Page last updated: 2024-08-24

triazoles and thiourea

triazoles has been researched along with thiourea in 41 studies

Research

Studies (41)

TimeframeStudies, this research(%)All Research%
pre-19909 (21.95)18.7374
1990's1 (2.44)18.2507
2000's10 (24.39)29.6817
2010's18 (43.90)24.3611
2020's3 (7.32)2.80

Authors

AuthorsStudies
Gibel, W; Schramm, T; Schwabe, K1
McNeill, JH; Verma, SC2
Matthey, K; Olthoff, U2
Jirousek, L; Soodak, M1
Blank, B; Nichols, DM; Vaidya, PD1
Aschbacher, PW; Feil, VJ; Zaylskie, RG1
Praphulla, HB; Puttaswamy, TL; Ramanathan, S; Rao, KV; Rao, PL1
Ahgren, C; Backro, K; Bell, FW; Cantrell, AS; Clemens, M; Colacino, JM; Deeter, JB; Engelhardt, JA; Hogberg, M; Jaskunas, SR1
Balzarini, J; Bird, LE; Diprose, J; Esnouf, RM; Ikemizu, S; Milton, J; Ren, J; Slater, M; Stammers, DK; Stuart, DI; Warren, J1
Kiraz, M; Küçükgüzel, I; Küçükgüzel, SG; Rollas, S1
Chen, C; Dagnino, R; Grigoriadis, DE; Huang, CQ; McCarthy, JR1
Katritzky, AR; Ledoux, S; Nair, SK; Witek, RM1
Benito, JJ; Criado, JJ; Hermosa, R; Manzano, JL; Monte, E; Rodríguez-Fernández, E1
Agrawal, RK; Ravichandran, V1
De Clercq, E; Küçükgüzel, I; Küçükgüzel, SG; Rollas, S; Tatar, E1
Akhtar, T; Choudhary, MI; Hameed, S; Khan, KM1
Chattopadhyaya, J; Dixit, SS; Kulkarni, GM; Sharma, V; Upadhayaya, RS; Vandavasi, JK; Vasireddy, NR1
Alberola, A; Cánoves, J; Chorro, FJ; Cinca, J; Hove-Madsen, L; Mainar, L; Pelechano, F; Such, L; Such-Miquel, L; Tormos, A; Trapero, I1
Liu, CJ; Wang, JD1
Azuma, T; Enkhtaivan, I; Takasu, K; Takemoto, Y1
Alcázar, J; Carrillo, JR; de Cózar, A; de la Hoz, A; Díaz-Ortiz, A; Fontana, A; Herrero, MA; Muñoz, Jde M; Prieto, P1
Güzeldemirci, NU; Küçükbasmacı, O; Satana, D1
Ali, A; Celen, AO; Khan, IA; Khan, SI; Kocyigit-Kaymakcioglu, B; Tabanca, N; Wedge, DE1
Completo, G; Damoiseaux, R; Du, L; Fike, F; Gatti, RA; Hu, H; Jung, ME; Ku, JM; Nahas, S; Piao, C1
Lavin, MF1
Arias-Montaño, JA; Escamilla-Sánchez, J; González-Pantoja, R; Márquez-Gómez, R; Morales-Figueroa, GE1
Ache, B; Bobkov, Y; Corey, E1
Arya, DP; Garneau-Tsodikova, S; Green, KD; Kumar, S; Watkins, D1
Dinnebier, RE; Friščić, T; Gracin, D; Magdysyuk, OV; Štrukil, V1
Bielenica, A; Iuliano, F; Jozwiak, M; Koziol, AE; Madeddu, S; Miroslaw, B; Sanna, G; Stefanska, J; Stepien, K; Struga, M; Szulczyk, D1
Camodeca, C; Carbotti, G; Ciccone, L; Cuffaro, D; D'Andrea, F; Dive, V; Fabbi, M; Ferrini, S; Nencetti, S; Nuti, E; Orlandini, E; Rosalia, L; Rossello, A; Santamaria, S; Stura, EA; Tepshi, L1
Collu, D; Iuliano, F; Jóźwiak, M; Kozioł, AE; Lis, T; Struga, M; Szulczyk, D; Tomaszewski, P1
Armstrong, A; De, W; Lin, JZ; Wang, ZJ; Wu, HF; Xu, WZ; Zheng, M; Zhu, JG1
Geng, PF; Guo, WG; Li, ZH; Liu, HM; Liu, XQ; Yu, B; Zhao, TQ1
Bale, S; Godugu, C; Janrao, IP; Kumar, NP; Senwar, KR; Shankaraiah, N; Tokala, R; Vennela, A1
Bogolyubsky, AV; Brovarets, VS; Doroshchuk, RO; Grishchenko, AV; Khomenko, DN; Konovets, AI; Moroz, YS; Pipko, SE; Savych, O; Vybornyi, M; Zhemera, AV1
Amanlou, M; Asadi, M; Asgari, MS; Azizian, H; Biglar, M; Larijani, B; Mahdavi, M; Mohammadi-Khanaposhtani, M; Nazari Montazer, M; Rahimi, R; Ranjbar, PR; Sepehri, S1
Balewski, Ł; Bednarski, PJ; Gdaniec, M; Kornicka, A; Nadworska, A; Sączewski, F; Wolff, L1
Denel-Bobrowska, M; Gaida, R; Iwan, D; Olejniczak, AB; Steppeler, F; Wojaczyńska, E1

