triazoles has been researched along with oxazoles in 77 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 8 (10.39) | 18.7374 |
1990's | 18 (23.38) | 18.2507 |
2000's | 17 (22.08) | 29.6817 |
2010's | 27 (35.06) | 24.3611 |
2020's | 7 (9.09) | 2.80 |
Authors | Studies |
---|---|
Fotsch, C; St Jean, DJ | 1 |
Kasahara, M; Konosu, T; Miyaoka, T; Oida, S; Tajima, Y; Takeda, N; Yasuda, H | 1 |
Allen, SD; Bennett, GA; Kinsolving, CR; Mitchell, JT; Mullen, GB; St Georgiev, V; Swift, PA | 1 |
Dunoff, RY; Graboyes, H; Jaffe, G; Karash, CB; Pachter, IJ; Snader, K; Weinstock, J | 1 |
Doorenbos, NJ; Dorn, CP | 1 |
Armstrong, DR; Breckenridge, RJ; Suckling, CJ | 1 |
Iwagami, H; Sasaki, Y; Yasuda, N | 1 |
Ban, TA | 1 |
Bischoff, M; Frederick, EK; Throssell, CS; Turco, RF | 1 |
Murphy, CT; Westwick, J | 1 |
Durham, SK; Heran, CL; Megill, JR; Schumacher, WA; Steinbacher, TE | 1 |
Dunkelberg, H; Edenharder, R; Gebel, T; Kevekordes, S; Pav, K | 1 |
Leidy, RB; Penmetsa, KV; Shea, D | 1 |
Chardigny, JM; Christie, WW; Dobson, G; Juanéda, P; Martin, JC; Ramilison, I; Sébédio, JL | 1 |
Ashby, J; Lefevre, PA | 1 |
Colpaert, FC; John, GW; Pagniez, F; Valentin, JP; Vieu, S | 1 |
Arditi, M; Kalra, VK; Kim, KS; Shen, Y; Sultana, C | 1 |
Bazzanini, R; Manfredini, S; Manfrini, M; Marongiu, ME; Musiu, C; Perra, G; Putzolu, M; Vicentini, CB | 1 |
Barba, A; Navarro, G; Navarro, S; Oliva, J | 1 |
Hopkins, B; McHarg, A; Melrose, H; Napier, C; Stewart, M; Wallis, R | 1 |
Birk, KL; Cohen, AF; De Puy, ME; De Smet, M; Fisher, AL; Goldberg, MR; Musson, DG; Sterrett, A; Van Gerven, JM; Van Haarst, AD | 1 |
Deleu, D; Hanssens, Y | 2 |
Goadsby, PJ | 1 |
Quinn, JV; Slotman, GJ | 1 |
Bartlett, MG; Stewart, JT; Vishwanathan, K | 1 |
Logemann, CD; Rankin, LM | 1 |
Chernyshev, O; Gentry, P; Kailasam, J; Mathew, NT | 1 |
Bartleson, JD | 1 |
Nagle, DG; Wedge, DE | 1 |
Dalvie, DK; Kalgutkar, AS; Khojasteh-Bakht, SC; O'Donnell, JP; Obach, RS | 1 |
Wang, JP | 1 |
BALLONOFF, LB; FEINSTEIN, RN; SEAHOLM, JE | 1 |
Abdel Aleem, AH; Abdel-Aal, MT; El Ashry, ES; El-Sayed, WA | 1 |
Cai, C; Katritzky, AR; Singh, SK; Suzuki, K | 1 |
Marriott, G; Miller, R; Petchprayoon, C; Sakata, T; Suwanborirux, K | 1 |
Heinzl, S | 1 |
Abramov, YA; Audoly, L; Bach, J; Barberia, JT; Braganza, JF; Carter, D; Carty, TJ; Cortina, SR; Dombroski, MA; Donahue, KM; Elliott, NC; Gabel, CA; Gibbons, CP; Jordan, CK; Kalgutkar, AS; Kuperman, AV; Labasi, JM; Laird, ER; Laliberte, RE; Letavic, MA; Lombardo, F; McClure, KF; McCoy, JM; Naiman, BM; Nelson, KL; Nguyen, HT; Peese, KM; Sweeney, FJ; Taylor, TJ; Trebino, CE; Volberg, WA; Zhou, J | 1 |
Ibrahim, WA; Naim, AA; Sanagi, MM; See, HH | 1 |
Bartoccini, F; Carminati, P; Castorina, M; Gallo, G; Ghirardi, O; Giorgi, F; Giorgi, L; Minetti, P; Piersanti, G; Tarzia, G | 1 |
Blasi, ER; Ecelbarger, CM; Heyen, JR; McHarg, AD; Tiwari, S | 1 |
Bryant, DN; Cummins, I; Edwards, R | 1 |
Andersen, HR; Kjaerstad, MB; Nellemann, C; Taxvig, C | 1 |
Hergenrother, PJ; Miller, MJ; Miller, PA; Moraski, GC; Palchaudhuri, R; Peterson, RJ; Stefely, JA | 1 |
Muralikrishna, A; Padmaja, A; Padmavathi, V; Rajasekhar, C | 1 |
Aldana, M; De Prado, R; Martínez, MJ | 1 |
Conrad, WE; Fettinger, JC; Haddadin, MJ; Kurth, MJ; Nguyen, HH; Rodriguez, KX | 1 |
Chen, J; Duan, W; He, F; Ma, Y; Song, C; Zhao, L | 1 |
Andréasson, E; Bylund, J; Christenson, K; Dahlgren, C; Forsman, H; Karlsson, A; Önnheim, K | 1 |
Baccei, CS; Bravo, Y; Broadhead, A; Bundey, R; Chen, A; Clark, R; Correa, L; Jacintho, JD; Lorrain, DS; Messmer, D; Prasit, P; Stebbins, K; Stock, N | 1 |
