triazoles has been researched along with glycine in 100 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 7 (7.00) | 18.7374 |
1990's | 4 (4.00) | 18.2507 |
2000's | 14 (14.00) | 29.6817 |
2010's | 57 (57.00) | 24.3611 |
2020's | 18 (18.00) | 2.80 |
Authors | Studies |
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Faden, AI; Tzendzalian, PA | 1 |
Ferro, AJ; Fitchen, JH; Johnson, LL; Riscoe, MK; Tower, PA | 1 |
Beattie, DS | 1 |
Baron, J; Tephly, TR | 1 |
Boguslawski, J; Klopotowski, T; Walczak, W | 1 |
Klopotowski, T; Rybicka, H | 1 |
Gnanam, A; Vivekanandhan, M | 1 |
Baron, J; Hasegawa, E; Tephly, TR | 1 |
Israels, LG; Levitt, M; Schacter, BA; Zipursky, A | 1 |
Braun, D; Chmielewski, PA; Kane, JM; Miller, JA | 1 |
Bend, JR; Halpert, JR; Hanna, IH; Hollenberg, PF; Kent, UM; Szklarz, GD; Vaz, AD | 1 |
Garry, VF; Lin, N | 1 |
Pèzzola, A; Pintor, A; Popoli, P; Quarta, D; Reggio, R | 1 |
Nikbakht, MR; Stone, TW | 1 |
Konishi, S; Rusakov, D; Saitow, F; Satake, S | 1 |
Domenici, MR; Martire, A; Pepponi, R; Popoli, P; Potenza, RL; Tebano, MT | 1 |
Syversen, N | 1 |
Franchi-Gazzola, R; Gaccioli, F; Lanfranchi, M; Marchiò, L; Metta, G; Pellinghelli, MA; Tardito, S; Tegoni, M | 1 |
Cheng, J; Feng, JX; Mao, XZ; Qin, YM; Shi, YH; Wang, ZY; Wei, LP; Zhang, L; Zhu, SW; Zhu, YX | 1 |
Heinzl, S | 1 |
Huang, WD; Liu, HT; Liu, YY; Pan, QH; Yang, HR; Zhan, JC | 1 |
Anziliero, D; Barcellos, LJ; Centenaro, L; Cericato, L; da Rosa, JG; Fagundes, M; Finco, J; Koakoski, G; Kreutz, LC; Neto, JG; Pottker, E; Quevedo, RM | 1 |
Barcellos, LJ; Centenaro, L; Cericato, L; da Rosa, JG; Koakoski, G; Kreutz, LC; Marqueze, A; Neto, JG; Pottker, E; Quevedo, RM | 1 |
Hata, M; Hikichi, H; Inoue, T; Ito, S; Kawagoe-Takaki, H; Kawamoto, H; Kimura, T; Maehara, S; Murai, T; Ohta, H; Ozaki, S; Satow, A; Suzuki, G | 1 |
Chen, JF; Chiodi, V; Domenici, MR; Ferrante, A; Frank, C; Ledent, C; Martire, A; Pepponi, R; Popoli, P; Tebano, MT | 1 |
Park, S; Perlin, DS; Procop, GW; Reja, V; Tuohy, MJ; Wnek, M; Yen-Lieberman, B | 1 |
Banerjee, S; Dhyani, MV; Korde, A; Kumar, C; Sarma, HD; Satpati, D | 1 |
Lenkowski, JR; McLaughlin, KA; Sanchez-Bravo, G | 1 |
Bartlett, SE; Engel, JA; Hyytiä, P; Jerlhag, E; Landgren, S; Simms, JA | 1 |
Engel, JA; Jerlhag, E | 1 |
Ahemad, M; Khan, MS | 1 |
Brunel, L; Clifford, PS; Eitan, S; Fehrentz, JA; Hart, N; Hughes, S; Kniffin, T; Martinez, J; Rodriguez, J; Schul, D; Wellman, PJ | 1 |
Brunel, L; Clifford, PS; Eitan, S; Fehrentz, JA; Hughes, S; Martinez, J; Rodriguez, J; Wellman, PJ | 1 |
Dell'anno, MT; Fisone, G; Pallottino, S | 1 |
Boeglin, D; Brunel, L; Demange, L; Denoyelle, S; Fehrentz, JA; M'Kadmi, C; Martinez, J; Moulin, A; Ryan, J | 1 |
Fukuzawa, S; Imae, K; Konno, T; Ogata, K | 1 |
Bahi, A; Brunel, L; Fehrentz, JA; Karam, SM; Martinez, J; Tolle, V; Tomasetto, CL | 1 |
Aslam, S; Benoit, P; Garnier, P; Parent, SE; Rumpel, C | 1 |
Chrysikos, D; Dimopoulos, MA; Papadimitriou, CA; Psaltopoulou, T; Sergentanis, TN; Zagouri, F | 1 |
Engel, JA; Fredriksson, I; Jerlhag, E; Steensland, P; Suchankova, P | 1 |
Havlickova, T; Jerabek, P; Kacer, P; Krsiak, M; Sustkova-Fiserova, M | 1 |
Gomez, JL; Ryabinin, AE | 1 |
Alletto, L; Benoit, P; Bergheaud, V; Cassigneul, A; Chuette, D; Dumény, V; Etiévant, V; Justes, E; Le Gac, AL; Rumpel, C | 1 |
Egecioglu, E; Jerlhag, E; Prieto-Garcia, L; Studer, E; Westberg, L | 2 |
Albertini, KM; Bohidar, AE; Buckley, LE; Buirkle, JM; Stevenson, JR; Young, KA | 1 |
Cunningham, CL; Fidler, TL; Finn, DA; Gomez, JL; Helpenstell, LK; Kosten, TA; Ryabinin, AE; Schuette, LM; Young, EA | 1 |
Belcastro, R; Jankov, RP; Kantores, C; Li, J; Lopez, L; Masood, A; Tanswell, AK; Yi, M | 1 |
Egecioglu, E; Engel, JA; Jerlhag, E; Smith, RG; Svensson, L | 1 |
Engel, JA; Jerlhag, E; Suchankova, P | 1 |
Anderberg, RH; Bergquist, F; Dickson, SL; Fenander, M; Hansson, C; Nissbrandt, H; Richard, JE; Skibicka, KP | 1 |
Havlickova, T; Jerabek, P; Kacer, P; Sustkova-Fiserova, M; Syslova, K | 1 |
Engel, JA; Jerlhag, E; Nylander, I | 1 |
Bartness, TJ; Ryu, V; Thomas, MA | 1 |
Bohidar, AE; Buirkle, JM; Francomacaro, LM; McMahon, EK; O'Bryan, CM; Pesarchick, BF; Stevenson, JR; Young, KA | 1 |
Aschrafi, A; Gioio, A; Kaplan, BB; Kos, A; Martens, GJ; Wanke, KA | 1 |
Bullmore, ET; Dodds, C; Fernando, D; Fletcher, PC; Hosking, LK; Korzeniowska, A; Maltby, K; Miller, SR; Nathan, PJ; Nestor, LJ; Richards, DB; Sarai, BK; Subramaniam, N; Vasist Johnson, L; Warren, L; Waterworth, D; Win, B; Ziauddeen, H | 1 |
Aourz, N; Coppens, J; De Bundel, D; Fehrentz, JA; Martinez, J; Portelli, J; Smolders, I; Walrave, L | 1 |
