triazoles has been researched along with 4,5,6,7-tetrabromo-2-azabenzimidazole in 77 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (2.60) | 18.2507 |
2000's | 34 (44.16) | 29.6817 |
2010's | 38 (49.35) | 24.3611 |
2020's | 3 (3.90) | 2.80 |
Authors | Studies |
---|---|
Boguszewska, A; Grankowski, N; Shugar, D; Szyszka, R | 1 |
Chaubet-Gigot, N; Combettes, B; Dot, J; Espunya, MC; Martínez, MC | 1 |
Davies, SP; Donella-Deana, A; Meggio, F; Pinna, LA; Reddy, H; Ruzzene, M; Sarno, S; Shugar, D | 1 |
Battistutta, R; De Moliner, E; Pinna, LA; Sarno, S; Zanotti, G | 1 |
Penzo, D; Pinna, LA; Ruzzene, M | 1 |
Chang, YS; Chi, LM; Yu, JS | 1 |
Bretner, M; Shugar, D; Szyszka, R; Zastapiło, K; Zień, P | 1 |
Abramczyk, O; Bretner, M; Domańska, K; Szyszka, R; Zień, P | 1 |
Camici, G; Gamberi, T; Magherini, F; Marchetta, M; Modesti, A; Pinna, LA; Raugei, G; Sarno, S | 1 |
Dunzendorfer, S; Lee, HK; Tobias, PS | 1 |
Andrzejewska, M; Kazimierczuk, Z; Meggio, F; Pagano, MA; Pinna, LA; Ruzzene, M | 1 |
Intine, RV; Maraia, RJ; Schwartz, EI | 1 |
Blanchette, M; Botchan, MR; Remus, D; Rio, DC | 1 |
Bretner, M; Duncan, JS; Litchfield, DW; Shugar, D; Skierski, J; Zien, P | 1 |
Allende-Vega, N; Dias, S; Meek, D; Milne, D | 1 |
Ahmad, KA; Ahmed, K; Wang, G | 1 |
Maathuis, FJ; Mariani, P; Moscatiello, R; Sanders, D | 1 |
Cai, LF; Erdjument-Bromage, H; Kaufman, AJ; Pandolfi, PP; Scaglioni, PP; Singh, B; Tempst, P; Teruya-Feldstein, J; Yung, TM | 1 |
Ahmed, K; He, H; Pamarthy, D; Sun, Y; Tan, M; Wang, G | 1 |
Leyton, L; Quest, AF; Rodriguez, DA; Tapia, JC; Torres, VA | 1 |
Bieberich, CJ; Guan, B; Hampton, BS; Li, X; Padmanabhan, A; Srivastava, MK | 1 |
Carneiro, AC; Fragel-Madeira, L; Linden, R; Silva-Neto, MA | 1 |
Aldehni, F; Almaça, J; Amaral, MD; Bachhuber, T; Kunzelmann, K; Mehta, A; Schreiber, R | 1 |
Kimura, R; Matsuki, N | 1 |
Boehning, D; Bucci, E; Doré, S; Koehler, RC; Kwansa, H; Qin, X; Shugar, D | 1 |
Bretner, M; Kilanowicz, A; Muszyńska, G; Najda-Bernatowicz, A; Sapota, A; Łebska, M | 1 |
Miyata, Y; Nishida, E | 1 |
Ahmad, KA; Ahmed, K; Harris, NH; Wang, G | 1 |
Bain, J; Cozza, G; Di Maira, G; Elliott, M; Kazimierczuk, Z; Meggio, F; Orzeszko, A; Pagano, MA; Pinna, LA; Ruzzene, M; Sarno, S | 1 |
Duncan, JS; Kerman, K; Kraatz, HB; Litchfield, DW; Song, H | 1 |
Chemnitz, J; Grüttner, C; Hauber, J; Pieper, D | 1 |
Isaeva, AR; Mitev, VI | 2 |
Götz, C; Hessenauer, A; Montenarh, M; Schneider, CC | 3 |
Jenkins, PM; Martens, JR; Thomas, G; Zhang, L | 1 |
Ahmad, KA; Ahmed, K; Hanif, IM; Pervaiz, S | 1 |
Fritz, G; Issinger, OG; Olsen, BB | 1 |
Götz, C; Gratz, A; Jose, J | 1 |
Barata, JT; Brandalise, SR; Jotta, PY; Ribeiro, D; Silva, A; Silveira, AB; Yunes, JA | 1 |
Jang, ER; Kim, W; Kim, YJ; Lee, CS; Myung, SC | 1 |
Ampofo, E; Götz, C; Jakupovic, M; Kietzmann, T; Montenarh, M; Zimmer, A | 1 |
Felczak, K; Poznański, J; Shugar, D; Wasik, R; Łebska, M | 1 |
Bovée, JV; Bruijn, IH; Hogendoorn, PC; Schrage, YM; Szuhai, K; Willems, SM | 1 |
Ahmed, K; Bdzhola, VG; Bretner, M; Golub, AG; Kramerov, AA; Ljubimov, AV; Yarmoluk, SM | 1 |
Debus, J; Ebert, M; Huber, PE; Weber, KJ; Zwicker, F | 1 |
Cala, SE; McFarland, TP; Sleiman, NH; Yaeger, DB | 1 |
Abe, S; Eto, K; Sonoda, Y | 1 |
Bilińska-Chomik, A; Bretner, M; Kuś, A; Makowska, M; Wińska, P; Łukowska-Chojnacka, E | 1 |
Götz, C; Günther, J; Hessenauer, A; Kartarius, S; Montenarh, M; Schneider, CC | 1 |
Kozłowska, E; Orzechowska, E; Staroń, K; Trzcińska-Danielewicz, J | 1 |
Alinger, B; Berr, F; Di Fazio, P; Fuereder, J; Kiesslich, T; Neureiter, D; Oberdanner, C; Ocker, M; Pichler, M; Wachter, J | 1 |
Ahmed, K; Kramerov, AA; Ljubimov, AV | 1 |
Horie, N; Hosoi, T; Korematsu, K; Nomura, Y; Okuma, Y; Ozawa, K; Suezawa, T | 1 |
Anand, M; Armanious, H; Gelebart, P; Lai, R | 1 |
Bretner, M; Gyenis, L; Litchfield, DW; Turowec, JP | 1 |
Cheng, Q; Jia, H; Li, D; Li, L; Zhang, G; Zhao, M; Zhao, T; Zheng, J | 1 |