Reviews

2 review(s) available for triazoles and thiourea

ArticleYear
[Recommendations for testing and evaluation of drugs as to carcinogenicity].
    Archiv fur Geschwulstforschung, 1971, Volume: 37, Issue:1

    Topics: Acridines; Alcohols; Alkylating Agents; Animals; Antithyroid Agents; Azo Compounds; Carbazoles; Carcinogens; Coal Tar; Dextrans; Estrogens; Immunosuppressive Agents; Iron; Lactones; Methylthiouracil; Naphthoquinones; Paraffin; Phenylbutazone; Reserpine; Sulfhydryl Compounds; Sulfonamides; Sulfonic Acids; Tannins; Thiourea; Toxicology; Triazoles; Urethane; World Health Organization

1971
Thiourea, triazole and thiadiazine compounds and their metal complexes as antifungal agents.
    Journal of inorganic biochemistry, 2005, Volume: 99, Issue:8

    Topics: Anti-Bacterial Agents; Antifungal Agents; Metals, Heavy; Thiadiazines; Thiourea; Triazoles

2005

Other Studies

39 other study(ies) available for triazoles and thiourea

ArticleYear
Blockade by burimamide of the effects of histamine and histamine analogs on cardiac contractility, phosphorylase activation and cyclic adenosine monophosphate.
    The Journal of pharmacology and experimental therapeutics, 1974, Volume: 188, Issue:1

    Topics: Adenylyl Cyclases; Animals; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Ethylamines; Guinea Pigs; Heart; Heparin; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Myocardium; Norepinephrine; Phosphorylases; Propranolol; Pyrazoles; Stimulation, Chemical; Theophylline; Thiourea; Time Factors; Triazoles

1974
Blockade by burimamide of the effects of histamine and histamine analogues on cardiac adenylate cyclase.
    The Journal of pharmacy and pharmacology, 1974, Volume: 26, Issue:5

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Guinea Pigs; Histamine; Histamine H1 Antagonists; Imidazoles; In Vitro Techniques; Myocardium; Pyrazoles; Thiourea; Triazoles

1974
[Stability of methallibure. 2. UV-spectrophotometric procedure for quantitative determination of methallibure derivatives related to methallibure].
    Die Pharmazie, 1974, Volume: 29, Issue:12

    Topics: Drug Stability; Hydrazines; Methallibure; Spectrophotometry, Ultraviolet; Sulfhydryl Compounds; Thiourea; Triazoles

1974
The reaction of N-iodosuccinimide with the goitrogens: a model for the active iodine of the thyroid gland.
    Proceedings of the National Academy of Sciences of the United States of America, 1973, Volume: 70, Issue:5

    Topics: Aminobenzoates; Aminosalicylic Acids; Antithyroid Agents; Barbiturates; Chemical Phenomena; Chemistry; Cysteine; Dimethyl Sulfoxide; Iodine; Mercaptoethanol; Methods; Models, Chemical; Nitrogen; Resorcinols; Salicylates; Spectrophotometry; Sulfadiazine; Sulfanilamides; Thiourea; Thyroid Gland; Triazoles; Uracil; Urea

1973
[Studies on stability of metallibure. 1. Structural delineation of the degradation products of metallibure].
    Die Pharmazie, 1974, Volume: 29, Issue:1

