Page last updated: 2024-08-16

triamterene and antipyrine

triamterene has been researched along with antipyrine in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19901 (12.50)18.7374
1990's1 (12.50)18.2507
2000's4 (50.00)29.6817
2010's2 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Weiss, M1
Dayton, PG; McNay, JL; Pruitt, AW; Steinhorst, J1
Hayashi, M; Sudo, R; Takahashi, M; Watanabe, E1

Other Studies

8 other study(ies) available for triamterene and antipyrine

ArticleYear
ElogD(oct): a tool for lipophilicity determination in drug discovery. 2. Basic and neutral compounds.
    Journal of medicinal chemistry, 2001, Jul-19, Volume: 44, Issue:15

    Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Water

2001
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Use of metabolite AUC data in bioavailability studies to discriminate between absorption and first-pass extraction.
    Clinical pharmacokinetics, 1990, Volume: 18, Issue:5

    Topics: Absorption; Antipyrine; Biological Availability; Caffeine; Diphenhydramine; Dose-Response Relationship, Drug; Humans; Ketanserin; Lidocaine; Liver Diseases; Metronidazole; Nomifensine; Triamterene

1990
Studies with triamterene, a substituted pteridine. Unusual brain to plasma ratio in mammals.
    Neuropharmacology, 1972, Volume: 11, Issue:3

    Topics: Adipose Tissue; Animals; Antipyrine; Biological Transport; Body Fluids; Brain; Carbon Isotopes; Eye; Female; Fetus; Guinea Pigs; Liver; Maternal-Fetal Exchange; Muscles; Myocardium; Omentum; Papio; Placenta; Pregnancy; Protein Binding; Solubility; Spectrometry, Fluorescence; Triamterene; Tritium

1972
Evaluation of absorbability of poorly water-soluble drugs: validity of the use of additives.
    Biological & pharmaceutical bulletin, 2000, Volume: 23, Issue:7

    Topics: Absorption; Animals; Anti-Inflammatory Agents, Non-Steroidal; Antipyrine; Cell Membrane Permeability; Chromogenic Compounds; Deoxycholic Acid; Detergents; Dextrans; Dimethyl Sulfoxide; Diuretics; Fluorescein-5-isothiocyanate; Indomethacin; Intestinal Mucosa; Intestines; Male; Phenolsulfonphthalein; Rats; Rats, Wistar; Reproducibility of Results; Solubility; Solvents; Triamterene

2000