torpedo has been researched along with phencyclidine in 82 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 47 (57.32) | 18.7374 |
1990's | 25 (30.49) | 18.2507 |
2000's | 10 (12.20) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Duvvuri, P; Johnson, DA; Kerr, JA; Valenzuela, CF | 1 |
Erlinger, T; Herz, JM; Kolb, SJ; Schmid, E | 1 |
Donnelly-Roberts, DL; Lentz, TL | 1 |
Cohen, JB; Cohen, SG; Howard, S; White, BH | 1 |
Johnson, RG; Unsworth, CD | 1 |
Adam, LP; Henderson, EG | 1 |
Li, LA; McNamee, MG; Ochoa, EL; Plummer, A | 1 |
Eterović, VA; Li, L; McNamee, MG; Palma, A | 1 |
Albuquerque, EX; Aronstam, RS; Daly, JW; Feigl, DM; King, CT | 1 |
Aronstam, RS; Hong, JS | 1 |
Hess, GP; Karpen, JW | 1 |
Durkin, JA; Henley, JM; Simasko, SM; Weiland, GA | 1 |
Eriksson, H; Häggblad, J; Hedlund, B; Heilbronn, E | 1 |
Kavanaugh, MP; Tester, BA; Weber, E | 1 |
Diebler, MF; Gaudry-Talarmain, YM; O'Regan, S | 1 |
Diebler, MF; Gaudry-Talarmain, YM | 1 |
Noremberg, K; Parsons, SM | 1 |
Fehlmann, C; Kaufman, R; Parsons, SM; Rogers, GA | 1 |
Anderson, DC; Bahr, BA; Jacobs, RS; Kaufman, R; Kirtman, B; Kornreich, WD; Nilsson, LM; Parsons, SM; Rogers, GA | 1 |
Herz, JM; Johnson, DA; Taylor, P | 2 |
Kornreich, WD; Parsons, SM | 1 |
Bahr, BA; Gracz, LM; Kaufman, R; Kornreich, WD; Nilsson, L; Parsons, SM; Rogers, GA | 1 |
Gracz, LM; Parsons, SM; Wang, WC | 1 |
Bakry, NM; Eldefrawi, ME; Schweizer, G; Valdes, JJ | 1 |
Gershoni, JM; Haring, R; Kloog, Y; Mosckovitz, R; Sokolovsky, M | 1 |
Bahr, BA; Parsons, SM | 2 |
Changeux, JP; Dennis, M; Giraudat, J; Haumont, PY; Heidmann, T; Lederer, F | 1 |
Andreasen, GL; Berman, HA; Brown, RD; Herz, JM; Johnson, DA; Taylor, P | 1 |
Burstein, M; Licht, R; Michaelson, DM | 1 |
McLaughlin, JT; Oswald, RE; Pennow, NN | 1 |
Anderson, DC; Bahr, BA; Parsons, SM | 1 |
Bigelow, J; Michel, L; Oswald, RE | 1 |
Goeldner, M; Hirth, C; Jaganathen, J; Kotzyba-Hibert, F; Lagenbuch-Cachat, J | 1 |
Burstein, M; Michaelson, DM | 1 |
Carroll, PT | 1 |
Alkadhi, KA; Branisteanu, DD; Epstein, PM; Henderson, EG; Lambert, JJ; Reynolds, LS; Smilowitz, H; Volle, RL | 1 |
Eldefrawi, AT; Eldefrawi, ME; Miller, ER; Murphy, DL | 1 |
Aronstam, RS; Narayanan, L; Wenger, DA | 1 |
Aronstam, RS; Graham, JL; Narayanan, L | 1 |
Abbassy, MA; Ei-Fakahany, EF; Eldefrawi, AT; Eldefrawi, ME; Miller, ER | 1 |
Aronstam, RS; King, CT | 1 |
Haring, R; Kalir, A; Sokolovsky, M; Theomy, S | 1 |
Oswald, RE | 2 |
Epstein, PM; Lambert, JJ | 1 |
Haring, R; Kloog, Y | 1 |
Haring, R; Kloog, Y; Sokolovsky, M | 1 |
Bamberger, MJ; McLaughlin, JT; Oswald, RE | 1 |
Anderson, DC; King, SC; Parsons, SM | 1 |
Haring, R; Kalir, A; Kloog, Y; Sokolovsky, M | 1 |
Changeux, JP; Heidmann, T; Oswald, RE | 2 |
Changeux, JP; Oswald, RE | 1 |
Hescheler, J; Krautwurst, D; Musgrave, IF; Schultz, G | 1 |
Chi, M; Sun, M | 1 |
Min, CK; Weiland, GA | 1 |
Koblin, DD; Lin, L; Wang, HH | 1 |
Eterović, VA; Ferchmin, PA; Hann, RM; Lee, YH; Li, L; McNamee, MG; Rodriguez, AD | 1 |
Arias, HR; Johnson, DA; Valenzuela, CF | 2 |
Papineni, RV; Pedersen, SE | 1 |
Arias, HR | 2 |
Eaton, MJ; Eterović, VA; Hann, RM; Pagán, OR | 1 |
Cortes, VI; Eldefrawi, AT; Eldefrawi, ME; Katz, EJ | 1 |
Eterović, VA; Ferchmin, PA; Gregory, L; Hann, RM; Jácome, T; Lu, R; Pagán, OR; Rodríguez, AD | 1 |
Eldefrawi, ME; Eterović, VA; Hann, RM; Hess, GP; Ippolito, JE; Lis, JT; Pagán, OR; Shi, H; Ulrich, H | 1 |
Lurtz, MM; Pedersen, SE | 1 |
Blanton, MP; Machu, TK; McCardy, EA; Sun, H | 1 |