Chen, X; Hu, J; Jin, J; Tian, Y; Wang, X; Xiao, Q; Yin, D; Zhou, W | 1 |
Bujak, A; Dymek, B; Dzwonek, K; Grygielewicz, P; Gunerka, P; Lamparska-Przybysz, M; Stanczak, A; Wieczorek, M; Zdzalik, D | 1 |
Buijsman, RC; de Man, J; de Roos, JA; de Vetter, JR; Prinsen, MB; Spijkers-Hagelstein, JA; Uitdehaag, JC; van Doornmalen, AM; Zaman, GJ | 1 |
Chen, H; Ding, HF; Dong, Z; Fang, D; Huang, S; Jing, Q; Lu, Y; Su, SB; Yang, L | 1 |
Bryant, DM; Farkas, JE; Freitas, PD; Monaghan, JR; Whited, JL | 1 |
Chang, GC; Chang, JS; Che, Y; Chen, JM; Conn, EL; Cook, JM; El Fakhri, G; Enerson, BE; Guehl, NJ; Haggarty, SJ; Holson, EB; Janat, F; Kurumbail, RG; Lanyon, LF; Lefker, BA; Liang, SH; Livni, E; Lopresti-Morrow, L; Nolan, CE; Normandin, MD; Para, KS; Patnaik, D; Perlis, R; Plummer, MS; Richter, KE; Schachter, JB; Shanmugasundaram, V; Taylor, CK; Trapa, P; Vasdev, N; Wagner, FF; Wang, L | 1 |
Baillie, TA; Cyrus Khojasteh, S; Dalvie, D; Rietjens, IM | 1 |
Cruz, HG; Dingemanse, J; Groenen, PM; Krause, A; Lott, D; Stalder, AK; Strasser, DS | 1 |
Akudugu, JM; Hamunyela, RH; Serafin, AM | 1 |
Rademacher, J; Welte, T | 1 |
Cao, S; Chen, L; Ge, RS; Huang, P; Mao, B; Su, Y; Wang, X; Wu, Y; Ye, L | 1 |
Chen, F; Chen, L; Ge, RS; Huang, P; Shen, X; Su, Y | 1 |
Afatsawo, C; Arabin, P; Bigaud, M; Cordier, V; Desrayaud, S; Hoffmann, L; Lehmann, D; Lowe, PJ; Risser, F; Stringer, R; Thiel, J; Widmer, T; Wipfli, P | 1 |
Geng, J; Li, Y; Najafov, A; Ofengeim, D; Ouchida, AT; Sun, X; Yu, Q; Yuan, J | 1 |
Carroll, AR; Leusch, FDL; Melvin, SD | 1 |
Hino, K; Horigome, K; Ikeya, M; Komura, S; Nagata, S; Nishio, M; Ohta, A; Okanishi, Y; Toguchida, J; Yamada, Y; Zhao, C | 1 |
Dahlgren, C; Forsman, H; Holmdahl, R; Lind, S; Olofsson, P; Sundqvist, M | 1 |
Baccelli, I; Bertomeu, T; Blouin-Chagnon, V; Boivin, I; Bordeleau, ME; Boucher, G; Corneau, S; Coulombe-Huntington, J; Frechette, M; Gareau, Y; Gingras, S; Girard, S; Hébert, J; Kanshin, E; Krosl, J; Lavallée, VP; Lehnertz, B; Lemieux, S; Leveillé, K; MacRae, T; Marinier, A; Mayotte, N; Roux, PP; Sauvageau, G; Spinella, JF; St-Denis, C; Thibault, P; Thiollier, C; Tyers, M | 1 |
Cao, M; Fang, YL; Tang, S; Wang, YC; Xi, ZW; Xu, XJ | 1 |
Allen, TE; Chung, I; Fischer, PM; Hardy, RE; Harvey, RF; Hirst, J; Kellam, B; MacFarlane, M; Mistry, S; Pryde, KR; Serreli, R; Stephenson, ZA; Stoneley, M; Willis, AE | 1 |
Ballard, J; Be, C; Berman, A; Biggart, A; Bursulaya, B; Caridha, D; Chen, YL; Chianelli, D; Davis, LC; Eggimann, FK; Gao, MY; Gibney, M; Glynne, RJ; Groessl, T; Hein, A; Jiricek, J; Johnson, K; Khare, S; Kreishman-Deitrick, M; Lai, YH; Lerario, I; Liang, F; Liu, X; Luneau, A; Mathison, CJN; Molteni, V; Nagle, A; Pybus, B; Rao, SPS; Richmond, W; Rudewicz, PJ; Sciotti, RJ; Shapiro, M; Smith, J; Spraggon, G; Srinivas, H; Supek, F; Thompson, C; Tuntland, T; Wiesmann, C; Xie, Y; Yeh, V | 1 |
Cantini, N; Cilibrizzi, A; Crocetti, L; Giovannoni, MP; Guerrini, G; Khlebnikov, AI; Kirpotina, LN; Paoli, P; Quinn, MT; Rossi, P; Schepetkin, IA; Vergelli, C | 1 |
Ge, S; He, H; Hou, Y; Lu, J; Lv, Y; Wang, C; Wang, X | 1 |
Beier, P; Motornov, V | 1 |
Chen, M; Dong, J; Gao, Y; Liu, W; Wang, T; Zhu, D | 1 |
10 review(s) available for triazoles and oxazoles
Article | Year |
---|---|
Mitigating heterocycle metabolism in drug discovery.
Topics: Animals; Biotransformation; Databases, Factual; Drug Discovery; Drug Interactions; Heterocyclic Compounds, 1-Ring; Heterocyclic Compounds, 4 or More Rings; Humans; Mice; Pharmaceutical Preparations; Rats | 2012 |
Monoamine uptake inhibitors.
