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torpedo and phencyclidine

torpedo has been researched along with phencyclidine in 82 studies

Research

Studies (82)

TimeframeStudies, this research(%)All Research%
pre-199047 (57.32)18.7374
1990's25 (30.49)18.2507
2000's10 (12.20)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Duvvuri, P; Johnson, DA; Kerr, JA; Valenzuela, CF1
Erlinger, T; Herz, JM; Kolb, SJ; Schmid, E1
Donnelly-Roberts, DL; Lentz, TL1
Cohen, JB; Cohen, SG; Howard, S; White, BH1
Johnson, RG; Unsworth, CD1
Adam, LP; Henderson, EG1
Li, LA; McNamee, MG; Ochoa, EL; Plummer, A1
Eterović, VA; Li, L; McNamee, MG; Palma, A1
Albuquerque, EX; Aronstam, RS; Daly, JW; Feigl, DM; King, CT1
Aronstam, RS; Hong, JS1
Hess, GP; Karpen, JW1
Durkin, JA; Henley, JM; Simasko, SM; Weiland, GA1
Eriksson, H; Häggblad, J; Hedlund, B; Heilbronn, E1
Kavanaugh, MP; Tester, BA; Weber, E1
Diebler, MF; Gaudry-Talarmain, YM; O'Regan, S1
Diebler, MF; Gaudry-Talarmain, YM1
Noremberg, K; Parsons, SM1
Fehlmann, C; Kaufman, R; Parsons, SM; Rogers, GA1
Anderson, DC; Bahr, BA; Jacobs, RS; Kaufman, R; Kirtman, B; Kornreich, WD; Nilsson, LM; Parsons, SM; Rogers, GA1
Herz, JM; Johnson, DA; Taylor, P2
Kornreich, WD; Parsons, SM1
Bahr, BA; Gracz, LM; Kaufman, R; Kornreich, WD; Nilsson, L; Parsons, SM; Rogers, GA1
Gracz, LM; Parsons, SM; Wang, WC1
Bakry, NM; Eldefrawi, ME; Schweizer, G; Valdes, JJ1
Gershoni, JM; Haring, R; Kloog, Y; Mosckovitz, R; Sokolovsky, M1
Bahr, BA; Parsons, SM2
Changeux, JP; Dennis, M; Giraudat, J; Haumont, PY; Heidmann, T; Lederer, F1
Andreasen, GL; Berman, HA; Brown, RD; Herz, JM; Johnson, DA; Taylor, P1
Burstein, M; Licht, R; Michaelson, DM1
McLaughlin, JT; Oswald, RE; Pennow, NN1
Anderson, DC; Bahr, BA; Parsons, SM1
Bigelow, J; Michel, L; Oswald, RE1
Goeldner, M; Hirth, C; Jaganathen, J; Kotzyba-Hibert, F; Lagenbuch-Cachat, J1
Burstein, M; Michaelson, DM1
Carroll, PT1
Alkadhi, KA; Branisteanu, DD; Epstein, PM; Henderson, EG; Lambert, JJ; Reynolds, LS; Smilowitz, H; Volle, RL1
Eldefrawi, AT; Eldefrawi, ME; Miller, ER; Murphy, DL1
Aronstam, RS; Narayanan, L; Wenger, DA1
Aronstam, RS; Graham, JL; Narayanan, L1
Abbassy, MA; Ei-Fakahany, EF; Eldefrawi, AT; Eldefrawi, ME; Miller, ER1
Aronstam, RS; King, CT1
Haring, R; Kalir, A; Sokolovsky, M; Theomy, S1
Oswald, RE2
Epstein, PM; Lambert, JJ1
Haring, R; Kloog, Y1
Haring, R; Kloog, Y; Sokolovsky, M1
Bamberger, MJ; McLaughlin, JT; Oswald, RE1
Anderson, DC; King, SC; Parsons, SM1
Haring, R; Kalir, A; Kloog, Y; Sokolovsky, M1
Changeux, JP; Heidmann, T; Oswald, RE2
Changeux, JP; Oswald, RE1
Hescheler, J; Krautwurst, D; Musgrave, IF; Schultz, G1
Chi, M; Sun, M1
Min, CK; Weiland, GA1
Koblin, DD; Lin, L; Wang, HH1
Eterović, VA; Ferchmin, PA; Hann, RM; Lee, YH; Li, L; McNamee, MG; Rodriguez, AD1
Arias, HR; Johnson, DA; Valenzuela, CF2
Papineni, RV; Pedersen, SE1
Arias, HR2
Eaton, MJ; Eterović, VA; Hann, RM; Pagán, OR1
Cortes, VI; Eldefrawi, AT; Eldefrawi, ME; Katz, EJ1
Eterović, VA; Ferchmin, PA; Gregory, L; Hann, RM; Jácome, T; Lu, R; Pagán, OR; Rodríguez, AD1
Eldefrawi, ME; Eterović, VA; Hann, RM; Hess, GP; Ippolito, JE; Lis, JT; Pagán, OR; Shi, H; Ulrich, H1
Lurtz, MM; Pedersen, SE1
Blanton, MP; Machu, TK; McCardy, EA; Sun, H1
Eakin, AE; Eterović, VA; Ferchmin, PA; Lu, R; Rodríguez, AD1
Blanton, MP; Fryer, JD; Liu, M; Lukas, RJ; McCardy, EA1
Chiara, DC; Cohen, JB; Gallagher, MJ1
Basilio, CM; Eterović, VA; Garcia, M; Hann, RM; Pagán, OR; Rodríguez, AD; Vergne, D1
Arias, HR; Bayer, EZ; Blanton, MP; Gallagher, MJ; McCardy, EA1
Arias, HR; Bayer, EZ; Blanton, MP; Hester, B; McCardy, EA; Trudell, JR1
Arias, HR; Bouzat, C; Gumilar, F; Spitzmaul, G1
Andreeva, IE; Cohen, JB; Nirthanan, S; Pedersen, SE1
Arias, HR; Bhumireddy, P; Bouzat, C; Spitzmaul, G; Trudell, JR1
Oswald, RE; Pagán, OR; Sivaprakasam, K1
Blanton, MP; Chiara, DC; Cohen, JB; Hamouda, AK1

