triazoles has been researched along with flunitrazepam in 16 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (18.75) | 18.7374 |
1990's | 12 (75.00) | 18.2507 |
2000's | 1 (6.25) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Beer, B; Benson, DI; Klepner, CA; Lippa, AS; Sano, MC | 1 |
Barbaz, BS; Bernard, PS; Braunwalder, AF; Cash, WD; Francis, JE; Friedmann, RC; Hyun, JL; Loo, PS; Lovell, RA; Mazzenga, GC | 1 |
Kabuto, M; Namura, I; Saitoh, Y | 1 |
Beer, B; Lippa, AS; Meyerson, LR | 1 |
Catarzi, D; Cecchi, L; Colotta, V; Giusti, L; Lucacchini, A; Martini, C; Valle, G | 1 |
Catarzi, D; Cecchi, L; Colotta, V; Filacchioni, G; Giusti, L; Lucacchini, A; Martini, C; Melani, F | 2 |
Bain, C; Wafford, KA; Whiting, PJ; Wingrove, PB | 1 |
Biagi, G; Giorgi, I; Livi, O; Lucacchini, A; Martini, C; Scartoni, V | 1 |
Ambrogi, V; Giusti, L; Grandolini, G; Lucacchini, A; Martini, C; Perioli, L | 1 |
Barton, JM; Olson, MS; Svetlov, SI | 1 |
Biggio, G; Ghiani, CA; Maciocco, E; Sanna, E; Serra, M; Tuligi, G | 1 |
Friend, JM; Gee, KW; Xue, BG | 1 |
Braun, D; Chmielewski, PA; Kane, JM; Miller, JA | 1 |
Simmonds, MA; Zhong, Y | 1 |
Bostwick, R; Chen, T; Huston, J; Knappenberger, K; Liu, J; Norris, T; Wood, M | 1 |
1 review(s) available for triazoles and flunitrazepam
Article | Year |
---|---|
Molecular substrates of anxiety: clues from the heterogeneity of benzodiazepine receptors.
Topics: Aging; Animals; Anxiety; Benzodiazepines; Binding, Competitive; Brain; Carbolines; Chemical Phenomena; Chemistry, Physical; Flunitrazepam; Humans; Muscles; Pentylenetetrazole; Pyridazines; Receptors, Drug; Receptors, GABA-A; Tissue Distribution; Triazoles | 1982 |
15 other study(ies) available for triazoles and flunitrazepam
Article | Year |
---|---|
Resolution of two biochemically and pharmacologically distinct benzodiazepine receptors.
Topics: Animals; Benzodiazepines; Dose-Response Relationship, Drug; Flunitrazepam; gamma-Aminobutyric Acid; Hippocampus; Male; Membranes; Rats; Receptors, Drug; Synaptosomes; Triazoles | 1979 |
Synthesis and benzodiazepine binding activity of a series of novel [1,2,4]triazolo[1,5-c]quinazolin-5(6H)-ones.
Topics: Animals; Binding, Competitive; Brain; Diazepam; Flunitrazepam; Indicators and Reagents; Molecular Structure; Quinazolines; Rats; Receptors, GABA-A; Structure-Activity Relationship; Triazoles | 1991 |
Nocturnal enhancement of plasma melatonin could be suppressed by benzodiazepines in humans.
Topics: Adult; Benzodiazepines; Circadian Rhythm; Flunitrazepam; Growth Hormone; Humans; Male; Melatonin; Prolactin; Sleep; Triazoles | 1986 |
Tricyclic heteroaromatic systems. 2-Phenyl-1,2,4-triazolo[1,5-c][1,3]benzoxazin-5-one: a novel benzodiazepine receptor ligand.
Topics: Animals; Benzoxazines; Binding, Competitive; Brain; Cattle; Crystallography, X-Ray; Flunitrazepam; In Vitro Techniques; Ligands; Magnetic Resonance Spectroscopy; Oxazines; Receptors, GABA-A; Triazoles | 1994 |
Structure-activity relationships of 1,2,4-triazolo[1,5-a] quinoxalines and their 1-deaza analogues imidazo[1,2-a]quinoxalines at the benzodiazepine receptor.
Topics: Animals; Binding Sites; Binding, Competitive; Brain; Cattle; Flunitrazepam; Imidazoles; In Vitro Techniques; Quinoxalines; Receptors, GABA-A; Structure-Activity Relationship; Triazoles | 1994 |
The modulatory action of loreclezole at the gamma-aminobutyric acid type A receptor is determined by a single amino acid in the beta 2 and beta 3 subunit.