Topics: Amines; Animals; Carboxylic Acids; Chemical Phenomena; Chemistry; Humans; Imidazoles; Indoles; Isoquinolines; Monoamine Oxidase Inhibitors; Oxazoles; Triazoles | 1982 |
Profiles of 5-HT 1B/1D agonists in acute migraine with special reference to second generation agents.
Topics: Acute Disease; Animals; Clinical Trials as Topic; Coronary Circulation; Coronary Vasospasm; Drug Design; Drug Interactions; Humans; Inactivation, Metabolic; Indoles; Meninges; Migraine Disorders; Molecular Structure; Nociceptors; Oxazoles; Oxazolidinones; Piperidines; Propranolol; Pyrrolidines; Randomized Controlled Trials as Topic; Rats; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Recurrence; Serotonin Receptor Agonists; Structure-Activity Relationship; Sumatriptan; Treatment Outcome; Triazoles; Tryptamines; Vasoconstrictor Agents | 1999 |
The scientific basis of medication choice in symptomatic migraine treatment.
Topics: Acute Disease; Choice Behavior; Dose-Response Relationship, Drug; Humans; Indoles; Migraine Disorders; Models, Biological; Oxazoles; Oxazolidinones; Piperidines; Serotonin Receptor Agonists; Severity of Illness Index; Sumatriptan; Triazoles; Tryptamines | 1999 |
Newer intranasal migraine medications.
Topics: Administration, Intranasal; Administration, Oral; Analgesics, Non-Narcotic; Clinical Trials as Topic; Dihydroergotamine; Half-Life; Humans; Indoles; Migraine Disorders; Oxazoles; Oxazolidinones; Piperidines; Recurrence; Serotonin Receptor Agonists; Sumatriptan; Triazoles; Tryptamines | 2000 |
Current and emerging second-generation triptans in acute migraine therapy: a comparative review.
Topics: Acute Disease; Carbazoles; Humans; Indoles; Migraine Disorders; Oxazoles; Oxazolidinones; Piperidines; Pyrrolidines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Receptor Agonists; Triazoles; Tryptamines | 2000 |
Biotransformation reactions of five-membered aromatic heterocyclic rings.
Topics: Animals; Cytochrome P-450 Enzyme System; Furans; Heterocyclic Compounds, 4 or More Rings; Humans; Imidazoles; Indoles; Isoxazoles; Models, Chemical; Molecular Structure; Oxadiazoles; Oxazoles; Pyrazoles; Pyrroles; Tetrazoles; Thiadiazoles; Thiazoles; Thiophenes; Triazoles; Xenobiotics | 2002 |
[Dipeptidylpeptidase IV inhibitors and dual action PPAR-agonists].
Topics: Adamantane; Adenosine Deaminase Inhibitors; Diabetes Mellitus, Type 2; Dipeptidyl Peptidase 4; Glycine; Glycoproteins; Humans; Hypoglycemic Agents; Nitriles; Oxazoles; Peroxisome Proliferator-Activated Receptors; Protease Inhibitors; Pyrazines; Pyrrolidines; Sitagliptin Phosphate; Triazoles; Vildagliptin | 2006 |
Biotransformation and bioactivation reactions - 2015 literature highlights.
Topics: Acetaminophen; Allylbenzene Derivatives; Aniline Compounds; Animals; Anisoles; Benzbromarone; Biotransformation; Humans; Imidazoles; Niacinamide; Nitroimidazoles; Nitrosamines; Oxazoles; Oxazolidinones; Peroxides; Pyrazines; Pyrazoles; Pyridazines; Pyridines; Pyridones; Pyrimidinones; Thiophenes; Triazoles | 2016 |
[New antibiotics - standstill or progress].
Topics: Anti-Bacterial Agents; Azabicyclo Compounds; Bacterial Infections; Ceftaroline; Ceftazidime; Cephalosporins; Clinical Trials as Topic; Drug Approval; Drug Combinations; Drug Resistance, Multiple, Bacterial; Ephedrine; Humans; Macrolides; Methicillin-Resistant Staphylococcus aureus; Organophosphates; Oxazoles; Penicillanic Acid; Phenobarbital; Staphylococcal Infections; Tazobactam; Theophylline; Triazoles | 2017 |
3 trial(s) available for triazoles and oxazoles
Article | Year |
---|---|
The effects of moclobemide on the pharmacokinetics of the 5-HT1B/1D agonist rizatriptan in healthy volunteers.
Topics: Adult; Area Under Curve; Benzamides; Biotransformation; Blood Pressure; Cross-Over Studies; Double-Blind Method; Female; Half-Life; Humans; Male; Methoxyhydroxyphenylglycol; Moclobemide; Monoamine Oxidase Inhibitors; Oxazoles; Oxazolidinones; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Receptor Agonists; Sumatriptan; Triazoles; Tryptamines | 1999 |
Treatment of nonresponders to oral sumatriptan with zolmitriptan and rizatriptan: a comparative open trial.
Topics: Administration, Oral; Cross-Over Studies; Drug Resistance; Humans; Migraine Disorders; Oxazoles; Oxazolidinones; Retreatment; Serotonin Receptor Agonists; Sumatriptan; Triazoles; Tryptamines; Vasoconstrictor Agents | 2000 |
Biomarker-guided clinical development of the first-in-class anti-inflammatory FPR2/ALX agonist ACT-389949.