Other Studies

82 other study(ies) available for torpedo and phencyclidine

ArticleYear
Modulation of phencyclidine-sensitive ethidium binding to the Torpedo acetylcholine receptor: interaction of noncompetitive inhibitors with carbamylcholine and cobra alpha-toxin.
    Molecular pharmacology, 1992, Volume: 41, Issue:2

    Topics: Anesthetics; Animals; Barbiturates; Binding Sites; Binding, Competitive; Carbachol; Cholinergic Antagonists; Cobra Neurotoxin Proteins; Drug Interactions; Ethidium; Phencyclidine; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo

1992
Channel permeant cations compete selectively with noncompetitive inhibitors of the nicotinic acetylcholine receptor.
    The Journal of biological chemistry, 1991, Sep-05, Volume: 266, Issue:25

    Topics: Animals; Binding, Competitive; Cations; Ethidium; Ion Channels; Kinetics; Nicotinic Antagonists; Phencyclidine; Torpedo

1991
Binding sites for alpha-bungarotoxin and the noncompetitive inhibitor phencyclidine on a synthetic peptide comprising residues 172-227 of the alpha-subunit of the nicotinic acetylcholine receptor.
    Biochemistry, 1991, Jul-30, Volume: 30, Issue:30

    Topics: Amino Acid Sequence; Animals; Binding Sites; Binding, Competitive; Bungarotoxins; Molecular Sequence Data; Peptide Fragments; Phencyclidine; Receptors, Nicotinic; Torpedo

1991
The hydrophobic photoreagent 3-(trifluoromethyl)-3-m-([125I] iodophenyl) diazirine is a novel noncompetitive antagonist of the nicotinic acetylcholine receptor.
    The Journal of biological chemistry, 1991, Nov-15, Volume: 266, Issue:32

    Topics: Affinity Labels; Amphibian Venoms; Animals; Azirines; Carbachol; Cell Membrane; Electric Organ; Iodine Radioisotopes; Kinetics; Macromolecular Substances; Nicotinic Antagonists; Phencyclidine; Receptors, Nicotinic; Sodium; Torpedo

1991
Acetylcholine and ATP are coreleased from the electromotor nerve terminals of Narcine brasiliensis by an exocytotic mechanism.
    Proceedings of the National Academy of Sciences of the United States of America, 1990, Volume: 87, Issue:2

    Topics: Acetylcholine; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Calcimycin; Electric Organ; Exocytosis; Ionomycin; Kinetics; Motor Neurons; Nerve Endings; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Potassium; Subcellular Fractions; Synaptosomes; Torpedo; Veratridine

1990
Calcium channel effectors are potent non-competitive blockers of acetylcholine receptors.
    Pflugers Archiv : European journal of physiology, 1990, Volume: 416, Issue:5

    Topics: Animals; Bepridil; Calcium Channel Agonists; Calcium Channels; Cell Membrane; Electric Conductivity; Electric Organ; Electrophysiology; Ion Channel Gating; Mice; Motor Endplate; Muscle Contraction; Nicardipine; Nicotinic Antagonists; Phencyclidine; Rana pipiens; Torpedo

1990
Direct effects of thymopentin (Arg-Lys-Asp-Val-Tyr) on cholinergic agonist-induced slow inactivation of nicotinic acetylcholine receptor function.
    Molecular pharmacology, 1990, Volume: 38, Issue:6

    Topics: Animals; Bungarotoxins; Calcitonin Gene-Related Peptide; Calcium; Carbachol; In Vitro Techniques; Parasympathomimetics; Phencyclidine; Receptors, Nicotinic; Thymopentin; Thymopoietins; Torpedo; Xenopus laevis

1990
Regulation of nicotinic acetylcholine receptor function by adenine nucleotides.
    Cellular and molecular neurobiology, 1990, Volume: 10, Issue:3

    Topics: Acetylcholine; Adenine Nucleotides; Animals; Calcium; Choline; Drug Interactions; Mice; Nicotine; Oocytes; Phencyclidine; Receptors, Nicotinic; Recombinant Proteins; Torpedo; Xenopus laevis

1990
Binding of [3H]perhydrohistrionicotoxin and [3H]phencyclidine to the nicotinic receptor-ion channel complex of Torpedo electroplax. Inhibition by histrionicotoxins and derivatives.
    Biochemical pharmacology, 1985, Sep-01, Volume: 34, Issue:17

    Topics: Amphibian Venoms; Animals; Binding, Competitive; Carbachol; Chemical Phenomena; Chemistry; Electric Organ; In Vitro Techniques; Ion Channels; Phencyclidine; Receptors, Nicotinic; Structure-Activity Relationship; Torpedo

1985
Interactions of chlordecone (kepone) and mirex with the nicotinic acetylcholine receptor--ion channel complex.
    Toxicology letters, 1986, Volume: 30, Issue:3

    Topics: Allosteric Regulation; Amphibian Venoms; Animals; Bungarotoxins; Carbachol; Chlordecone; Electric Organ; In Vitro Techniques; Insecticides; Ion Channels; Mirex; Phencyclidine; Receptors, Nicotinic; Torpedo