Beyer, C; Dees, C; Distler, A; Distler, JH; Distler, O; Kreuter, A; Lin, NY; Palumbo, K; Schett, G; Susok, L; Zerr, P; Zhang, Y | 1 |
Chen, H; Chen, SR; Hu, YM; Pan, HL | 1 |
Borowiecki, P; Bretner, M; Wawro, AM; Wielechowska, M; Wińska, P | 1 |
Ahmed, K; Kren, BT; Naveed, AK; Qaiser, F; Trembley, JH; Wu, JJ | 1 |
Chen, L; Fang, L; Hu, Z; Huang, Y; Li, D; Li, H; Li, J; Song, H; Wei, C | 1 |
Bretner, M; Maj, P; Makowska, M; Poznański, J; Shugar, D; Wielechowska, M; Winiewska, M | 1 |
Chen, BC; Lin, CH; Shih, CH | 1 |
Bailey, TD; Bobek, G; Buskila, Y; Johnson, AJ; Kersaitis, C; Kueh, S; Wu, MJ; Zaman, MS | 1 |
Ahmad, F; Dixit, D; Ghildiyal, R; Joshi, SD; Sen, E | 1 |
Gao, Y; Liu, L; Liu, S; Luo, Z; Shi, J; Yu, X; Zhao, B; Zhao, Y | 1 |
Chung, WT; Kim, HY; Lee, SW; Lee, SY; Rho, JH; Yoo, SH; Yoo, YH | 1 |
Jung, I; Koš, M; Kos-Braun, IC | 1 |
Beyreis, M; Helm, K; Jakab, M; Kiesslich, T; Mayr, C; Plaetzer, K; Ritter, M | 1 |
Berman, JM; Mironova, E; Stockand, JD | 1 |
Kim, K; Kim, KM; Park, YC; Sohn, DH | 1 |
He, P; Liu, C; Luan, Z; Song, W; Zhang, X; Zhao, L | 1 |
Adade, CM; Atella, GC; Coelho, FS; Dutra, FL; Lopes, AH; Silva Neto, MAC; Vieira, DP | 1 |
Afzal, M; Ahmed, K; Kren, BT; Naveed, AK; Trembley, JH | 1 |
Aiello, G; Kobeissy, F; Kurup, M; Lin, F; Torres, I; Wang, KK; Yadikar, H; Yang, Z; Yost, R | 1 |
2 review(s) available for triazoles and 4,5,6,7-tetrabromo-2-azabenzimidazole
Article | Year |
---|---|
Tetrabromobenzotriazole (TBBt) and tetrabromobenzimidazole (TBBz) as selective inhibitors of protein kinase CK2: evaluation of their effects on cells and different molecular forms of human CK2.
Topics: Apoptosis; Benzimidazoles; Casein Kinase II; Cell Membrane Permeability; Cell Proliferation; Evaluation Studies as Topic; HeLa Cells; Humans; Protein Isoforms; Triazoles | 2005 |
Chemical proteomics and functional proteomics strategies for protein kinase inhibitor validation and protein kinase substrate identification: applications to protein kinase CK2.
Topics: Adenosine Triphosphate; Casein Kinase II; Humans; Models, Molecular; Protein Binding; Protein Kinase Inhibitors; Protein Kinases; Proteomics; Substrate Specificity; Triazoles | 2013 |
75 other study(ies) available for triazoles and 4,5,6,7-tetrabromo-2-azabenzimidazole
Article | Year |
---|---|
Halogenated benzimidazole inhibitors of phosphorylation, in vitro and in vivo, of the surface acidic proteins of the yeast ribosomal 60S subunit by endogenous protein kinases CK-II and PK60S.
Topics: Benzimidazoles; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Fungal Proteins; Halogens; Peptide Fragments; Phosphorylation; Protein Serine-Threonine Kinases; Ribosomal Proteins; Ribosomes; Saccharomyces cerevisiae; Triazoles | 1996 |
Cell-cycle modulation of CK2 activity in tobacco BY-2 cells.
Topics: Antibody Specificity; Casein Kinase II; Cell Cycle; Cell Cycle Proteins; Cell Line; Gene Expression Regulation, Enzymologic; Gene Expression Regulation, Plant; Nicotiana; Periodicity; Plants, Toxic; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; RNA, Messenger; RNA, Plant; Triazoles | 1999 |
Selectivity of 4,5,6,7-tetrabromobenzotriazole, an ATP site-directed inhibitor of protein kinase CK2 ('casein kinase-2').
Topics: Adenosine Triphosphate; Amino Acid Substitution; Binding Sites; Binding, Competitive; Casein Kinase II; Emodin; Enzyme Inhibitors; Humans; Jurkat Cells; Protein Kinases; Protein Serine-Threonine Kinases; Staurosporine; Substrate Specificity; Triazoles | 2001 |
Structural features underlying selective inhibition of protein kinase CK2 by ATP site-directed tetrabromo-2-benzotriazole.
Topics: Adenosine Triphosphate; Binding Sites; Casein Kinase II; Emodin; Enzyme Inhibitors; Guanosine Triphosphate; Models, Molecular; Protein Serine-Threonine Kinases; Triazoles; Zea mays | 2001 |
Protein kinase CK2 inhibitor 4,5,6,7-tetrabromobenzotriazole (TBB) induces apoptosis and caspase-dependent degradation of haematopoietic lineage cell-specific protein 1 (HS1) in Jurkat cells.
