Page last updated: 2024-08-24

triazoles and 11-cis-retinal

triazoles has been researched along with 11-cis-retinal in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (80.00)29.6817
2010's1 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baraldi, PG; Borea, PA; Braiuca, P; Cacciari, B; Deflorian, F; Ferrari, C; Moro, S; Pastorin, G; Spalluto, G; Varani, K1
Bacilieri, M; Deflorian, F; Moro, S; Spalluto, G1
Catarzi, D; Ciampi, O; Colotta, V; Filacchioni, G; Lenzi, O; Martini, C; Morizzo, E; Moro, S; Pedata, F; Pugliese, AM; Traini, C; Trincavelli, L; Varano, F1
Maass, A; Müller, CE; Schiedel, AC; Sherbiny, FF1
Cherezov, V; Gao, ZG; Han, GW; Jacobson, KA; Katritch, V; Stevens, RC; Wu, H; Xu, F1

Reviews

1 review(s) available for triazoles and 11-cis-retinal

ArticleYear
Ligand-based homology modeling as attractive tool to inspect GPCR structural plasticity.
    Current pharmaceutical design, 2006, Volume: 12, Issue:17

    Topics: Adenosine A3 Receptor Antagonists; Computer Simulation; Computer-Aided Design; Crystallography, X-Ray; Drug Design; Ligands; Models, Molecular; Molecular Structure; Protein Binding; Protein Conformation; Pyrimidines; Receptor, Adenosine A3; Receptors, G-Protein-Coupled; Rhodopsin; Structural Homology, Protein; Structure-Activity Relationship; Triazoles

2006

Other Studies

4 other study(ies) available for triazoles and 11-cis-retinal

ArticleYear
Combined target-based and ligand-based drug design approach as a tool to define a novel 3D-pharmacophore model of human A3 adenosine receptor antagonists: pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine derivatives as a key study.
    Journal of medicinal chemistry, 2005, Jan-13, Volume: 48, Issue:1

    Topics: Adenosine A3 Receptor Antagonists; Animals; Binding Sites; Combinatorial Chemistry Techniques; Cricetinae; Drug Design; Drug Evaluation, Preclinical; Humans; Ligands; Models, Molecular; Models, Theoretical; Protein Conformation; Pyrimidines; Quantitative Structure-Activity Relationship; Receptor, Adenosine A3; Reproducibility of Results; Rhodopsin; Static Electricity; Triazoles

2005
Synthesis, ligand-receptor modeling studies and pharmacological evaluation of novel 4-modified-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-one derivatives as potent and selective human A3 adenosine receptor antagonists.
    Bioorganic & medicinal chemistry, 2008, Jun-01, Volume: 16, Issue:11

    Topics: Adenosine A3 Receptor Antagonists; Animals; Binding, Competitive; Brain Ischemia; Cattle; Cell Membrane; Cerebral Cortex; Disease Models, Animal; Humans; Hydrogen Bonding; Ligands; Models, Molecular; Protein Binding; Quinoxalines; Rats; Receptor, Adenosine A3; Rhodopsin; Structural Homology, Protein; Structure-Activity Relationship; Triazoles; Xanthines

2008
Homology modelling of the human adenosine A2B receptor based on X-ray structures of bovine rhodopsin, the beta2-adrenergic receptor and the human adenosine A2A receptor.
    Journal of computer-aided molecular design, 2009, Volume: 23, Issue:11

    Topics: Animals; Cattle; Humans; Models, Molecular; Molecular Structure; Mutagenesis, Site-Directed; Protein Binding; Protein Conformation; Receptor, Adenosine A2B; Receptors, Adrenergic, beta-2; Rhodopsin; Triazines; Triazoles; X-Rays

2009
Structure of an agonist-bound human A2A adenosine receptor.
    Science (New York, N.Y.), 2011, Apr-15, Volume: 332, Issue:6027

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Binding Sites; Crystallography, X-Ray; Humans; Hydrogen Bonding; Ligands; Models, Molecular; Opsins; Protein Conformation; Protein Structure, Secondary; Receptor, Adenosine A2A; Rhodopsin; Triazines; Triazoles

2011