1986
Cocaine, phencyclidine, and procaine inhibition of the acetylcholine receptor: characterization of the binding site by stopped-flow measurements of receptor-controlled ion flux in membrane vesicles.
    Biochemistry, 1986, Apr-08, Volume: 25, Issue:7

    Topics: Animals; Cell Membrane; Cocaine; Electric Organ; Electrophorus; Ion Channels; Kinetics; Mathematics; Membrane Potentials; Models, Biological; Phencyclidine; Procaine; Receptors, Cholinergic; Torpedo

1986
Effects of substance P on the binding of ligands to nicotinic acetylcholine receptors.
    Molecular pharmacology, 1987, Volume: 32, Issue:5

    Topics: Acetylcholine; Animals; Brain; Bungarotoxins; Electric Organ; Kinetics; Ligands; Nicotine; Phencyclidine; Receptors, Nicotinic; Substance P; Torpedo

1987
Forskolin blocks carbachol-mediated ion-permeability of chick myotube nicotinic receptors and inhibits binding of 3H-phencyclidine to Torpedo microsac nicotinic receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 336, Issue:4

    Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Chick Embryo; Cholera Toxin; Colforsin; Ethidium; In Vitro Techniques; Ion Channels; Microtubules; Phencyclidine; Receptors, Nicotinic; Rubidium Radioisotopes; Torpedo

1987
Interaction of MK-801 with the nicotinic acetylcholine receptor-associated ion channel from electroplax.
    European journal of pharmacology, 1989, May-19, Volume: 164, Issue:2

    Topics: Animals; Anticonvulsants; Dibenzocycloheptenes; Dizocilpine Maleate; Electric Organ; In Vitro Techniques; Ion Channels; Phencyclidine; Receptors, Cholinergic; Receptors, Nicotinic; Torpedo

1989
Compared effects of two vesicular acetylcholine uptake blockers, AH5183 and cetiedil, on cholinergic functions in Torpedo synaptosomes: acetylcholine synthesis, choline transport, vesicular uptake, and evoked acetylcholine release.
    Journal of neurochemistry, 1989, Volume: 52, Issue:3

    Topics: Acetylcholine; Animals; Azepines; Biological Transport; Calcimycin; Choline; Electric Organ; Hydrogen-Ion Concentration; Kinetics; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Synaptic Vesicles; Synaptosomes; Torpedo

1989
AH5183 and cetiedil: two potent inhibitors of acetylcholine uptake into isolated synaptic vesicles from Torpedo marmorata.
    Journal of neurochemistry, 1989, Volume: 52, Issue:3

    Topics: Acetylcholine; Adenosine Triphosphate; Animals; Azepines; Binding, Competitive; Biological Transport; Ca(2+) Mg(2+)-ATPase; Calcium; Electric Organ; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Synaptic Vesicles; Torpedo

1989
Regulation of the vesamicol receptor in cholinergic synaptic vesicles by acetylcholine and an endogenous factor.
    Journal of neurochemistry, 1989, Volume: 52, Issue:3

    Topics: Acetylcholine; Animals; Binding, Competitive; Biological Transport, Active; Electric Organ; Kinetics; Neuromuscular Depolarizing Agents; Osmolar Concentration; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Phencyclidine; Synaptic Vesicles; Torpedo

1989
Fractional vesamicol receptor occupancy and acetylcholine active transport inhibition in synaptic vesicles.
    Molecular pharmacology, 1989, Volume: 36, Issue:3

    Topics: Acetylcholine; Animals; Binding, Competitive; Biological Transport, Active; In Vitro Techniques; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Phencyclidine; Structure-Activity Relationship; Synaptic Vesicles; Torpedo

1989
Synthesis, in vitro acetylcholine-storage-blocking activities, and biological properties of derivatives and analogues of trans-2-(4-phenylpiperidino)cyclohexanol (vesamicol).
    Journal of medicinal chemistry, 1989, Volume: 32, Issue:6

    Topics: Acetylcholine; Animals; Biological Transport; Chemical Phenomena; Chemistry; Electric Organ; Lethal Dose 50; Mice; Molecular Structure; Narcotics; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Stereoisomerism; Structure-Activity Relationship; Synaptic Vesicles; Torpedo; X-Ray Diffraction

1989
Distance between the agonist and noncompetitive inhibitor sites on the nicotinic acetylcholine receptor.
    The Journal of biological chemistry, 1989, Jul-25, Volume: 264, Issue:21

    Topics: Animals; Binding Sites; Bungarotoxins; Choline; Dansyl Compounds; Electric Organ; Energy Transfer; Kinetics; Macromolecular Substances; Mathematics; Models, Biological; Models, Theoretical; Phencyclidine; Quaternary Ammonium Compounds; Receptors, Nicotinic; Torpedo

1989
Sidedness and chemical and kinetic properties of the vesamicol receptor of cholinergic synaptic vesicles.
    Biochemistry, 1988, Jul-12, Volume: 27, Issue:14

    Topics: Acetylcholine; Algorithms; Animals; Cholinergic Fibers; Electric Organ; Hydrogen-Ion Concentration; Kinetics; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Phencyclidine; Synaptic Vesicles; Time Factors; Torpedo

1988
Acetylcholine transport: fundamental properties and effects of pharmacologic agents.
    Annals of the New York Academy of Sciences, 1987, Volume: 493

    Topics: Acetylcholine; Adenosine Triphosphatases; Animals; Biological Transport, Active; Electric Organ; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Receptors, Neurotransmitter; Receptors, Phencyclidine; Synaptic Vesicles; Torpedo

1987
Cholinergic synaptic vesicle heterogeneity: evidence for regulation of acetylcholine transport.
    Biochemistry, 1988, Jul-12, Volume: 27, Issue:14