Topics: Adaptor Proteins, Signal Transducing; Apoptosis; Blood Proteins; Casein Kinase II; Caspase 3; Caspases; Cell Death; Cell Survival; Cytochrome c Group; DNA Fragmentation; Dose-Response Relationship, Drug; Enzyme Inhibitors; Etoposide; Humans; Jurkat Cells; Phosphorylation; Poly(ADP-ribose) Polymerases; Precipitin Tests; Protein Binding; Protein Serine-Threonine Kinases; Serine; Threonine; Time Factors; Triazoles; Tyrosine | 2002 |
Identification of protein kinase CK2 as a potent kinase of Epstein-Barr virus latent membrane protein 1.
Topics: Amino Acid Sequence; Casein Kinase II; Enzyme Inhibitors; Humans; Molecular Sequence Data; Phosphorylation; Protein Serine-Threonine Kinases; Substrate Specificity; Triazoles; Tumor Cells, Cultured; Viral Matrix Proteins | 2002 |
Selectivity of 4,5,6,7-tetrabromobenzimidazole as an ATP-competitive potent inhibitor of protein kinase CK2 from various sources.
Topics: Adenosine Triphosphate; Animals; Benzimidazoles; Binding, Competitive; Candida tropicalis; Casein Kinase II; Enzyme Inhibitors; In Vitro Techniques; Kinetics; Liver; Neurospora crassa; Protein Serine-Threonine Kinases; Rats; Saccharomyces cerevisiae; Triazoles | 2003 |
TBBz but not TBBt discriminates between two molecular forms of CK2 in vivo and its implications.
Topics: Benzimidazoles; Binding, Competitive; Casein Kinase II; Cell Division; Dose-Response Relationship, Drug; Enzyme Activation; Protein Biosynthesis; Protein Serine-Threonine Kinases; Protozoan Proteins; Ribosomal Proteins; Saccharomyces cerevisiae; Structure-Activity Relationship; Triazoles | 2003 |
Expression of the Stp1 LMW-PTP and inhibition of protein CK2 display a cooperative effect on immunophilin Fpr3 tyrosine phosphorylation and Saccharomyces cerevisiae growth.
Topics: Casein Kinase II; Cell Cycle; Cell Division; Enzyme Inhibitors; Immunoblotting; Immunophilins; Nuclear Proteins; Phenotype; Phosphorylation; Plasmids; Precipitin Tests; Protein Serine-Threonine Kinases; RNA-Binding Proteins; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Time Factors; Transcription Factors; Triazoles; Tyrosine | 2004 |
Flow-dependent regulation of endothelial Toll-like receptor 2 expression through inhibition of SP1 activity.
Topics: Arteriosclerosis; Carrier Proteins; Casein Kinase II; Cells, Cultured; Coronary Vessels; DNA-Binding Proteins; Endothelial Cells; Endothelium, Vascular; Gene Expression Regulation; Hemorheology; Humans; Lipopeptides; Lipopolysaccharides; Membrane Glycoproteins; Oligopeptides; Phosphorylation; Protein Processing, Post-Translational; Receptors, Cell Surface; Recombinant Proteins; RNA, Messenger; Sp1 Transcription Factor; Sp3 Transcription Factor; Stress, Mechanical; Toll-Like Receptor 2; Toll-Like Receptors; Transcription Factors; Triazoles; Tumor Necrosis Factor-alpha | 2004 |
2-Dimethylamino-4,5,6,7-tetrabromo-1H-benzimidazole: a novel powerful and selective inhibitor of protein kinase CK2.
Topics: Animals; Apoptosis; Benzimidazoles; Casein Kinase II; Casein Kinases; Enzyme Inhibitors; Humans; In Vitro Techniques; Jurkat Cells; Kinetics; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Rats; Triazoles | 2004 |
CK2 is responsible for phosphorylation of human La protein serine-366 and can modulate rpL37 5'-terminal oligopyrimidine mRNA metabolism.
Topics: Alanine; Apoptosis; Autoantigens; Casein Kinase II; Cell Line; Humans; Mutation; Phosphorylation; Phosphoserine; Polyribosomes; Protein Processing, Post-Translational; Pyrimidines; Ribonucleoproteins; Ribosomal Proteins; RNA, Messenger; Serine; SS-B Antigen; Triazoles | 2004 |
CDK phosphorylation inhibits the DNA-binding and ATP-hydrolysis activities of the Drosophila origin recognition complex.
Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Amino Acid Motifs; Animals; Cell Nucleus; Cell Proliferation; Cross-Linking Reagents; Cyclin B; Cyclin E; Cyclin-Dependent Kinases; DNA; DNA Replication; Drosophila melanogaster; Hydrolysis; Immunoprecipitation; Mass Spectrometry; Models, Genetic; Origin Recognition Complex; Phosphorylation; Protein Binding; Protein Kinases; Purines; Silver Staining; Time Factors; Triazoles | 2005 |
Phosphorylation of the acidic domain of Mdm2 by protein kinase CK2.
Topics: Casein Kinase II; Cell Line; Humans; Phosphorylation; Protein Structure, Tertiary; Proto-Oncogene Proteins c-mdm2; Recombinant Fusion Proteins; Serine; Signal Transduction; Triazoles; Tumor Suppressor Protein p53 | 2005 |
Role of protein kinase CK2 in the regulation of tumor necrosis factor-related apoptosis inducing ligand-induced apoptosis in prostate cancer cells.
Topics: Androgens; Apoptosis; Apoptosis Regulatory Proteins; bcl-X Protein; Casein Kinase II; Cell Line, Tumor; Drug Synergism; Humans; Lamin Type A; Male; Membrane Glycoproteins; Mitochondria; Neoplasms, Hormone-Dependent; Prostatic Neoplasms; Proto-Oncogene Proteins c-bcl-2; TNF-Related Apoptosis-Inducing Ligand; Transfection; Triazoles; Tumor Necrosis Factor-alpha | 2006 |
Transcriptional analysis of calcium-dependent and calcium-independent signalling pathways induced by oligogalacturonides.
Topics: Arabidopsis; Arabidopsis Proteins; Calcium; Calcium Signaling; Cells, Cultured; Gene Expression Profiling; Gene Expression Regulation, Plant; Hexuronic Acids; Lanthanum; Oligonucleotide Array Sequence Analysis; Oligosaccharides; RNA, Messenger; Signal Transduction; Triazoles | 2006 |
A CK2-dependent mechanism for degradation of the PML tumor suppressor.