Topics: Adolescent; Adult; Animals; Biomarkers; Cell Migration Assays; Cytokines; Disease Models, Animal; Dose-Response Relationship, Drug; Double-Blind Method; Humans; Inflammation; Lipopolysaccharides; Male; Middle Aged; Neutrophils; Oxazoles; Receptors, Formyl Peptide; Receptors, Lipoxin; Triazoles; Young Adult | 2017 |
64 other study(ies) available for triazoles and oxazoles
Article | Year |
---|---|
Triazole antifungals. II. Synthesis and antifungal activities of 3-acyl-4-methyloxazolidine derivatives.
Topics: Animals; Antifungal Agents; Male; Mice; Oxazoles; Triazoles | 1990 |
In vitro antifungal activity of novel substituted 3,5-diphenyl-3-(1H-1,2,4-triazol-1-ylmethyl)-2- methylisoxazolidine derivatives.
Topics: Antifungal Agents; Fungi; Isoxazoles; Microbial Sensitivity Tests; Molecular Structure; Oxazoles; Structure-Activity Relationship; Triazoles | 1988 |
[Comparative studies on various compounds with trichomonacidal activity].
Topics: Antiprotozoal Agents; Bacteria; Female; Fungi; Humans; In Vitro Techniques; Infant, Newborn; Metronidazole; Oxazoles; Pregnancy; Triazoles; Trichomonas | 1970 |
Pteridines. 8. Some 2,4,7-triamino-6-heteroarylpteridines.
Topics: Chromatography, Paper; Furans; Hydrogen-Ion Concentration; Imidazoles; Oxazoles; Pteridines; Pyrazoles; Pyridines; Pyrimidines; Pyrroles; Spectrum Analysis; Thiazoles; Thiophenes; Triazoles; Ultraviolet Rays | 1968 |
Steroids 23. Synthesis fo some ring A-fused heterocyclic steroids.
Topics: Anabolic Agents; Chemical Phenomena; Chemistry; Heterocyclic Compounds; Imidazoles; Oxazoles; Pyrazoles; Thiazoles; Triazoles | 1965 |
Muscimol and some aza analogues: molecular orbital calculations relating to their potency as GABA mimetics.
Topics: Binding Sites; Chemical Phenomena; Chemistry; Electrons; gamma-Aminobutyric Acid; Humans; Molecular Conformation; Muscimol; Oxazoles; Pyrazoles; Pyrazolones; Receptors, Neurotransmitter; Rotation; Structure-Activity Relationship; Triazoles | 1982 |
Synthesis and antibacterial activity of triazole and isoxazole derivatives of ampicillin.
Topics: Ampicillin; Anti-Bacterial Agents; Bacteria; Indicators and Reagents; Isoxazoles; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Oxazoles; Pseudomonas aeruginosa; Spectrophotometry, Infrared; Structure-Activity Relationship; Triazoles | 1983 |
Degradation of chloroneb, triadimefon, and vinclozolin in soil, thatch, and grass clippings.
Topics: Biodegradation, Environmental; Chlorobenzenes; Chromatography, Gas; Fungicides, Industrial; Indiana; Oxazoles; Poaceae; Soil; Triazoles | 1994 |
Role of type 1 and type 2A phosphatases in signal transduction of platelet-activating-factor-stimulated rabbit platelets.
Topics: Animals; Azepines; Blood Platelets; Calcium; Cations, Divalent; Indoles; Inositol 1,4,5-Trisphosphate; Ionomycin; Maleimides; Manganese; Marine Toxins; Oxazoles; Phosphoprotein Phosphatases; Phosphoproteins; Phosphorylation; Platelet Activating Factor; Protein Kinase C; Rabbits; Signal Transduction; Triazoles | 1994 |
Effects of antithrombotic drugs in a rat model of aspirin-insensitive arterial thrombosis.
Topics: Amino Acid Chloromethyl Ketones; Animals; Aspirin; Azepines; Bridged Bicyclo Compounds, Heterocyclic; Carotid Artery Thrombosis; Dipyridamole; Fibrinolytic Agents; Heparin; Male; Oxazoles; Propionates; Rats; Rats, Sprague-Dawley; Thrombolytic Therapy; Ticlopidine; Triazoles; Warfarin | 1993 |
Genotoxicity of selected pesticides in the mouse bone-marrow micronucleus test and in the sister-chromatid exchange test with human lymphocytes in vitro.
Topics: Adult; Aldicarb; Allyl Compounds; Animals; Bone Marrow; Cells, Cultured; Female; Humans; Hydrocarbons, Chlorinated; Lymphocytes; Male; Mice; Micronuclei, Chromosome-Defective; Micronucleus Tests; Organothiophosphorus Compounds; Oxazoles; Parathion; Pesticides; Sister Chromatid Exchange; Triazoles | 1996 |
Separation of fungicides by micellar electrokinetic capillary chromatography.
Topics: Alanine; Benzimidazoles; Buffers; Carbamates; Chromatography; Electrophoresis, Capillary; Fungicides, Industrial; Micelles; Oxazoles; Surface-Active Agents; Triazoles | 1997 |
Metabolites of conjugated isomers of linoleic acid (CLA) in the rat.
Topics: Animals; Chromatography, High Pressure Liquid; Diet, Fat-Restricted; Gas Chromatography-Mass Spectrometry; Isomerism; Linoleic Acids; Lipids; Liver; Male; Oxazoles; Rats; Rats, Wistar; Triazoles | 1997 |
The weanling male rat as an assay for endocrine disruption: preliminary observations.
Topics: Anastrozole; Androgen Antagonists; Animals; Body Weight; Cyproterone Acetate; Drug Evaluation, Preclinical; Endocrine System Diseases; Female; Lactose; Male; Methylcellulose; Nitriles; Organ Size; Oxazines; Oxazoles; Rats; Rats, Inbred Strains; Toxicology; Triazoles; Uterus; Weaning | 1997 |
Pharmacological analysis of the haemodynamic effects of 5-HT1B/D receptor agonists in the normotensive rat.