Eakin, AE; Eterović, VA; Ferchmin, PA; Lu, R; Rodríguez, AD | 1 |
Blanton, MP; Fryer, JD; Liu, M; Lukas, RJ; McCardy, EA | 1 |
Chiara, DC; Cohen, JB; Gallagher, MJ | 1 |
Basilio, CM; Eterović, VA; Garcia, M; Hann, RM; Pagán, OR; Rodríguez, AD; Vergne, D | 1 |
Arias, HR; Bayer, EZ; Blanton, MP; Gallagher, MJ; McCardy, EA | 1 |
Arias, HR; Bayer, EZ; Blanton, MP; Hester, B; McCardy, EA; Trudell, JR | 1 |
Arias, HR; Bouzat, C; Gumilar, F; Spitzmaul, G | 1 |
Andreeva, IE; Cohen, JB; Nirthanan, S; Pedersen, SE | 1 |
Arias, HR; Bhumireddy, P; Bouzat, C; Spitzmaul, G; Trudell, JR | 1 |
Oswald, RE; Pagán, OR; Sivaprakasam, K | 1 |
Blanton, MP; Chiara, DC; Cohen, JB; Hamouda, AK | 1 |
82 other study(ies) available for torpedo and phencyclidine
Article | Year |
---|---|
Modulation of phencyclidine-sensitive ethidium binding to the Torpedo acetylcholine receptor: interaction of noncompetitive inhibitors with carbamylcholine and cobra alpha-toxin.
Topics: Anesthetics; Animals; Barbiturates; Binding Sites; Binding, Competitive; Carbachol; Cholinergic Antagonists; Cobra Neurotoxin Proteins; Drug Interactions; Ethidium; Phencyclidine; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo | 1992 |
Channel permeant cations compete selectively with noncompetitive inhibitors of the nicotinic acetylcholine receptor.
Topics: Animals; Binding, Competitive; Cations; Ethidium; Ion Channels; Kinetics; Nicotinic Antagonists; Phencyclidine; Torpedo | 1991 |
Binding sites for alpha-bungarotoxin and the noncompetitive inhibitor phencyclidine on a synthetic peptide comprising residues 172-227 of the alpha-subunit of the nicotinic acetylcholine receptor.
Topics: Amino Acid Sequence; Animals; Binding Sites; Binding, Competitive; Bungarotoxins; Molecular Sequence Data; Peptide Fragments; Phencyclidine; Receptors, Nicotinic; Torpedo | 1991 |
The hydrophobic photoreagent 3-(trifluoromethyl)-3-m-([125I] iodophenyl) diazirine is a novel noncompetitive antagonist of the nicotinic acetylcholine receptor.
Topics: Affinity Labels; Amphibian Venoms; Animals; Azirines; Carbachol; Cell Membrane; Electric Organ; Iodine Radioisotopes; Kinetics; Macromolecular Substances; Nicotinic Antagonists; Phencyclidine; Receptors, Nicotinic; Sodium; Torpedo | 1991 |
Acetylcholine and ATP are coreleased from the electromotor nerve terminals of Narcine brasiliensis by an exocytotic mechanism.
Topics: Acetylcholine; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Calcimycin; Electric Organ; Exocytosis; Ionomycin; Kinetics; Motor Neurons; Nerve Endings; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Potassium; Subcellular Fractions; Synaptosomes; Torpedo; Veratridine | 1990 |
Calcium channel effectors are potent non-competitive blockers of acetylcholine receptors.
Topics: Animals; Bepridil; Calcium Channel Agonists; Calcium Channels; Cell Membrane; Electric Conductivity; Electric Organ; Electrophysiology; Ion Channel Gating; Mice; Motor Endplate; Muscle Contraction; Nicardipine; Nicotinic Antagonists; Phencyclidine; Rana pipiens; Torpedo | 1990 |
Direct effects of thymopentin (Arg-Lys-Asp-Val-Tyr) on cholinergic agonist-induced slow inactivation of nicotinic acetylcholine receptor function.
Topics: Animals; Bungarotoxins; Calcitonin Gene-Related Peptide; Calcium; Carbachol; In Vitro Techniques; Parasympathomimetics; Phencyclidine; Receptors, Nicotinic; Thymopentin; Thymopoietins; Torpedo; Xenopus laevis | 1990 |
Regulation of nicotinic acetylcholine receptor function by adenine nucleotides.