Topics: Amino Acid Sequence; Amino Acid Substitution; Animals; Apoptosis; Carcinoma, Non-Small-Cell Lung; Casein Kinase II; Cell Line; Cell Line, Transformed; Cell Line, Tumor; Enzyme Activation; Enzyme Inhibitors; Genes, Tumor Suppressor; Green Fluorescent Proteins; Hemagglutinins; Humans; Leupeptins; Lung Neoplasms; Mice; Mice, Transgenic; Molecular Sequence Data; Neoplasm Proteins; NIH 3T3 Cells; Nuclear Proteins; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Promyelocytic Leukemia Protein; Proteasome Endopeptidase Complex; Protein Structure, Tertiary; Protein Subunits; RNA, Small Interfering; Sequence Deletion; Serine; Sorbitol; Transcription Factors; Transcriptional Activation; Triazoles; Tumor Suppressor Proteins; Ubiquitin | 2006 |
CK2 phosphorylation of SAG at Thr10 regulates SAG stability, but not its E3 ligase activity.
Topics: Antibodies, Phospho-Specific; Casein Kinase II; Cell Hypoxia; Cobalt; Enzyme Activation; Enzyme Stability; Half-Life; HeLa Cells; Humans; Phosphoproteins; Phosphorylation; Phosphothreonine; Proteasome Inhibitors; Protein Transport; RNA-Binding Proteins; Subcellular Fractions; Thermodynamics; Triazoles; Ubiquitin-Protein Ligases | 2007 |
Casein kinase 2 (CK2) increases survivin expression via enhanced beta-catenin-T cell factor/lymphoid enhancer binding factor-dependent transcription.
Topics: beta Catenin; Casein Kinase II; Cell Line; HT29 Cells; Humans; Inhibitor of Apoptosis Proteins; Lymphoid Enhancer-Binding Factor 1; Microtubule-Associated Proteins; Neoplasm Proteins; Survivin; TCF Transcription Factors; Transcription, Genetic; Triazoles; Up-Regulation | 2006 |
The reverse in-gel kinase assay to profile physiological kinase substrates.
Topics: Acrylic Resins; Animals; Casein Kinase II; Caseins; Catalysis; Cell Extracts; Cell Line, Tumor; Cyclic AMP-Dependent Protein Kinases; Electrophoresis, Gel, Two-Dimensional; Electrophoresis, Polyacrylamide Gel; Humans; Intramolecular Oxidoreductases; Male; Mice; Phosphoric Monoester Hydrolases; Phosphorylation; Prostaglandin-E Synthases; Protein Denaturation; Protein Folding; Protein Kinases; Reproducibility of Results; Seminal Vesicles; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Triazoles | 2007 |
A role for CK2 upon interkinetic nuclear migration in the cell cycle of retinal progenitor cells.
Topics: Animals; Animals, Newborn; Antimetabolites; Blotting, Western; Bromodeoxyuridine; Casein Kinase II; Cell Cycle; Cell Nucleus; Cytoskeleton; Fluorescent Antibody Technique; Immunohistochemistry; Nucleotides; Rats; Retina; Stem Cells; Triazoles; Tubulin | 2008 |
Regulation of the epithelial Na+ channel by the protein kinase CK2.
Topics: Animals; Casein Kinase II; Cell Membrane; Electrophysiology; Enzyme Activation; Epithelial Cells; Epithelial Sodium Channels; Female; Mice; Mice, Inbred C57BL; Oocytes; Patch-Clamp Techniques; Protein Kinase Inhibitors; Protein Transport; Rats; Sodium; Substrate Specificity; Triazoles; Xenopus laevis | 2008 |
Protein kinase CK2 modulates synaptic plasticity by modification of synaptic NMDA receptors in the hippocampus.
Topics: Animals; Casein Kinase II; Cells, Cultured; Dichlororibofuranosylbenzimidazole; Enzyme Inhibitors; Hippocampus; Membrane Potentials; Neuronal Plasticity; Neurons; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Synapses; Triazoles | 2008 |
Role of heme oxygenase-2 in pial arteriolar response to acetylcholine in mice with and without transfusion of cell-free hemoglobin polymers.
Topics: Acetylcholine; Animals; Arterioles; Blood Component Transfusion; Blood Substitutes; Carbon Dioxide; Casein Kinase II; Cerebrovascular Circulation; Cerebrum; Dose-Response Relationship, Drug; Enzyme Inhibitors; Heme Oxygenase (Decyclizing); Hemoglobins; Metalloporphyrins; Mice; Mice, Inbred C57BL; Mice, Knockout; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Protoporphyrins; Triazoles; Vasodilation; Vasodilator Agents | 2008 |
New inhibitors of protein kinase CK2, analogues of benzimidazole and benzotriazole.
Topics: Benzimidazoles; Casein Kinase II; Humans; Protein Kinase Inhibitors; Triazoles | 2008 |
Evaluating CK2 activity with the antibody specific for the CK2-phosphorylated form of a kinase-targeting cochaperone Cdc37.
Topics: Animals; Antibodies, Phospho-Specific; Antibody Specificity; Carrier Proteins; Casein Kinase II; Cell Cycle Proteins; Chlorocebus aethiops; COS Cells; Holoenzymes; Humans; Intercellular Signaling Peptides and Proteins; Molecular Chaperones; Phosphorylation; Phosphoserine; Protein Subunits; Rats; Swine; Triazoles | 2008 |
Impact of protein kinase CK2 on inhibitor of apoptosis proteins in prostate cancer cells.
Topics: Apigenin; Apoptosis; Apoptosis Regulatory Proteins; Casein Kinase II; Caspases; Cell Line, Tumor; Humans; Male; Prostatic Neoplasms; Protein Kinase Inhibitors; Subcellular Fractions; Triazoles | 2008 |
The selectivity of inhibitors of protein kinase CK2: an update.
