Page last updated: 2024-08-23

torpedo and carbachol

torpedo has been researched along with carbachol in 115 studies

Research

Studies (115)

TimeframeStudies, this research(%)All Research%
pre-199066 (57.39)18.7374
1990's39 (33.91)18.2507
2000's8 (6.96)29.6817
2010's1 (0.87)24.3611
2020's1 (0.87)2.80

Authors

AuthorsStudies
Min, CK; Weiland, GA2
Arrondo, JL; Castresana, J; Fernandez, AM; Fernandez-Ballester, G; Ferragut, JA; Gonzalez-Ros, JM; Laynez, JL1
Chen, L; Martin, GB; Rechnitz, GA1
Arrondo, JL; Castresana, J; Fernandez-Ballester, G; Ferragut, JA; Gonzalez-Ros, JM1
Barth, A; Görne-Tschelnokow, U; Hucho, F; Mäntele, W; Naumann, D1
Duvvuri, P; Johnson, DA; Kerr, JA; Valenzuela, CF1
Baenziger, JE; Miller, KW; Rothschild, KJ1
Baenziger, JE; McCarthy, MP; Miller, KW; Rothschild, KJ1
Eterović, VA; Ferchmin, PA; Hann, RM; Szczawinska, K1
Cohen, JB; White, BH1
Forman, SA; Miller, KW; Wood, SC1
Cohen, JB; Cohen, SG; Howard, S; White, BH1
Chen, XJ; Li, L; McNamee, M; Palma, A; Pappone, P1
Li, LA; McNamee, MG; Ochoa, EL; Plummer, A1
Albuquerque, EX; Aracava, Y; Eldefrawi, ME; Sherby, SM; VanMeter, WG; Varanda, WA1
Aoshima, H; Cash, DJ; Hess, GP; Pasquale, EB1
Albuquerque, EX; Aronstam, RS; Daly, JW; Feigl, DM; King, CT1
Aronstam, RS; Hong, JS1
Fels, G; Maelicke, A; Plümer-Wilk, R; Schreiber, M1
Diebler, MF; Dolezal, V; Israël, M; Lazereg, S; Tucek, S1
Eriksson, H; Häggblad, J; Hedlund, B; Heilbronn, E1
Braswell, LM; Forman, SA; Miller, KW; Roth, SH1
Fahr, A; Heyn, MP; Hucho, F; Lauffer, L; Schmidt, D1
Forman, SA; Miller, KW; Righi, DL1
McCarthy, MP; Stroud, RM1
McCarthy, MP; Mitra, AK; Stroud, RM1
Mielke, DL; Wallace, BA1
Bachy, A; Changeux, JP; Chemouilli, P; Heidmann, T; Morre, M1
Fong, TM; McNamee, MG1
Firestone, LL; Forman, SA; Miller, KW1
Bakry, NM; Eldefrawi, ME; Schweizer, G; Valdes, JJ1
Abood, LG; Kanne, DB1
Behling, RW; Jelinski, LW; Navon, G; Sammon, MJ; Yamane, T1
Mihovilovic, M; Richman, DP2
Herz, JM; Johnson, DA; Taylor, P1
Changeux, JP; Dennis, M; Giraudat, J; Haumont, PY; Heidmann, T; Lederer, F1
Lindstrom, JM; Whiting, PJ1
Clarke, JH; Martinez-Carrion, M1
Baumann, H; Hucho, F; Lottspeich, F; Muhn, P; Oberthür, W; Wittmann-Liebold, B1
Nuske, JH1
Bigelow, J; Michel, L; Oswald, RE1
Albuquerque, EX; Eldefrawi, AT; Eldefrawi, ME; Sherby, SM1
Goeldner, M; Hirth, C; Jaganathen, J; Kotzyba-Hibert, F; Lagenbuch-Cachat, J1
Raftery, MA; Zabrecky, JR1
Lindstrom, JM; Wan, KK1
McNamee, MG; Richardson, CA; Walker, JW1
Martinez-Carrion, M; Mattingly, JR; Soler, G1
Huganir, RL; Racker, E1