Topics: Allosteric Site; Amino Acid Sequence; Animals; Anticonvulsants; Base Sequence; DNA Primers; DNA, Complementary; Dose-Response Relationship, Drug; Female; Flunitrazepam; gamma-Aminobutyric Acid; Humans; Macromolecular Substances; Molecular Sequence Data; Mutagenesis, Site-Directed; Oocytes; Point Mutation; Polymerase Chain Reaction; Receptors, GABA-A; Recombinant Fusion Proteins; Triazoles; Xenopus | 1994 |
Tricyclic heteroaromatic systems 1,2,4-triazolo[1,5-a]quinoxalines: synthesis and benzodiazepine receptor activity.
Topics: Animals; Binding, Competitive; Cattle; Cerebral Cortex; Chlordiazepoxide; Flunitrazepam; In Vitro Techniques; Quinoxalines; Receptors, GABA-A; Triazoles | 1993 |
Studies on specific inhibition of benzodiazepine receptor binding by some C-benzoyl-1,2,3-triazole derivatives.
Topics: Animals; Binding, Competitive; Cattle; Cerebral Cortex; Chemical Phenomena; Chemistry, Physical; Flunitrazepam; GABA-A Receptor Antagonists; Hydrogen Bonding; In Vitro Techniques; Receptors, GABA-A; Triazoles | 1993 |
Studies on annelated 1,4-benzothiazines and 1,5-benzothiazepines. VII. Synthesis and inhibition of benzodiazepine receptor binding of some 4,5-dihydro-tetrazolo[5,1-d]-1,5-benzothiazepines and 5-phenyl-s-triazolo[3,4-d]-1,5-benzothiazepines.
Topics: Animals; Binding Sites; Binding, Competitive; Brain; Cattle; Flunitrazepam; Receptors, GABA-A; Structure-Activity Relationship; Thiazepines; Triazoles | 1993 |
The specific binding of the platelet-activating factor (PAF) receptor antagonist WEB 2086 and the benzodiazepine flunitrazepam to rat hepatocytes.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Azepines; Benzodiazepinones; Bicuculline; Cells, Cultured; Clonazepam; Convulsants; Flunitrazepam; Kinetics; Liver; Male; Platelet Aggregation Inhibitors; Platelet Membrane Glycoproteins; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Triazoles; Tritium | 1996 |
Biochemical evaluations of the effects of loreclezole and propofol on the GABAA receptor in rat brain.
Topics: Anesthetics; Animals; Anticonvulsants; Brain; Bridged Bicyclo Compounds, Heterocyclic; Diazepam; Flunitrazepam; GABA Modulators; gamma-Aminobutyric Acid; Hypnotics and Sedatives; In Vitro Techniques; Male; Muscimol; Pentobarbital; Pregnanediones; Propofol; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Sulfur Radioisotopes; Triazoles; Tritium | 1996 |
Loreclezole modulates [35S]t-butylbicyclophosphorothionate and [3H]flunitrazepam binding via a distinct site on the GABAA receptor complex.
Topics: Animals; Anticonvulsants; Benzodiazepinones; Binding Sites; Brain; Bridged Bicyclo Compounds, Heterocyclic; Convulsants; Drug Interactions; Flunitrazepam; Male; Rats; Rats, Sprague-Dawley; Receptors, GABA; Triazoles | 1996 |
The enhancement of muscimol-stimulated 36C1 influx by the antispastic 5-aryl-3-(alkylsulfonyl)-4H-1,2,4-triazole (MDL 27,531) in rat brain membrane vesicles.
Topics: Animals; Brain Chemistry; Chloride Channels; Chlorine; Flunitrazepam; GABA Agonists; GABA Modulators; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Ion Channel Gating; Male; Membranes; Muscimol; Radioisotopes; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Triazoles | 1995 |
Interactions between loreclezole, chlormethiazole and pentobarbitone at GABA(A) receptors: functional and binding studies.
Topics: Animals; Anticonvulsants; Bicuculline; Chlormethiazole; Flunitrazepam; In Vitro Techniques; Male; Medulla Oblongata; Pentobarbital; Rats; Rats, Wistar; Receptors, GABA-A; Triazoles | 1997 |
A high-throughput functional assay for characterization of gamma-aminobutyric acid(A) channel modulators using cryopreserved transiently transfected cells.
Topics: Carbolines; Cell Culture Techniques; Cell Line; Cell Membrane; Cryopreservation; Diazepam; DNA; Dose-Response Relationship, Drug; Drug Discovery; Flumazenil; Flunitrazepam; Fluorescent Dyes; Fluorobenzenes; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Humans; Membrane Potentials; Receptors, GABA-A; Reproducibility of Results; Spectrometry, Fluorescence; Transfection; Triazoles; Tritium | 2008 |