Page last updated: 2024-08-23

torpedo and donepezil

torpedo has been researched along with donepezil in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (25.00)18.2507
2000's2 (25.00)29.6817
2010's4 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hopfinger, AJ; Inoue, A; Kawai, T; Kawakami, Y; Sugimoto, H; Wakita, M1
Kryger, G; Silman, I; Sussman, JL1
Koellner, G; Kryger, G; Millard, CB; Silman, I; Steiner, T; Sussman, JL1
Contreras, JM; Parrot, I; Rival, YM; Sippl, W; Wermuth, CG1
Burshteyn, F; Cassidy, MS; Cheung, J; Franklin, MC; Gary, EN; Height, JJ; Love, J; Rudolph, MJ1
Cheng, S; Song, W; Xu, Y; Yuan, X1
Ali, MR; Boutajangout, A; Mezei, M; Møller, SG; Sadoqi, M1
Caliandro, R; Cariati, L; Lamba, D; Oliverio, M; Pesaresi, A; Procopio, A1

Other Studies

8 other study(ies) available for torpedo and donepezil

ArticleYear
The rationale for E2020 as a potent acetylcholinesterase inhibitor.
    Bioorganic & medicinal chemistry, 1996, Volume: 4, Issue:9

    Topics: Acetylcholinesterase; Animals; Cholinesterase Inhibitors; Crystallography, X-Ray; Donepezil; Indans; Models, Molecular; Piperidines; Protein Conformation; Software; Torpedo

1996
Structure of acetylcholinesterase complexed with E2020 (Aricept): implications for the design of new anti-Alzheimer drugs.
    Structure (London, England : 1993), 1999, Mar-15, Volume: 7, Issue:3

    Topics: Acetylcholinesterase; Alzheimer Disease; Animals; Binding Sites; Cholinesterase Inhibitors; Crystallography, X-Ray; Donepezil; Drug Design; Indans; Macromolecular Substances; Mice; Models, Molecular; Nootropic Agents; Piperidines; Protein Conformation; Solvents; Structure-Activity Relationship; Substrate Specificity; Torpedo

1999
Active-site gorge and buried water molecules in crystal structures of acetylcholinesterase from Torpedo californica.
    Journal of molecular biology, 2000, Feb-18, Volume: 296, Issue:2

    Topics: Acetylcholinesterase; Alkaloids; Amino Acid Sequence; Animals; Binding Sites; Cholinesterase Inhibitors; Crystallization; Crystallography, X-Ray; Donepezil; Edrophonium; Hydrogen Bonding; Indans; Ligands; Models, Molecular; Molecular Sequence Data; Piperidines; Protein Structure, Secondary; Reproducibility of Results; Sesquiterpenes; Static Electricity; Torpedo; Water

2000
Structure-based 3D QSAR and design of novel acetylcholinesterase inhibitors.
    Journal of computer-aided molecular design, 2001, Volume: 15, Issue:5

    Topics: Acetylcholinesterase; Alzheimer Disease; Animals; Binding Sites; Cholinesterase Inhibitors; Computer Simulation; Crystallography, X-Ray; Donepezil; Drug Design; Humans; Indans; Models, Molecular; Piperidines; Protein Conformation; Quantitative Structure-Activity Relationship; Thermodynamics; Torpedo

2001
Structures of human acetylcholinesterase in complex with pharmacologically important ligands.
    Journal of medicinal chemistry, 2012, Nov-26, Volume: 55, Issue:22

    Topics: Acetylcholinesterase; Acetylthiocholine; Animals; Cholinesterase Inhibitors; Crystallography, X-Ray; Donepezil; Humans; Indans; Models, Molecular; Piperidines; Protein Conformation; Torpedo

2012
Gorge Motions of Acetylcholinesterase Revealed by Microsecond Molecular Dynamics Simulations.
    Scientific reports, 2017, 06-12, Volume: 7, Issue:1

    Topics: Acetylcholinesterase; Allosteric Regulation; Animals; Biocatalysis; Catalytic Domain; Cholinesterase Inhibitors; Donepezil; Fish Proteins; Molecular Dynamics Simulation; Motion; Protein Binding; Protein Domains; Protein Multimerization; Torpedo

2017
Assessing the binding of cholinesterase inhibitors by docking and molecular dynamics studies.
    Journal of molecular graphics & modelling, 2017, Volume: 76

    Topics: Acetylcholinesterase; Alzheimer Disease; Animals; Cholinesterase Inhibitors; Donepezil; Galantamine; Humans; Hydrogen Bonding; Indans; Molecular Conformation; Molecular Dynamics Simulation; Piperidines; Rivastigmine; Torpedo

2017
Kinetic and structural studies on the interactions of Torpedo californica acetylcholinesterase with two donepezil-like rigid analogues.
    Journal of enzyme inhibition and medicinal chemistry, 2018, Volume: 33, Issue:1

    Topics: Acetylcholinesterase; Animals; Cholinesterase Inhibitors; Crystallography, X-Ray; Donepezil; Dose-Response Relationship, Drug; Indans; Kinetics; Molecular Docking Simulation; Molecular Structure; Piperidines; Structure-Activity Relationship; Torpedo

2018