Abbassy, MA; Eldefrawi, AT; Eldefrawi, ME1
McNamee, MG; Takeyasu, K; Walker, JW1
Abbassy, MA; Ei-Fakahany, EF; Eldefrawi, AT; Eldefrawi, ME; Miller, ER1
Hucho, F; Muhn, P1
Kaldany, RR; Karlin, A1
Lindstrom, J; Montal, M; Suarez-Isla, BA; Wan, K1
Gonzalez-Ros, JM; Martinez-Carrion, M; Paraschos, A2
Changeux, JP; Heidmann, T1
Fredkin, DR; Labarca, P; Montal, M; Suarez-Isla, BA1
Albuquerque, EX; Aronstam, RS; Daly, JW; Souccar, C; Varanda, WA1
Oswald, RE1
Hirose, S; Vieth, WR1
Farach, MC; Gonzalez-Ros, JM; Martinez-Carrion, M1
Haring, R; Kloog, Y1
Haring, R; Kloog, Y; Sokolovsky, M1
Covarrubias, M; Maelicke, A; Prinz, H1
Bamberger, MJ; McLaughlin, JT; Oswald, RE1
Barrantes, FJ; Criado, M; Eibl, H1
Dalziel, AW; McNamee, MG; Ochoa, EL1
Sigman, DS; Young, AP1
Hess, GP; McNamee, MG; Pasquale, EB; Walker, JW1
Doerge, DR; Ingraham, LL; McNamee, MG1
Dunn, SM; Raftery, MA5
Anholt, R; Deerinck, T; Ellisman, M; Fredkin, DR; Lindstrom, J; Montal, M1
El-Fakahany, EF; Eldefrawi, AT; Eldefrawi, ME1
Bakry, NM; Eldefrawi, AT; Eldefrawi, ME; Riker, WF1
Cartaud, J; Changeux, JP; Popot, JL1
Blanchard, SG; Dunn, SM; Raftery, MA1
Oshiki, JR; Sigman, DS; Young, AP1
Min, CK; Owens, J; Weiland, GA1
Baenziger, JE; McCarthy, MP; Méthot, N1
Baenziger, JE; Demers, CN; Méthot, N1
Alifimoff, JK; Bugge, B; Forman, SA; Miller, KW1
Arias, HR; Johnson, DA1
Kessler, P; Ménez, A; Servent, D1
Blanton, MP; Cohen, JB1
Bugge, B; de Armendi, AJ; Miller, KW; Tonner, PH1
Hill, WA; Miller, KW; Wood, SC1
Donnelly-Roberts, DL; Lentz, TL1
Claudio, T; Wang, YD1
Aslanian, D; Changeux, JP; Galzi, JL; Grof, P1
Tasaki, I1
Ayres, S; Johnson, DA1
Goeldner, M; Peng, L; Silman, I; Sussman, J1
Butler, DH; Lasalde, JA; McNamee, MG; Tamamizu, S1
Dreger, M; Herrmann, A; Hucho, F; Krauss, M1
Cortes, VI; Eldefrawi, AT; Eldefrawi, ME; Katz, EJ1
Addona, GH; Bugge, B; Kloczewiak, MA; Miller, KW; Rankin, SE1
Fairclough, RH; Gudipati, E; Lin, MY; Richman, DP; Twaddle, GM1
Baenziger, JE; Ryan, SE1
Baenziger, JE; Nguyen, HP; Ryan, SE1
Pedersen, SE; Song, XZ1
Biscoglio de Jiménez Bonino, MJ; Cortez, LM; del Canto, SG; Testai, FD1
Chiara, DC; Cohen, JB; Dangott, LJ; Eckenhoff, RG1
Braekman, JC; Kem, WR; LeFrancois, S; Marszalec, W; Raja, M; Wildeboer, K1
Ivorra, I; Morales, A; Olivera-Bravo, S1
Martin, JL; Négrerie, M; Nghiêm, HO1
Chuang, AR; Doniach, S; Fairclough, RH; Lee, TE; Marek, MS1
Barrantes, FJ; Bonini, IC; Diaz, C; Maza, E; Pissinis, DE; Salvarezza, RC; Schilardi, PL1
Hibbs, RE; Karlin, A; Lee, M; Noviello, CM; Rahman, MM; Stowell, MHB; Teng, J; Worrell, BT1