Topics: Animals; Autonomic Nervous System; Blood Pressure; Drug Interactions; Heart Rate; Hemodynamics; Male; Oxazoles; Oxazolidinones; Parasympathetic Nervous System; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Receptor Agonists; Sumatriptan; Triazoles; Tryptamines | 1998 |
Endotoxin-induced migration of monocytes and PECAM-1 phosphorylation are abrogated by PAF receptor antagonists.
Topics: Azepines; Cell Differentiation; Cells, Cultured; Chemotaxis, Leukocyte; Endothelium, Vascular; Endotoxins; Escherichia coli; Gene Expression Regulation; HL-60 Cells; Humans; Indoles; Lipopolysaccharide Receptors; Lipopolysaccharides; Maleimides; Marine Toxins; Monocytes; Oxazoles; Phosphorylation; Platelet Endothelial Cell Adhesion Molecule-1; Platelet Membrane Glycoproteins; Pyridinium Compounds; Receptors, Cell Surface; Receptors, G-Protein-Coupled; RNA, Messenger; Transcription, Genetic; Triazoles; Umbilical Veins | 1998 |
New "triptans" and other drugs for migraine.
Topics: Adrenergic beta-Antagonists; Amitriptyline; Anti-Inflammatory Agents, Non-Steroidal; Antidepressive Agents, Tricyclic; Calcium Channel Blockers; Dihydroergotamine; Drug Interactions; Ergotamine; Humans; Indoles; Methysergide; Migraine Disorders; Naproxen; Oxazoles; Oxazolidinones; Piperidines; Propranolol; Selective Serotonin Reuptake Inhibitors; Serotonin Receptor Agonists; Sumatriptan; Time Factors; Timolol; Triazoles; Tryptamines; Valproic Acid; Vasoconstrictor Agents | 1998 |
Synthesis and biological evaluation of a series of substituted pyrazolo[3,4-d]-1,2,3-triazoles and pyrazolo[3,4-d]oxazoles.
Topics: Anti-Bacterial Agents; Anti-HIV Agents; Antifungal Agents; Bacteria; Humans; Microbial Sensitivity Tests; Oxazoles; Triazoles | 1998 |
Determination of chlorpyrifos, penconazole, fenarimol, vinclozolin and metalaxyl in grapes, must and wine by on-line microextraction and gas chromatography.
Topics: Alanine; Chlorpyrifos; Chromatography, Gas; Fungicides, Industrial; Insecticides; Oxazoles; Pyrimidines; Reproducibility of Results; Rosales; Sensitivity and Specificity; Triazoles; Wine | 1999 |
Characterisation of the 5-HT receptor binding profile of eletriptan and kinetics of [3H]eletriptan binding at human 5-HT1B and 5-HT1D receptors.
Topics: Animals; Binding, Competitive; Cell Line; Cold Temperature; COS Cells; HeLa Cells; Humans; Indoles; Kinetics; Oxazoles; Oxazolidinones; Piperidines; Pyrrolidines; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Sumatriptan; Triazoles; Tritium; Tryptamines | 1999 |
Platelet-activating factor and arachidonic acid metabolites mediate tumor necrosis factor and eicosanoid kinetics and cardiopulmonary dysfunction during bacteremic shock.
Topics: Aeromonas hydrophila; Animals; Arachidonic Acid; Azepines; Bridged Bicyclo Compounds, Heterocyclic; Eicosanoids; Female; Gram-Negative Bacterial Infections; Heart Diseases; Hemodynamics; Hypertension, Pulmonary; Lipoxygenase Inhibitors; Masoprocol; Oxazoles; Oxygen; Oxygen Consumption; Platelet Activating Factor; Prostaglandin-Endoperoxide Synthases; Shock, Septic; Swine; Thromboxane A2; Triazoles; Tumor Necrosis Factor-alpha | 1999 |
Determination of antimigraine compounds rizatriptan, zolmitriptan, naratriptan and sumatriptan in human serum by liquid chromatography/electrospray tandem mass spectrometry.
Topics: Bufotenin; Chromatography, High Pressure Liquid; Humans; Indoles; Mass Spectrometry; Migraine Disorders; Molecular Structure; Oxazoles; Oxazolidinones; Piperidines; Sensitivity and Specificity; Serotonin Receptor Agonists; Sumatriptan; Triazoles; Tryptamines; Vasoconstrictor Agents | 2000 |
Triptans to the rescue: effective therapy for migraine headaches in the workplace.
Topics: Absenteeism; Adult; Cost-Benefit Analysis; Efficiency; Female; Humans; Indoles; Injections, Subcutaneous; Male; Migraine Disorders; Oxazoles; Oxazolidinones; Piperidines; Randomized Controlled Trials as Topic; Self Administration; Serotonin Receptor Agonists; Sumatriptan; Treatment Outcome; Triazoles; Tryptamines; Workplace | 2000 |
A new 2D-TLC bioautography method for the discovery of novel antifungal agents To control plant pathogens.
Topics: Acrylates; Aniline Compounds; Antifungal Agents; Ascomycota; Benzimidazoles; Biological Assay; Captan; Carbamates; Chromatography, Thin Layer; Colletotrichum; Dimethyldithiocarbamate; Fungicides, Industrial; Guanidines; Maneb; Methacrylates; Nitriles; Nitrobenzenes; Oxazoles; Piperazines; Plant Diseases; Plants; Pyrimidines; Strobilurins; Thiabendazole; Thiophanate; Triazoles | 2000 |
GEA3162 stimulates Ca2+ entry in neutrophils.