Topics: Acetylcholine; Adenine Nucleotides; Animals; Calcium; Choline; Drug Interactions; Mice; Nicotine; Oocytes; Phencyclidine; Receptors, Nicotinic; Recombinant Proteins; Torpedo; Xenopus laevis | 1990 |
Binding of [3H]perhydrohistrionicotoxin and [3H]phencyclidine to the nicotinic receptor-ion channel complex of Torpedo electroplax. Inhibition by histrionicotoxins and derivatives.
Topics: Amphibian Venoms; Animals; Binding, Competitive; Carbachol; Chemical Phenomena; Chemistry; Electric Organ; In Vitro Techniques; Ion Channels; Phencyclidine; Receptors, Nicotinic; Structure-Activity Relationship; Torpedo | 1985 |
Interactions of chlordecone (kepone) and mirex with the nicotinic acetylcholine receptor--ion channel complex.
Topics: Allosteric Regulation; Amphibian Venoms; Animals; Bungarotoxins; Carbachol; Chlordecone; Electric Organ; In Vitro Techniques; Insecticides; Ion Channels; Mirex; Phencyclidine; Receptors, Nicotinic; Torpedo | 1986 |
Cocaine, phencyclidine, and procaine inhibition of the acetylcholine receptor: characterization of the binding site by stopped-flow measurements of receptor-controlled ion flux in membrane vesicles.
Topics: Animals; Cell Membrane; Cocaine; Electric Organ; Electrophorus; Ion Channels; Kinetics; Mathematics; Membrane Potentials; Models, Biological; Phencyclidine; Procaine; Receptors, Cholinergic; Torpedo | 1986 |
Effects of substance P on the binding of ligands to nicotinic acetylcholine receptors.
Topics: Acetylcholine; Animals; Brain; Bungarotoxins; Electric Organ; Kinetics; Ligands; Nicotine; Phencyclidine; Receptors, Nicotinic; Substance P; Torpedo | 1987 |
Forskolin blocks carbachol-mediated ion-permeability of chick myotube nicotinic receptors and inhibits binding of 3H-phencyclidine to Torpedo microsac nicotinic receptors.
Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Chick Embryo; Cholera Toxin; Colforsin; Ethidium; In Vitro Techniques; Ion Channels; Microtubules; Phencyclidine; Receptors, Nicotinic; Rubidium Radioisotopes; Torpedo | 1987 |
Interaction of MK-801 with the nicotinic acetylcholine receptor-associated ion channel from electroplax.
Topics: Animals; Anticonvulsants; Dibenzocycloheptenes; Dizocilpine Maleate; Electric Organ; In Vitro Techniques; Ion Channels; Phencyclidine; Receptors, Cholinergic; Receptors, Nicotinic; Torpedo | 1989 |
Compared effects of two vesicular acetylcholine uptake blockers, AH5183 and cetiedil, on cholinergic functions in Torpedo synaptosomes: acetylcholine synthesis, choline transport, vesicular uptake, and evoked acetylcholine release.
Topics: Acetylcholine; Animals; Azepines; Biological Transport; Calcimycin; Choline; Electric Organ; Hydrogen-Ion Concentration; Kinetics; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Synaptic Vesicles; Synaptosomes; Torpedo | 1989 |
AH5183 and cetiedil: two potent inhibitors of acetylcholine uptake into isolated synaptic vesicles from Torpedo marmorata.
Topics: Acetylcholine; Adenosine Triphosphate; Animals; Azepines; Binding, Competitive; Biological Transport; Ca(2+) Mg(2+)-ATPase; Calcium; Electric Organ; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Synaptic Vesicles; Torpedo | 1989 |
Regulation of the vesamicol receptor in cholinergic synaptic vesicles by acetylcholine and an endogenous factor.
Topics: Acetylcholine; Animals; Binding, Competitive; Biological Transport, Active; Electric Organ; Kinetics; Neuromuscular Depolarizing Agents; Osmolar Concentration; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Phencyclidine; Synaptic Vesicles; Torpedo | 1989 |
Fractional vesamicol receptor occupancy and acetylcholine active transport inhibition in synaptic vesicles.
Topics: Acetylcholine; Animals; Binding, Competitive; Biological Transport, Active; In Vitro Techniques; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Phencyclidine; Structure-Activity Relationship; Synaptic Vesicles; Torpedo | 1989 |
Synthesis, in vitro acetylcholine-storage-blocking activities, and biological properties of derivatives and analogues of trans-2-(4-phenylpiperidino)cyclohexanol (vesamicol).
Topics: Acetylcholine; Animals; Biological Transport; Chemical Phenomena; Chemistry; Electric Organ; Lethal Dose 50; Mice; Molecular Structure; Narcotics; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Stereoisomerism; Structure-Activity Relationship; Synaptic Vesicles; Torpedo; X-Ray Diffraction | 1989 |
Distance between the agonist and noncompetitive inhibitor sites on the nicotinic acetylcholine receptor.
Topics: Animals; Binding Sites; Bungarotoxins; Choline; Dansyl Compounds; Electric Organ; Energy Transfer; Kinetics; Macromolecular Substances; Mathematics; Models, Biological; Models, Theoretical; Phencyclidine; Quaternary Ammonium Compounds; Receptors, Nicotinic; Torpedo | 1989 |
Sidedness and chemical and kinetic properties of the vesamicol receptor of cholinergic synaptic vesicles.