Reviews

1 review(s) available for torpedo and carbachol

ArticleYear
Acetylcholine-receptor-mediated ion fluxes in Electrophorus electricus and Torpedo california membrane vesicles.
    Reviews of physiology, biochemistry and pharmacology, 1985, Volume: 102

    Topics: Acetylcholine; Animals; Biological Transport; Calcium; Carbachol; Cations, Monovalent; Cell Membrane; Cell Membrane Permeability; Electric Conductivity; Electric Organ; Electrophorus; Electrophysiology; Ion Channels; Kinetics; Lithium; Mathematics; Models, Biological; Muscles; Potassium; Radioisotopes; Receptors, Cholinergic; Rubidium; Sodium; Torpedo

1985

Other Studies

114 other study(ies) available for torpedo and carbachol

ArticleYear
Substance P inhibits carbamylcholine-stimulated 22Na+ efflux from acetylcholine receptor-enriched Torpedo electroplaque membrane vesicles.
    Brain research, 1992, Jul-24, Volume: 586, Issue:2

    Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Kinetics; Receptors, Nicotinic; Sodium; Sodium Radioisotopes; Substance P; Torpedo

1992
Protein structural effects of agonist binding to the nicotinic acetylcholine receptor.
    FEBS letters, 1992, Dec-14, Volume: 314, Issue:2

    Topics: Animals; Calorimetry, Differential Scanning; Carbachol; Fourier Analysis; Hot Temperature; Protein Structure, Secondary; Receptors, Nicotinic; Spectrophotometry, Infrared; Torpedo

1992
Microtiter plate binding assay for cholinergic compounds utilizing the nicotinic acetylcholine receptor.
    Analytical chemistry, 1992, Dec-01, Volume: 64, Issue:23

    Topics: Animals; Avidin; Binding, Competitive; Biotin; Bungarotoxins; Carbachol; Enzyme-Linked Immunosorbent Assay; Horseradish Peroxidase; Parasympathomimetics; Receptors, Nicotinic; Torpedo

1992
Protein stability and interaction of the nicotinic acetylcholine receptor with cholinergic ligands studied by Fourier-transform infrared spectroscopy.
    The Biochemical journal, 1992, Dec-01, Volume: 288 ( Pt 2)

    Topics: Amides; Animals; Carbachol; Detergents; Fourier Analysis; In Vitro Techniques; Ligands; Protein Denaturation; Protein Structure, Secondary; Receptors, Nicotinic; Spectrophotometry, Infrared; Temperature; Torpedo; Trehalose; Tubocurarine

1992
Fourier transform infrared (FTIR) spectroscopic investigation of the nicotinic acetylcholine receptor (nAChR). Investigation of agonist binding and receptor conformational changes by flash-induced release of 'caged' carbamoylcholine.
    FEBS letters, 1992, Sep-07, Volume: 309, Issue:2

    Topics: Animals; Carbachol; Fourier Analysis; Protein Conformation; Receptors, Nicotinic; Spectrophotometry, Infrared; Torpedo

1992
Modulation of phencyclidine-sensitive ethidium binding to the Torpedo acetylcholine receptor: interaction of noncompetitive inhibitors with carbamylcholine and cobra alpha-toxin.
    Molecular pharmacology, 1992, Volume: 41, Issue:2

    Topics: Anesthetics; Animals; Barbiturates; Binding Sites; Binding, Competitive; Carbachol; Cholinergic Antagonists; Cobra Neurotoxin Proteins; Drug Interactions; Ethidium; Phencyclidine; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo

1992
Incorporation of the nicotinic acetylcholine receptor into planar multilamellar films: characterization by fluorescence and Fourier transform infrared difference spectroscopy.
    Biophysical journal, 1992, Volume: 61, Issue:4

    Topics: Animals; Biophysical Phenomena; Biophysics; Carbachol; Ethidium; Fourier Analysis; Membranes, Artificial; Protein Conformation; Receptors, Nicotinic; Spectrometry, Fluorescence; Spectrophotometry, Infrared; Torpedo

1992
Probing conformational changes in the nicotinic acetylcholine receptor by Fourier transform infrared difference spectroscopy.
    Biophysical journal, 1992, Volume: 62, Issue:1

    Topics: Animals; Biophysical Phenomena; Biophysics; Carbachol; In Vitro Techniques; Kinetics; Membranes, Artificial; Protein Conformation; Receptors, Nicotinic; Spectrophotometry, Infrared; Torpedo

1992
Electric organ polyamines and their effects on the acetylcholine receptor.
    Cellular and molecular neurobiology, 1992, Volume: 12, Issue:2

    Topics: Animals; Binding, Competitive; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Polyamines; Receptors, Cholinergic; Rubidium; Spermine; Torpedo

1992
Agonist-induced changes in the structure of the acetylcholine receptor M2 regions revealed by photoincorporation of an uncharged nicotinic noncompetitive antagonist.
    The Journal of biological chemistry, 1992, Aug-05, Volume: 267, Issue:22

    Topics: Amino Acid Sequence; Animals; Azirines; Binding Sites; Carbachol; Cell Membrane; Cyanogen Bromide; Electric Organ; Iodine Radioisotopes; Macromolecular Substances; Models, Structural; Molecular Sequence Data; Peptide Fragments; Protein Conformation; Receptors, Nicotinic; Torpedo; Trypsin

1992
Short chain and long chain alkanols have different sites of action on nicotinic acetylcholine receptor channels from Torpedo.
    Molecular pharmacology, 1991, Volume: 39, Issue:3

    Topics: Acetylcholine; Alcohols; Animals; Carbachol; Dose-Response Relationship, Drug; In Vitro Techniques; Ion Channel Gating; Ion Channels; Receptors, Nicotinic; Rubidium; Structure-Activity Relationship; Synaptic Membranes; Torpedo

