triazoles has been researched along with ds 4574 in 12 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 12 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Kurebayashi, Y; Tabuchi, Y | 1 |
Aibara, S; Iwamoto, T; Mori, M; Tsubokawa, M; Tsukada, W | 1 |
Aibara, S; Fujiwara, H; Iwamoto, T; Matsumoto, H; Miwa, T; Mori, M; Moroi, R; Nakayama, K; Tsukada, W; Yokohama, S | 1 |
Furuhama, K; Kawarabayashi, K; Tabuchi, Y | 1 |
Aibara, S; Mori, M; Tsukada, W | 1 |
Furuhama, K; Tabuchi, Y | 2 |
Hakusui, H; Murayama, N; Nakaoka, M; Nomura, H | 2 |
Furuhama, K; Kawarabayashi, K; Komada, T; Tabuchi, Y | 1 |
Kokue, E; Tabuchi, Y; Yamashika, Y | 1 |
Aibara, S; Iwamoto, T; Mori, M; Takamori, H; Tsubokawa, M; Tsukada, W | 1 |
2 trial(s) available for triazoles and ds 4574
Article | Year |
---|---|
Radioimmunoassay for DS-4574, an antiallergic agent: development, evaluation, and application to human plasma samples.
Topics: Adult; Animals; Antibody Specificity; Cross Reactions; Haptens; Humans; Leukotriene Antagonists; Magnetic Resonance Spectroscopy; Male; Ovalbumin; Pyrimidines; Quality Control; Rabbits; Radioimmunoassay; Triazoles | 1994 |
Radioimmunoassay for DS-4574, an anti-allergic agent: development, evaluation and application to human plasma samples.
Topics: Half-Life; Humans; Hypersensitivity; Leukotriene Antagonists; Male; Pyrimidines; Radioimmunoassay; Triazoles | 1995 |
10 other study(ies) available for triazoles and ds 4574
Article | Year |
---|---|
Effect of DS-4574, a novel peptidoleukotriene antagonist with mast cell stabilizing action, on acute gastric lesions and gastric secretion in rats.
Topics: Animals; Anti-Ulcer Agents; Aspirin; Cimetidine; Dose-Response Relationship, Drug; Ethanol; Gastric Acid; Gastric Mucosa; Hydrochloric Acid; Immersion; Leukotriene Antagonists; Male; Mast Cells; Pylorus; Pyrimidines; Rats; Rats, Sprague-Dawley; Restraint, Physical; Stomach Ulcer; Triazoles | 1992 |
Antiallergic activity of 6-(2-cyclohexylethyl)-[1,3,4]thiadiazolo- [3,2-a]-1,2,3-triazolo-[4,5-d]pyrimidin-9(3H)-one (DS-4574) in rats.
Topics: Adrenalectomy; Anaphylaxis; Animals; Capillary Permeability; Histamine; Histamine Release; Hypersensitivity; Leukotriene Antagonists; Lung; Male; Passive Cutaneous Anaphylaxis; Peritoneal Cavity; Pyrimidines; Rats; Rats, Inbred Strains; Serotonin; Time Factors; Triazoles | 1992 |
Synthesis and antiallergy activity of [1,3,4]thiadiazolo[3,2-a]-1,2,3-triazolo[4,5-d]pyrimidin-9(3H)-one derivatives. II. 6-Alkyl- and 6-cycloalkylalkyl derivatives.
Topics: Animals; Female; Guinea Pigs; Hypersensitivity; In Vitro Techniques; Lung; Muscle Contraction; Ovalbumin; Passive Cutaneous Anaphylaxis; Pyrimidines; Rats; Rats, Sprague-Dawley; SRS-A; Thiadiazoles; Triazoles; X-Ray Diffraction | 1992 |
Inhibitory effect of DS-4574, a peptidoleukotriene antagonist with mast cell stabilizing action, on compound 48/80-induced gastric mucosal lesions in rats.
Topics: Acetophenones; Administration, Oral; Animals; Cimetidine; Cromolyn Sodium; Gastric Mucosa; Histamine; Histamine Release; Injections, Intraperitoneal; Injections, Subcutaneous; Leukotriene Antagonists; Male; Mast Cells; p-Methoxy-N-methylphenethylamine; Pyrimidines; Rats; Rats, Sprague-Dawley; Tetrazoles; Triazoles | 1994 |
Inhibitory effect of DS-4574 on leukotriene- or antigen-induced bronchoconstriction in guinea pigs.
Topics: Animals; Antigens; Asthma; Atropine; Bronchoconstriction; Guinea Pigs; Histamine Release; Immunization; Indomethacin; Leukotriene Antagonists; Leukotriene E4; Male; Pyrilamine; Pyrimidines; SRS-A; Triazoles | 1993 |
Protective effect of DS-4574, a peptidoleukotriene receptor antagonist, against endotoxin-induced intestinal injury in rats.
Topics: Animals; Capillary Permeability; Endotoxins; Escherichia coli; Gastrointestinal Hemorrhage; Hematocrit; Intestinal Diseases; Intestinal Mucosa; Leukotriene Antagonists; Lipopolysaccharides; Male; Pyrimidines; Rats; Rats, Sprague-Dawley; Triazoles | 1995 |
Protective effect of DS-4574 on gastric mucosal injury induced by acidified ethanol in rats.
Topics: Acetophenones; Animals; Autacoids; Cell Degranulation; Edema; Ethanol; Gastric Mucosa; Hydrogen-Ion Concentration; Leukotriene Antagonists; Male; Mast Cells; Necrosis; Pyrimidines; Rats; Rats, Sprague-Dawley; Tetrazoles; Triazoles | 1993 |
Inhibitory effect of DS-4574, a mast cell stabilizer with peptidoleukotriene receptor antagonism, on gastric acid secretion in rats.
Topics: Animals; Bucladesine; Carbachol; Fistula; Gastric Acid; H(+)-K(+)-Exchanging ATPase; Histamine; Leukotriene Antagonists; Male; Mast Cells; Pentagastrin; Pyrimidines; Rats; Rats, Sprague-Dawley; Stomach; Triazoles | 1994 |
Antisecretory effect of DS-4574, a mast cell stabilizer with peptidoleukotriene antagonism, on gastric acid secretion in the pig.
Topics: Adenosine Triphosphatases; Animals; Carbachol; Cation Transport Proteins; Female; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Injections, Intramuscular; Leukotriene Antagonists; Male; Pyrimidines; Swine; Swine, Miniature; Tetragastrin; Triazoles | 1994 |
Effects of DS-4574, a new orally active antiallergic agent, in experimental allergic and inflammatory models.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Female; Guinea Pigs; Hypersensitivity; Immunoglobulin E; Male; Mice; Mice, Inbred C57BL; Passive Cutaneous Anaphylaxis; Pyrimidines; Rats; Rats, Inbred Lew; Rats, Sprague-Dawley; Triazoles | 1993 |