Topics: Acetylcholine; Algorithms; Animals; Cholinergic Fibers; Electric Organ; Hydrogen-Ion Concentration; Kinetics; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Phencyclidine; Synaptic Vesicles; Time Factors; Torpedo | 1988 |
Acetylcholine transport: fundamental properties and effects of pharmacologic agents.
Topics: Acetylcholine; Adenosine Triphosphatases; Animals; Biological Transport, Active; Electric Organ; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Phencyclidine; Synaptic Vesicles; Torpedo | 1987 |
Cholinergic synaptic vesicle heterogeneity: evidence for regulation of acetylcholine transport.
Topics: Acetylcholine; Animals; Biological Transport, Active; Cholinergic Fibers; Electric Organ; Nigericin; Phencyclidine; Piperidines; Synaptic Vesicles; Torpedo | 1988 |
Desensitization of the nicotinic acetylcholine receptor by diisopropylfluorophosphate.
Topics: Acetylcholine; Acetylcholinesterase; Animals; Bungarotoxins; Carbachol; Electric Organ; Isoflurophate; Kinetics; Phencyclidine; Receptors, Nicotinic; Torpedo | 1988 |
Localization of azidophencyclidine-binding site on the nicotinic acetylcholine receptor alpha-subunit.
Topics: Affinity Labels; Animals; Azides; Cyanogen Bromide; Endopeptidases; Macromolecular Substances; Molecular Weight; Peptide Fragments; Phencyclidine; Photochemistry; Receptors, Cholinergic; Serine Endopeptidases; Torpedo | 1987 |
Demonstration of a receptor in Torpedo synaptic vesicles for the acetylcholine storage blocker L-trans-2-(4-phenyl[3,4-3H]-piperidino) cyclohexanol.
Topics: Acetylcholine; Animals; Binding, Competitive; Choline; Electric Organ; Kinetics; Phencyclidine; Piperidines; Receptors, Drug; Stereoisomerism; Synaptic Vesicles; Torpedo | 1986 |
Interaction of noncompetitive inhibitors with the acetylcholine receptor. The site specificity and spectroscopic properties of ethidium binding.
Topics: Acetylcholine; Allosteric Site; Animals; Binding Sites; Binding, Competitive; Carbachol; Cell Membrane; Electric Organ; Ethidium; Fluorescence; Fluorescence Polarization; Phencyclidine; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo | 1987 |
Structure of the high-affinity binding site for noncompetitive blockers of the acetylcholine receptor: [3H]chlorpromazine labels homologous residues in the beta and delta chains.
Topics: Amino Acid Sequence; Amino Acids; Animals; Carbachol; Cell Membrane; Chlorpromazine; Macromolecular Substances; Models, Molecular; Peptide Fragments; Phencyclidine; Receptors, Cholinergic; Torpedo | 1987 |
Decidium. A novel fluorescent probe of the agonist/antagonist and noncompetitive inhibitor sites on the nicotinic acetylcholine receptor.
Topics: Animals; Binding, Competitive; Cell Line; Cell Membrane; Electric Organ; Kinetics; Phenanthridines; Phencyclidine; Receptors, Nicotinic; Spectrometry, Fluorescence; Torpedo | 1987 |
Translocation of cytosolic acetylcholine into synaptic vesicles and demonstration of vesicular release.
Topics: Acetylcholine; Animals; Biological Transport; Cytosol; Electric Organ; Kinetics; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Synaptic Vesicles; Synaptosomes; Torpedo | 1986 |
Demonstration and affinity labeling of a stereoselective binding site for a benzomorphan opiate on acetylcholine receptor-rich membranes from Torpedo electroplaque.
Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Electric Organ; Electrophoresis, Polyacrylamide Gel; Kinetics; Phenazocine; Phencyclidine; Photochemistry; Receptors, Cholinergic; Torpedo | 1985 |
Stoichiometries of acetylcholine uptake, release, and drug inhibition in Torpedo synaptic vesicles: heterogeneity in acetylcholine transport and storage.
Topics: Acetylcholine; Animals; Biological Transport, Active; Electric Organ; Hemicholinium 3; Phencyclidine; Piperidines; Quinacrine; Synaptic Vesicles; Torpedo | 1986 |
Acetylcholine transport and drug inhibition kinetics in Torpedo synaptic vesicles.
Topics: Acetylcholine; Allosteric Regulation; Animals; Biological Transport, Active; Electric Organ; Kinetics; Phencyclidine; Piperidines; Synaptic Vesicles; Torpedo | 1986 |
Mechanism of binding of a benzomorphan opiate to the acetylcholine receptor from Torpedo electroplaque.
Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Carbachol; Decamethonium Compounds; In Vitro Techniques; Kinetics; Phenazocine; Phencyclidine; Receptors, Cholinergic; Structure-Activity Relationship; Tetracaine; Torpedo; Tritium; Tubocurarine | 1986 |
Aryldiazonium salts as photoaffinity labels of the nicotinic acetylcholine receptor PCP binding site.
Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Carbachol; Diazonium Compounds; Electric Organ; Phencyclidine; Photochemistry; Receptors, Nicotinic; Torpedo | 1985 |
Biochemical evidence that acetylcholine release from cholinergic nerve terminals is mostly vesicular.
Topics: Acetates; Acetylcholine; Animals; Electric Organ; In Vitro Techniques; Phencyclidine; Piperidines; Synaptic Vesicles; Synaptosomes; Torpedo | 1985 |
The effect of the acetylcholine transport blocker 2-(4-phenylpiperidino) cyclohexanol (AH5183) on the subcellular storage and release of acetylcholine in mouse brain.
Topics: Acetylcholine; Animals; Biological Transport; Brain; Electric Organ; Mice; Mice, Inbred ICR; Phencyclidine; Piperidines; Potassium; Synaptic Vesicles; Torpedo; Veratridine | 1985 |
Ketamine and ditran block end-plate ion conductance and [3H]phencyclidine binding to electric organ membrane.
Topics: Animals; Drug Combinations; Electric Organ; Glycolates; Hydrogen-Ion Concentration; In Vitro Techniques; Ion Channels; Ketamine; Neurotransmitter Agents; Phencyclidine; Piperidines; Pyrrolidines; Rana pipiens; Receptors, Cholinergic; Torpedo | 1982 |
[3H]Phencyclidine interactions with the nicotinic acetylcholine receptor channel and its inhibition by psychotropic, antipsychotic, opiate, antidepressant, antibiotic, antiviral, and antiarrhythmic drugs.
Topics: Allosteric Site; Animals; Anti-Arrhythmia Agents; Anti-Bacterial Agents; Antidepressive Agents; Antipsychotic Agents; Antiviral Agents; Binding, Competitive; Electric Organ; In Vitro Techniques; Ion Channels; Narcotics; Phencyclidine; Psychotropic Drugs; Receptors, Cholinergic; Receptors, Nicotinic; Torpedo | 1982 |
Ketamine inhibition of ligand binding to cholinergic receptors and ion channels.
Topics: Acetylcholine; Animals; Electric Organ; In Vitro Techniques; Ion Channels; Ketamine; Ligands; N-Methylscopolamine; Phencyclidine; Receptors, Cholinergic; Scopolamine Derivatives; Torpedo; Tubocurarine | 1982 |
Receptor--ion channel interactions in Torpedo electric organ: influence of thiol group modification.
Topics: Animals; Dithionitrobenzoic Acid; Dithiothreitol; Electric Organ; Ethylmaleimide; Ion Channels; Nitrobenzoates; Phencyclidine; Receptors, Cholinergic; Receptors, Nicotinic; Torpedo | 1982 |
Alcohol modulation of drug binding to the channel sites of the nicotinic acetylcholine receptor.
Topics: Alcohols; Amphibian Venoms; Animals; Carbachol; Drug Interactions; Imipramine; Ion Channels; Membranes; Naphthols; Phencyclidine; Receptors, Cholinergic; Torpedo | 1983 |
Benzomorphan interactions with acetylcholine receptor complexes from Torpedo.
Topics: Amphibian Venoms; Animals; Benzomorphans; Drug Interactions; Ion Channels; Morphinans; Parasympatholytics; Phencyclidine; Receptors, Cholinergic; Receptors, Nicotinic; Receptors, Opioid; Torpedo | 1983 |
Characterization of the interaction of phencyclidine and its derivatives with the ionic channel of the nicotinic receptor.
Topics: Animals; Electric Organ; In Vitro Techniques; Ion Channels; Kinetics; Phencyclidine; Receptors, Nicotinic; Torpedo | 1983 |
Effects of calcium on the binding of phencyclidine to acetylcholine receptor-rich membrane fragments from Torpedo californica electroplaque.
Topics: Animals; Calcium; Carbachol; Cations, Divalent; Cell Membrane; Egtazic Acid; Electric Organ; Phencyclidine; Receptors, Cholinergic; Torpedo | 1983 |
Displacement of [3H]phencyclidine binding to Torpedo electric organ membrane by calcium channel antagonists.
Topics: Animals; Calcium Channel Blockers; Calcium Chloride; Cell Membrane; Electric Organ; In Vitro Techniques; Phencyclidine; Torpedo; Tritium | 1984 |
Multiple binding sites for phencyclidine on the nicotinic acetylcholine receptor from Torpedo ocellata electric organ.
Topics: Acetylcholine; Animals; Binding Sites; Bungarotoxins; Carbachol; Dibucaine; Electric Organ; Kinetics; Phencyclidine; Receptors, Cholinergic; Tetracaine; Torpedo; Tubocurarine | 1984 |
Localization of phencyclidine binding sites on alpha and beta subunits of the nicotinic acetylcholine receptor from Torpedo ocellata electric organ using azido phencyclidine.
Topics: Affinity Labels; Animals; Azides; Binding Sites; Binding, Competitive; Carbachol; Cell Membrane; Electric Organ; Macromolecular Substances; Molecular Weight; Phencyclidine; Photochemistry; Receptors, Nicotinic; Torpedo | 1984 |
Mechanism of phencyclidine binding to the acetylcholine receptor from Torpedo electroplaque.