1991
The hydrophobic photoreagent 3-(trifluoromethyl)-3-m-([125I] iodophenyl) diazirine is a novel noncompetitive antagonist of the nicotinic acetylcholine receptor.
    The Journal of biological chemistry, 1991, Nov-15, Volume: 266, Issue:32

    Topics: Affinity Labels; Amphibian Venoms; Animals; Azirines; Carbachol; Cell Membrane; Electric Organ; Iodine Radioisotopes; Kinetics; Macromolecular Substances; Nicotinic Antagonists; Phencyclidine; Receptors, Nicotinic; Sodium; Torpedo

1991
Effects of pH on acetylcholine receptor function.
    The Journal of membrane biology, 1991, Volume: 120, Issue:1

    Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane Permeability; Electric Conductivity; Electrophysiology; Hydrogen-Ion Concentration; Ion Channel Gating; Liposomes; Membrane Potentials; Microelectrodes; Oocytes; Receptors, Nicotinic; RNA, Messenger; Torpedo; Xenopus laevis

1991
Direct effects of thymopentin (Arg-Lys-Asp-Val-Tyr) on cholinergic agonist-induced slow inactivation of nicotinic acetylcholine receptor function.
    Molecular pharmacology, 1990, Volume: 38, Issue:6

    Topics: Animals; Bungarotoxins; Calcitonin Gene-Related Peptide; Calcium; Carbachol; In Vitro Techniques; Parasympathomimetics; Phencyclidine; Receptors, Nicotinic; Thymopentin; Thymopoietins; Torpedo; Xenopus laevis

1990
The acetylcholine receptor of the neuromuscular junction recognizes mecamylamine as a noncompetitive antagonist.
    Molecular pharmacology, 1985, Volume: 28, Issue:2

    Topics: Amphibian Venoms; Animals; Bungarotoxins; Carbachol; Electric Conductivity; In Vitro Techniques; Ion Channels; Mecamylamine; Muscle Contraction; Neuromuscular Junction; Rana pipiens; Receptors, Nicotinic; Synaptic Transmission; Torpedo; Tubocurarine

1985
Binding of [3H]perhydrohistrionicotoxin and [3H]phencyclidine to the nicotinic receptor-ion channel complex of Torpedo electroplax. Inhibition by histrionicotoxins and derivatives.
    Biochemical pharmacology, 1985, Sep-01, Volume: 34, Issue:17

    Topics: Amphibian Venoms; Animals; Binding, Competitive; Carbachol; Chemical Phenomena; Chemistry; Electric Organ; In Vitro Techniques; Ion Channels; Phencyclidine; Receptors, Nicotinic; Structure-Activity Relationship; Torpedo

1985
Interactions of chlordecone (kepone) and mirex with the nicotinic acetylcholine receptor--ion channel complex.
    Toxicology letters, 1986, Volume: 30, Issue:3

    Topics: Allosteric Regulation; Amphibian Venoms; Animals; Bungarotoxins; Carbachol; Chlordecone; Electric Organ; In Vitro Techniques; Insecticides; Ion Channels; Mirex; Phencyclidine; Receptors, Nicotinic; Torpedo

1986
A monoclonal antibody interfering with binding and response of the acetylcholine receptor.
    The Journal of biological chemistry, 1986, Nov-25, Volume: 261, Issue:33

    Topics: Acetylcholine; Animals; Antibodies, Monoclonal; Antibody Affinity; Antibody Specificity; Binding, Competitive; Carbachol; Cobra Neurotoxin Proteins; Enzyme-Linked Immunosorbent Assay; Hybridomas; Ion Channels; Kinetics; Mice; Parasympathomimetics; Receptors, Nicotinic; Torpedo

1986
Calcium-independent release of acetylcholine from electric organ synaptosomes and its changes by depolarization and cholinergic drugs.
    Journal of neurochemistry, 1988, Volume: 50, Issue:2

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Calcimycin; Calcium; Carbachol; Choline; Electric Organ; Electrophysiology; Gramicidin; Hydrogen-Ion Concentration; Luminescent Measurements; Potassium; Synaptosomes; Torpedo; Valinomycin

1988
Forskolin blocks carbachol-mediated ion-permeability of chick myotube nicotinic receptors and inhibits binding of 3H-phencyclidine to Torpedo microsac nicotinic receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 336, Issue:4

    Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Chick Embryo; Cholera Toxin; Colforsin; Ethidium; In Vitro Techniques; Ion Channels; Microtubules; Phencyclidine; Receptors, Nicotinic; Rubidium Radioisotopes; Torpedo

1987
Actions of pentobarbital enantiomers on nicotinic cholinergic receptors.
    Molecular pharmacology, 1989, Volume: 36, Issue:6

