Page last updated: 2024-08-16

triazolam and cimetidine

triazolam has been researched along with cimetidine in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19906 (37.50)18.7374
1990's0 (0.00)18.2507
2000's6 (37.50)29.6817
2010's4 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Topliss, JG; Yoshida, F1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY1
Andricopulo, AD; Moda, TL; Montanari, CA1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chen, L; He, Z; Li, H; Liu, J; Liu, X; Sui, X; Sun, J; Wang, Y; Zhang, W1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Desager, JP; Harvengt, C; Hulhoven, R; Pourbaix, S; Smith, RB1
Burstein, ES; Friedman, H; Greenblatt, DJ; Harmatz, JS; Scavone, JM; Shader, RI1
Britton, ML; Waller, ES1
Greenblatt, DJ1
Abernethy, DR; Divoll, M; Greenblatt, DJ; Harmatz, JS; Moschitto, LJ; Shader, RI1
MacLachlan, RA; Parker, WA1

Reviews

1 review(s) available for triazolam and cimetidine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Trials

1 trial(s) available for triazolam and cimetidine

ArticleYear
Interaction of cimetidine with the triazolobenzodiazepines alprazolam and triazolam.
    Psychopharmacology, 1983, Volume: 80, Issue:3

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Cimetidine; Drug Interactions; Female; Guanidines; Humans; Male; Metabolic Clearance Rate; Middle Aged; Triazolam

1983

Other Studies

14 other study(ies) available for triazolam and cimetidine

ArticleYear
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Hologram QSAR model for the prediction of human oral bioavailability.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Administration, Oral; Biological Availability; Holography; Humans; Models, Biological; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Prediction of volume of distribution values in human using immobilized artificial membrane partitioning coefficients, the fraction of compound ionized and plasma protein binding data.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:11

    Topics: Blood Proteins; Chemistry, Physical; Computer Simulation; Humans; Membranes, Artificial; Models, Biological; Pharmaceutical Preparations; Protein Binding; Tissue Distribution

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Pharmacokinetic consequences of long term coadministration of cimetidine and triazolobenzodiazepines, alprazolam and triazolam, in healthy subjects.
    International journal of clinical pharmacology, therapy, and toxicology, 1985, Volume: 23, Issue:8

    Topics: Adult; Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Cimetidine; Drug Interactions; Female; Half-Life; Humans; Kinetics; Male; Time Factors; Triazolam

1985
Triazolam kinetics: interaction with cimetidine, propranolol, and the combination.
    Journal of clinical pharmacology, 1988, Volume: 28, Issue:3

    Topics: Adult; Cimetidine; Drug Interactions; Female; Humans; Male; Middle Aged; Propranolol; Triazolam

1988
Central nervous system toxicity associated with concurrent use of triazolam and cimetidine.
    Drug intelligence & clinical pharmacy, 1985, Volume: 19, Issue:9

    Topics: Central Nervous System Diseases; Cimetidine; Drug Interactions; Female; Humans; Middle Aged; Triazolam; Zollinger-Ellison Syndrome

1985
Comment: Triazolam-cimetidine reaction.
    Drug intelligence & clinical pharmacy, 1985, Volume: 19, Issue:9

    Topics: Cimetidine; Drug Interactions; Humans; Triazolam

1985
Prolonged hypnotic response to triazolam-cimetidine combination in an elderly patient.
    Drug intelligence & clinical pharmacy, 1984, Volume: 18, Issue:12

    Topics: Aged; Anti-Anxiety Agents; Cimetidine; Drug Interactions; Female; Humans; Hypnotics and Sedatives; Microsomes, Liver; Time Factors; Triazolam

1984