Desai, A; Gong, T; Lu, P; Wang, M; Zeng, D; Zhang, K | 1 |
Block, GA; Fishbane, S; Locatelli, F; Macdougall, IC | 1 |
Gupta, N; Wish, JB | 1 |
Cao, Z; Fu, W; Gao, F; Liu, W; Wang, H; Xu, B; Zhang, Y; Zhu, H | 1 |
Aparicio, VC; Costa, JL; De Gerónimo, E; Menone, ML; Okada, E; Pérez, DJ | 1 |
de Oliveira, M; Elias, MC; Hoffmann, JF; Lang, GH; Lindemann, IDS; Rombaldi, CV; Vanier, NL | 1 |
Hajnal, A; Horvath, N; Jamis, C; Orellana, ER | 1 |
Cruz, RA; Fernandes, FL; Lacerda, MC; Sediyama, CS; Soares, MA; Tavares, WS; Wilcken, CF; Zanuncio, JC | 1 |
Charalambous, C; Havlickova, T; Jerabek, P; Kacer, P; Lapka, M; Puskina, N; Sustkova-Fiserova, M | 1 |
Ben Haj Salah, K; Fehrentz, JA; Martinez, J; Rodriguez, JA; Wellman, PJ | 1 |
Charalambous, C; Havlickova, T; Jerabek, P; Lapka, M; Puskina, N; Sustkova-Fiserova, M; Syslova, K | 1 |
Maske, CB; Medina, ND; Terrill, SJ; Wall, KD; Williams, DL | 1 |
Gu, J; Jiang, Z; Li, Z; Wu, Y; You, Q; Zhang, X | 1 |
Abtahi, S; Currie, PJ; Howell, E | 1 |
Alfenas, AC; Rodrigues, FÁ; Sant'Anna-Santos, BF; Santos, SAD; Tanaka, FAO; Tuffi-Santos, LD | 1 |
Allard, PM; Chahtane, H; Falquet, J; Ferreira Queiroz, E; Lopez-Molina, L; Marcourt, L; Nogueira Füller, T; Shanmugabalaji, V; Wolfender, JL | 1 |
Charalambous, C; Havlickova, T; Jerabek, P; Lapka, M; Puskina, N; Sustkova-Fiserova, M | 1 |
Anckarsäter, H; Hovey, D; Jerlhag, E; Lichtenstein, P; Lundström, S; Studer, E; Suchankova, P; Vestlund, J; Westberg, L; Winsa-Jörnulf, J | 1 |
Adermark, L; Bergquist, F; Eckernäs, D; Jerlhag, E; Licheri, V; Vestlund, J | 1 |
Ben Haj Salah, K; Buckinx, A; Cottone, E; De Bundel, D; Fehrentz, JA; Kooijman, R; Pierre, A; Smolders, I; Van Den Herrewegen, Y | 1 |
Oliveira, GT; Valgas, AAN; Wilkens, ALL | 1 |
Abtahi, S; Bastacky, JMR; Currie, PJ; Dunn, DP; Gray, CC | 1 |
Castrogiovanni, D; Cornejo, MP; Fehrentz, JA; Marie, J; Perello, M; Reynaldo, M; Schiöth, HB | 1 |
Burade, S; Dhavale, DD; Kumbhar, N; Patil, R; Pawar, SV; Upadhyay, PK | 1 |
Charalambous, C; Havlickova, T; Lapka, M; Pohorala, V; Puskina, N; Sustkova-Fiserova, M; Syslova, K | 1 |
Abizaid, A; Edwards, A; Hay, RE; Hill, MN; Hyland, L; Karatsoreos, I; Klein, M; MacDonald, D | 1 |
Chung, D; Diab, V; Drullinsky, P; Giralt, S; Hassoun, H; Hultcrantz, M; Korde, N; Lahoud, O; Landau, H; Landgren, O; Lendvai, N; Lesokhin, A; Mailankody, S; Mastey, D; Salcedo, M; Schlossman, J; Scordo, M; Shah, G; Shah, U; Smith, E; Werner, K | 1 |
Ashrafi Tafreshi, F; Esfandiari, N; Fatahi, Z; Ghasemi, SF; Taherian, A | 1 |
De Wilde, L; Deventer, K; Roels, K; Van Eenoo, P | 1 |
Almasri, H; Belzunces, LP; Brunet, JL; Cousin, M; Pioz, M; Sené, D; Tavares, DA; Tchamitchian, S | 1 |
Barraja, P; Barreca, M; Galietta, LJV; Genovese, M; Montalbano, A; Raimondi, MV; Spanò, V; Venturini, A | 1 |
Borges-Martins, M; da Silva, PR; Oliveira, GT | 1 |
Prosser, RS; Skanes, B; Warriner, K | 1 |
Charalambous, C; Havlickova, T; Lapka, M; Sustkova-Fiserova, M; Syslova, K | 1 |
Bertrand, M; Boutin, JA; Dupuis, P; Ferry, G; Frankiewicz, L; Galibert, M; Gloanec, P; Jullian, M; Ko, A; Le Diguarher, T; Pecquery, A; Puget, K; Ripoll, L | 1 |
Charalambous, C; Havlickova, T; Kuchar, M; Lapka, M; Puskina, N; Šlamberová, R; Sustkova-Fiserova, M | 1 |
Edvardsson, CE; Jerlhag, E; Vestlund, J | 1 |
Alamil, M; Almasri, H; Belzunces, LP; Brunet, JL; Cousin, M; Diogon, M; Pioz, M; Sené, D; Tavares, DA; Tchamitchian, S | 1 |
Jensen, BL | 1 |
Chuang, TJ; Fuh, MT; Li, SM; Lu, CH; Tsai, HJ; Tsai, SE; Tseng, CC; Wong, FF; Yang, YC | 1 |
de Aguiar Marciano, LP; Lima Brigagão, MRP; Machado Viana, AL; Machado, SC; Martins, I; Rodrigues, MR; Souza Pereira, AF; Souza, BM | 1 |
Alcaraz, MR; Altamirano, GA; Bosquiazzo, VL; Culzoni, MJ; Gomez, AL; Kass, L; Montemurro, M; Muñoz-de-Toro, M; Oddi, SL; Schierano-Marotti, G | 1 |
7 review(s) available for triazoles and glycine
Article | Year |
---|---|
[Dipeptidylpeptidase IV inhibitors and dual action PPAR-agonists].
Topics: Adamantane; Adenosine Deaminase Inhibitors; Diabetes Mellitus, Type 2; Dipeptidyl Peptidase 4; Glycine; Glycoproteins; Humans; Hypoglycemic Agents; Nitriles; Oxazoles; Peroxisome Proliferator-Activated Receptors; Protease Inhibitors; Pyrazines; Pyrrolidines; Sitagliptin Phosphate; Triazoles; Vildagliptin | 2006 |
The 1,2,4-triazole as a scaffold for the design of ghrelin receptor ligands: development of JMV 2959, a potent antagonist.
Topics: Animals; Drug Design; Glycine; Humans; Ligands; Molecular Structure; Receptors, Ghrelin; Triazoles | 2013 |
Hsp90 inhibitors in breast cancer: a systematic review.