Topics: Animals; Benzimidazoles; Casein Kinase II; Humans; Indazoles; Jurkat Cells; Kinetics; Models, Molecular; Protein Kinase Inhibitors; Rats; Structure-Activity Relationship; Triazoles | 2008 |
Peptide biosensors for the electrochemical measurement of protein kinase activity.
Topics: Adenosine Triphosphate; Benzimidazoles; Biosensing Techniques; Bone Neoplasms; Casein Kinase II; Catalysis; Electrochemistry; Ferrous Compounds; fms-Like Tyrosine Kinase 3; Humans; Kinetics; Metallocenes; Mutation; Osteosarcoma; Oxidation-Reduction; Peptide Fragments; Phosphorylation; Protein Kinase C; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-abl; Receptor, ErbB-2; Staurosporine; Triazoles; Tumor Cells, Cultured | 2008 |
Phosphorylation of the HuR ligand APRIL by casein kinase 2 regulates CD83 expression.
Topics: Animals; Antigens, CD; Antigens, Surface; Casein Kinase II; CD83 Antigen; Cell Line, Tumor; ELAV Proteins; ELAV-Like Protein 1; Exportin 1 Protein; Genetic Vectors; HeLa Cells; Humans; Immunoglobulins; Jurkat Cells; Karyopherins; Membrane Glycoproteins; Mice; NIH 3T3 Cells; Nuclear Proteins; Phosphorylation; Receptors, Cytoplasmic and Nuclear; RNA-Binding Proteins; Transfection; Triazoles | 2009 |
Inhibition of protein kinase CK2 induces E2F1 nuclear export, formation of p21/E2F1 complexes and suppression of DNA synthesis in normal human epidermal keratinocytes.
Topics: Active Transport, Cell Nucleus; Casein Kinase II; Cell Proliferation; Cells, Cultured; Cyclin-Dependent Kinase Inhibitor p21; DNA Replication; Dose-Response Relationship, Drug; Down-Regulation; E2F1 Transcription Factor; Epidermis; Humans; Keratinocytes; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-myc; Signal Transduction; Triazoles | 2009 |
DMAT, an inhibitor of protein kinase CK2 induces reactive oxygen species and DNA double strand breaks.
Topics: Antineoplastic Agents; Apoptosis; Benzimidazoles; Casein Kinase II; Cell Line, Tumor; Cell Survival; DNA Breaks, Double-Stranded; Humans; Male; Oxidative Stress; Prostatic Neoplasms; Protein Kinase Inhibitors; Reactive Oxygen Species; Time Factors; Triazoles; Up-Regulation | 2009 |
PACS-1 mediates phosphorylation-dependent ciliary trafficking of the cyclic-nucleotide-gated channel in olfactory sensory neurons.
Topics: Alanine; Animals; Casein Kinase II; Cell Line, Transformed; Cilia; Cyclic Nucleotide-Gated Cation Channels; Dogs; Enzyme Inhibitors; Green Fluorescent Proteins; Humans; Immunoprecipitation; Mice; Mice, Transgenic; Mutation; Olfactory Mucosa; Phosphorylation; Protein Subunits; Protein Transport; RNA Interference; RNA, Messenger; Sensory Receptor Cells; Serine; Transfection; Triazoles; Vesicular Transport Proteins | 2009 |
Involvement of reactive oxygen species in apoptosis induced by pharmacological inhibition of protein kinase CK2.
Topics: Apoptosis; Casein Kinase II; Cell Line, Tumor; DNA Fragmentation; Dose-Response Relationship, Drug; Flow Cytometry; Humans; Hydrogen Peroxide; Intracellular Space; Reactive Oxygen Species; Superoxides; Time Factors; Triazoles | 2009 |
p53 is dispensable for the induction of apoptosis after inhibition of protein kinase CK2.
Topics: Apoptosis; Casein Kinase II; Cell Line, Tumor; Cell Proliferation; Cell Survival; Enzyme Inhibitors; Humans; Male; Prostatic Neoplasms; Triazoles; Tumor Suppressor Protein p53 | 2010 |
Selectivity analysis of protein kinase CK2 inhibitors DMAT, TBB and resorufin in cisplatin-induced stress responses.
Topics: Antineoplastic Agents; Benzimidazoles; Blotting, Western; Casein Kinase II; Cell Line, Tumor; Cell Survival; Cisplatin; Enzyme Inhibitors; Humans; Oxazines; Signal Transduction; Stress, Physiological; Triazoles | 2009 |
A FRET-based microplate assay for human protein kinase CK2, a target in neoplastic disease.
Topics: Casein Kinase II; Emodin; Enzyme Assays; Fluorescence; Fluorescence Resonance Energy Transfer; Humans; Naphthalenesulfonates; Neoplasms; p-Dimethylaminoazobenzene; Pancreatic Elastase; Peptides; Phosphorylation; Protein Kinase Inhibitors; Sensitivity and Specificity; Triazoles | 2010 |
Regulation of PTEN by CK2 and Notch1 in primary T-cell acute lymphoblastic leukemia: rationale for combined use of CK2- and gamma-secretase inhibitors.
Topics: Amyloid Precursor Protein Secretases; Blotting, Western; Casein Kinase II; Cell Proliferation; Cell Size; Child; Dichlororibofuranosylbenzimidazole; Drug Therapy, Combination; Enzyme Inhibitors; Gene Expression Regulation, Leukemic; Humans; Mutation; Precursor T-Cell Lymphoblastic Leukemia-Lymphoma; PTEN Phosphohydrolase; Receptor, Notch1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Triazoles | 2010 |
Casein kinase 2 inhibition differentially modulates apoptotic effect of trichostatin A against epithelial ovarian carcinoma cell lines.
Topics: Animals; Apigenin; Apoptosis; Casein Kinase II; Cell Line, Tumor; Cell Nucleus; DNA Fragmentation; Epithelium; Female; Histone Deacetylase Inhibitors; Humans; Hydroxamic Acids; Ovarian Neoplasms; Signal Transduction; Triazoles | 2010 |
Phosphorylation of the von Hippel-Lindau protein (VHL) by protein kinase CK2 reduces its protein stability and affects p53 and HIF-1alpha mediated transcription.