Topics: Adenylyl Cyclase Inhibitors; Animals; Barium; Boron Compounds; Calcium; Calcium Signaling; Calcium-Transporting ATPases; Cell Membrane Permeability; Dose-Response Relationship, Drug; Enzyme Inhibitors; Genistein; Imines; Indoles; Manganese; Marine Toxins; Neutrophils; Nitric Oxide Donors; Oxazoles; Phosphoprotein Phosphatases; Rats; Rats, Sprague-Dawley; S-Nitrosothiols; Strontium; Triazoles | 2003 |
EFFECT ON CATALASE IN VIVO AND IN VITRO OF COMPOUNDS RELATED TO AMINOTRIAZOLE. ANL-6823.
Topics: Amitrole; Azides; Azoles; Catalase; Enzyme Inhibitors; Erythrocytes; Imidazoles; In Vitro Techniques; Isoniazid; Kidney; Liver; Oxadiazoles; Oxazoles; Oxidation-Reduction; Pentylenetetrazole; Pharmacology; Pyrazoles; Rats; Research; Thiazoles; Triazoles | 1964 |
Synthesis of some functionalized arylaminomethyl-1 ,2,4-triazoles, 1,3,4-oxa- and thiadiazoles.
Topics: Antiviral Agents; Cell Line; Cell Survival; Drug Screening Assays, Antitumor; Enzyme-Linked Immunosorbent Assay; Hepatitis B virus; Humans; Indicators and Reagents; Magnetic Resonance Spectroscopy; Methylation; Oxazoles; Reverse Transcriptase Polymerase Chain Reaction; Thiazoles; Triazoles | 2003 |
Facile syntheses of oxazolines and thiazolines with N-acylbenzotriazoles under microwave irradiation.
Topics: Microwaves; Oxazoles; Thiazoles; Triazoles | 2004 |
Synthesis and characterization of the 7-(4-aminomethyl-1H-1,2,3-triazol-1-yl) analogue of kabiramide C.
Topics: Actins; Animals; HeLa Cells; Humans; Molecular Structure; Oxazoles; Porifera; Rabbits; Thailand; Triazoles | 2005 |
Structure-activity relationships of triazolopyridine oxazole p38 inhibitors: identification of candidates for clinical development.
Topics: Chemistry, Pharmaceutical; Drug Design; Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Kinetics; Models, Chemical; Oxazoles; p38 Mitogen-Activated Protein Kinases; Pyridines; Solubility; Structure-Activity Relationship; Triazoles | 2006 |
Determination of pesticides in water by cone-shaped membrane protected liquid phase microextraction prior to micro-liquid chromatography.
Topics: Analytic Sample Preparation Methods; Bridged Bicyclo Compounds; Chromatography, Liquid; Humic Substances; Hydrogen-Ion Concentration; Microchemistry; Organothiophosphorus Compounds; Oxazoles; Pesticides; Reproducibility of Results; Triazoles; Uncertainty; Water Pollutants, Chemical | 2007 |
Synthesis of benzo[1,2-d;3,4-d']diimidazole and 1H-pyrazolo[4,3-b]pyridine as putative A2A receptor antagonists.
Topics: Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Antagonists; Benzimidazoles; Binding Sites; Binding, Competitive; Molecular Structure; Oxazoles; Pyrazoles; Stereoisomerism; Triazoles | 2007 |
Time course of AQP-2 and ENaC regulation in the kidney in response to PPAR agonists associated with marked edema in rats.
Topics: Adiponectin; Animals; Aquaporin 2; Blood Pressure; Edema; Epithelial Sodium Channels; Insulin; Kidney; Male; Natriuresis; Oxazoles; PPAR gamma; Rats; Rats, Sprague-Dawley; Rosiglitazone; Thiazolidinediones; Triazoles; Water-Electrolyte Balance | 2008 |
Safener responsiveness and multiple herbicide resistance in the weed black-grass (Alopecurus myosuroides).
Topics: Glutathione; Glutathione Transferase; Herbicide Resistance; Herbicides; Oxazoles; Plant Proteins; Poaceae; Propionates; Triazoles; Triticum | 2009 |
Mixture effects of endocrine disrupting compounds in vitro.
Topics: Androgen Antagonists; Animals; Bridged Bicyclo Compounds; Cell Line, Tumor; CHO Cells; Cricetinae; Cricetulus; Drug Combinations; Endocrine Disruptors; Estradiol; Flutamide; Fungicides, Industrial; Genes, Reporter; Humans; Oxazoles; Parabens; Receptors, Androgen; Testosterone; Triazoles | 2010 |
N-((1-benzyl-1H-1,2,3-triazol-4-yl)methyl)arylamide as a new scaffold that provides rapid access to antimicrotubule agents: synthesis and evaluation of antiproliferative activity against select cancer cell lines.
Topics: Acrylamides; Cell Division; Cell Line, Tumor; Drug Screening Assays, Antitumor; G2 Phase; Humans; Microtubules; Oxazoles; Structure-Activity Relationship; Triazoles; Tubulin; Tubulin Modulators | 2010 |
Synthesis and antimicrobial activity of pyrrolyl/pyrazolyl arylaminosulfonylmethyl 1,3,4-oxadiazoles, 1,3,4-thiadiazoles and 1,2,4-triazoles.
Topics: Anti-Infective Agents; Bacteria; Bacterial Infections; Fungi; Humans; Microbial Sensitivity Tests; Mycoses; Oxazoles; Thiadiazoles; Triazoles | 2011 |
Leaching of oxadyxil and tebuconazole in Colombian soil.
Topics: Acetamides; Colombia; Environmental Monitoring; Fungicides, Industrial; Oxazoles; Triazoles; Water Pollutants, Chemical | 2011 |
A one-pot-three-step route to triazolotriazepinoindazolones from oxazolino-2H-indazoles.