Topics: Adenine; Antineoplastic Agents; Benzamides; Benzoquinones; Biomarkers, Tumor; Female; Glycine; HSP70 Heat-Shock Proteins; HSP90 Heat-Shock Proteins; Humans; Indazoles; Isoxazoles; Lactams, Macrocyclic; Pyridines; Resorcinols; Triazoles; Triple Negative Breast Neoplasms | 2013 |
Magic year for multiple myeloma therapeutics: Key takeaways from the ASH 2015 annual meeting.
Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents, Immunological; Boron Compounds; Congresses as Topic; Glycine; Humans; Hydrazines; Molecular Targeted Therapy; Multiple Myeloma; Proteasome Inhibitors; Protein Kinase Inhibitors; Signal Transduction; Thiadiazoles; Treatment Outcome; Triazoles | 2017 |
Targeting Hypoxia-Inducible Factors for the Treatment of Anemia in Chronic Kidney Disease Patients.
Topics: Anemia; Animals; Barbiturates; Blood Pressure; Disease Models, Animal; Drug Design; Drug Interactions; Glycine; Hepcidins; Humans; Hypoxia-Inducible Factor 1; Inflammation; Isoquinolines; Kidney Failure, Chronic; Picolinic Acids; Protein Domains; Pyrazoles; Triazoles | 2017 |
Hypoxia-Inducible Factor Prolyl Hydroxylase Inhibitors: A Potential New Treatment for Anemia in Patients With CKD.
Topics: Anemia; Barbiturates; Clinical Trials as Topic; Enzyme Inhibitors; Erythropoietin; Glycine; Humans; Hypoxia-Inducible Factor-Proline Dioxygenases; Isoquinolines; Pyrazoles; Renal Insufficiency, Chronic; Triazoles | 2017 |
Current development of CFTR potentiators in the last decade.
Topics: Aminophenols; Cystic Fibrosis Transmembrane Conductance Regulator; Glycine; Humans; Mutation; Quinolones; Small Molecule Libraries; Structure-Activity Relationship; Triazoles | 2020 |
2 trial(s) available for triazoles and glycine
Article | Year |
---|---|
Opioid Antagonists and the A118G Polymorphism in the μ-Opioid Receptor Gene: Effects of GSK1521498 and Naltrexone in Healthy Drinkers Stratified by OPRM1 Genotype.
Topics: Adolescent; Adult; Aged; Alanine; Cross-Over Studies; Dose-Response Relationship, Drug; Double-Blind Method; Drinking; Eating; Female; Glycine; Humans; Indans; Male; Middle Aged; Naltrexone; Narcotic Antagonists; Pharmacogenomic Testing; Polymorphism, Single Nucleotide; Receptors, Opioid, mu; Triazoles; Young Adult | 2016 |
Phase I Study of Selinexor, Ixazomib, and Low-dose Dexamethasone in Patients With Relapsed or Refractory Multiple Myeloma.
Topics: Adult; Aged; Antineoplastic Combined Chemotherapy Protocols; Boron Compounds; Dexamethasone; Female; Glycine; Humans; Hydrazines; Male; Middle Aged; Multiple Myeloma; Neoplasm Recurrence, Local; Triazoles | 2020 |
91 other study(ies) available for triazoles and glycine
Article | Year |
---|---|
Platelet-activating factor antagonists limit glycine changes and behavioral deficits after brain trauma.
Topics: Animals; Azepines; Behavior, Animal; Body Water; Brain; Brain Injuries; Cations; Dialysis; Diterpenes; Ginkgolides; Glycine; Lactones; Male; Platelet Activating Factor; Rats; Rats, Sprague-Dawley; Triazoles | 1992 |
Synergistic activity of 5-trifluoromethylthioribose and inhibitors of methionine synthesis against Klebsiella pneumoniae.
Topics: Alkynes; Azaserine; Drug Synergism; Glycine; Klebsiella pneumoniae; Methionine; Pargyline; Thioglycosides; Triazoles | 1991 |
The possible relationship between heme synthesis and mitochondrial biogenesis.
Topics: Acetamides; Acyltransferases; Allyl Compounds; Animals; Carbon Isotopes; Cytochromes; Electron Transport Complex IV; Enzyme Induction; Glycine; Heme; Leucine; Levulinic Acids; Male; Mitochondria, Liver; Rats; Stimulation, Chemical; Succinates; Triazoles; Tritium | 1971 |
The role of heme synthesis during the induction of hepatic microsomal cytochrome P-450 and drug metabolism produced by benzpyrene.
Topics: Acyltransferases; Amino Acids; Animals; Azo Compounds; Benzopyrenes; Carbon Isotopes; Cytochromes; Depression, Chemical; Enzyme Induction; Glycine; Heme; Levulinic Acids; Liver; Male; Microsomes; NADP; Oxidoreductases; Phenobarbital; Rats; Stimulation, Chemical; Time Factors; Transferases; Triazoles | 1969 |
Reversal by serine and potentiation by glycine of the inhibitory effect of 1,2,4-triazole on growth of Salmonella typhimurium.
Topics: Adenine; Amino Acids; Cysteine; Drug Resistance, Microbial; Drug Synergism; Glycine; Homocysteine; Methionine; Mutation; Salmonella typhimurium; Serine; Triazoles | 1967 |
Purine metabolism in wheat shoots treated with aminotriazole.
Topics: Adenine; Adenine Nucleotides; Amines; Carbon Isotopes; Chromatography, Ion Exchange; Chromatography, Paper; Glycine; Guanine; Histidine; Light; Plants; Polynucleotides; Purines; Radiation Effects; Triazoles | 1972 |
3-amino-1,4-triazole, a herbicide affecting chloroplast development.
Topics: Carbon Isotopes; Chloroplasts; Glycine; Herbicides; Mitochondria; Photosynthesis; Seeds; Triazoles | 1972 |
Effect of drugs on heme synthesis in the liver.
Topics: Acyltransferases; Animals; Benzopyrenes; Cytochromes; Depression, Chemical; Glycine; Heme; Lead; Levulinic Acids; Liver; Lyases; Microsomes, Liver; Mitochondria; Oxidoreductases; Phenobarbital; Pyridines; Rats; Stimulation, Chemical; Succinates; Triazoles | 1971 |
The nonerythropoietic component of early bilirubin.
Topics: Amides; Amino Acids; Animals; Bile Ducts; Biliary Fistula; Bilirubin; Carbon Isotopes; Catalase; Cycloheximide; Cytochromes; Erythropoiesis; Glycine; Heme; Infusions, Parenteral; Kidney; Lead Poisoning; Levulinic Acids; Male; Nephrectomy; Phenobarbital; Porphyrins; Protein Biosynthesis; Rats; Triazoles | 1968 |
The enhancement of muscimol-stimulated 36C1 influx by the antispastic 5-aryl-3-(alkylsulfonyl)-4H-1,2,4-triazole (MDL 27,531) in rat brain membrane vesicles.
Topics: Animals; Brain Chemistry; Chloride Channels; Chlorine; Flunitrazepam; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Ion Channel Gating; Male; Membranes; Muscimol; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Triazoles | 1995 |
Significance of glycine 478 in the metabolism of N-benzyl-1-aminobenzotriazole to reactive intermediates by cytochrome P450 2B1.