    Topics: Acetylcholine; Allosteric Regulation; Animals; Binding Sites; Carbachol; In Vitro Techniques; Ion Channels; Pentobarbital; Receptors, GABA-A; Receptors, Nicotinic; Rubidium; Stereoisomerism; Torpedo

1989
Covalent labeling of functional states of the acetylcholine receptor. Effects of antagonists on the receptor conformation.
    European journal of biochemistry, 1985, Mar-15, Volume: 147, Issue:3

    Topics: Acetylcholine; Affinity Labels; Animals; Carbachol; Chemical Phenomena; Chemistry; Choline; Electric Organ; Gallamine Triethiodide; Hexamethonium; Hexamethonium Compounds; In Vitro Techniques; Ion Channels; Kinetics; Lasers; Onium Compounds; Photochemistry; Protein Conformation; Receptors, Cholinergic; Torpedo; Trityl Compounds; Tubocurarine

1985
Ethanol increases agonist affinity for nicotinic receptors from Torpedo.
    Biochimica et biophysica acta, 1989, Dec-11, Volume: 987, Issue:1

    Topics: Acetylcholine; Animals; Carbachol; Ethanol; Receptors, Nicotinic; Rubidium Radioisotopes; Synaptic Membranes; Torpedo

1989
Conformational states of the nicotinic acetylcholine receptor from Torpedo californica induced by the binding of agonists, antagonists, and local anesthetics. Equilibrium measurements using tritium-hydrogen exchange.
    Biochemistry, 1989, Jan-10, Volume: 28, Issue:1

    Topics: Animals; Binding, Competitive; Bungarotoxins; Carbachol; Electric Organ; Hydrogen; In Vitro Techniques; Procaine; Protein Conformation; Receptors, Nicotinic; Tetracaine; Torpedo; Tritium

1989
Three-dimensional structure of the nicotinic acetylcholine receptor and location of the major associated 43-kD cytoskeletal protein, determined at 22 A by low dose electron microscopy and x-ray diffraction to 12.5 A.
    The Journal of cell biology, 1989, Volume: 109, Issue:2

    Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Crystallization; Cytoplasm; Cytoskeletal Proteins; Electric Organ; Image Processing, Computer-Assisted; Lipids; Microscopy, Electron; Molecular Structure; Molecular Weight; Receptors, Cholinergic; Receptors, Nicotinic; Torpedo; X-Ray Diffraction

1989
Secondary structural analyses of the nicotinic acetylcholine receptor as a test of molecular models.
    The Journal of biological chemistry, 1988, Mar-05, Volume: 263, Issue:7

    Topics: Animals; Carbachol; Cholic Acid; Cholic Acids; Circular Dichroism; Electrophoresis, Polyacrylamide Gel; Hexamethonium; Hexamethonium Compounds; Liposomes; Protein Conformation; Receptors, Nicotinic; Solubility; Torpedo

1988
Allosteric effects of diprobutine on acetylcholine receptors.
    European journal of pharmacology, 1985, Nov-05, Volume: 117, Issue:2

    Topics: Allosteric Site; Animals; Antiparkinson Agents; Binding, Competitive; Brain; Butylamines; Carbachol; Electric Organ; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Permeability; Rats; Receptors, Cholinergic; Receptors, Neurotransmitter; Receptors, Nicotinic; Receptors, Phencyclidine; Sodium; Torpedo

1985
Correlation between acetylcholine receptor function and structural properties of membranes.
    Biochemistry, 1986, Feb-25, Volume: 25, Issue:4

    Topics: Animals; Biological Transport, Active; Bungarotoxins; Carbachol; Cell Membrane; Chromatography, Affinity; Electric Organ; Electron Spin Resonance Spectroscopy; Kinetics; Membrane Fluidity; Membrane Lipids; Membrane Proteins; Phospholipids; Receptors, Cholinergic; Rubidium; Torpedo

1986
Is agonist self-inhibition at the nicotinic acetylcholine receptor a nonspecific action?
    Biochemistry, 1987, May-19, Volume: 26, Issue:10

    Topics: Acetylcholine; Animals; Carbachol; Choline; Electric Organ; Electron Spin Resonance Spectroscopy; Isoflurophate; Kinetics; Nicotine; Quaternary Ammonium Compounds; Receptors, Nicotinic; Rubidium; Synaptic Membranes; Torpedo

1987
Desensitization of the nicotinic acetylcholine receptor by diisopropylfluorophosphate.
    Journal of biochemical toxicology, 1988,Spring, Volume: 3

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Bungarotoxins; Carbachol; Electric Organ; Isoflurophate; Kinetics; Phencyclidine; Receptors, Nicotinic; Torpedo

1988
Synthesis and biological characterization of pyridohomotropanes. Structure-activity relationships of conformationally restricted nicotinoids.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:3