    Topics: Alkanes; Allyl Compounds; Buffers; Chemical Phenomena; Chemistry; Chromatography, Thin Layer; Drug Stability; Gonadotropins; Hydrazines; Hydrochloric Acid; Isomerism; Sodium Hydroxide; Spectrophotometry, Infrared; Thiadiazoles; Thiourea; Triazoles

1974
Synthesis of 1,2,4-triazoles as potential hypoglycemic agents.
    Journal of medicinal chemistry, 1972, Volume: 15, Issue:6

    Topics: Hypoglycemic Agents; Thiourea; Triazoles

1972
Metabolism of 1-( -methylallylthiocarbamoyl)-2-methylthiocarbamoylhydrazine (methallibure) in cattle.
    Journal of animal science, 1972, Volume: 35, Issue:1

    Topics: Allyl Compounds; Animals; Carbon Isotopes; Cattle; Chromatography, Gel; Chromatography, Paper; Feces; Female; Hydrazines; Mass Spectrometry; Methods; Milk; Thiadiazoles; Thiourea; Triazoles

1972
Structure and antiviral activity of substituted potassium benzylaminothiomethane-sulphonates and allied compounds.
    British journal of pharmacology and chemotherapy, 1967, Volume: 31, Issue:1

    Topics: Animals; Antiviral Agents; Chemical Phenomena; Chemistry; Mice; Orthomyxoviridae; Rabbits; Sulfonic Acids; Thiocyanates; Thiosemicarbazones; Thiourea; Triazoles; Vaccinia virus

1967
The PETT series, a new class of potent nonnucleoside inhibitors of human immunodeficiency virus type 1 reverse transcriptase.
    Antimicrobial agents and chemotherapy, 1995, Volume: 39, Issue:6

    Topics: Animals; Antiviral Agents; Base Sequence; Benzodiazepines; Brain; Cattle; Cells, Cultured; DNA-Directed DNA Polymerase; Drug Resistance, Microbial; HIV-1; Humans; Imidazoles; Intercalating Agents; Male; Molecular Sequence Data; Pyridines; Rats; Rats, Inbred F344; Reverse Transcriptase Inhibitors; Structure-Activity Relationship; Thiazoles; Thiourea; Triazoles

1995
Phenylethylthiazolylthiourea (PETT) non-nucleoside inhibitors of HIV-1 and HIV-2 reverse transcriptases. Structural and biochemical analyses.
    The Journal of biological chemistry, 2000, Feb-25, Volume: 275, Issue:8

    Topics: Binding, Competitive; Crystallography, X-Ray; Deoxyguanine Nucleotides; DNA Primers; Dose-Response Relationship, Drug; HIV Reverse Transcriptase; Inhibitory Concentration 50; Intercalating Agents; Kinetics; Models, Chemical; Models, Molecular; Protein Binding; Pyridines; Regression Analysis; Reverse Transcriptase Inhibitors; RNA-Directed DNA Polymerase; Thiazoles; Thiourea; Triazoles

2000
Some 3-thioxo/alkylthio-1,2,4-triazoles with a substituted thiourea moiety as possible antimycobacterials.
    Bioorganic & medicinal chemistry letters, 2001, Jul-09, Volume: 11, Issue:13

    Topics: Animals; Antitubercular Agents; Chlorocebus aethiops; Microbial Sensitivity Tests; Mycobacterium fortuitum; Mycobacterium tuberculosis; Thiourea; Triazoles; Vero Cells

2001
1-Alkyl-3-amino-5-aryl-1H-[1,2,4]triazoles: novel synthesis via cyclization of N-acyl-S-methylisothioureas with alkylhydrazines and their potent corticotropin-releasing factor-1 (CRF(1)) receptor antagonist activities.
    Bioorganic & medicinal chemistry letters, 2001, Dec-17, Volume: 11, Issue:24

    Topics: Humans; Hydrazines; Magnetic Resonance Spectroscopy; Receptors, Corticotropin-Releasing Hormone; Thiourea; Triazoles

2001
1-(Alkyl/arylthiocarbamoyl)benzotriazoles as stable isothiocyanate equivalents: synthesis of Di- and trisubstituted thioureas.
    The Journal of organic chemistry, 2004, Apr-30, Volume: 69, Issue:9

    Topics: Isothiocyanates; Molecular Structure; Tetrazoles; Thiocarbamates; Thiourea; Triazoles