    Topics: Acetylcholine; Animals; Biological Transport, Active; Cholinergic Fibers; Electric Organ; Nigericin; Phencyclidine; Piperidines; Synaptic Vesicles; Torpedo

1988
Desensitization of the nicotinic acetylcholine receptor by diisopropylfluorophosphate.
    Journal of biochemical toxicology, 1988,Spring, Volume: 3

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Bungarotoxins; Carbachol; Electric Organ; Isoflurophate; Kinetics; Phencyclidine; Receptors, Nicotinic; Torpedo

1988
Localization of azidophencyclidine-binding site on the nicotinic acetylcholine receptor alpha-subunit.
    Biochemical and biophysical research communications, 1987, Jun-15, Volume: 145, Issue:2

    Topics: Affinity Labels; Animals; Azides; Cyanogen Bromide; Endopeptidases; Macromolecular Substances; Molecular Weight; Peptide Fragments; Phencyclidine; Photochemistry; Receptors, Cholinergic; Serine Endopeptidases; Torpedo

1987
Demonstration of a receptor in Torpedo synaptic vesicles for the acetylcholine storage blocker L-trans-2-(4-phenyl[3,4-3H]-piperidino) cyclohexanol.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:7

    Topics: Acetylcholine; Animals; Binding, Competitive; Choline; Electric Organ; Kinetics; Phencyclidine; Piperidines; Receptors, Drug; Stereoisomerism; Synaptic Vesicles; Torpedo

1986
Interaction of noncompetitive inhibitors with the acetylcholine receptor. The site specificity and spectroscopic properties of ethidium binding.
    The Journal of biological chemistry, 1987, May-25, Volume: 262, Issue:15

    Topics: Acetylcholine; Allosteric Site; Animals; Binding Sites; Binding, Competitive; Carbachol; Cell Membrane; Electric Organ; Ethidium; Fluorescence; Fluorescence Polarization; Phencyclidine; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo

1987
Structure of the high-affinity binding site for noncompetitive blockers of the acetylcholine receptor: [3H]chlorpromazine labels homologous residues in the beta and delta chains.
    Biochemistry, 1987, May-05, Volume: 26, Issue:9

    Topics: Amino Acid Sequence; Amino Acids; Animals; Carbachol; Cell Membrane; Chlorpromazine; Macromolecular Substances; Models, Molecular; Peptide Fragments; Phencyclidine; Receptors, Cholinergic; Torpedo

1987
Decidium. A novel fluorescent probe of the agonist/antagonist and noncompetitive inhibitor sites on the nicotinic acetylcholine receptor.
    The Journal of biological chemistry, 1987, Oct-15, Volume: 262, Issue:29

    Topics: Animals; Binding, Competitive; Cell Line; Cell Membrane; Electric Organ; Kinetics; Phenanthridines; Phencyclidine; Receptors, Nicotinic; Spectrometry, Fluorescence; Torpedo

1987
Translocation of cytosolic acetylcholine into synaptic vesicles and demonstration of vesicular release.
    The Journal of biological chemistry, 1986, May-25, Volume: 261, Issue:15

    Topics: Acetylcholine; Animals; Biological Transport; Cytosol; Electric Organ; Kinetics; Neuromuscular Depolarizing Agents; Phencyclidine; Piperidines; Synaptic Vesicles; Synaptosomes; Torpedo

1986
Demonstration and affinity labeling of a stereoselective binding site for a benzomorphan opiate on acetylcholine receptor-rich membranes from Torpedo electroplaque.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:3

    Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Electric Organ; Electrophoresis, Polyacrylamide Gel; Kinetics; Phenazocine; Phencyclidine; Photochemistry; Receptors, Cholinergic; Torpedo

1985
Stoichiometries of acetylcholine uptake, release, and drug inhibition in Torpedo synaptic vesicles: heterogeneity in acetylcholine transport and storage.
    Journal of neurochemistry, 1986, Volume: 46, Issue:4

    Topics: Acetylcholine; Animals; Biological Transport, Active; Electric Organ; Hemicholinium 3; Phencyclidine; Piperidines; Quinacrine; Synaptic Vesicles; Torpedo

1986
Acetylcholine transport and drug inhibition kinetics in Torpedo synaptic vesicles.
    Journal of neurochemistry, 1986, Volume: 46, Issue:4

    Topics: Acetylcholine; Allosteric Regulation; Animals; Biological Transport, Active; Electric Organ; Kinetics; Phencyclidine; Piperidines; Synaptic Vesicles; Torpedo

1986
Mechanism of binding of a benzomorphan opiate to the acetylcholine receptor from Torpedo electroplaque.
    Molecular pharmacology, 1986, Volume: 29, Issue:2

    Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Carbachol; Decamethonium Compounds; In Vitro Techniques; Kinetics; Phenazocine; Phencyclidine; Receptors, Cholinergic; Structure-Activity Relationship; Tetracaine; Torpedo; Tritium; Tubocurarine

1986
Aryldiazonium salts as photoaffinity labels of the nicotinic acetylcholine receptor PCP binding site.
    FEBS letters, 1985, Mar-25, Volume: 182, Issue:2

    Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Carbachol; Diazonium Compounds; Electric Organ; Phencyclidine; Photochemistry; Receptors, Nicotinic; Torpedo

1985
Biochemical evidence that acetylcholine release from cholinergic nerve terminals is mostly vesicular.
    FEBS letters, 1985, Sep-02, Volume: 188, Issue:2

    Topics: Acetates; Acetylcholine; Animals; Electric Organ; In Vitro Techniques; Phencyclidine; Piperidines; Synaptic Vesicles; Synaptosomes; Torpedo

1985
The effect of the acetylcholine transport blocker 2-(4-phenylpiperidino) cyclohexanol (AH5183) on the subcellular storage and release of acetylcholine in mouse brain.
    Brain research, 1985, Dec-09, Volume: 358, Issue:1-2

