Page last updated: 2024-08-26

tretazicar and apaziquone

tretazicar has been researched along with apaziquone in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (57.14)18.2507
2000's3 (42.86)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Phillips, RM; Seville, S; Shnyder, SD; Wright, CW1
Sugget, N; Walton, MI; Workman, P1
Riley, RJ; Workman, P1
Chen, S; Deng, PS; Ebenstein, D; Friedlos, F; Fung, M; Knox, R; Lewis, AD; Tsai, TM; Workman, P; Wu, K1
Melo, T; Misra, V; Rauth, AM1
Celli, CM; Jaiswal, AK; Knox, R; Tran, N1
Boyle, RG; Travers, S1

Reviews

2 review(s) available for tretazicar and apaziquone

ArticleYear
DT-diaphorase and cancer chemotherapy.
    Biochemical pharmacology, 1992, Apr-15, Volume: 43, Issue:8

    Topics: Animals; Antineoplastic Agents; Aziridines; Benzoquinones; Dihydrolipoamide Dehydrogenase; Drug Design; Enzyme Induction; Gene Expression Regulation, Enzymologic; Humans; Indolequinones; Indoles; Mitomycin; Neoplasms; Precancerous Conditions; Tirapazamine; Triazines

1992
Hypoxia: targeting the tumour.
    Anti-cancer agents in medicinal chemistry, 2006, Volume: 6, Issue:4

    Topics: Anthraquinones; Antineoplastic Agents; Aziridines; Benzoquinones; Cell Hypoxia; Clinical Trials, Phase III as Topic; Drug Screening Assays, Antitumor; Humans; Imidazoles; Indolequinones; Neoplasms; Prodrugs; Quinolines; Radiation-Sensitizing Agents; Tirapazamine; Triazines

2006

Other Studies

5 other study(ies) available for tretazicar and apaziquone

ArticleYear
Synthesis of cryptolepine analogues as potential bioreducible anticancer agents.
    Bioorganic & medicinal chemistry, 2007, Oct-01, Volume: 15, Issue:19

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cytosol; Drug Screening Assays, Antitumor; Humans; Indole Alkaloids; Inhibitory Concentration 50; Prodrugs; Quinolines; Quinone Reductases; Structure-Activity Relationship

2007
The role of human and rodent DT-diaphorase in the reductive metabolism of hypoxic cell cytotoxins.
    International journal of radiation oncology, biology, physics, 1992, Volume: 22, Issue:4

    Topics: Animals; Antineoplastic Agents; Aziridines; Carcinoma 256, Walker; Cell Hypoxia; Colonic Neoplasms; Humans; In Vitro Techniques; Indolequinones; Indoles; Mitomycin; NAD(P)H Dehydrogenase (Quinone); Oxidation-Reduction; Prodrugs; Rats; Tirapazamine; Triazines

1992
Catalytic properties of NAD(P)H:quinone acceptor oxidoreductase: study involving mouse, rat, human, and mouse-rat chimeric enzymes.
    Molecular pharmacology, 1995, Volume: 47, Issue:5

    Topics: Amino Acid Sequence; Animals; Aziridines; Base Sequence; DNA Damage; DNA Primers; Escherichia coli; Humans; In Vitro Techniques; Indolequinones; Indoles; Kinetics; Mice; Molecular Sequence Data; NAD(P)H Dehydrogenase (Quinone); Prodrugs; Rats; Recombinant Fusion Proteins; Sequence Homology, Amino Acid; Species Specificity

1995
Bioreductive therapies: an overview of drugs and their mechanisms of action.
    International journal of radiation oncology, biology, physics, 1998, Nov-01, Volume: 42, Issue:4

    Topics: Animals; Antineoplastic Agents; Aziridines; Cell Hypoxia; DNA, Neoplasm; Forecasting; Humans; Indolequinones; Indoles; Misonidazole; Mitomycin; Nitrofurans; Nitroimidazoles; Oxidation-Reduction; Prodrugs; Radiation-Sensitizing Agents; Tirapazamine; Triazines

1998
NRH:quinone oxidoreductase 2 (NQO2) catalyzes metabolic activation of quinones and anti-tumor drugs.
    Biochemical pharmacology, 2006, Jul-28, Volume: 72, Issue:3

    Topics: Animals; Antineoplastic Agents; Aziridines; Benzopyrenes; Biotransformation; Cell Survival; Cells, Cultured; CHO Cells; Cricetinae; Cricetulus; Cross-Linking Reagents; DNA, Complementary; Dose-Response Relationship, Drug; Hydroquinones; Indolequinones; Keratinocytes; Mice; Mice, Knockout; Mitomycin; Mitomycins; Quinone Reductases; Quinones; Transfection; Vitamin K 3

2006