Page last updated: 2024-08-24

triazoles and 4,5,6,7-tetrabromobenzimidazole

triazoles has been researched along with 4,5,6,7-tetrabromobenzimidazole in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (60.00)29.6817
2010's2 (40.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bretner, M; Shugar, D; Szyszka, R; Zastapiło, K; Zień, P1
Abramczyk, O; Bretner, M; Domańska, K; Szyszka, R; Zień, P1
Bretner, M; Duncan, JS; Litchfield, DW; Shugar, D; Skierski, J; Zien, P1
Bilińska-Chomik, A; Bretner, M; Kuś, A; Makowska, M; Wińska, P; Łukowska-Chojnacka, E1
Bretner, M; Maj, P; Makowska, M; Poznański, J; Shugar, D; Wielechowska, M; Winiewska, M1

Reviews

1 review(s) available for triazoles and 4,5,6,7-tetrabromobenzimidazole

ArticleYear
Tetrabromobenzotriazole (TBBt) and tetrabromobenzimidazole (TBBz) as selective inhibitors of protein kinase CK2: evaluation of their effects on cells and different molecular forms of human CK2.
    Biochimica et biophysica acta, 2005, Dec-30, Volume: 1754, Issue:1-2

    Topics: Apoptosis; Benzimidazoles; Casein Kinase II; Cell Membrane Permeability; Cell Proliferation; Evaluation Studies as Topic; HeLa Cells; Humans; Protein Isoforms; Triazoles

2005

Other Studies

4 other study(ies) available for triazoles and 4,5,6,7-tetrabromobenzimidazole

ArticleYear
Selectivity of 4,5,6,7-tetrabromobenzimidazole as an ATP-competitive potent inhibitor of protein kinase CK2 from various sources.
    Biochemical and biophysical research communications, 2003, Jun-20, Volume: 306, Issue:1

    Topics: Adenosine Triphosphate; Animals; Benzimidazoles; Binding, Competitive; Candida tropicalis; Casein Kinase II; Enzyme Inhibitors; In Vitro Techniques; Kinetics; Liver; Neurospora crassa; Protein Serine-Threonine Kinases; Rats; Saccharomyces cerevisiae; Triazoles

2003
TBBz but not TBBt discriminates between two molecular forms of CK2 in vivo and its implications.
    Biochemical and biophysical research communications, 2003, Dec-19, Volume: 312, Issue:3

    Topics: Benzimidazoles; Binding, Competitive; Casein Kinase II; Cell Division; Dose-Response Relationship, Drug; Enzyme Activation; Protein Biosynthesis; Protein Serine-Threonine Kinases; Protozoan Proteins; Ribosomal Proteins; Saccharomyces cerevisiae; Structure-Activity Relationship; Triazoles

2003
Design and synthesis of CK2 inhibitors.
    Molecular and cellular biochemistry, 2011, Volume: 356, Issue:1-2

    Topics: Benzimidazoles; Casein Kinase II; Drug Design; Humans; Inhibitory Concentration 50; Protein Kinase Inhibitors; Triazoles

2011
Thermodynamic parameters for binding of some halogenated inhibitors of human protein kinase CK2.
    Biochemical and biophysical research communications, 2015, Jan-02, Volume: 456, Issue:1

    Topics: Benzimidazoles; Binding Sites; Calorimetry; Calorimetry, Differential Scanning; Casein Kinase II; Drug Design; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Inhibitory Concentration 50; Ligands; Methylation; Microscopy, Fluorescence; Protein Binding; Static Electricity; Temperature; Thermodynamics; Triazoles

2015