Topics: Casein Kinase II; Down-Regulation; HEK293 Cells; Humans; Hypoxia-Inducible Factor 1, alpha Subunit; Mutagenesis, Site-Directed; Mutant Proteins; Phosphorylation; Protein Binding; Protein Stability; Transcriptional Activation; Transgenes; Triazoles; Tumor Suppressor Protein p53; Von Hippel-Lindau Tumor Suppressor Protein | 2010 |
Relative role of halogen bonds and hydrophobic interactions in inhibition of human protein kinase CK2α by tetrabromobenzotriazole and some C5-substituted analogues.
Topics: Casein Kinase II; Enzyme Inhibitors; Halogens; Humans; Hydrophobic and Hydrophilic Interactions; Models, Molecular; Molecular Structure; Protein Conformation; Triazoles | 2010 |
CK2 inhibition induces apoptosis via the ER stress response.
Topics: Apoptosis; Casein Kinase II; Caspase 9; Cell Line, Tumor; Cytochromes c; Endoplasmic Reticulum; Humans; Proto-Oncogene Proteins c-bcl-2; Receptors, TNF-Related Apoptosis-Inducing Ligand; Transcription Factor CHOP; Triazoles; Unfolded Protein Response | 2011 |
Kinome profiling of myxoid liposarcoma reveals NF-kappaB-pathway kinase activity and casein kinase II inhibition as a potential treatment option.
Topics: Casein Kinase II; Cell Line; Cell Line, Tumor; Cell Survival; Cells, Cultured; Dasatinib; HeLa Cells; Humans; Immunoblotting; Jurkat Cells; Karyotyping; Liposarcoma, Myxoid; NF-kappa B; Oncogene Proteins, Fusion; Protein Kinase Inhibitors; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; Thiazoles; Triazoles | 2010 |
Treatment of cultured human astrocytes and vascular endothelial cells with protein kinase CK2 inhibitors induces early changes in cell shape and cytoskeleton.
Topics: Animals; Astrocytes; Casein Kinase II; Cattle; Cell Line, Tumor; Cell Shape; Culture Media; Cytoskeleton; Endothelial Cells; Enzyme Activation; Humans; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Triazoles | 2011 |
A specific inhibitor of protein kinase CK2 delays gamma-H2Ax foci removal and reduces clonogenic survival of irradiated mammalian cells.
Topics: Animals; Casein Kinase II; Cell Survival; Cells, Cultured; DNA Breaks, Double-Stranded; DNA Repair; Drug Evaluation, Preclinical; Fibroblasts; Histones; Humans; Mammals; Neoplastic Stem Cells; Protein Kinase Inhibitors; Substrate Specificity; Time Factors; Triazoles; Tumor Stem Cell Assay | 2011 |
The cytosolic protein kinase CK2 phosphorylates cardiac calsequestrin in intact cells.
Topics: Amino Acid Substitution; Animals; Benzimidazoles; Calsequestrin; Casein Kinase II; Cells, Cultured; Chlorocebus aethiops; Cinnamates; COS Cells; Cytosol; Electrophoresis, Polyacrylamide Gel; Endoplasmic Reticulum; Mutation; Myocytes, Cardiac; Phosphorylation; Protein Serine-Threonine Kinases; Protein Subunits; Rats; RNA Interference; Triazoles | 2011 |
The kinase DYRKIA regulates pre-mRNA splicing in spermatogonia and proliferation of spermatogonia and Sertoli cells by phosphorylating a spliceosomal component, SAP155, in postnatal murine testes.
Topics: Animals; Animals, Newborn; Cell Line; Cell Proliferation; Cyclin-Dependent Kinase 2; Dyrk Kinases; Male; Mice; Phosphoproteins; Phosphorylation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Pyrans; Ribonucleoprotein, U2 Small Nuclear; RNA Precursors; RNA Splicing; RNA Splicing Factors; Sertoli Cells; Spermatogonia; Spiro Compounds; Spliceosomes; Testis; Triazoles | 2011 |
The protein kinase CK2 inhibitor TBB mediates up-regulation of MEK3/6 and p38δ activities, down-regulation of ERK1/2 activity and induction of G1/S arrest in normal human epidermal autocrine proliferating keratinocytes.
Topics: Autocrine Communication; Casein Kinase II; Cell Cycle; Cell Proliferation; Cells, Cultured; Down-Regulation; Epidermis; Humans; Keratinocytes; MAP Kinase Kinase 3; MAP Kinase Kinase 6; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 13; Mitogen-Activated Protein Kinase 3; Protein Kinase Inhibitors; Triazoles; Up-Regulation | 2011 |
Design and synthesis of CK2 inhibitors.
Topics: Benzimidazoles; Casein Kinase II; Drug Design; Humans; Inhibitory Concentration 50; Protein Kinase Inhibitors; Triazoles | 2011 |
Down-regulation of CK2 activity results in a decrease in the level of cdc25C phosphatase in different prostate cancer cell lines.
Topics: Anthraquinones; Apoptosis; Benzimidazoles; Casein Kinase II; CDC2 Protein Kinase; cdc25 Phosphatases; Cell Line, Tumor; Down-Regulation; Genes, Dominant; Humans; Male; Mutant Proteins; Prostatic Neoplasms; Protein Kinase Inhibitors; Transfection; Triazoles | 2011 |
Time schedule-dependent effect of the CK2 inhibitor TBB on PC-3 human prostate cancer cell viability.
Topics: Antineoplastic Agents; Apoptosis; Camptothecin; Cell Line, Tumor; Cell Survival; Checkpoint Kinase 2; Enzyme Inhibitors; Humans; Male; Prostatic Neoplasms; Protein Serine-Threonine Kinases; TNF-Related Apoptosis-Inducing Ligand; Triazoles | 2012 |
Influence of five potential anticancer drugs on wnt pathway and cell survival in human biliary tract cancer cells.