    Topics: Acetylcholine; Animals; Biological Transport; Brain; Electric Organ; Mice; Mice, Inbred ICR; Phencyclidine; Piperidines; Potassium; Synaptic Vesicles; Torpedo; Veratridine

1985
Ketamine and ditran block end-plate ion conductance and [3H]phencyclidine binding to electric organ membrane.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 221, Issue:3

    Topics: Animals; Drug Combinations; Electric Organ; Glycolates; Hydrogen-Ion Concentration; In Vitro Techniques; Ion Channels; Ketamine; Neurotransmitter Agents; Phencyclidine; Piperidines; Pyrrolidines; Rana pipiens; Receptors, Cholinergic; Torpedo

1982
[3H]Phencyclidine interactions with the nicotinic acetylcholine receptor channel and its inhibition by psychotropic, antipsychotic, opiate, antidepressant, antibiotic, antiviral, and antiarrhythmic drugs.
    Molecular pharmacology, 1982, Volume: 22, Issue:1

    Topics: Allosteric Site; Animals; Anti-Arrhythmia Agents; Anti-Bacterial Agents; Antidepressive Agents; Antipsychotic Agents; Antiviral Agents; Binding, Competitive; Electric Organ; In Vitro Techniques; Ion Channels; Narcotics; Phencyclidine; Psychotropic Drugs; Receptors, Cholinergic; Receptors, Nicotinic; Torpedo

1982
Ketamine inhibition of ligand binding to cholinergic receptors and ion channels.
    European journal of pharmacology, 1982, Mar-12, Volume: 78, Issue:3

    Topics: Acetylcholine; Animals; Electric Organ; In Vitro Techniques; Ion Channels; Ketamine; Ligands; N-Methylscopolamine; Phencyclidine; Receptors, Cholinergic; Scopolamine Derivatives; Torpedo; Tubocurarine

1982
Receptor--ion channel interactions in Torpedo electric organ: influence of thiol group modification.
    Neuroscience letters, 1982, Jul-20, Volume: 31, Issue:1

    Topics: Animals; Dithionitrobenzoic Acid; Dithiothreitol; Electric Organ; Ethylmaleimide; Ion Channels; Nitrobenzoates; Phencyclidine; Receptors, Cholinergic; Receptors, Nicotinic; Torpedo

1982
Alcohol modulation of drug binding to the channel sites of the nicotinic acetylcholine receptor.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:2

    Topics: Alcohols; Amphibian Venoms; Animals; Carbachol; Drug Interactions; Imipramine; Ion Channels; Membranes; Naphthols; Phencyclidine; Receptors, Cholinergic; Torpedo

1983
Benzomorphan interactions with acetylcholine receptor complexes from Torpedo.
    European journal of pharmacology, 1983, Jun-17, Volume: 90, Issue:4

    Topics: Amphibian Venoms; Animals; Benzomorphans; Drug Interactions; Ion Channels; Morphinans; Parasympatholytics; Phencyclidine; Receptors, Cholinergic; Receptors, Nicotinic; Receptors, Opioid; Torpedo

1983
Characterization of the interaction of phencyclidine and its derivatives with the ionic channel of the nicotinic receptor.
    Archives of toxicology. Supplement. = Archiv fur Toxikologie. Supplement, 1983, Volume: 6

    Topics: Animals; Electric Organ; In Vitro Techniques; Ion Channels; Kinetics; Phencyclidine; Receptors, Nicotinic; Torpedo

1983
Effects of calcium on the binding of phencyclidine to acetylcholine receptor-rich membrane fragments from Torpedo californica electroplaque.
    Journal of neurochemistry, 1983, Volume: 41, Issue:4

    Topics: Animals; Calcium; Carbachol; Cations, Divalent; Cell Membrane; Egtazic Acid; Electric Organ; Phencyclidine; Receptors, Cholinergic; Torpedo

1983
Displacement of [3H]phencyclidine binding to Torpedo electric organ membrane by calcium channel antagonists.
    Biochemical pharmacology, 1984, Dec-15, Volume: 33, Issue:24

    Topics: Animals; Calcium Channel Blockers; Calcium Chloride; Cell Membrane; Electric Organ; In Vitro Techniques; Phencyclidine; Torpedo; Tritium

1984
Multiple binding sites for phencyclidine on the nicotinic acetylcholine receptor from Torpedo ocellata electric organ.
    Life sciences, 1984, Mar-12, Volume: 34, Issue:11

    Topics: Acetylcholine; Animals; Binding Sites; Bungarotoxins; Carbachol; Dibucaine; Electric Organ; Kinetics; Phencyclidine; Receptors, Cholinergic; Tetracaine; Torpedo; Tubocurarine

1984
Localization of phencyclidine binding sites on alpha and beta subunits of the nicotinic acetylcholine receptor from Torpedo ocellata electric organ using azido phencyclidine.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1984, Volume: 4, Issue:3

    Topics: Affinity Labels; Animals; Azides; Binding Sites; Binding, Competitive; Carbachol; Cell Membrane; Electric Organ; Macromolecular Substances; Molecular Weight; Phencyclidine; Photochemistry; Receptors, Nicotinic; Torpedo

1984
Mechanism of phencyclidine binding to the acetylcholine receptor from Torpedo electroplaque.
    Molecular pharmacology, 1984, Volume: 25, Issue:3

    Topics: Animals; Carbachol; Cell Membrane; Electric Organ; Glycerol; Kinetics; Phencyclidine; Receptors, Cholinergic; Temperature; Thermodynamics; Torpedo