Topics: Alkynes; Catalysis; Cyclization; Hydrocarbons, Brominated; Indazoles; Molecular Structure; Oxazoles; Palladium; Triazoles | 2012 |
Asymmetric β-boration of α,β-unsaturated N-acyloxazolidinones by [2.2]paracyclophane-based bifunctional catalyst.
Topics: Boron Compounds; Catalysis; Copper; Esters; Molecular Structure; Oxazoles; Stereoisomerism; Triazoles | 2012 |
Reactivation of desensitized formyl peptide receptors by platelet activating factor: a novel receptor cross talk mechanism regulating neutrophil superoxide anion production.
Topics: Actins; Azepines; Bridged Bicyclo Compounds, Heterocyclic; Calcium; Cells, Cultured; Cyclosporine; Cytochalasin B; Cytoskeleton; Gelsolin; Humans; Marine Toxins; NADPH Oxidases; Neutrophils; Oligopeptides; Oxazoles; Peptide Fragments; Platelet Activating Factor; Receptors, Formyl Peptide; Superoxides; Thiazolidines; Triazoles | 2013 |
Identification of the first potent, selective and bioavailable PPARα antagonist.
Topics: Animals; Butyrates; Humans; Mice; Molecular Structure; Oxazoles; Phenylurea Compounds; PPAR alpha; Propionates; Structure-Activity Relationship; Sulfonamides; Triazoles; Tyrosine | 2014 |
Discovery of oxazole and triazole derivatives as potent and selective S1P(1) agonists through pharmacophore-guided design.
Topics: Animals; CHO Cells; Cricetinae; Cricetulus; Drug Design; Heart Rate; Lymphocytes; Male; Models, Molecular; Molecular Conformation; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Lysosphingolipid; Structure-Activity Relationship; Triazoles | 2014 |
Epithelial-mesenchymal transition confers resistance to selective FGFR inhibitors in SNU-16 gastric cancer cells.
Topics: Antineoplastic Agents; Benzamides; Cell Line, Tumor; Drug Resistance, Neoplasm; Epithelial-Mesenchymal Transition; Humans; Isoxazoles; Molecular Targeted Therapy; Oxazoles; Phenylurea Compounds; Piperazines; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Receptor, Fibroblast Growth Factor, Type 2; Receptors, Fibroblast Growth Factor; Resorcinols; Stomach Neoplasms; Transforming Growth Factor beta1; Triazoles | 2016 |
Selective Targeting of CTNBB1-, KRAS- or MYC-Driven Cell Growth by Combinations of Existing Drugs.
Topics: Antineoplastic Combined Chemotherapy Protocols; Aza Compounds; Benzimidazoles; beta Catenin; Cell Line, Tumor; Cell Proliferation; Humans; Imidazoles; Indazoles; Indoles; Melanoma; Molecular Targeted Therapy; Mutation; Oxazoles; Oximes; Proto-Oncogene Proteins B-raf; Proto-Oncogene Proteins c-myc; Proto-Oncogene Proteins p21(ras); Pyridones; Pyrimidinones; Quinolines; Sulfonamides; Triazoles; Vemurafenib | 2015 |
Cyclin-dependent kinase 2 is an ideal target for ovary tumors with elevated cyclin E1 expression.
Topics: Animals; Apoptosis; CDC2 Protein Kinase; Cell Line, Tumor; Cyclin E; Cyclin-Dependent Kinase 2; Cyclin-Dependent Kinases; Female; Gene Expression Profiling; Gene Expression Regulation, Neoplastic; Humans; Mice; Mice, Nude; Neoplasm Metastasis; Neoplasm Transplantation; Oncogene Proteins; Ovarian Neoplasms; Oxazoles; RNA, Small Interfering; Thiazoles; Triazoles | 2015 |
Neuregulin-1 signaling is essential for nerve-dependent axolotl limb regeneration.
Topics: Ambystoma mexicanum; Animals; Blotting, Western; Extremities; Immunohistochemistry; In Situ Hybridization; Nerve Regeneration; Neuregulin-1; Oxazoles; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Triazoles | 2016 |
Discovery of a Highly Selective Glycogen Synthase Kinase-3 Inhibitor (PF-04802367) That Modulates Tau Phosphorylation in the Brain: Translation for PET Neuroimaging.
Topics: Brain; Crystallography, X-Ray; Dose-Response Relationship, Drug; Glycogen Synthase Kinase 3; Humans; Models, Molecular; Molecular Structure; Neuroimaging; Oxazoles; Phosphorylation; Positron-Emission Tomography; Protein Kinase Inhibitors; tau Proteins; Triazoles | 2016 |
Strong synergism between small molecule inhibitors of HER2, PI3K, mTOR and Bcl-2 in human breast cancer cells.
Topics: Aniline Compounds; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Cell Line, Tumor; Cell Survival; Drug Synergism; Humans; Imidazoles; Oxazoles; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-bcl-2; Quinolines; Receptor, ErbB-2; Sulfonamides; TOR Serine-Threonine Kinases; Triazoles | 2017 |
The Effects of Fungicides on Human 3β-Hydroxysteroid Dehydrogenase 1 and Aromatase in Human Placental Cell Line JEG-3.
Topics: Aromatase; Aromatase Inhibitors; Cell Line, Tumor; Endocrine Disruptors; Estradiol; Female; Fungicides, Industrial; Humans; Multienzyme Complexes; Organotin Compounds; Oxazoles; Placenta; Pregnancy; Progesterone; Progesterone Reductase; Steroid Isomerases; Trialkyltin Compounds; Triazoles | 2017 |
Effects of Fungicides on Rat's Neurosteroid Synthetic Enzymes.
