Page last updated: 2024-08-24

triazoles and thienopyrimidine

triazoles has been researched along with thienopyrimidine in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (66.67)24.3611
2020's2 (33.33)2.80

Authors

AuthorsStudies
Gayatri, G; Narsaiah, B; Prasad, MR; Rao, AR; Sastry, GN; Sirisha, B; Yakaiah, T1
El-Ashmawy, IM; Rizk, OH; Shaaban, OG1
Ahn, J; Ahn, S; Cechetto, J; Choi, I; Choi, J; Han, SJ; Hwang, JY; Jo, S; Ju, MK; Kim, J; Kim, TH; Ko, Y; Kwon, J; Lee, D; Lee, J; Liuzzi, M; Nam, J; No, Z; Park, DS; Park, E; Sommer, P1
Chen, X; Hou, S; Liu, X; Tang, Q; Wang, L; Xiong, H; Xu, S; Zheng, P; Zhu, W; Zou, W1
Geronikaki, A; Glamoclija, J; Hakobyan, EK; Hovakimyan, AA; Ivanov, M; Kartsev, VG; Petrou, A; Sirakanyan, SN; Sokovic, M; Spinelli, D1
Alshamari, AK; Awad, HM; El-Sayed, WA; Elganzory, HH; Hassan, AA; Hassan, NA; Khattab, RR; Nossier, ES1

Other Studies

6 other study(ies) available for triazoles and thienopyrimidine

ArticleYear
Synthesis and theoretical studies on energetics of novel N- and O- perfluoroalkyl triazole tagged thienopyrimidines--their potential as adenosine receptor ligands.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:5

    Topics: Animals; Binding Sites; Computer Simulation; Cyclization; Drug Design; Ligands; Models, Molecular; Pyrimidines; Rats; Receptors, Purinergic P1; Structure-Activity Relationship; Thermodynamics; Triazoles

2010
Design, synthesis and biological evaluation of some novel thienopyrimidines and fused thienopyrimidines as anti-inflammatory agents.
    European journal of medicinal chemistry, 2012, Volume: 55

    Topics: Animals; Anti-Inflammatory Agents; Chemistry Techniques, Synthetic; Drug Design; Edema; Formaldehyde; Granuloma; Male; Pyrimidines; Rats; Triazoles; Turpentine; Ulcer

2012
Synthesis and biological evaluation of triazolothienopyrimidine derivatives as novel HIV-1 replication inhibitors.
    Bioorganic & medicinal chemistry letters, 2013, Jan-01, Volume: 23, Issue:1

    Topics: Anti-HIV Agents; Cell Line; Drug Evaluation, Preclinical; High-Throughput Screening Assays; HIV-1; Humans; Pyrimidines; Structure-Activity Relationship; Triazoles; Virus Replication

2013
Discovery of thinopyrimidine-triazole conjugates as c-Met targeting and apoptosis inducing agents.
    Bioorganic chemistry, 2018, Volume: 77

    Topics: Apoptosis; Cell Line, Tumor; Dose-Response Relationship, Drug; Drug Discovery; Hep G2 Cells; Humans; MCF-7 Cells; Molecular Docking Simulation; Molecular Structure; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-met; Pyrimidines; Structure-Activity Relationship; Triazoles

2018
Synthesis and Evaluation of Antimicrobial Activity and Molecular Dock - ing of New N-1,3-thiazol-2-ylacetamides of Condensed Pyrido[3',2':4,5] furo(thieno)[3,2-d]pyrimidines.
    Current topics in medicinal chemistry, 2020, Volume: 20, Issue:24

    Topics: Alkylation; Anti-Bacterial Agents; Antifungal Agents; Biofilms; Drug Design; Humans; Microbial Sensitivity Tests; Molecular Conformation; Molecular Docking Simulation; Protein Binding; Pyrimidines; Structure-Activity Relationship; Triazoles

2020
Click chemistry based synthesis, cytotoxic activity and molecular docking of novel triazole-thienopyrimidine hybrid glycosides targeting EGFR.
    Journal of enzyme inhibition and medicinal chemistry, 2021, Volume: 36, Issue:1

    Topics: Antineoplastic Agents; Cell Proliferation; Cell Survival; Click Chemistry; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; ErbB Receptors; Glycosides; Humans; Molecular Docking Simulation; Molecular Structure; Protein Kinase Inhibitors; Pyrimidines; Structure-Activity Relationship; Triazoles; Tumor Cells, Cultured

2021