Triphosphate; Amino Acid Sequence; Amino Acid Substitution; Aurora Kinases; Binding Sites; Crystallography, X-Ray; Cyclic AMP-Dependent Protein Kinases; Cyclin-Dependent Kinases; Enzyme Inhibitors; Humans; Kinetics; Molecular Sequence Data; Piperazines; Protein Serine-Threonine Kinases; Recombinant Fusion Proteins; Sequence Alignment; Triazoles	2011

Article

Year

Crystal structures of ABL-related gene (ABL2) in complex with imatinib, tozasertib (VX-680), and a type I inhibitor of the triazole carbothioamide class.

Journal of medicinal chemistry, 2011, Apr-14, Volume: 54, Issue:7

Topics: Amino Acid Motifs; Benzamides; Crystallography, X-Ray; Humans; Imatinib Mesylate; Models, Molecular; Piperazines; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; Protein-Tyrosine Kinases; Pyrimidines; Triazoles

2011

Mutants of protein kinase A that mimic the ATP-binding site of Aurora kinase.

The Biochemical journal, 2011, Nov-15, Volume: 440, Issue:1

Topics: Adenosine Triphosphate; Amino Acid Sequence; Amino Acid Substitution; Aurora Kinases; Binding Sites; Crystallography, X-Ray; Cyclic AMP-Dependent Protein Kinases; Cyclin-Dependent Kinases; Enzyme Inhibitors; Humans; Kinetics; Molecular Sequence Data; Piperazines; Protein Serine-Threonine Kinases; Recombinant Fusion Proteins; Sequence Alignment; Triazoles

2011