triazoles has been researched along with 4,5,6,7-tetrabromobenzimidazole in 5 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 3 (60.00) | 29.6817 |
2010's | 2 (40.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Bretner, M; Shugar, D; Szyszka, R; Zastapiło, K; Zień, P | 1 |
Abramczyk, O; Bretner, M; Domańska, K; Szyszka, R; Zień, P | 1 |
Bretner, M; Duncan, JS; Litchfield, DW; Shugar, D; Skierski, J; Zien, P | 1 |
Bilińska-Chomik, A; Bretner, M; Kuś, A; Makowska, M; Wińska, P; Łukowska-Chojnacka, E | 1 |
Bretner, M; Maj, P; Makowska, M; Poznański, J; Shugar, D; Wielechowska, M; Winiewska, M | 1 |
1 review(s) available for triazoles and 4,5,6,7-tetrabromobenzimidazole
Article | Year |
---|---|
Tetrabromobenzotriazole (TBBt) and tetrabromobenzimidazole (TBBz) as selective inhibitors of protein kinase CK2: evaluation of their effects on cells and different molecular forms of human CK2.
Topics: Apoptosis; Benzimidazoles; Casein Kinase II; Cell Membrane Permeability; Cell Proliferation; Evaluation Studies as Topic; HeLa Cells; Humans; Protein Isoforms; Triazoles | 2005 |
4 other study(ies) available for triazoles and 4,5,6,7-tetrabromobenzimidazole
Article | Year |
---|---|
Selectivity of 4,5,6,7-tetrabromobenzimidazole as an ATP-competitive potent inhibitor of protein kinase CK2 from various sources.
Topics: Adenosine Triphosphate; Animals; Benzimidazoles; Binding, Competitive; Candida tropicalis; Casein Kinase II; Enzyme Inhibitors; In Vitro Techniques; Kinetics; Liver; Neurospora crassa; Protein Serine-Threonine Kinases; Rats; Saccharomyces cerevisiae; Triazoles | 2003 |
TBBz but not TBBt discriminates between two molecular forms of CK2 in vivo and its implications.
Topics: Benzimidazoles; Binding, Competitive; Casein Kinase II; Cell Division; Dose-Response Relationship, Drug; Enzyme Activation; Protein Biosynthesis; Protein Serine-Threonine Kinases; Protozoan Proteins; Ribosomal Proteins; Saccharomyces cerevisiae; Structure-Activity Relationship; Triazoles | 2003 |
Design and synthesis of CK2 inhibitors.
Topics: Benzimidazoles; Casein Kinase II; Drug Design; Humans; Inhibitory Concentration 50; Protein Kinase Inhibitors; Triazoles | 2011 |
Thermodynamic parameters for binding of some halogenated inhibitors of human protein kinase CK2.
Topics: Benzimidazoles; Binding Sites; Calorimetry; Calorimetry, Differential Scanning; Casein Kinase II; Drug Design; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Inhibitory Concentration 50; Ligands; Methylation; Microscopy, Fluorescence; Protein Binding; Static Electricity; Temperature; Thermodynamics; Triazoles | 2015 |