Topics: Animals; Binding Sites; Chromatography, High Pressure Liquid; Cytochrome P-450 CYP2B1; Glycine; Heme; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Microsomes, Liver; Models, Chemical; Models, Molecular; Mutagenesis, Site-Directed; Rats; Rats, Inbred F344; Rats, Wistar; Triazoles | 1997 |
In vitro studies of cellular and molecular developmental toxicity of adjuvants, herbicides, and fungicides commonly used in Red River Valley, Minnesota.
Topics: 2,4-Dichlorophenoxyacetic Acid; Agrochemicals; Apoptosis; Cell Division; Cell Line; Cell Survival; Congenital Abnormalities; Female; Flow Cytometry; Fungicides, Industrial; Glycine; Glyphosate; Herbicides; Humans; Male; Maneb; Minnesota; Organotin Compounds; Ploidies; Regression Analysis; Surface-Active Agents; Triazoles; Tumor Cells, Cultured; Zineb | 2000 |
The mGlu5 receptor agonist CHPG stimulates striatal glutamate release: possible involvement of A2A receptors.
Topics: Animals; Corpus Striatum; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Male; Microdialysis; Neuroprotective Agents; Phenylacetates; Pyridines; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, Purinergic P1; Triazoles | 2000 |
Suppression of presynaptic responses to adenosine by activation of NMDA receptors.
Topics: Action Potentials; Adenosine; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Baclofen; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; GABA Agonists; Glycine; Hippocampus; In Vitro Techniques; Kainic Acid; Long-Term Potentiation; Male; N-Methylaspartate; Phenethylamines; Presynaptic Terminals; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, N-Methyl-D-Aspartate; Time Factors; Triazines; Triazoles | 2001 |
AMPA receptor-mediated presynaptic inhibition at cerebellar GABAergic synapses: a characterization of molecular mechanisms.
Topics: Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Benzoxazines; Calcium; Calcium Channel Blockers; Cerebellum; Chelating Agents; Colforsin; Cyclopropanes; Drug Interactions; Egtazic Acid; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Morpholines; Naphthalenes; Neural Inhibition; Neurons; Piperidines; Presynaptic Terminals; Pyrazoles; Rats; Rats, Wistar; Receptors, AMPA; Ryanodine; Synapses; Triazines; Triazoles | 2004 |
Permissive role of adenosine A2A receptors on metabotropic glutamate receptor 5 (mGluR5)-mediated effects in the striatum.
Topics: Adenosine; Animals; Carbazoles; Cells, Cultured; Corpus Striatum; Dose-Response Relationship, Drug; Drug Interactions; Electrophysiology; Embryo, Mammalian; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Female; Glycine; In Vitro Techniques; Indoles; Male; Membrane Potentials; N-Methylaspartate; Phenethylamines; Phenylacetates; Pregnancy; Purinergic P1 Receptor Agonists; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Adenosine A2; Receptors, Metabotropic Glutamate; Triazines; Triazoles | 2004 |
Cold-climate vegetative buffer zones as pesticide-filters for surface runoff.
Topics: Adsorption; Cold Climate; Glycine; Glyphosate; Morpholines; Norway; Particle Size; Pesticides; Rain; Seasons; Snow; Triazoles; Water Movements; Water Pollutants, Chemical | 2005 |
Synthesis, solution equilibria and antiproliferative activity of copper(II) aminomethyltriazole and aminomethylthioxotriazoline complexes.
Topics: Cell Proliferation; Cells, Cultured; Chlorides; Crystallography, X-Ray; Glycine; Humans; Hydrogen-Ion Concentration; Lactones; Molecular Structure; Organometallic Compounds; Solubility; Triazoles | 2005 |
Transcriptome profiling, molecular biological, and physiological studies reveal a major role for ethylene in cotton fiber cell elongation.
Topics: Amino Acids, Cyclic; Cell Enlargement; Cell Wall; Cytoskeleton; Ethylenes; Flowers; Gene Expression Profiling; Glycine; Gossypium; Molecular Sequence Data; Oligonucleotide Array Sequence Analysis; Triazoles; Up-Regulation | 2006 |
Novel interrelationship between salicylic acid, abscisic acid, and PIP2-specific phospholipase C in heat acclimation-induced thermotolerance in pea leaves.
Topics: Abscisic Acid; Acclimatization; Anisoles; Antioxidants; Benzoates; Glucosyltransferases; Glycine; Hot Temperature; Models, Biological; Neomycin; Phosphoinositide Phospholipase C; Phosphoric Diester Hydrolases; Pisum sativum; Plant Leaves; Protein Synthesis Inhibitors; Salicylic Acid; Triazoles | 2006 |
Cortisol response to acute stress in jundiá Rhamdia quelen acutely exposed to sub-lethal concentrations of agrichemicals.
Topics: Agrochemicals; Animals; Atrazine; Catfishes; Female; Glycine; Glyphosate; Hydrocortisone; Male; Methyl Parathion; Simazine; Stress, Physiological; Triazoles; Water Pollutants, Chemical | 2008 |
Responsiveness of the interrenal tissue of Jundiá (Rhamdia quelen) to an in vivo ACTH test following acute exposure to sublethal concentrations of agrichemicals.
Topics: Adrenocorticotropic Hormone; Agrochemicals; Animals; Atrazine; Catfishes; Endocrine Disruptors; Female; Glycine; Glyphosate; Hydrocortisone; Hypothalamo-Hypophyseal System; Injections, Intraperitoneal; Interrenal Gland; Male; Methyl Parathion; Pituitary-Adrenal Function Tests; Simazine; Triazoles; Water Pollutants, Chemical | 2009 |
Correlation of receptor occupancy of metabotropic glutamate receptor subtype 1 (mGluR1) in mouse brain with in vivo activity of allosteric mGluR1 antagonists.
Topics: Allosteric Regulation; Animals; Behavior, Animal; Brain; CHO Cells; Cricetinae; Cricetulus; Glycine; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Mice, Knockout; Protein Binding; Receptors, Metabotropic Glutamate; Recombinant Proteins; Resorcinols; Triazoles | 2009 |
Adenosine A2A receptors enable the synaptic effects of cannabinoid CB1 receptors in the rodent striatum.
Topics: Action Potentials; Animals; Benzoxazines; Biophysics; Calcium; Calcium Channel Blockers; Cerebral Cortex; Corpus Striatum; Electric Stimulation; Embryo, Mammalian; Excitatory Amino Acid Agonists; Female; Glycine; In Vitro Techniques; L-Lactate Dehydrogenase; Male; Mice; Mice, Knockout; Morpholines; N-Methylaspartate; Naphthalenes; Neurons; Phenylacetates; Piperidines; Pregnancy; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptors, Adenosine A2; Synapses; Triazines; Triazoles | 2009 |
Use of a high-resolution melt assay to characterize codon 54 of the cyp51A gene of Aspergillus fumigatus on a Rotor-Gene 6000 instrument.
Topics: Antifungal Agents; Aspergillus fumigatus; Codon; Cytochrome P-450 Enzyme System; Drug Resistance, Fungal; Fungal Proteins; Genes, Fungal; Genetic Testing; Glycine; Itraconazole; Microbial Sensitivity Tests; Nucleic Acid Denaturation; Sequence Analysis, DNA; Triazoles | 2010 |
Preparation and preliminary bioevaluation of 99mTc(CO)3-11β-progesterone derivative prepared via click chemistry route.