Topics: Animals; Carbachol; Cell Membrane; Electric Organ; Glycerol; Kinetics; Phencyclidine; Receptors, Cholinergic; Temperature; Thermodynamics; Torpedo | 1984 |
Binding of phencyclidine to the detergent solubilized acetylcholine receptor from Torpedo marmorata.
Topics: Animals; Cholic Acid; Cholic Acids; Electric Organ; Kinetics; Phencyclidine; Polysorbates; Receptors, Cholinergic; Solubility; Torpedo | 1983 |
Pharmacological characterization of the acetylcholine transport system in purified Torpedo electric organ synaptic vesicles.
Topics: Acetylcholine; Animals; Binding Sites; Biological Transport, Active; Electric Organ; In Vitro Techniques; Phencyclidine; Piperidines; Receptors, Cholinergic; Synaptic Vesicles; Torpedo | 1983 |
Species differences determine azido phencyclidine labeling pattern in desensitized nicotinic acetylcholine receptors.
Topics: Affinity Labels; Animals; Azides; Electrophoresis, Polyacrylamide Gel; Isotope Labeling; Phencyclidine; Photochemistry; Receptors, Cholinergic; Receptors, Nicotinic; Species Specificity; Torpedo; Tritium | 1983 |
Multiple sites of action for noncompetitive blockers on acetylcholine receptor rich membrane fragments from torpedo marmorata.
Topics: Alkanes; Allosteric Regulation; Amphibian Venoms; Animals; Binding Sites; Chlorpromazine; Electric Organ; Isoquinolines; Membrane Lipids; Neuromuscular Junction; Parasympatholytics; Phencyclidine; Polyethylene Glycols; Proadifen; Receptors, Cholinergic; Torpedo | 1983 |
Multiple affinity states for noncompetitive blockers revealed by [3H]phencyclidine binding to acetylcholine receptor rich membrane fragments from Torpedo marmorata.
Topics: Allosteric Regulation; Animals; Binding Sites; Electric Organ; Kinetics; Neuromuscular Junction; Phencyclidine; Protein Binding; Protein Conformation; Receptors, Cholinergic; Torpedo | 1983 |
Selective labeling of the delta subunit of the acetylcholine receptor by a covalent local anesthetic.
Topics: Acetylcholine; Affinity Labels; Animals; Azides; Binding, Competitive; Cell Membrane; Electric Organ; Isoquinolines; Kinetics; Macromolecular Substances; Phencyclidine; Receptors, Cholinergic; Torpedo | 1981 |
Clonidine and cirazoline inhibit activation of nicotinic channels in PC-12 cells.
Topics: Adrenergic alpha-Agonists; Animals; Binding Sites; Calcium; Clonidine; Imidazoles; Ion Channels; Nicotinic Antagonists; PC12 Cells; Phencyclidine; Radioligand Assay; Rats; Receptors, Nicotinic; Torpedo; Tritium | 1995 |
Action of organophosphate anticholinesterases on the three conformational states of nicotinic receptor.
Topics: Animals; Cholinesterase Inhibitors; Cobra Neurotoxin Proteins; Organophosphorus Compounds; Phencyclidine; Protein Conformation; Receptors, Nicotinic; Soman; Torpedo; Tubocurarine | 1995 |
Effects of substance P on the binding of agonists to the nicotinic acetylcholine receptor of Torpedo electroplaque.
Topics: Acetylcholine; Animals; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Kinetics; Least-Squares Analysis; Mathematics; Models, Theoretical; Phencyclidine; Receptors, Nicotinic; Substance P; Time Factors; Torpedo | 1993 |
Effects of halothane on the nicotinic acetylcholine receptor from Torpedo californica.
Topics: Animals; Binding, Competitive; Halothane; Kinetics; Nicotinic Antagonists; Phencyclidine; Receptors, Nicotinic; Torpedo | 1995 |
The ion channel of muscle and electric organ acetylcholine receptors: differing affinities for noncompetitive inhibitors.
Topics: Amino Acid Sequence; Animals; Cell Line; Diterpenes; Electric Organ; Ion Channel Gating; Magnesium; Membrane Potentials; Mice; Molecular Sequence Data; Muscle Proteins; Nerve Tissue Proteins; Nicotinic Antagonists; Oocytes; Organ Specificity; Phencyclidine; Recombinant Proteins; Sequence Homology, Amino Acid; Sodium Channels; Tetracaine; Torpedo; Xenopus laevis | 1993 |
Transverse localization of the quinacrine binding site on the Torpedo acetylcholine receptor.
Topics: Animals; Binding Sites; Cell Membrane; Iodides; Kinetics; Phencyclidine; Quinacrine; Receptors, Cholinergic; Rhodamines; Stearates; Torpedo | 1993 |
Quinacrine and ethidium bind to different loci on the Torpedo acetylcholine receptor.