1984
Binding of phencyclidine to the detergent solubilized acetylcholine receptor from Torpedo marmorata.
    Life sciences, 1983, Mar-07, Volume: 32, Issue:10

    Topics: Animals; Cholic Acid; Cholic Acids; Electric Organ; Kinetics; Phencyclidine; Polysorbates; Receptors, Cholinergic; Solubility; Torpedo

1983
Pharmacological characterization of the acetylcholine transport system in purified Torpedo electric organ synaptic vesicles.
    Molecular pharmacology, 1983, Volume: 24, Issue:1

    Topics: Acetylcholine; Animals; Binding Sites; Biological Transport, Active; Electric Organ; In Vitro Techniques; Phencyclidine; Piperidines; Receptors, Cholinergic; Synaptic Vesicles; Torpedo

1983
Species differences determine azido phencyclidine labeling pattern in desensitized nicotinic acetylcholine receptors.
    Biochemical and biophysical research communications, 1983, Jun-15, Volume: 113, Issue:2

    Topics: Affinity Labels; Animals; Azides; Electrophoresis, Polyacrylamide Gel; Isotope Labeling; Phencyclidine; Photochemistry; Receptors, Cholinergic; Receptors, Nicotinic; Species Specificity; Torpedo; Tritium

1983
Multiple sites of action for noncompetitive blockers on acetylcholine receptor rich membrane fragments from torpedo marmorata.
    Biochemistry, 1983, Jun-21, Volume: 22, Issue:13

    Topics: Alkanes; Allosteric Regulation; Amphibian Venoms; Animals; Binding Sites; Chlorpromazine; Electric Organ; Isoquinolines; Membrane Lipids; Neuromuscular Junction; Parasympatholytics; Phencyclidine; Polyethylene Glycols; Proadifen; Receptors, Cholinergic; Torpedo

1983
Multiple affinity states for noncompetitive blockers revealed by [3H]phencyclidine binding to acetylcholine receptor rich membrane fragments from Torpedo marmorata.
    Biochemistry, 1983, Jun-21, Volume: 22, Issue:13

    Topics: Allosteric Regulation; Animals; Binding Sites; Electric Organ; Kinetics; Neuromuscular Junction; Phencyclidine; Protein Binding; Protein Conformation; Receptors, Cholinergic; Torpedo

1983
Selective labeling of the delta subunit of the acetylcholine receptor by a covalent local anesthetic.
    Biochemistry, 1981, Dec-08, Volume: 20, Issue:25

    Topics: Acetylcholine; Affinity Labels; Animals; Azides; Binding, Competitive; Cell Membrane; Electric Organ; Isoquinolines; Kinetics; Macromolecular Substances; Phencyclidine; Receptors, Cholinergic; Torpedo

1981
Clonidine and cirazoline inhibit activation of nicotinic channels in PC-12 cells.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Adrenergic alpha-Agonists; Animals; Binding Sites; Calcium; Clonidine; Imidazoles; Ion Channels; Nicotinic Antagonists; PC12 Cells; Phencyclidine; Radioligand Assay; Rats; Receptors, Nicotinic; Torpedo; Tritium

1995
Action of organophosphate anticholinesterases on the three conformational states of nicotinic receptor.
    Advances in experimental medicine and biology, 1995, Volume: 363

    Topics: Animals; Cholinesterase Inhibitors; Cobra Neurotoxin Proteins; Organophosphorus Compounds; Phencyclidine; Protein Conformation; Receptors, Nicotinic; Soman; Torpedo; Tubocurarine

1995
Effects of substance P on the binding of agonists to the nicotinic acetylcholine receptor of Torpedo electroplaque.
    Journal of neurochemistry, 1993, Volume: 60, Issue:6

    Topics: Acetylcholine; Animals; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Kinetics; Least-Squares Analysis; Mathematics; Models, Theoretical; Phencyclidine; Receptors, Nicotinic; Substance P; Time Factors; Torpedo

1993
Effects of halothane on the nicotinic acetylcholine receptor from Torpedo californica.
    Biochemical pharmacology, 1995, Apr-18, Volume: 49, Issue:8

    Topics: Animals; Binding, Competitive; Halothane; Kinetics; Nicotinic Antagonists; Phencyclidine; Receptors, Nicotinic; Torpedo

1995
The ion channel of muscle and electric organ acetylcholine receptors: differing affinities for noncompetitive inhibitors.
    Cellular and molecular neurobiology, 1993, Volume: 13, Issue:2

    Topics: Amino Acid Sequence; Animals; Cell Line; Diterpenes; Electric Organ; Ion Channel Gating; Magnesium; Membrane Potentials; Mice; Molecular Sequence Data; Muscle Proteins; Nerve Tissue Proteins; Nicotinic Antagonists; Oocytes; Organ Specificity; Phencyclidine; Recombinant Proteins; Sequence Homology, Amino Acid; Sodium Channels; Tetracaine; Torpedo; Xenopus laevis

1993
Transverse localization of the quinacrine binding site on the Torpedo acetylcholine receptor.
    The Journal of biological chemistry, 1993, Mar-25, Volume: 268, Issue:9

    Topics: Animals; Binding Sites; Cell Membrane; Iodides; Kinetics; Phencyclidine; Quinacrine; Receptors, Cholinergic; Rhodamines; Stearates; Torpedo

1993
Quinacrine and ethidium bind to different loci on the Torpedo acetylcholine receptor.
    Biochemistry, 1993, Jun-22, Volume: 32, Issue:24

    Topics: Animals; Binding Sites; Cell Membrane; Ethidium; Phencyclidine; Quinacrine; Receptors, Cholinergic; Spectrometry, Fluorescence; Spin Labels; Torpedo