2004
Predicting anti-HIV activity of PETT derivatives: CoMFA approach.
    Bioorganic & medicinal chemistry letters, 2007, Apr-15, Volume: 17, Issue:8

    Topics: Anti-HIV Agents; Computational Biology; Drug Design; Humans; Models, Molecular; Quantitative Structure-Activity Relationship; Reverse Transcriptase Inhibitors; Static Electricity; Thiazoles; Thiourea; Triazoles

2007
Synthesis of some novel thiourea derivatives obtained from 5-[(4-aminophenoxy)methyl]-4-alkyl/aryl-2,4-dihydro-3H-1,2,4-triazole-3-thiones and evaluation as antiviral/anti-HIV and anti-tuberculosis agents.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:2

    Topics: Animals; Antitubercular Agents; Antiviral Agents; Cell Line; Drug Evaluation, Preclinical; Humans; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Thiourea; Triazoles

2008
Syntheses, urease inhibition, and antimicrobial studies of some chiral 3-substituted-4-amino-5-thioxo-1H,4H-1,2,4-triazoles.
    Medicinal chemistry (Shariqah (United Arab Emirates)), 2008, Volume: 4, Issue:6

    Topics: Anti-Infective Agents; Bacteria; Cyclization; Enzyme Inhibitors; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Spectrophotometry, Infrared; Spectrophotometry, Ultraviolet; Structure-Activity Relationship; Thiourea; Triazoles; Urease

2008
Design, synthesis and biological evaluation of novel triazole, urea and thiourea derivatives of quinoline against Mycobacterium tuberculosis.
    Bioorganic & medicinal chemistry, 2009, Jul-01, Volume: 17, Issue:13

    Topics: Animals; Antitubercular Agents; ATP Synthetase Complexes; Bacterial Proteins; Cell Survival; Macrophages; Models, Molecular; Molecular Structure; Murinae; Mycobacterium tuberculosis; Protein Binding; Quinolines; Structure-Activity Relationship; Thiourea; Triazoles; Tuberculosis; Urea

2009
Pharmacological modifications of the stretch-induced effects on ventricular fibrillation in perfused rabbit hearts.
    American journal of physiology. Heart and circulatory physiology, 2009, Volume: 297, Issue:5

    Topics: Action Potentials; Adenosine A2 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Anti-Arrhythmia Agents; Calcium Signaling; Disease Models, Animal; Electrophysiologic Techniques, Cardiac; Fourier Analysis; Heart Conduction System; In Vitro Techniques; Muscle Spindles; Myocardium; Perfusion; Propranolol; Pyrimidines; Rabbits; Receptors, Adenosine A2; Sodium-Calcium Exchanger; Thiourea; Time Factors; Triazoles; Ventricular Fibrillation

2009
Ultrasound-assisted synthesis of novel 4-(2-phenyl-1,2,3-triazol-4-yl)-3,4-dihydropyrimidin-(1H)-(thio)ones catalyzed by Sm(ClO(4))(3).
    Molecules (Basel, Switzerland), 2010, Mar-24, Volume: 15, Issue:4

    Topics: Anti-Bacterial Agents; Anti-Inflammatory Agents, Non-Steroidal; Antineoplastic Agents; Antiviral Agents; Catalysis; Perchlorates; Pyrimidinones; Samarium; Thiourea; Triazoles; Ultrasonics; Urea

2010
Synthesis and properties of chiral thioureas bearing an additional function at a remote position tethered by a 1,5-disubstituted triazole.
    Molecules (Basel, Switzerland), 2010, Nov-15, Volume: 15, Issue:11

    Topics: Molecular Structure; Stereoisomerism; Thiourea; Triazoles

2010
Influence of polarity on the scalability and reproducibility of solvent-free microwave-assisted reactions.
    Combinatorial chemistry & high throughput screening, 2011, Volume: 14, Issue:2

    Topics: Alkylation; Aniline Compounds; Bromides; Chemistry, Organic; Combinatorial Chemistry Techniques; Microwaves; Oxidation-Reduction; Pyridines; Reproducibility of Results; Temperature; Thiourea; Triazoles; Urea

2011
Synthesis, characterization, and antimicrobial evaluation of some new hydrazinecarbothioamide, 1,2,4-triazole and 1,3,4-thiadiazole derivatives.
    Journal of enzyme inhibition and medicinal chemistry, 2013, Volume: 28, Issue:5