Topics: Animals; Binding Sites; Cell Membrane; Ethidium; Phencyclidine; Quinacrine; Receptors, Cholinergic; Spectrometry, Fluorescence; Spin Labels; Torpedo | 1993 |
Interaction of d-tubocurarine analogs with the Torpedo nicotinic acetylcholine receptor. Methylation and stereoisomerization affect site-selective competitive binding and binding to the noncompetitive site.
Topics: Animals; Binding, Competitive; Methylation; Nicotinic Agonists; Nicotinic Antagonists; Phencyclidine; Receptors, Nicotinic; Stereoisomerism; Torpedo; Tritium; Tubocurarine | 1995 |
Temperature and ionic strength dependence of quinacrine binding and quinacrine displacement elicited by high concentrations of agonists on the nicotinic acetylcholine receptor.
Topics: Animals; Binding Sites; Electric Organ; In Vitro Techniques; Kinetics; Models, Biological; Nicotinic Agonists; Osmolar Concentration; Phencyclidine; Quinacrine; Receptors, Nicotinic; Sodium Chloride; Temperature; Thermodynamics; Torpedo | 1996 |
Differential effects of dimethyl sulfoxide on nicotinic acetylcholine receptors from mouse muscle and Torpedo electrocytes.
Topics: Administration, Topical; Animals; Anti-Inflammatory Agents; Bungarotoxins; Dimethyl Sulfoxide; Excitatory Amino Acid Antagonists; Female; Iodine Radioisotopes; Ion Channel Gating; Mice; Oocytes; Patch-Clamp Techniques; Phencyclidine; Radioligand Assay; Receptors, Nicotinic; Torpedo; Tritium; Xenopus laevis | 1997 |
Chlorpyrifos, parathion, and their oxons bind to and desensitize a nicotinic acetylcholine receptor: relevance to their toxicities.
Topics: Animals; Binding, Competitive; Bungarotoxins; Carbachol; Chlorpyrifos; Cholinesterase Inhibitors; Cholinesterases; Dose-Response Relationship, Drug; Insecticides; Iodine Radioisotopes; Lethal Dose 50; Nicotinic Agonists; Paraoxon; Parathion; Phencyclidine; Receptors, Nicotinic; Structure-Activity Relationship; Torpedo; Tritium | 1997 |
Characterization of cembranoid interaction with the nicotinic acetylcholine receptor.
Topics: Acetylcholine; Animals; Binding Sites; Bungarotoxins; Diterpenes; Female; Phencyclidine; Receptors, Nicotinic; Torpedo; Xenopus laevis | 1998 |
In vitro selection of RNA molecules that displace cocaine from the membrane-bound nicotinic acetylcholine receptor.
Topics: Animals; Base Sequence; Binding Sites; Binding, Competitive; Cell Membrane; Cocaine; Consensus Sequence; Electric Organ; Illicit Drugs; Kinetics; Ligands; Molecular Sequence Data; Nucleic Acid Conformation; Oligodeoxyribonucleotides; Phencyclidine; Receptors, Nicotinic; RNA; Sequence Alignment; Torpedo | 1998 |
Aminotriarylmethane dyes are high-affinity noncompetitive antagonists of the nicotinic acetylcholine receptor.
Topics: Animals; Binding Sites; Binding, Competitive; Coloring Agents; Gentian Violet; Nicotinic Antagonists; Phencyclidine; Protein Conformation; Receptors, Nicotinic; Sodium; Spectrometry, Fluorescence; Structure-Activity Relationship; Torpedo | 1999 |
Characterization of interaction of 3,4,5-trimethoxybenzoic acid 8-(diethylamino)octyl ester with Torpedo californica nicotinic acetylcholine receptor and 5-hydroxytryptamine3 receptor.
Topics: Amino Acid Sequence; Animals; Binding, Competitive; Cell Membrane; Electrophysiology; Gallic Acid; Humans; In Vitro Techniques; Iodine Radioisotopes; Mice; Molecular Sequence Data; Nicotinic Antagonists; Oocytes; Phencyclidine; Radioligand Assay; Receptors, Nicotinic; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Torpedo; Xenopus laevis | 1999 |
Determinants of phencyclidine potency on the nicotinic acetylcholine receptors from muscle and electric organ.
Topics: Acetylcholine; Amino Acid Sequence; Amino Acid Substitution; Animals; Atropine; Binding Sites; Diterpenes; DNA, Complementary; Dose-Response Relationship, Drug; Electric Organ; Ion Channel Gating; Ion Channels; Kinetics; Mice; Molecular Sequence Data; Muscle Proteins; Muscle, Skeletal; Mutagenesis, Site-Directed; Nerve Tissue Proteins; Nicotinic Antagonists; Patch-Clamp Techniques; Phencyclidine; Point Mutation; Protein Multimerization; Receptors, Nicotinic; Recombinant Fusion Proteins; Sequence Alignment; Sequence Homology, Amino Acid; Torpedo; Xenopus laevis | 1999 |
5-Doxylstearate-induced displacement of phencyclidine from its low-affinity binding sites on the nicotinic acetylcholine receptor.