    Topics: Animals; Brain; Carbachol; Electric Organ; Ganglionic Stimulants; In Vitro Techniques; Nicotine; Pyridines; Rats; Receptors, Nicotinic; Structure-Activity Relationship; Torpedo; Tropanes

1988
Measuring relative acetylcholine receptor agonist binding by selective proton nuclear magnetic resonance relaxation experiments.
    Biophysical journal, 1988, Volume: 53, Issue:6

    Topics: Acetylcholine; Animals; Binding, Competitive; Carbachol; Cell Membrane; Electric Organ; Magnetic Resonance Spectroscopy; Muscarine; Nicotine; Receptors, Cholinergic; Torpedo

1988
Monoclonal antibodies as probes of the alpha-bungarotoxin and cholinergic binding regions of the acetylcholine receptor.
    The Journal of biological chemistry, 1987, Apr-15, Volume: 262, Issue:11

    Topics: Animals; Antibodies, Monoclonal; Binding Sites; Bungarotoxins; Carbachol; Centrifugation, Density Gradient; Enzyme-Linked Immunosorbent Assay; Molecular Weight; Receptors, Cholinergic; Torpedo; Tubocurarine

1987
Interaction of noncompetitive inhibitors with the acetylcholine receptor. The site specificity and spectroscopic properties of ethidium binding.
    The Journal of biological chemistry, 1987, May-25, Volume: 262, Issue:15

    Topics: Acetylcholine; Allosteric Site; Animals; Binding Sites; Binding, Competitive; Carbachol; Cell Membrane; Electric Organ; Ethidium; Fluorescence; Fluorescence Polarization; Phencyclidine; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo

1987
Structure of the high-affinity binding site for noncompetitive blockers of the acetylcholine receptor: [3H]chlorpromazine labels homologous residues in the beta and delta chains.
    Biochemistry, 1987, May-05, Volume: 26, Issue:9

    Topics: Amino Acid Sequence; Amino Acids; Animals; Carbachol; Cell Membrane; Chlorpromazine; Macromolecular Substances; Models, Molecular; Peptide Fragments; Phencyclidine; Receptors, Cholinergic; Torpedo

1987
Purification and characterization of a nicotinic acetylcholine receptor from chick brain.
    Biochemistry, 1986, Apr-22, Volume: 25, Issue:8

    Topics: Acetylcholine; Animals; Antibodies, Monoclonal; Antigen-Antibody Complex; Brain; Bungarotoxins; Carbachol; Chick Embryo; Chickens; Chromatography, Affinity; Electric Organ; Kinetics; Macromolecular Substances; Molecular Weight; Muscles; Peptide Fragments; Receptors, Nicotinic; Torpedo

1986
Labeling of functionally sensitive sulfhydryl-containing domains of acetylcholine receptor from Torpedo californica membranes.
    The Journal of biological chemistry, 1986, Aug-05, Volume: 261, Issue:22

    Topics: Alkylation; Animals; Binding, Competitive; Bungarotoxins; Carbachol; Cell Membrane; Cell Membrane Permeability; Cysteine; Electric Organ; Ethylmaleimide; Fluorescent Dyes; Humans; Hydrogen-Ion Concentration; Maleimides; Receptors, Cholinergic; Spectrometry, Fluorescence; Sulfhydryl Compounds; Sulfhydryl Reagents; Torpedo

1986
The reaction site of a non-competitive antagonist in the delta-subunit of the nicotinic acetylcholine receptor.
    The EMBO journal, 1986, Volume: 5, Issue:8

    Topics: Amino Acid Sequence; Amphibian Venoms; Animals; Binding Sites; Carbachol; Electric Organ; Kinetics; Macromolecular Substances; Onium Compounds; Receptors, Nicotinic; Torpedo; Trityl Compounds

1986
Stimulation of protein methylase II from Torpedo marmorata by cholinergic effectors.
    Biochimica et biophysica acta, 1986, Jan-16, Volume: 854, Issue:1

    Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Cytosol; Electric Organ; Gallamine Triethiodide; Kinetics; Methylation; Phosphates; Phospholipases A; Phospholipases A2; Protein Methyltransferases; Protein O-Methyltransferase; Receptors, Cholinergic; S-Adenosylmethionine; Torpedo

1986
Mechanism of binding of a benzomorphan opiate to the acetylcholine receptor from Torpedo electroplaque.
    Molecular pharmacology, 1986, Volume: 29, Issue:2

    Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Carbachol; Decamethonium Compounds; In Vitro Techniques; Kinetics; Phenazocine; Phencyclidine; Receptors, Cholinergic; Structure-Activity Relationship; Tetracaine; Torpedo; Tritium; Tubocurarine

1986
Comparison of the actions of carbamate anticholinesterases on the nicotinic acetylcholine receptor.
    Molecular pharmacology, 1985, Volume: 27, Issue:3

