Page last updated: 2024-08-24

triazoles and geldanamycin

triazoles has been researched along with geldanamycin in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (80.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Cicero, G; Gorska, M; Knap, N; Kuban-Jankowska, A; Popowska, U; Sawczuk, W; Sielicka-Dudzin, A; Wozniak, F1
Anderson, GP; Asselin-Labat, ML; Bozinovski, S; Burns, CJ; Donald, A; Dousha, L; Lilja, A; McArthur, K; Nguyen, T; Vlahos, R; Weeden, CE; Wong, ZX1
Alarcon, S; Beebe, K; Khamit-Kush, K; Kijima, T; Lee, S; Neckers, L; Prince, TL; Rivas, C; Schwartz, H; Scroggins, BT; Tatokoro, M; Trepel, JB; Tsutsumi, S; Yim, K1
Badali, H; Chowdhary, A; Daie Ghazvini, R; Diba, K; Foroumadi, A; Hashemi, SJ; Khodavaisy, S; Mahmoudi, S; Meis, JF; Rezaie, S1
Alzebari, AM; Bartl, F; Bohusz, W; Buczkowski, A; Gdaniec, M; Leśniewska, A; Nowak, E; Przybylski, P; Ruszkowski, P; Skrzypczak, N; Tokarska, K1

Reviews

1 review(s) available for triazoles and geldanamycin

ArticleYear
Geldanamycin and its derivatives as Hsp90 inhibitors.
    Frontiers in bioscience (Landmark edition), 2012, 06-01, Volume: 17, Issue:6

    Topics: Animals; Antineoplastic Agents; Benzoquinones; Cyclin-Dependent Kinases; HSP90 Heat-Shock Proteins; Humans; Indoles; Lactams, Macrocyclic; Macrolides; Models, Biological; Mutation; Novobiocin; Proto-Oncogene Proteins c-raf; src-Family Kinases; Transforming Growth Factor beta; Triazoles; Tumor Suppressor Protein p53

2012

Other Studies

4 other study(ies) available for triazoles and geldanamycin

ArticleYear
HSP90 inhibition suppresses lipopolysaccharide-induced lung inflammation in vivo.
    PloS one, 2015, Volume: 10, Issue:1

    Topics: Animals; B-Lymphocytes; Benzoquinones; Cytokines; HSP90 Heat-Shock Proteins; Inflammation; Killer Cells, Natural; Lactams, Macrocyclic; Lipopolysaccharides; Lung; Male; Matrix Metalloproteinase 9; Mice; Mice, Inbred BALB C; Neutrophils; Triazoles

2015
Client Proteins and Small Molecule Inhibitors Display Distinct Binding Preferences for Constitutive and Stress-Induced HSP90 Isoforms and Their Conformationally Restricted Mutants.
    PloS one, 2015, Volume: 10, Issue:10

    Topics: Adenosine Triphosphate; Amino Acid Sequence; Benzoquinones; Binding Sites; DNA-Binding Proteins; GTP-Binding Proteins; Heat Shock Transcription Factors; HEK293 Cells; HSP90 Heat-Shock Proteins; Humans; Hypoxia-Inducible Factor 1, alpha Subunit; Intracellular Signaling Peptides and Proteins; Kelch-Like ECH-Associated Protein 1; Lactams, Macrocyclic; Molecular Sequence Data; Mutation; Protein Binding; Protein Conformation; Protein Isoforms; Protein Kinase Inhibitors; Receptor, ErbB-2; Transcription Factors; Triazoles; Tumor Suppressor Proteins

2015
In Vitro Interaction of Geldanamycin with Triazoles and Echinocandins Against Common and Emerging Candida Species.
    Mycopathologia, 2019, Volume: 184, Issue:5

    Topics: Antifungal Agents; Benzoquinones; Candida; Drug Interactions; Echinocandins; Lactams, Macrocyclic; Microbial Sensitivity Tests; Triazoles

2019
Modifications of geldanamycin via CuAAC altering affinity to chaperone protein Hsp90 and cytotoxicity.
    European journal of medicinal chemistry, 2023, Aug-05, Volume: 256

    Topics: Alkynes; Antineoplastic Agents; Azides; Benzoquinones; HSP90 Heat-Shock Proteins; Structure-Activity Relationship; Triazoles

2023