Topics: Antineoplastic Agents; Benzimidazoles; beta Catenin; Biliary Tract Neoplasms; Cadherins; Cell Line, Tumor; Cell Survival; Clinical Trials as Topic; Cyclin D1; Flavonoids; Gene Expression Regulation, Neoplastic; Genes, p53; Humans; Ki-67 Antigen; Proliferating Cell Nuclear Antigen; Quercetin; RNA, Messenger; Sulfonamides; Triazoles; Vimentin; Wnt Signaling Pathway | 2012 |
Cell rounding in cultured human astrocytes and vascular endothelial cells upon inhibition of CK2 is mediated by actomyosin cytoskeleton alterations.
Topics: Actomyosin; Animals; Astrocytes; Casein Kinase II; Cattle; Cell Shape; Cinnamates; Cytoskeleton; Endothelial Cells; Humans; Myosin Light Chains; Phosphorylation; Rats; Triazoles | 2012 |
Inhibition of casein kinase 2 modulates XBP1-GRP78 arm of unfolded protein responses in cultured glial cells.
Topics: Activating Transcription Factor 6; Animals; Casein Kinase II; Cells, Cultured; DNA-Binding Proteins; Endoplasmic Reticulum; Endoplasmic Reticulum Chaperone BiP; Endoplasmic Reticulum Stress; Eukaryotic Initiation Factor-2; Gene Knockdown Techniques; Heat-Shock Proteins; Mice; Mice, Inbred C57BL; Neuroglia; Protein Kinase Inhibitors; Protein Transport; Regulatory Factor X Transcription Factors; RNA Splicing; Subcellular Fractions; Transcription Factor CHOP; Transcription Factors; Triazoles; Unfolded Protein Response; X-Box Binding Protein 1 | 2012 |
Identification of a novel crosstalk between casein kinase 2α and NPM-ALK in ALK-positive anaplastic large cell lymphoma.
Topics: beta Catenin; Casein Kinase II; Cell Communication; Cell Line, Tumor; Cell Proliferation; Cell Transformation, Neoplastic; Down-Regulation; Enzyme Inhibitors; Humans; Lymphoma, Large-Cell, Anaplastic; Phosphorylation; Protein-Tyrosine Kinases; RNA Interference; RNA, Small Interfering; Signal Transduction; Triazoles; Wnt Proteins | 2013 |
Inhibition of CK2 enhances UV-triggered apoptotic cell death in lung cancer cell lines.
Topics: Apoptosis; Casein Kinase II; Caspase 3; Cell Line, Tumor; Cell Survival; Cytochromes c; Humans; Lung Neoplasms; Nuclear Proteins; Poly(ADP-ribose) Polymerases; Promyelocytic Leukemia Protein; RNA Interference; RNA, Small Interfering; Transcription Factors; Triazoles; Tumor Suppressor Proteins; Ultraviolet Rays | 2013 |
Inhibition of casein kinase II reduces TGFβ induced fibroblast activation and ameliorates experimental fibrosis.
Topics: Adult; Aged; Animals; Casein Kinase II; Disease Models, Animal; Female; Fibroblasts; Fibrosis; Humans; Janus Kinase 2; Male; Mice; Middle Aged; Scleroderma, Systemic; Signal Transduction; Skin; STAT3 Transcription Factor; Transforming Growth Factor beta; Triazoles; Young Adult | 2015 |
Casein kinase II inhibition reverses pain hypersensitivity and potentiated spinal N-methyl-D-aspartate receptor activity caused by calcineurin inhibitor.
Topics: Animals; Calcineurin Inhibitors; Casein Kinase II; Dichlororibofuranosylbenzimidazole; Excitatory Postsynaptic Potentials; Hyperalgesia; Male; Miniature Postsynaptic Potentials; N-Methylaspartate; Physical Stimulation; Posterior Horn Cells; Rats, Sprague-Dawley; Spinal Cord; Tacrolimus; Touch; Triazoles | 2014 |
Synthesis of novel chiral TBBt derivatives with hydroxyl moiety. Studies on inhibition of human protein kinase CK2α and cytotoxicity properties.
Topics: Antineoplastic Agents; Casein Kinase II; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; MCF-7 Cells; Molecular Docking Simulation; Molecular Structure; Protein Kinase Inhibitors; Structure-Activity Relationship; Triazoles; Tumor Cells, Cultured | 2014 |
Protein kinase CK2 inhibition induces cell death via early impact on mitochondrial function.
Topics: Apoptosis; Calcium Signaling; Casein Kinase II; Catalase; Cell Line, Tumor; Egtazic Acid; Humans; Membrane Potential, Mitochondrial; Mitochondria; Mitochondrial Membrane Transport Proteins; Mitochondrial Permeability Transition Pore; Triazoles | 2014 |
Alterations of microRNAs are associated with impaired growth of MCF-7 breast cancer cells induced by inhibition of casein kinase 2.
Topics: Apoptosis; Breast Neoplasms; Casein Kinase II; Cell Cycle; Cell Proliferation; Cell Survival; Flow Cytometry; Gene Expression Regulation, Neoplastic; Humans; MCF-7 Cells; MicroRNAs; Oligonucleotide Array Sequence Analysis; Real-Time Polymerase Chain Reaction; Triazoles | 2014 |
Thermodynamic parameters for binding of some halogenated inhibitors of human protein kinase CK2.
Topics: Benzimidazoles; Binding Sites; Calorimetry; Calorimetry, Differential Scanning; Casein Kinase II; Drug Design; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Inhibitory Concentration 50; Ligands; Methylation; Microscopy, Fluorescence; Protein Binding; Static Electricity; Temperature; Thermodynamics; Triazoles | 2015 |
Thrombin-induced IL-8/CXCL8 release is mediated by CK2, MSK1, and NF-κB pathways in human lung epithelial cells.
Topics: Animals; Apigenin; Casein Kinase II; Cells, Cultured; Epithelial Cells; Humans; Indoles; Interleukin-8; Lung; NF-kappa B; Phosphorylation; Pyrroles; Ribosomal Protein S6 Kinases, 90-kDa; RNA, Small Interfering; Signal Transduction; Thrombin; Transcription Factor RelA; Triazoles | 2015 |
Protein kinase CK2 regulates metal toxicity in neuronal cells.