    Topics: Acetylcholine; Amphibian Venoms; Animals; Binding, Competitive; Bungarotoxins; Carbachol; Electric Organ; Kinetics; Neostigmine; Physostigmine; Pyridostigmine Bromide; Receptors, Cholinergic; Torpedo

1985
Aryldiazonium salts as photoaffinity labels of the nicotinic acetylcholine receptor PCP binding site.
    FEBS letters, 1985, Mar-25, Volume: 182, Issue:2

    Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Carbachol; Diazonium Compounds; Electric Organ; Phencyclidine; Photochemistry; Receptors, Nicotinic; Torpedo

1985
The role of lipids in the function of the acetylcholine receptor.
    Journal of receptor research, 1985, Volume: 5, Issue:5-6

    Topics: Animals; Carbachol; Cholesterol; In Vitro Techniques; Kinetics; Liposomes; Membrane Fusion; Membrane Lipids; Microscopy, Electron; Phospholipids; Receptors, Cholinergic; Torpedo

1985
Effects of monoclonal antibodies on the function of acetylcholine receptors purified from Torpedo californica and reconstituted into vesicles.
    Biochemistry, 1985, Feb-26, Volume: 24, Issue:5

    Topics: Animals; Antibodies, Monoclonal; Binding, Competitive; Bungarotoxins; Carbachol; Cell Line; Electric Organ; Immunoglobulin Fab Fragments; Kinetics; Mice; Plasmacytoma; Rats; Receptors, Cholinergic; Torpedo

1985
Effects of thio-group modifications of Torpedo californica acetylcholine receptor on ion flux activation and inactivation kinetics.
    Biochemistry, 1984, May-22, Volume: 23, Issue:11

    Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Disulfides; Dithiothreitol; Electric Organ; Electrophorus; Ion Channels; Kinetics; Receptors, Cholinergic; Rubidium; Torpedo

1984
Effects of heating on the ion-gating function and structural domains of the acetylcholine receptor.
    Biochemistry, 1984, Sep-25, Volume: 23, Issue:20

    Topics: Animals; Carbachol; Cell Membrane; Electric Organ; Hot Temperature; Ion Channels; Kinetics; Macromolecular Substances; Molecular Weight; Receptors, Cholinergic; Thermodynamics; Torpedo

1984
Properties of proteoliposomes reconstituted with acetylcholine receptor from Torpedo californica.
    The Journal of biological chemistry, 1982, Aug-25, Volume: 257, Issue:16

    Topics: Animals; Biological Transport; Bungarotoxins; Carbachol; Centrifugation, Density Gradient; Electric Organ; Ion Channels; Kinetics; Liposomes; Receptors, Cholinergic; Torpedo

1982
Allethrin interactions with the nicotinic acetylcholine receptor channel.
    Life sciences, 1982, Oct-11, Volume: 31, Issue:15

    Topics: Acetylcholine; Allethrins; Allosteric Site; Amphibian Venoms; Animals; Binding, Competitive; Carbachol; Electric Organ; Ion Channels; Neurotoxins; Parasympatholytics; Receptors, Cholinergic; Receptors, Nicotinic; Temperature; Torpedo

1982
Activation and inactivation kinetics of Torpedo californica acetylcholine receptor in reconstituted membranes.
    Biochemistry, 1982, Oct-26, Volume: 21, Issue:22

    Topics: Acetylcholine; Animals; Carbachol; Cations; Dose-Response Relationship, Drug; In Vitro Techniques; Ion Channels; Kinetics; Liposomes; Receptors, Cholinergic; Rubidium; Torpedo

1982
Alcohol modulation of drug binding to the channel sites of the nicotinic acetylcholine receptor.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:2

    Topics: Alcohols; Amphibian Venoms; Animals; Carbachol; Drug Interactions; Imipramine; Ion Channels; Membranes; Naphthols; Phencyclidine; Receptors, Cholinergic; Torpedo

1983
Covalent labeling of the acetylcholine receptor from Torpedo electric tissue with the channel blocker [3H]triphenylmethylphosphonium by ultraviolet irradiation.
    Biochemistry, 1983, Jan-18, Volume: 22, Issue:2

    Topics: Acetylcholine; Affinity Labels; Animals; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Hydrogen-Ion Concentration; Ion Channels; Macromolecular Substances; Onium Compounds; Receptors, Cholinergic; Torpedo; Trityl Compounds; Tubocurarine; Ultraviolet Rays

1983
Reaction of quinacrine mustard with the acetylcholine receptor from Torpedo californica.
    The Journal of biological chemistry, 1983, May-25, Volume: 258, Issue:10

    Topics: Animals; Carbachol; Cell Membrane Permeability; Cobra Neurotoxin Proteins; Electric Organ; Ion Channels; Proadifen; Quinacrine; Quinacrine Mustard; Radioisotopes; Receptors, Cholinergic; Rubidium; Torpedo; Tritium; Tubocurarine