1993
Interaction of d-tubocurarine analogs with the Torpedo nicotinic acetylcholine receptor. Methylation and stereoisomerization affect site-selective competitive binding and binding to the noncompetitive site.
    The Journal of biological chemistry, 1995, Dec-29, Volume: 270, Issue:52

    Topics: Animals; Binding, Competitive; Methylation; Nicotinic Agonists; Nicotinic Antagonists; Phencyclidine; Receptors, Nicotinic; Stereoisomerism; Torpedo; Tritium; Tubocurarine

1995
Temperature and ionic strength dependence of quinacrine binding and quinacrine displacement elicited by high concentrations of agonists on the nicotinic acetylcholine receptor.
    Archives of biochemistry and biophysics, 1996, Sep-01, Volume: 333, Issue:1

    Topics: Animals; Binding Sites; Electric Organ; In Vitro Techniques; Kinetics; Models, Biological; Nicotinic Agonists; Osmolar Concentration; Phencyclidine; Quinacrine; Receptors, Nicotinic; Sodium Chloride; Temperature; Thermodynamics; Torpedo

1996
Differential effects of dimethyl sulfoxide on nicotinic acetylcholine receptors from mouse muscle and Torpedo electrocytes.
    Neuroscience letters, 1997, Jul-25, Volume: 230, Issue:3

    Topics: Administration, Topical; Animals; Anti-Inflammatory Agents; Bungarotoxins; Dimethyl Sulfoxide; Excitatory Amino Acid Antagonists; Female; Iodine Radioisotopes; Ion Channel Gating; Mice; Oocytes; Patch-Clamp Techniques; Phencyclidine; Radioligand Assay; Receptors, Nicotinic; Torpedo; Tritium; Xenopus laevis

1997
Chlorpyrifos, parathion, and their oxons bind to and desensitize a nicotinic acetylcholine receptor: relevance to their toxicities.
    Toxicology and applied pharmacology, 1997, Volume: 146, Issue:2

    Topics: Animals; Binding, Competitive; Bungarotoxins; Carbachol; Chlorpyrifos; Cholinesterase Inhibitors; Cholinesterases; Dose-Response Relationship, Drug; Insecticides; Iodine Radioisotopes; Lethal Dose 50; Nicotinic Agonists; Paraoxon; Parathion; Phencyclidine; Receptors, Nicotinic; Structure-Activity Relationship; Torpedo; Tritium

1997
Characterization of cembranoid interaction with the nicotinic acetylcholine receptor.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 287, Issue:1

    Topics: Acetylcholine; Animals; Binding Sites; Bungarotoxins; Diterpenes; Female; Phencyclidine; Receptors, Nicotinic; Torpedo; Xenopus laevis

1998
In vitro selection of RNA molecules that displace cocaine from the membrane-bound nicotinic acetylcholine receptor.
    Proceedings of the National Academy of Sciences of the United States of America, 1998, Nov-24, Volume: 95, Issue:24

    Topics: Animals; Base Sequence; Binding Sites; Binding, Competitive; Cell Membrane; Cocaine; Consensus Sequence; Electric Organ; Illicit Drugs; Kinetics; Ligands; Molecular Sequence Data; Nucleic Acid Conformation; Oligodeoxyribonucleotides; Phencyclidine; Receptors, Nicotinic; RNA; Sequence Alignment; Torpedo

1998
Aminotriarylmethane dyes are high-affinity noncompetitive antagonists of the nicotinic acetylcholine receptor.
    Molecular pharmacology, 1999, Volume: 55, Issue:1

    Topics: Animals; Binding Sites; Binding, Competitive; Coloring Agents; Gentian Violet; Nicotinic Antagonists; Phencyclidine; Protein Conformation; Receptors, Nicotinic; Sodium; Spectrometry, Fluorescence; Structure-Activity Relationship; Torpedo

1999
Characterization of interaction of 3,4,5-trimethoxybenzoic acid 8-(diethylamino)octyl ester with Torpedo californica nicotinic acetylcholine receptor and 5-hydroxytryptamine3 receptor.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:1

    Topics: Amino Acid Sequence; Animals; Binding, Competitive; Cell Membrane; Electrophysiology; Gallic Acid; Humans; In Vitro Techniques; Iodine Radioisotopes; Mice; Molecular Sequence Data; Nicotinic Antagonists; Oocytes; Phencyclidine; Radioligand Assay; Receptors, Nicotinic; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Torpedo; Xenopus laevis

1999
Determinants of phencyclidine potency on the nicotinic acetylcholine receptors from muscle and electric organ.
    Cellular and molecular neurobiology, 1999, Volume: 19, Issue:6

    Topics: Acetylcholine; Amino Acid Sequence; Amino Acid Substitution; Animals; Atropine; Binding Sites; Diterpenes; DNA, Complementary; Dose-Response Relationship, Drug; Electric Organ; Ion Channel Gating; Ion Channels; Kinetics; Mice; Molecular Sequence Data; Muscle Proteins; Muscle, Skeletal; Mutagenesis, Site-Directed; Nerve Tissue Proteins; Nicotinic Antagonists; Patch-Clamp Techniques; Phencyclidine; Point Mutation; Protein Multimerization; Receptors, Nicotinic; Recombinant Fusion Proteins; Sequence Alignment; Sequence Homology, Amino Acid; Torpedo; Xenopus laevis

1999
5-Doxylstearate-induced displacement of phencyclidine from its low-affinity binding sites on the nicotinic acetylcholine receptor.
    Archives of biochemistry and biophysics, 1999, Nov-01, Volume: 371, Issue:1

    Topics: Animals; Binding Sites; Binding, Competitive; Cell Membrane; Cyclic N-Oxides; Electric Organ; Ethidium; Kinetics; Phencyclidine; Quinacrine; Receptors, Nicotinic; Spin Labels; Torpedo; Tritium