Topics: Alkynes; Animals; Biological Transport; Cell Line, Tumor; Click Chemistry; Female; Glycine; Humans; Hydroxyprogesterones; Mice; Organotechnetium Compounds; Progesterone; Receptors, Progesterone; Triazoles | 2010 |
Low concentrations of atrazine, glyphosate, 2,4-dichlorophenoxyacetic acid, and triadimefon exposures have diverse effects on Xenopus laevis organ morphogenesis.
Topics: 2,4-Dichlorophenoxyacetic Acid; Animals; Atrazine; Glycine; Glyphosate; Herbicides; Larva; Morphogenesis; Triazoles; Xenopus laevis | 2010 |
Ghrelin receptor (GHS-R1A) antagonism suppresses both operant alcohol self-administration and high alcohol consumption in rats.
Topics: Alcohol Drinking; Alcoholism; Analysis of Variance; Animals; Central Nervous System Depressants; Choice Behavior; Conditioning, Operant; Disease Models, Animal; Ethanol; Glycine; Male; Rats; Rats, Long-Evans; Receptors, Ghrelin; Self Administration; Signal Transduction; Triazoles | 2012 |
Ghrelin receptor antagonism attenuates nicotine-induced locomotor stimulation, accumbal dopamine release and conditioned place preference in mice.
Topics: Animals; Conditioning, Psychological; Dopamine; Dose-Response Relationship, Drug; Glycine; Male; Mice; Microdialysis; Motor Activity; Nicotine; Nicotinic Agonists; Nucleus Accumbens; Receptors, Ghrelin; Triazoles | 2011 |
Effect of pesticides on plant growth promoting traits of greengram-symbiont, Bradyrhizobium sp. strain MRM6.
Topics: Alanine; Bradyrhizobium; Dose-Response Relationship, Drug; Fabaceae; Fungicides, Industrial; Glycine; Glyphosate; Herbicides; Imidazoles; Insecticides; Neonicotinoids; Nitro Compounds; Organothiophosphorus Compounds; Oxazines; Symbiosis; Thiamethoxam; Thiazoles; Triazines; Triazoles | 2011 |
Attenuation of cocaine-induced locomotor sensitization in rats sustaining genetic or pharmacologic antagonism of ghrelin receptors.
Topics: Animals; Behavior, Animal; Cocaine; Dopamine Uptake Inhibitors; Gene Knockout Techniques; Glycine; Locomotion; Male; Motor Activity; Rats; Rats, Sprague-Dawley; Receptors, Ghrelin; Triazoles | 2012 |
Pharmacologic antagonism of ghrelin receptors attenuates development of nicotine induced locomotor sensitization in rats.
Topics: Animals; Glycine; Male; Motor Activity; Nicotine; Rats; Rats, Sprague-Dawley; Receptors, Ghrelin; Triazoles | 2011 |
mGlu5R promotes glutamate AMPA receptor phosphorylation via activation of PKA/DARPP-32 signaling in striatopallidal medium spiny neurons.
Topics: Animals; Corpus Striatum; Cyclic AMP-Dependent Protein Kinases; Dopamine and cAMP-Regulated Phosphoprotein 32; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Neurons; Phosphorylation; Purinergic P1 Receptor Antagonists; Pyridines; Receptor, Adenosine A2A; Receptor, Metabotropic Glutamate 5; Receptors, AMPA; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Metabotropic Glutamate; Resorcinols; Signal Transduction; Triazines; Triazoles | 2013 |
Silver/ThioClickFerrophos-catalyzed enantioselective conjugate addition and cycloaddition of glycine imino ester with nitroalkenes.
Topics: Alkenes; Catalysis; Esters; Ferrous Compounds; Glycine; Imines; Molecular Structure; Nitro Compounds; Organometallic Compounds; Pyrrolidines; Silver; Stereoisomerism; Triazoles | 2012 |
Ghrelin knockout mice show decreased voluntary alcohol consumption and reduced ethanol-induced conditioned place preference.
Topics: Alcohol Drinking; Animals; Conditioning, Operant; Ethanol; Ghrelin; Glycine; Locomotion; Mice; Mice, Inbred C57BL; Mice, Knockout; Receptors, Ghrelin; Structure-Activity Relationship; Triazoles | 2013 |
Adsorption and desorption behavior of selected pesticides as influenced by decomposition of maize mulch.
Topics: Acetamides; Adsorption; Climate; Environmental Exposure; Environmental Monitoring; Epoxy Compounds; Fungicides, Industrial; Glycine; Glyphosate; Herbicides; Light; Magnetic Resonance Spectroscopy; Models, Chemical; Plant Stems; Rain; Soil Pollutants; Triazoles; Zea mays | 2013 |
Ghrelin receptor (GHS-R1A) antagonism suppresses both alcohol consumption and the alcohol deprivation effect in rats following long-term voluntary alcohol consumption.
Topics: Administration, Oral; Alcohol Drinking; Alcoholism; Animals; CpG Islands; DNA Methylation; Gene Expression Regulation; Ghrelin; Glycine; Male; Rats; Rats, Wistar; Receptors, Ghrelin; Self Administration; Signal Transduction; Substance Withdrawal Syndrome; Triazoles; Ventral Tegmental Area | 2013 |
Ghrelin receptor antagonism of morphine-induced accumbens dopamine release and behavioral stimulation in rats.
Topics: 3,4-Dihydroxyphenylacetic Acid; Analgesics, Opioid; Animals; Behavior, Animal; Dopamine; Dose-Response Relationship, Drug; Ghrelin; Glycine; Homovanillic Acid; Male; Microdialysis; Morphine; Nucleus Accumbens; Rats; Rats, Wistar; Receptors, Ghrelin; Reward; Stereotyped Behavior; Triazoles | 2014 |
The effects of ghrelin antagonists [D-Lys(3) ]-GHRP-6 or JMV2959 on ethanol, water, and food intake in C57BL/6J mice.
Topics: Alcohol Drinking; Animals; Drinking; Eating; Ethanol; Glycine; Male; Mice; Mice, Inbred C57BL; Oligopeptides; Random Allocation; Receptors, Ghrelin; Treatment Outcome; Triazoles | 2014 |
Nature and decomposition degree of cover crops influence pesticide sorption: quantification and modelling.
Topics: Acetamides; Adsorption; Carbon Isotopes; Crops, Agricultural; Epoxy Compounds; Glycine; Glyphosate; Magnetic Resonance Spectroscopy; Models, Chemical; Pesticides; Soil Pollutants; Time Factors; Triazoles | 2015 |
The role of ghrelin signalling for sexual behaviour in male mice.
Topics: 5-Hydroxytryptophan; Analysis of Variance; Animals; Central Nervous System Agents; Conditioning, Psychological; Dopamine Agents; Female; Ghrelin; Glycine; Levodopa; Male; Mating Preference, Animal; Mice; Mice, Knockout; Motivation; Reaction Time; Receptors, Ghrelin; Sexual Behavior, Animal; Signal Transduction; Triazoles | 2016 |
GHS-R1A antagonism reduces alcohol but not sucrose preference in prairie voles.