Topics: Animals; Binding Sites; Binding, Competitive; Cell Membrane; Cyclic N-Oxides; Electric Organ; Ethidium; Kinetics; Phencyclidine; Quinacrine; Receptors, Nicotinic; Spin Labels; Torpedo; Tritium | 1999 |
5-hydroxytryptamine interaction with the nicotinic acetylcholine receptor.
Topics: Animals; Binding Sites; Bungarotoxins; Cells, Cultured; Dose-Response Relationship, Drug; Humans; Phencyclidine; Photoaffinity Labels; Receptors, Nicotinic; Serotonin; Torpedo | 2000 |
Interactions between 3-(Trifluoromethyl)-3-(m-[(125)I]iodophenyl)diazirine and tetracaine, phencyclidine, or histrionicotoxin in the Torpedo series nicotinic acetylcholine receptor ion channel.
Topics: Affinity Labels; Amphibian Venoms; Anesthetics, Local; Animals; Azirines; Ceramides; Drug Interactions; Excitatory Amino Acid Antagonists; Iodine Radioisotopes; Membrane Proteins; Phencyclidine; Receptors, Nicotinic; Tetracaine; Torpedo | 2001 |
Cembranoid and long-chain alkanol sites on the nicotinic acetylcholine receptor and their allosteric interaction.
Topics: Allosteric Regulation; Anesthetics; Animals; Binding Sites; Binding, Competitive; Diterpenes; Fatty Alcohols; Hexanols; Models, Theoretical; Nicotinic Antagonists; Octanols; Phencyclidine; Procaine; Receptors, Nicotinic; Torpedo | 2001 |
Allosterically linked noncompetitive antagonist binding sites in the resting nicotinic acetylcholine receptor ion channel.
Topics: Allosteric Site; Amobarbital; Anesthetics, Local; Animals; Binding Sites; Binding, Competitive; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Modulators; Inhibitory Concentration 50; Ions; Ketamine; Kinetics; Light; Models, Molecular; Phencyclidine; Protein Binding; Protein Conformation; Receptors, Nicotinic; Tetracaine; Torpedo | 2002 |
Noncompetitive antagonist binding sites in the torpedo nicotinic acetylcholine receptor ion channel. Structure-activity relationship studies using adamantane derivatives.
Topics: Adamantane; Allosteric Site; Anesthetics, Local; Animals; Binding Sites; Binding, Competitive; Excitatory Amino Acid Antagonists; Iodine Isotopes; Ion Channels; Models, Molecular; Nicotinic Antagonists; Phencyclidine; Protein Binding; Receptors, Nicotinic; Structure-Activity Relationship; Thermodynamics; Torpedo; Tritium | 2003 |
Molecular mechanisms of inhibition of nicotinic acetylcholine receptors by tricyclic antidepressants.
Topics: Acetylcholine; Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Cell Membrane; Doxepin; Excitatory Amino Acid Antagonists; Humans; Imipramine; In Vitro Techniques; Kidney; Kinetics; Membrane Potentials; Mice; Nicotinic Antagonists; Patch-Clamp Techniques; Phencyclidine; Receptors, Nicotinic; Torpedo | 2003 |
Site specificity of agonist-induced opening and desensitization of the Torpedo californica nicotinic acetylcholine receptor.
Topics: Animals; Binding Sites; Calcium Channel Blockers; Conotoxins; Dansyl Compounds; Enzyme Inhibitors; Fluorescent Dyes; Kinetics; Nicotinic Agonists; Phencyclidine; Proadifen; Quaternary Ammonium Compounds; Receptors, Nicotinic; Spectrometry, Fluorescence; Structure-Activity Relationship; Torpedo; Tubocurarine | 2006 |
Molecular mechanisms and binding site location for the noncompetitive antagonist crystal violet on nicotinic acetylcholine receptors.
Topics: Allosteric Regulation; Amobarbital; Animals; Binding Sites; Fluorescent Dyes; Gentian Violet; Ion Channels; Models, Molecular; Nicotinic Agonists; Nicotinic Antagonists; Pentobarbital; Phencyclidine; Protein Binding; Protein Conformation; Quaternary Ammonium Compounds; Receptors, Nicotinic; Temperature; Tetracaine; Thiophenes; Torpedo; Tritium | 2006 |
Molecular properties of local anesthetics as predictors of affinity for nicotinic acetylcholine receptors.
Topics: Anesthetics, Local; Animals; Binding, Competitive; Bungarotoxins; Cell Membrane; Electric Organ; Neuroprotective Agents; Phencyclidine; Predictive Value of Tests; Protein Conformation; Receptors, Nicotinic; Torpedo; Tritium | 2007 |
Probing the structure of the affinity-purified and lipid-reconstituted torpedo nicotinic acetylcholine receptor.
Topics: Affinity Labels; Animals; Azirines; Binding Sites; Cholates; Iodine Radioisotopes; Ion Channels; Lipid Metabolism; Models, Molecular; Nicotinic Antagonists; Phencyclidine; Protein Structure, Secondary; Protein Structure, Tertiary; Receptors, Nicotinic; Solubility; Spectroscopy, Fourier Transform Infrared; Staining and Labeling; Substrate Specificity; Torpedo | 2008 |