1999
5-hydroxytryptamine interaction with the nicotinic acetylcholine receptor.
    European journal of pharmacology, 2000, Feb-18, Volume: 389, Issue:2-3

    Topics: Animals; Binding Sites; Bungarotoxins; Cells, Cultured; Dose-Response Relationship, Drug; Humans; Phencyclidine; Photoaffinity Labels; Receptors, Nicotinic; Serotonin; Torpedo

2000
Interactions between 3-(Trifluoromethyl)-3-(m-[(125)I]iodophenyl)diazirine and tetracaine, phencyclidine, or histrionicotoxin in the Torpedo series nicotinic acetylcholine receptor ion channel.
    Molecular pharmacology, 2001, Volume: 59, Issue:6

    Topics: Affinity Labels; Amphibian Venoms; Anesthetics, Local; Animals; Azirines; Ceramides; Drug Interactions; Excitatory Amino Acid Antagonists; Iodine Radioisotopes; Membrane Proteins; Phencyclidine; Receptors, Nicotinic; Tetracaine; Torpedo

2001
Cembranoid and long-chain alkanol sites on the nicotinic acetylcholine receptor and their allosteric interaction.
    Biochemistry, 2001, Sep-18, Volume: 40, Issue:37

    Topics: Allosteric Regulation; Anesthetics; Animals; Binding Sites; Binding, Competitive; Diterpenes; Fatty Alcohols; Hexanols; Models, Theoretical; Nicotinic Antagonists; Octanols; Phencyclidine; Procaine; Receptors, Nicotinic; Torpedo

2001
Allosterically linked noncompetitive antagonist binding sites in the resting nicotinic acetylcholine receptor ion channel.
    Archives of biochemistry and biophysics, 2002, Jul-01, Volume: 403, Issue:1

    Topics: Allosteric Site; Amobarbital; Anesthetics, Local; Animals; Binding Sites; Binding, Competitive; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Modulators; Inhibitory Concentration 50; Ions; Ketamine; Kinetics; Light; Models, Molecular; Phencyclidine; Protein Binding; Protein Conformation; Receptors, Nicotinic; Tetracaine; Torpedo

2002
Noncompetitive antagonist binding sites in the torpedo nicotinic acetylcholine receptor ion channel. Structure-activity relationship studies using adamantane derivatives.
    Biochemistry, 2003, Jun-24, Volume: 42, Issue:24

    Topics: Adamantane; Allosteric Site; Anesthetics, Local; Animals; Binding Sites; Binding, Competitive; Excitatory Amino Acid Antagonists; Iodine Isotopes; Ion Channels; Models, Molecular; Nicotinic Antagonists; Phencyclidine; Protein Binding; Receptors, Nicotinic; Structure-Activity Relationship; Thermodynamics; Torpedo; Tritium

2003
Molecular mechanisms of inhibition of nicotinic acetylcholine receptors by tricyclic antidepressants.
    Neuropharmacology, 2003, Volume: 45, Issue:7

    Topics: Acetylcholine; Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Cell Membrane; Doxepin; Excitatory Amino Acid Antagonists; Humans; Imipramine; In Vitro Techniques; Kidney; Kinetics; Membrane Potentials; Mice; Nicotinic Antagonists; Patch-Clamp Techniques; Phencyclidine; Receptors, Nicotinic; Torpedo

2003
Site specificity of agonist-induced opening and desensitization of the Torpedo californica nicotinic acetylcholine receptor.
    Biochemistry, 2006, Jan-10, Volume: 45, Issue:1

    Topics: Animals; Binding Sites; Calcium Channel Blockers; Conotoxins; Dansyl Compounds; Enzyme Inhibitors; Fluorescent Dyes; Kinetics; Nicotinic Agonists; Phencyclidine; Proadifen; Quaternary Ammonium Compounds; Receptors, Nicotinic; Spectrometry, Fluorescence; Structure-Activity Relationship; Torpedo; Tubocurarine

2006
Molecular mechanisms and binding site location for the noncompetitive antagonist crystal violet on nicotinic acetylcholine receptors.
    Biochemistry, 2006, Feb-21, Volume: 45, Issue:7

    Topics: Allosteric Regulation; Amobarbital; Animals; Binding Sites; Fluorescent Dyes; Gentian Violet; Ion Channels; Models, Molecular; Nicotinic Agonists; Nicotinic Antagonists; Pentobarbital; Phencyclidine; Protein Binding; Protein Conformation; Quaternary Ammonium Compounds; Receptors, Nicotinic; Temperature; Tetracaine; Thiophenes; Torpedo; Tritium

2006
Molecular properties of local anesthetics as predictors of affinity for nicotinic acetylcholine receptors.
    Journal of neuroscience research, 2007, Volume: 85, Issue:13

    Topics: Anesthetics, Local; Animals; Binding, Competitive; Bungarotoxins; Cell Membrane; Electric Organ; Neuroprotective Agents; Phencyclidine; Predictive Value of Tests; Protein Conformation; Receptors, Nicotinic; Torpedo; Tritium

2007
Probing the structure of the affinity-purified and lipid-reconstituted torpedo nicotinic acetylcholine receptor.
    Biochemistry, 2008, Dec-02, Volume: 47, Issue:48

    Topics: Affinity Labels; Animals; Azirines; Binding Sites; Cholates; Iodine Radioisotopes; Ion Channels; Lipid Metabolism; Models, Molecular; Nicotinic Antagonists; Phencyclidine; Protein Structure, Secondary; Protein Structure, Tertiary; Receptors, Nicotinic; Solubility; Spectroscopy, Fourier Transform Infrared; Staining and Labeling; Substrate Specificity; Torpedo

2008