Topics: Alcohol Drinking; Animals; Arvicolinae; Choice Behavior; Dose-Response Relationship, Drug; Drinking; Drinking Behavior; Ethanol; Female; Food Preferences; Glycine; Receptors, Ghrelin; Self Administration; Sucrose; Triazoles | 2015 |
Differential effects of ghrelin antagonists on alcohol drinking and reinforcement in mouse and rat models of alcohol dependence.
Topics: Alcohol Drinking; Alcoholism; Animals; Central Nervous System Agents; Conditioning, Operant; Disease Models, Animal; Dose-Response Relationship, Drug; Ethanol; Food Preferences; Ghrelin; Glycine; Male; Mice, Inbred C57BL; Random Allocation; Rats, Wistar; Receptors, Ghrelin; Reinforcement, Psychology; Self Administration; Triazoles | 2015 |
Neutrophil elastase-induced elastin degradation mediates macrophage influx and lung injury in 60% O2-exposed neonatal rats.
Topics: Animals; Animals, Newborn; Cell Movement; Elafin; Elastin; Female; Glycine; Leukocyte Elastase; Lung; Lung Injury; Macrophages; Maternal Exposure; Neutrophils; Oxygen; Peroxynitrous Acid; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptors, Interleukin-8B; Sulfonamides; Triazoles; Vascular Remodeling | 2015 |
Blockade of growth hormone secretagogue receptor 1A signaling by JMV 2959 attenuates the NMDAR antagonist, phencyclidine-induced impairments in prepulse inhibition.
Topics: Animals; Dose-Response Relationship, Drug; Glycine; Male; Phencyclidine; Prepulse Inhibition; Rats; Rats, Sprague-Dawley; Receptors, Ghrelin; Receptors, N-Methyl-D-Aspartate; Reflex, Startle; Schizophrenia; Sensory Gating; Signal Transduction; Triazoles | 2015 |
Sub-chronic Ghrelin Receptor Blockade Attenuates Alcohol- and Amphetamine-Induced Locomotor Stimulation in Mice.
Topics: Amphetamine; Animals; Central Nervous System Stimulants; Ethanol; Glycine; Locomotion; Male; Mice; Nucleus Accumbens; Receptors, Ghrelin; Triazoles; Ventral Tegmental Area | 2016 |
Ghrelin and GHS-R1A signaling within the ventral and laterodorsal tegmental area regulate sexual behavior in sexually naïve male mice.
Topics: Animals; Ghrelin; Glycine; Male; Mice; Receptors, Ghrelin; Reward; Sexual Behavior, Animal; Signal Transduction; Triazoles; Ventral Tegmental Area | 2015 |
The Stomach-Derived Hormone Ghrelin Increases Impulsive Behavior.
Topics: Animals; Corpus Striatum; Delay Discounting; Dopamine; Ghrelin; Glycine; Impulsive Behavior; Male; Motor Activity; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Receptors, Ghrelin; Reward; RNA, Messenger; Triazoles; Ventral Tegmental Area | 2016 |
Ghrelin and endocannabinoids participation in morphine-induced effects in the rat nucleus accumbens.
Topics: Animals; Arachidonic Acids; Dose-Response Relationship, Drug; Endocannabinoids; Extracellular Space; Ghrelin; Glycerides; Glycine; Male; Morphine; Narcotics; Nucleus Accumbens; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptors, Ghrelin; Receptors, Somatotropin; Stereotyped Behavior; Triazoles | 2016 |
A ghrelin receptor (GHS-R1A) antagonist attenuates the rewarding properties of morphine and increases opioid peptide levels in reward areas in mice.
Topics: Analgesics, Opioid; Animals; Brain; Conditioning, Operant; Dopamine; Dynorphins; Endorphins; Extracellular Fluid; Glycine; Male; Mice; Microdialysis; Morphine; Motor Activity; Opioid Peptides; Receptors, Ghrelin; Reward; Triazoles | 2015 |
Central ghrelin increases food foraging/hoarding that is blocked by GHSR antagonism and attenuates hypothalamic paraventricular nucleus neuronal activation.
Topics: Animals; Appetitive Behavior; Consummatory Behavior; Eating; Feeding Behavior; Food Deprivation; Ghrelin; Glycine; Injections, Intraperitoneal; Injections, Intraventricular; Male; Paraventricular Hypothalamic Nucleus; Phodopus; Proto-Oncogene Proteins c-fos; Receptors, Ghrelin; Time Factors; Triazoles | 2016 |
Ghrelin receptor (GHS-R1A) antagonism alters preference for ethanol and sucrose in a concentration-dependent manner in prairie voles.
Topics: Animals; Arvicolinae; Central Nervous System Agents; Choice Behavior; Dietary Sucrose; Dose-Response Relationship, Drug; Drinking Behavior; Drinking Water; Ethanol; Female; Follow-Up Studies; Glycine; Random Allocation; Receptors, Ghrelin; Taste Perception; Triazoles | 2016 |
Monitoring mRNA Translation in Neuronal Processes Using Fluorescent Non-Canonical Amino Acid Tagging.
Topics: Alanine; Alkynes; Amino Acids; Animals; Axons; Azides; Cerebral Cortex; Click Chemistry; Dendrites; Disks Large Homolog 4 Protein; Embryo, Mammalian; Fluorescent Dyes; Glycine; Intracellular Signaling Peptides and Proteins; Lab-On-A-Chip Devices; Membrane Proteins; Neurons; Primary Cell Culture; Protein Biosynthesis; Rats, Wistar; RNA, Messenger; Triazoles | 2016 |
Anticonvulsant effect of a ghrelin receptor agonist in 6Hz corneally kindled mice.
Topics: Animals; Anticonvulsants; Cornea; Disease Models, Animal; Electric Stimulation; Glycine; Indoles; Kindling, Neurologic; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Oligopeptides; Receptors, Ghrelin; Status Epilepticus; Triazoles; Tryptophan | 2016 |
A High Strength Self-Healable Antibacterial and Anti-Inflammatory Supramolecular Polymer Hydrogel.
Topics: Animals; Anti-Bacterial Agents; Anti-Inflammatory Agents; Bacteria; Cell Survival; Glycine; Hydrogel, Polyethylene Glycol Dimethacrylate; Male; Mice; Polymers; Triazoles | 2017 |
Spatial and temporal trends and flow dynamics of glyphosate and other pesticides within an agricultural watershed in Argentina.
Topics: Argentina; Atrazine; Crops, Agricultural; Environmental Monitoring; Geologic Sediments; Glycine; Glyphosate; Herbicides; Isoxazoles; Neonicotinoids; Nitro Compounds; Organophosphonates; Pesticides; Rain; Rivers; Tetrazoles; Triazoles; Water Movements; Water Pollutants, Chemical | 2017 |
Foliar Desiccators Glyphosate, Carfentrazone, and Paraquat Affect the Technological and Chemical Properties of Cowpea Grains.
Topics: Glycine; Glyphosate; Herbicides; Paraquat; Seeds; Triazoles; Vigna | 2017 |
Effect of vertical sleeve gastrectomy on alcohol consumption and preferences in dietary obese rats and mice: A plausible role for altered ghrelin signaling.
