Page last updated: 2024-08-24

triazoles and aprepitant

triazoles has been researched along with aprepitant in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's2 (50.00)24.3611
2020's1 (25.00)2.80

Authors

AuthorsStudies
Elipe, MV; Huskey, SE; Zhu, B1
Kast, RE1
Preskorn, SH1
Alluri, RV; Basu, S; Dodd, S; Emami Riedmaier, A; Huckle, JE; Parrott, N; Pepin, XJH1

Reviews

1 review(s) available for triazoles and aprepitant

ArticleYear
Glioblastoma: synergy of growth promotion between CCL5 and NK-1R can be thwarted by blocking CCL5 with miraviroc, an FDA approved anti-HIV drug and blocking NK-1R with aprepitant, an FDA approved anti-nausea drug.
    Journal of clinical pharmacy and therapeutics, 2010, Volume: 35, Issue:6

    Topics: Anti-HIV Agents; Antiemetics; Antineoplastic Agents; Aprepitant; CCR5 Receptor Antagonists; Cyclohexanes; Drug Approval; Drug Interactions; Glioblastoma; Humans; Maraviroc; Mitogen-Activated Protein Kinase 3; Morpholines; Neurokinin-1 Receptor Antagonists; Phosphorylation; Signal Transduction; Triazoles; United States; United States Food and Drug Administration

2010

Other Studies

3 other study(ies) available for triazoles and aprepitant

ArticleYear
Application of LC-NMR for the study of the volatile metabolite of MK-0869, a substance P receptor antagonist.
    Journal of pharmaceutical and biomedical analysis, 2003, Jan-01, Volume: 30, Issue:5

    Topics: Animals; Antiemetics; Aprepitant; Chromatography, Liquid; Cytochrome P-450 Enzyme System; Humans; Isoenzymes; Magnetic Resonance Spectroscopy; Microsomes, Liver; Morpholines; Neurokinin-1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Triazoles

2003
CNS drug development: lessons from the development of ondansetron, aprepitant, ramelteon, varenicline, lorcaserin, and suvorexant. Part I.
    Journal of psychiatric practice, 2014, Volume: 20, Issue:6

    Topics: Aprepitant; Azepines; Benzazepines; Central Nervous System Agents; Drug Discovery; History, 20th Century; History, 21st Century; Humans; Indenes; Morpholines; Neurotransmitter Agents; Ondansetron; Quinoxalines; Triazoles; Varenicline

2014
Understanding Mechanisms of Food Effect and Developing Reliable PBPK Models Using a Middle-out Approach.
    The AAPS journal, 2021, 01-04, Volume: 23, Issue:1

    Topics: Administration, Oral; Aprepitant; Computer Simulation; Drug Liberation; Food-Drug Interactions; Furosemide; Hepatobiliary Elimination; Humans; Intestinal Absorption; Intestinal Elimination; Intestinal Mucosa; Models, Biological; Permeability; Piperazines; Solubility; Triazoles

2021