    Topics: Anti-Bacterial Agents; Antifungal Agents; Bacteria; Dose-Response Relationship, Drug; Fungi; Hydrazines; Microbial Sensitivity Tests; Molecular Structure; Structure-Activity Relationship; Thiadiazoles; Thiourea; Triazoles

2013
Synthesis and biological activity of substituted urea and thiourea derivatives containing 1,2,4-triazole moieties.
    Molecules (Basel, Switzerland), 2013, Mar-19, Volume: 18, Issue:3

    Topics: Animals; Anopheles; Botrytis; Fungicides, Industrial; Fusarium; Humans; Insect Repellents; Insecticides; Larva; Lethal Dose 50; Microbial Sensitivity Tests; Plant Diseases; Thiourea; Triazoles; Urea

2013
A new series of small molecular weight compounds induce read through of all three types of nonsense mutations in the ATM gene.
    Molecular therapy : the journal of the American Society of Gene Therapy, 2013, Volume: 21, Issue:9

    Topics: Acetanilides; Ataxia Telangiectasia; Ataxia Telangiectasia Mutated Proteins; Benzodioxoles; Cells, Cultured; Codon, Nonsense; Codon, Terminator; DNA-Binding Proteins; High-Throughput Screening Assays; Humans; Molecular Targeted Therapy; Molecular Weight; Small Molecule Libraries; Structure-Activity Relationship; Thiourea; Triazoles

2013
Generating SM(a)RTer compounds for translation termination suppression in A-T and other genetic disorders.
    Molecular therapy : the journal of the American Society of Gene Therapy, 2013, Volume: 21, Issue:9

    Topics: Acetanilides; Ataxia Telangiectasia; Ataxia Telangiectasia Mutated Proteins; Benzodioxoles; Codon, Nonsense; Codon, Terminator; Humans; Thiourea; Triazoles

2013
Histamine H3 receptor activation counteracts adenosine A2A receptor-mediated enhancement of depolarization-evoked [3H]-GABA release from rat globus pallidus synaptosomes.
    ACS chemical neuroscience, 2014, Aug-20, Volume: 5, Issue:8

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Animals; Biphenyl Compounds; gamma-Aminobutyric Acid; Globus Pallidus; Histamine Agonists; Histamine H3 Antagonists; Imidazoles; Male; Membrane Potentials; Nitriles; Phenethylamines; Piperidines; Potassium; Pyrrolidines; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Histamine H3; Synaptosomes; Thiourea; Triazines; Triazoles; Tritium

2014
An inhibitor of Na(+)/Ca(2+) exchange blocks activation of insect olfactory receptors.
    Biochemical and biophysical research communications, 2014, Jul-25, Volume: 450, Issue:2

    Topics: Animals; Anopheles; HEK293 Cells; Humans; Insect Proteins; Ion Channel Gating; Protein Multimerization; Receptors, Odorant; Sodium-Calcium Exchanger; Thioglycolates; Thiourea; Triazoles

2014
Influence of linker length and composition on enzymatic activity and ribosomal binding of neomycin dimers.
    Antimicrobial agents and chemotherapy, 2015, Volume: 59, Issue:7

    Topics: Anti-Bacterial Agents; Bacteria; Binding Sites; Binding, Competitive; Dimerization; Humans; Microbial Sensitivity Tests; Neomycin; Protein Conformation; Ribosomes; RNA, Ribosomal; Structure-Activity Relationship; Thiourea; Triazoles; Urea

2015
Trapping Reactive Intermediates by Mechanochemistry: Elusive Aryl N-Thiocarbamoylbenzotriazoles as Bench-Stable Reagents.
    Angewandte Chemie (International ed. in English), 2015, Jul-13, Volume: 54, Issue:29

    Topics: Crystallography, X-Ray; Indicators and Reagents; Isothiocyanates; Models, Molecular; Spectrum Analysis, Raman; Thiourea; Triazoles

2015
Antimicrobial and Anti-biofilm Activity of Thiourea Derivatives Bearing 3-amino-1H-1,2,4-triazole Scaffold.
    Medicinal chemistry (Shariqah (United Arab Emirates)), 2016, Volume: 12, Issue:5

    Topics: Anti-Bacterial Agents; Biofilms; Methicillin Resistance; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Staphylococcus epidermidis; Thioamides; Thiourea; Triazoles