Topics: Alcohol Drinking; Analysis of Variance; Animals; Blood Glucose; Central Nervous System Depressants; Choice Behavior; Diet, High-Fat; Disease Models, Animal; Dose-Response Relationship, Drug; Ethanol; Food Preferences; Gastrectomy; Ghrelin; Glycine; Male; Mice; Mice, Inbred C57BL; Obesity; Rats; Rats, Sprague-Dawley; Signal Transduction; Triazoles | 2018 |
Side-effects of pesticides on the generalist endoparasitoid Palmistichus elaeisis (Hymenoptera: Eulophidae).
Topics: Animals; Benzamides; Diflubenzuron; Female; Glycine; Glycine max; Glyphosate; Herbicides; Hymenoptera; Insecticides; Larva; Lepidoptera; Longevity; Malathion; Male; Plant Leaves; Pupa; Triazoles | 2017 |
Ghrelin receptor antagonism of morphine-induced conditioned place preference and behavioral and accumbens dopaminergic sensitization in rats.
Topics: Analgesics, Opioid; Animals; Conditioning, Operant; Dopamine; Glycine; Male; Microdialysis; Morphine; Nucleus Accumbens; Rats; Rats, Wistar; Receptors, Ghrelin; Triazoles | 2017 |
The GHR-R antagonist JMV 2959 neither induces malaise nor alters the malaise property of LiCl in the adult male rat.
Topics: Animals; Appetite; Avoidance Learning; Conditioning, Psychological; Feeding Behavior; Glycine; Lithium Chloride; Male; Nicotine; Psychotropic Drugs; Random Allocation; Rats, Sprague-Dawley; Receptors, Ghrelin; Reinforcement, Psychology; Saccharin; Sodium, Dietary; Taste Perception; Triazoles | 2018 |
Alterations in Rat Accumbens Endocannabinoid and GABA Content during Fentanyl Treatment: The Role of Ghrelin.
Topics: Animals; Behavior, Animal; Endocannabinoids; Extracellular Space; Fentanyl; gamma-Aminobutyric Acid; Ghrelin; Glycine; Male; Nucleus Accumbens; Rats; Receptors, Ghrelin; Triazoles; Ventral Tegmental Area | 2017 |
Lateral septum growth hormone secretagogue receptor affects food intake and motivation for sucrose reinforcement.
Topics: Animals; Behavior, Animal; Conditioning, Operant; Eating; Food Preferences; Ghrelin; Glycine; Hormone Antagonists; Male; Motivation; Oligopeptides; Rats, Wistar; Receptors, Ghrelin; Reinforcement, Psychology; Septal Nuclei; Signal Transduction; Sucrose; Time Factors; Triazoles | 2018 |
Click Chemistry-Based Discovery of [3-Hydroxy-5-(1 H-1,2,3-triazol-4-yl)picolinoyl]glycines as Orally Active Hypoxia-Inducing Factor Prolyl Hydroxylase Inhibitors with Favorable Safety Profiles for the Treatment of Anemia.
Topics: Administration, Oral; Anemia; Animals; Cisplatin; Click Chemistry; Erythropoietin; Female; Fluorescence Polarization; Glycine; Hemoglobins; Humans; Hypoxia-Inducible Factor-Proline Dioxygenases; Male; Mice, Inbred C57BL; Molecular Docking Simulation; Prolyl-Hydroxylase Inhibitors; Rats, Sprague-Dawley; Structure-Activity Relationship; Triazoles | 2018 |
Accumbal ghrelin and glucagon-like peptide 1 signaling in alcohol reward in female rats.
Topics: Alcohol Drinking; Animals; Ethanol; Female; Ghrelin; Glucagon-Like Peptide 1; Glycine; Microinjections; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Reward; Signal Transduction; Triazoles | 2018 |
Carfentrazone-ethyl and glyphosate drift inhibits uredinial formation of Austropuccinia psidii on Eucalyptus grandis leaves.
Topics: Basidiomycota; Eucalyptus; Glycine; Glyphosate; Herbicides; Plant Diseases; Plant Leaves; Triazoles | 2019 |
The plant pathogen
Topics: Abscisic Acid; Aminobutyrates; Antibody Specificity; Arabidopsis; Arabidopsis Proteins; Discriminant Analysis; Gene Expression Regulation, Plant; Germination; Gibberellins; Glycine; Least-Squares Analysis; Metabolomics; Pseudomonas aeruginosa; Seeds; Signal Transduction; Triazoles | 2018 |
Ghrelin Receptor Antagonism of Methamphetamine-Induced Conditioned Place Preference and Intravenous Self-Administration in Rats.
Topics: Administration, Intravenous; Analysis of Variance; Animals; Body Weight; Central Nervous System Stimulants; Conditioning, Psychological; Glycine; Male; Methamphetamine; Rats, Wistar; Receptors, Ghrelin; Self Administration; Spatial Behavior; Time Factors; Triazoles | 2018 |
Ghrelin and aggressive behaviours-Evidence from preclinical and human genetic studies.
Topics: Adolescent; Aggression; Amygdala; Animals; Dopamine; Ghrelin; Glycine; Humans; Male; Mice; Mice, Inbred C57BL; Receptors, Ghrelin; Secretagogues; Serotonin; Signal Transduction; Triazoles | 2019 |
Ghrelin signalling within the rat nucleus accumbens and skilled reach foraging.
Topics: Animals; Feeding Behavior; Ghrelin; Glycine; Male; Nucleus Accumbens; Rats; Rats, Wistar; Receptors, Ghrelin; Signal Transduction; Triazoles; Ventral Tegmental Area | 2019 |
Differential Effects of a Full and Biased Ghrelin Receptor Agonist in a Mouse Kindling Model.
Topics: Animals; Benzazepines; beta-Arrestins; Brain; Dopamine Agonists; Glycine; Indoles; Kindling, Neurologic; Male; Mice; Mice, Inbred C57BL; Piperidines; Quinazolinones; Receptors, Ghrelin; Triazoles; Tryptophan | 2019 |
Effects of ecologically relevant concentrations of Boral® 500 SC, Glifosato® Biocarb, and a blend of both herbicides on markers of metabolism, stress, and nutritional condition factors in bullfrog tadpoles.
Topics: Animals; Biomarkers; Dose-Response Relationship, Drug; Glycine; Glyphosate; Herbicides; Larva; Liver; Muscles; Oxidative Stress; Rana catesbeiana; Sulfonamides; Triazoles; Water Pollutants, Chemical | 2019 |
Role of mesolimbic ghrelin in the acquisition of cocaine reward.
Topics: Animals; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Synergism; Ghrelin; Glycine; Injections, Intraventricular; Male; Nucleus Accumbens; Rats; Rats, Sprague-Dawley; Reward; Triazoles; Ventral Tegmental Area | 2019 |
Growth hormone secretagogue receptor signalling affects high-fat intake independently of plasma levels of ghrelin and LEAP2, in a 4-day binge eating model.
Topics: Animals; Antimicrobial Cationic Peptides; Bulimia; Diet, High-Fat; Ghrelin; Glycine; Infusions, Intraventricular; Male; Mice; Oligopeptides; Receptors, Ghrelin; Time Factors; Triazoles | 2019 |
Synthesis and anti-leishmanial activity of TRIS-glycine-β-alanine dipeptidic triazole dendron coated with nonameric mannoside glycocluster.