Topics: Animals; Anthraquinones; Calcium; Casein Kinase II; Cell Line, Tumor; Gene Knockdown Techniques; Heavy Metal Poisoning; Inhibitory Concentration 50; Intracellular Space; Ions; Metals; Mice; Microscopy, Confocal; Neurons; Poisoning; Protein Kinase Inhibitors; Reproducibility of Results; RNA, Small Interfering; Saccharomyces cerevisiae; Triazoles; Zinc | 2016 |
CK2 inhibition induced PDK4-AMPK axis regulates metabolic adaptation and survival responses in glioma.
Topics: Adenosine Triphosphate; AMP-Activated Protein Kinases; Animals; Brain Neoplasms; Casein Kinase II; Cell Line, Tumor; Cell Proliferation; Cell Survival; Cellular Senescence; Cyclic AMP Response Element-Binding Protein; Glioma; Glucose; Humans; Mice, Nude; Phenotype; Phosphorylation; Protein Serine-Threonine Kinases; Pyruvate Dehydrogenase Acetyl-Transferring Kinase; RNA, Messenger; Signal Transduction; Sirtuin 1; Triazoles; Tumor Suppressor Protein p53; Xenograft Model Antitumor Assays | 2016 |
Annexin-1 Mediates Microglial Activation and Migration via the CK2 Pathway during Oxygen-Glucose Deprivation/Reperfusion.
Topics: alpha Catenin; Amino Acid Sequence; Animals; Annexin A1; Casein Kinase II; Cell Hypoxia; Cell Line; Cell Movement; Female; Gene Expression Regulation; Glucose; Hippocampus; Male; Microglia; Neurons; Oligopeptides; Patch-Clamp Techniques; Peptides; Phosphorylation; Rats; Rats, Sprague-Dawley; Receptors, Formyl Peptide; RNA, Small Interfering; Tissue Culture Techniques; Triazoles | 2016 |
Alpha B-Crystallin Protects Rat Articular Chondrocytes against Casein Kinase II Inhibition-Induced Apoptosis.
Topics: alpha-Crystallin B Chain; Animals; Apigenin; Apoptosis; Benzimidazoles; Cartilage, Articular; Casein Kinase II; Chondrocytes; Cytoprotection; Disease Models, Animal; Gene Knockdown Techniques; Gene Silencing; Male; Osteoarthritis; Phenotype; Phosphorylation; Protein Transport; Rats, Sprague-Dawley; Subcellular Fractions; Triazoles | 2016 |
Tor1 and CK2 kinases control a switch between alternative ribosome biogenesis pathways in a growth-dependent manner.
Topics: Casein Kinase II; Heat-Shock Response; Mutation; Organelle Biogenesis; Oxidative Stress; Phosphatidylinositol 3-Kinases; Phosphorylation; Proteomics; Ribosomes; RNA Polymerase I; RNA Precursors; RNA Processing, Post-Transcriptional; Saccharomyces cerevisiae; Saccharomyces cerevisiae Proteins; Sirolimus; Triazoles | 2017 |
In Vitro Cell Death Discrimination and Screening Method by Simple and Cost-Effective Viability Analysis.
Topics: Apoptosis; Biological Assay; Biomarkers; Caspase 3; Caspase 7; Cell Line, Tumor; Cell Survival; Dactinomycin; Dose-Response Relationship, Drug; Epidermis; Gene Expression; Humans; Hydrogen Peroxide; Indicators and Reagents; Indoles; Light; Necrosis; Oxazines; Triazoles; Xanthenes | 2017 |
Physiological regulation of the epithelial Na
Topics: Amiloride; Animals; Casein Kinase II; CHO Cells; Cricetulus; Epithelial Sodium Channel Blockers; Epithelial Sodium Channels; Kidney Tubules, Collecting; Membrane Potentials; Mice; Mutation; Natriuresis; Phosphorylation; Protein Kinase Inhibitors; Sodium; Triazoles | 2018 |
Inhibition of protein kinase CK2 facilitates cellular senescence by inhibiting the expression of HO-1 in articular chondrocytes.
Topics: Animals; Cartilage, Articular; Casein Kinase II; Cellular Senescence; Chondrocytes; Gene Expression Regulation; Heme Oxygenase-1; Male; Rats; Triazoles | 2019 |
Detection of casein kinase II by aggregation-induced emission.
Topics: Benzylidene Compounds; Biosensing Techniques; Casein Kinase II; Cathepsin A; Enzyme Assays; Fluorescent Dyes; HeLa Cells; Humans; Oligopeptides; Phosphorylation; Protein Kinase Inhibitors; Proteolysis; Spectrometry, Fluorescence; Triazoles | 2019 |
Lysophosphatidylcholine triggers cell differentiation in the protozoan parasite Herpetomonas samuelpessoai through the CK2 pathway.
Topics: Animals; Casein Kinase II; Cell Differentiation; Dichlororibofuranosylbenzimidazole; Enzyme Inhibitors; Hemiptera; Lysophosphatidylcholines; Metabolic Networks and Pathways; Phospholipases A2; Triazoles; Trypanosomatina | 2020 |
Protein kinase CK2 impact on intracellular calcium homeostasis in prostate cancer.
Topics: Animals; Apoptosis; Calcium; Casein Kinase II; Cell Line, Tumor; Cell Survival; Cytosol; Endoplasmic Reticulum; Homeostasis; Humans; Male; Membrane Potential, Mitochondrial; Mice; Mice, Nude; Naphthyridines; Phenazines; Prostatic Neoplasms; Triazoles | 2020 |
Screening of tau protein kinase inhibitors in a tauopathy-relevant cell-based model of tau hyperphosphorylation and oligomerization.
Topics: Animals; Cell Line; Cyclosporine; Glycogen Synthase Kinase 3; Lithium Chloride; Mice; Models, Biological; Okadaic Acid; Phosphorylation; Protein Kinase Inhibitors; Protein Multimerization; Rats; Tauopathies; Triazoles | 2020 |