2016
Sugar-Based Arylsulfonamide Carboxylates as Selective and Water-Soluble Matrix Metalloproteinase-12 Inhibitors.
    ChemMedChem, 2016, 08-05, Volume: 11, Issue:15

    Topics: Acetylglucosamine; Catalytic Domain; Glucosides; Humans; Matrix Metalloproteinase 12; Matrix Metalloproteinase 9; Matrix Metalloproteinase Inhibitors; Solubility; Sulfonamides; Thiourea; Triazoles; Water

2016
Synthesis and Biological Activities of Ethyl 2-(2-pyridylacetate) Derivatives Containing Thiourea, 1,2,4-triazole, Thiadiazole and Oxadiazole Moieties.
    Molecules (Basel, Switzerland), 2017, Mar-06, Volume: 22, Issue:3

    Topics: Anti-Infective Agents; Bacteria; Cell Line; Cells, Cultured; Crystallography, X-Ray; Fungi; HIV-1; Humans; Microbial Sensitivity Tests; Models, Molecular; Molecular Structure; Oxadiazoles; Structure-Activity Relationship; Thiadiazoles; Thiourea; Triazoles

2017
Targeting AXL overcomes resistance to docetaxel therapy in advanced prostate cancer.
    Oncotarget, 2017, Jun-20, Volume: 8, Issue:25

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Axl Receptor Tyrosine Kinase; Benzocycloheptenes; Cell Line, Tumor; Docetaxel; Drug Resistance, Neoplasm; Epithelial-Mesenchymal Transition; Gene Expression Regulation, Neoplastic; Humans; Male; Mice, Nude; Piperazines; Prostatic Neoplasms; Protein Kinase Inhibitors; Proto-Oncogene Proteins; Pyrimidines; Receptor Protein-Tyrosine Kinases; RNA Interference; Taxoids; Thiourea; Triazoles; Xenograft Model Antitumor Assays

2017
Design, synthesis and preliminary biological evaluation of new [1,2,3]triazolo[4,5-d]pyrimidine/thiourea hybrids as antiproliferative agents.
    European journal of medicinal chemistry, 2017, Oct-20, Volume: 139

    Topics: Apoptosis; Cell Line; Cell Proliferation; Dose-Response Relationship, Drug; Drug Design; Humans; Molecular Structure; Structure-Activity Relationship; Thiourea; Triazoles

2017
Synthesis of 1,2,4-triazole-linked urea/thiourea conjugates as cytotoxic and apoptosis inducing agents.
    Bioorganic & medicinal chemistry letters, 2018, 06-01, Volume: 28, Issue:10

    Topics: A549 Cells; Animals; Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Drug Screening Assays, Antitumor; G1 Phase Cell Cycle Checkpoints; Humans; MCF-7 Cells; Mice; Structure-Activity Relationship; Thiourea; Triazoles; Urea

2018
Facile One-Pot Parallel Synthesis of 3-Amino-1,2,4-triazoles.
    ACS combinatorial science, 2018, 07-09, Volume: 20, Issue:7

    Topics: Alkylation; Molecular Structure; Small Molecule Libraries; Temperature; Thiophenes; Thiourea; Time Factors; Triazoles

2018
New 1,2,3-triazole-(thio)barbituric acid hybrids as urease inhibitors: Design, synthesis, in vitro urease inhibition, docking study, and molecular dynamic simulation.
    Archiv der Pharmazie, 2020, Volume: 353, Issue:9

    Topics: Anti-Bacterial Agents; Enzyme Inhibitors; Helicobacter pylori; Molecular Docking Simulation; Molecular Dynamics Simulation; Structure-Activity Relationship; Thiobarbiturates; Thiourea; Triazoles; Urease

2020
Synthesis, Structure and Cytotoxicity Testing of Novel 7-(4,5-dihydro-1
    Molecules (Basel, Switzerland), 2020, Dec-14, Volume: 25, Issue:24

    Topics: Apoptosis; Cell Line, Tumor; Cell Proliferation; Cytotoxins; Humans; Imidazoles; Imines; Inhibitory Concentration 50; Structure-Activity Relationship; Sulfonamides; Thiourea; Triazoles; Urea

2020
Chiral 2-azabicycloalkanes bearing 1,2,3-triazole, thiourea, and ebselen moieties - Synthesis and biological activity.
    Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2023, Volume: 164

    Topics: Antiviral Agents; Organoselenium Compounds; Structure-Activity Relationship; Thiourea; Triazoles

2023