Topics: Antiprotozoal Agents; beta-Alanine; Chemistry Techniques, Synthetic; Dendrimers; Dipeptides; Glycine; Leishmania; Mannosides; Metalloendopeptidases; Molecular Docking Simulation; Molecular Dynamics Simulation; Protein Conformation; Triazoles | 2019 |
Ghrelin receptor antagonism of fentanyl-induced conditioned place preference, intravenous self-administration, and dopamine release in the nucleus accumbens in rats.
Topics: Administration, Intravenous; Animals; Conditioning, Operant; Dopamine; Fentanyl; Ghrelin; Glycine; Male; Narcotics; Nucleus Accumbens; Rats; Rats, Wistar; Receptors, Ghrelin; Self Administration; Triazoles | 2020 |
Ghrelin Receptor Signaling Is Not Required for Glucocorticoid-Induced Obesity in Male Mice.
Topics: Adiposity; Animals; Eating; Glucocorticoids; Glycine; Hippocampus; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Obesity; Prefrontal Cortex; Receptors, Ghrelin; Triazoles; Weight Gain | 2020 |
Ultrasensitive fluorescent detection of pesticides in real sample by using green carbon dots.
Topics: Carbon; Diazinon; Environmental Monitoring; Food Contamination; Glycine; Glyphosate; Limit of Detection; Pesticides; Quantum Dots; Solanum lycopersicum; Spectrometry, Fluorescence; Triazoles | 2020 |
Automated sample preparation for the detection and confirmation of hypoxia-inducible factor stabilizers in urine.
Topics: Chromatography, Liquid; Doping in Sports; Glycine; Humans; Hypoxia-Inducible Factor 1; Isoquinolines; Limit of Detection; Linear Models; Pyrazoles; Reproducibility of Results; Solid Phase Extraction; Substance Abuse Detection; Tandem Mass Spectrometry; Triazoles | 2021 |
Mixtures of an insecticide, a fungicide and a herbicide induce high toxicities and systemic physiological disturbances in winter Apis mellifera honey bees.
Topics: Animals; Bees; Dioxolanes; Drug Synergism; Fungicides, Industrial; Glycine; Glyphosate; Herbicides; Insecticides; Neonicotinoids; Nitro Compounds; Pesticides; Pollination; Triazoles | 2020 |
Melanophryniscus admirabilis tadpoles' responses to sulfentrazone and glyphosate-based herbicides: an approach on metabolism and antioxidant defenses.
Topics: Animals; Antioxidants; Brazil; Glycine; Glyphosate; Herbicides; Larva; Sulfonamides; Triazoles | 2021 |
Hazard assessment using an in-silico toxicity assessment of the transformation products of boscalid, pyraclostrobin, fenbuconazole and glyphosate generated by exposure to an advanced oxidative process.
Topics: Animals; Biphenyl Compounds; Computer Simulation; Decision Trees; Dietary Exposure; Fruit; Fungicides, Industrial; Glycine; Glyphosate; Herbicides; Niacinamide; Nitriles; Oxidation-Reduction; Quantitative Structure-Activity Relationship; Rats; Risk Assessment; Software; Strobilurins; Toxicity Tests; Triazoles; Vegetables | 2021 |
Alterations in Rat Accumbens Dopamine, Endocannabinoids and GABA Content During WIN55,212-2 Treatment: The Role of Ghrelin.
Topics: Animals; Arachidonic Acids; Benzoxazines; Dopamine; Drug Evaluation, Preclinical; Endocannabinoids; gamma-Aminobutyric Acid; Ghrelin; Glycerides; Glycine; Male; Morpholines; Naphthalenes; Nucleus Accumbens; Polyunsaturated Alkamides; Rats, Wistar; Triazoles | 2020 |
MCH-R1 Antagonist GPS18169, a Pseudopeptide, Is a Peripheral Anti-Obesity Agent in Mice.
Topics: Adipose Tissue; Alkynes; Aminobutyrates; Animals; Anti-Obesity Agents; Appetite; Aspartic Acid; Disease Models, Animal; Drug Discovery; Glutamic Acid; Glycine; HEK293 Cells; Hepatocytes; Homeostasis; Humans; Insulin; Lactams; Male; Mice; Mice, Inbred C57BL; Obesity; Rats; Receptors, Pituitary Hormone; Structure-Activity Relationship; Tissue Distribution; Triazoles | 2021 |
Cannabinoid-Induced Conditioned Place Preference, Intravenous Self-Administration, and Behavioral Stimulation Influenced by Ghrelin Receptor Antagonism in Rats.
Topics: Administration, Intravenous; Animals; Behavior, Animal; Cannabinoids; Conditioning, Operant; Conditioning, Psychological; Glycine; Male; Rats; Rats, Wistar; Receptors, Ghrelin; Reinforcement, Psychology; Self Administration; Triazoles | 2021 |
A ghrelin receptor antagonist reduces the ability of ghrelin, alcohol or amphetamine to induce a dopamine release in the ventral tegmental area and in nucleus accumbens shell in rats.
Topics: Amphetamine; Animals; Behavior, Animal; Dopamine; Ethanol; Ghrelin; Glycine; Hormone Antagonists; Locomotion; Male; Mice; Nucleus Accumbens; Rats, Wistar; Receptors, Dopamine D1; Receptors, Ghrelin; Reward; Triazoles; Ventral Tegmental Area | 2021 |
Physiological effects of the interaction between Nosema ceranae and sequential and overlapping exposure to glyphosate and difenoconazole in the honey bee Apis mellifera.
Topics: Animals; Bees; Dioxolanes; Fungicides, Industrial; Glycine; Glyphosate; Herbicides; Nosema; Pesticides; Triazoles | 2021 |
Get use to the -dustats: Roxadustat and molidustat, members of the hypoxia-inducible factor (HIF) prolyl hydroxylase (PHD) inhibitor drug class promote kidney function, perfusion and oxygenation in rats through nitric oxide.
Topics: Animals; Glycine; Hypoxia; Isoquinolines; Kidney; Nitric Oxide; Perfusion; Pharmaceutical Preparations; Prolyl Hydroxylases; Prolyl-Hydroxylase Inhibitors; Pyrazoles; Rats; Triazoles | 2021 |
Design, synthesis and biological evaluation of glycolamide, glycinamide, and β-amino carbonyl 1,2,4-triazole derivatives as DPP-4 inhibitors.
Topics: Dipeptidyl Peptidase 4; Dipeptidyl-Peptidase IV Inhibitors; Dose-Response Relationship, Drug; Drug Design; Glycine; Glycolates; Humans; Molecular Structure; Structure-Activity Relationship; Triazoles | 2021 |
Endpoints as human biomarkers in exposure assessment of triazoles fungicides.
Topics: Adult; Androstenedione; Bile Acids and Salts; Biological Monitoring; Biomarkers; Endocrine Disruptors; Fungicides, Industrial; Glycine; Humans; Middle Aged; Occupational Exposure; Oxidative Stress; Rural Population; Testosterone; Triazoles; Urban Population | 2021 |
Mammary gland development in male rats perinatally exposed to propiconazole, glyphosate, or their mixture.
Topics: Animals; Female; Glycine; Glyphosate; Humans; Hyperplasia; Male; Mammary Glands, Animal; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Triazoles | 2023 |