Topics: 3-Oxo-5-alpha-Steroid 4-Dehydrogenase; Alcohol Oxidoreductases; Animals; Chlorocebus aethiops; COS Cells; Endocrine Disruptors; Fungicides, Industrial; Gene Expression Regulation, Enzymologic; Humans; Neurotransmitter Agents; Oxazoles; Rats; Triazoles | 2017 |
Utility of food pellets containing 1-aminobenzotriazole for longer term in vivo inhibition of cytochrome P450 in mice.
Topics: Administration, Oral; Animals; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Mice; Oxazoles; Pyrazoles; Triazoles | 2019 |
Synergistic effect of a novel autophagy inhibitor and Quizartinib enhances cancer cell death.
Topics: Apoptosis; Autophagy; Benzothiazoles; Cell Line, Tumor; Cell Proliferation; Drug Synergism; Humans; Neoplasms; Oxazoles; Phenylurea Compounds; Receptor, ErbB-2; Signal Transduction; Triazoles | 2018 |
Metabolite profiles of striped marsh frog (Limnodynastes peronii) larvae exposed to the anti-androgenic fungicides vinclozolin and propiconazole are consistent with altered steroidogenesis and oxidative stress.
Topics: Androgen Antagonists; Animals; Anura; Discriminant Analysis; Fungicides, Industrial; Larva; Least-Squares Analysis; Magnetic Resonance Spectroscopy; Metabolome; Metabolomics; Multivariate Analysis; Oxazoles; Oxidative Stress; Principal Component Analysis; Steroids; Survival Analysis; Triazoles; Water Pollutants, Chemical; Wetlands | 2018 |
An mTOR Signaling Modulator Suppressed Heterotopic Ossification of Fibrodysplasia Ossificans Progressiva.
Topics: Activin Receptors, Type I; Animals; Benzodioxoles; High-Throughput Screening Assays; Humans; Induced Pluripotent Stem Cells; Mice, SCID; Mice, Transgenic; Myositis Ossificans; Ossification, Heterotopic; Oxazoles; Pyrimidines; Quinazolines; Reproducibility of Results; Signal Transduction; TOR Serine-Threonine Kinases; Triazoles; Urea | 2018 |
Functional and signaling characterization of the neutrophil FPR2 selective agonist Act-389949.
Topics: Cells, Cultured; Dose-Response Relationship, Drug; Humans; Neutrophils; Oxazoles; Receptors, Formyl Peptide; Receptors, Lipoxin; Signal Transduction; Triazoles | 2019 |
Mubritinib Targets the Electron Transport Chain Complex I and Reveals the Landscape of OXPHOS Dependency in Acute Myeloid Leukemia.
Topics: Animals; Antineoplastic Agents; Biomarkers; Cell Line, Tumor; Cell Survival; Disease Models, Animal; Dose-Response Relationship, Drug; Electron Transport Complex I; Female; Hematopoiesis; Humans; Leukemia, Myeloid, Acute; Mice; Models, Biological; Oxazoles; Oxidative Phosphorylation; Protein Kinase Inhibitors; Receptor, ErbB-2; Triazoles | 2019 |
Ce(OTf)
Topics: Alkynes; Azides; Carboxylic Acids; Catalysis; Crystallography, X-Ray; Mesylates; Models, Molecular; Molecular Structure; Nitriles; Oxazoles; Triazoles | 2020 |
Identification of a novel toxicophore in anti-cancer chemotherapeutics that targets mitochondrial respiratory complex I.
Topics: Adenosine Triphosphate; Antineoplastic Agents; Cell Death; Cell Line; Cell Proliferation; Electron Transport Complex I; Gene Expression Regulation; Humans; Mitochondria; Mitochondria, Heart; Myocytes, Cardiac; Oxazoles; Oxidative Phosphorylation; Protein Binding; Receptor, ErbB-2; Triazoles | 2020 |
Discovery and Characterization of Clinical Candidate LXE408 as a Kinetoplastid-Selective Proteasome Inhibitor for the Treatment of Leishmaniases.
Topics: Animals; Antiprotozoal Agents; Dogs; Humans; Leishmania donovani; Leishmania major; Leishmaniasis, Visceral; Liver; Macaca fascicularis; Mice; Mice, Inbred BALB C; Oxazoles; Proteasome Inhibitors; Pyrimidines; Rats; Rats, Sprague-Dawley; Triazoles | 2020 |
Synthesis, biological evaluation, molecular modeling, and structural analysis of new pyrazole and pyrazolone derivatives as N-formyl peptide receptors agonists.
Topics: Acetamides; Binding Sites; Humans; Models, Molecular; Neutrophils; Oxazoles; Protein Binding; Pyrazoles; Pyrazolones; Pyridones; Receptors, Formyl Peptide; Structure-Activity Relationship; Triazoles | 2021 |
Synthesis and evaluation of new potential anti-pseudo-allergic agents.
Topics: Anaphylaxis; Anti-Allergic Agents; Cell Line; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Hypersensitivity; Molecular Structure; Nerve Tissue Proteins; Oxazoles; Receptors, G-Protein-Coupled; Receptors, Neuropeptide; Structure-Activity Relationship; Triazoles | 2022 |
Access to Fluoroalkylated Azoles and 2-Acylaminoketones via Fluorinated Anhydride-Mediated Cleavage of NH-1,2,3-Triazoles.
Topics: Amines; Anhydrides; Azoles; Oxazoles; Triazoles | 2022 |
Mubritinib enhanced the inhibiting function of cisplatin in lung cancer by interfering with mitochondrial function.
Topics: Animals; Apoptosis; Carcinoma, Non-Small-Cell Lung; Cell Line, Tumor; Cell Proliferation; Cisplatin; Humans; Lung Neoplasms; Mice; Mitochondria; Oxazoles; Phosphatidylinositol 3-Kinases; Proto-Oncogene Proteins c-akt; Reactive Oxygen Species; Triazoles | 2022 |