1983
Single-channel recordings from purified acetylcholine receptors reconstituted in bilayers formed at the tip of patch pipets.
    Biochemistry, 1983, May-10, Volume: 22, Issue:10

    Topics: Acetylcholine; Animals; Carbachol; Choline; Electric Conductivity; Electric Organ; Ion Channels; Lipid Bilayers; Methods; Receptors, Cholinergic; Torpedo

1983
Absorption filtration. A tool for the measurement of ion tracer flux in native membranes and reconstituted lipid vesicles.
    Biochimica et biophysica acta, 1983, Sep-07, Volume: 733, Issue:2

    Topics: Absorption; Animals; Carbachol; Cell Membrane; Electric Organ; Ion Channels; Kinetics; Liposomes; Receptors, Cholinergic; Sodium; Torpedo

1983
Time-resolved photolabeling by the noncompetitive blocker chlorpromazine of the acetylcholine receptor in its transiently open and closed ion channel conformations.
    Proceedings of the National Academy of Sciences of the United States of America, 1984, Volume: 81, Issue:6

    Topics: Acetylcholine; Animals; Carbachol; Chlorpromazine; Ion Channels; Kinetics; Photochemistry; Receptors, Cholinergic; Torpedo; Tubocurarine

1984
Channel properties of the purified acetylcholine receptor from Torpedo californica reconstituted in planar lipid bilayer membranes.
    Biophysical journal, 1984, Volume: 45, Issue:1

    Topics: Animals; Carbachol; Electric Organ; Ion Channels; Lipid Bilayers; Membrane Potentials; Receptors, Nicotinic; Software; Torpedo

1984
Interactions of gephyrotoxin with the acetylcholine receptor-ionic channel complex. II. Enhancement of desensitization.
    Molecular pharmacology, 1984, Volume: 25, Issue:3

    Topics: Acetylcholine; Alkaloids; Amphibian Venoms; Animals; Carbachol; Drug Synergism; Electric Organ; Evoked Potentials; Ion Channels; Kinetics; Motor Endplate; Muscle Denervation; Muscles; Ranidae; Rats; Receptors, Nicotinic; Torpedo

1984
Effects of calcium on the binding of phencyclidine to acetylcholine receptor-rich membrane fragments from Torpedo californica electroplaque.
    Journal of neurochemistry, 1983, Volume: 41, Issue:4

    Topics: Animals; Calcium; Carbachol; Cations, Divalent; Cell Membrane; Egtazic Acid; Electric Organ; Phencyclidine; Receptors, Cholinergic; Torpedo

1983
Transport of acetylcholine in a membrane. Laminate model of the neuromuscular junction.
    Applied biochemistry and biotechnology, 1984, Volume: 9, Issue:1

    Topics: Acetylcholine; Animals; Biological Transport, Active; Carbachol; Collagen; Electric Organ; Kinetics; Membranes, Artificial; Models, Neurological; Neuromuscular Junction; Sodium; Synaptic Membranes; Torpedo

1984
Modification of alpha-bungarotoxin and cholinergic ligand-binding properties of Torpedo acetylcholine receptor by a monoclonal anti-acetylcholine receptor antibody.
    The Journal of biological chemistry, 1984, Dec-25, Volume: 259, Issue:24

    Topics: Animals; Antibodies, Monoclonal; Antigen-Antibody Complex; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Kinetics; Ligands; Receptors, Cholinergic; Torpedo; Tubocurarine

1984
Ligand-induced effects at regions of acetylcholine receptor accessible to membrane lipids.
    Biochemistry, 1983, Aug-02, Volume: 22, Issue:16

    Topics: Animals; Azides; Carbachol; Cell Membrane; Electric Organ; Kinetics; Ligands; Membrane Lipids; Methane; Nitroparaffins; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo

1983
Multiple binding sites for phencyclidine on the nicotinic acetylcholine receptor from Torpedo ocellata electric organ.
    Life sciences, 1984, Mar-12, Volume: 34, Issue:11

    Topics: Acetylcholine; Animals; Binding Sites; Bungarotoxins; Carbachol; Dibucaine; Electric Organ; Kinetics; Phencyclidine; Receptors, Cholinergic; Tetracaine; Torpedo; Tubocurarine

1984
Localization of phencyclidine binding sites on alpha and beta subunits of the nicotinic acetylcholine receptor from Torpedo ocellata electric organ using azido phencyclidine.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1984, Volume: 4, Issue:3

    Topics: Affinity Labels; Animals; Azides; Binding Sites; Binding, Competitive; Carbachol; Cell Membrane; Electric Organ; Macromolecular Substances; Molecular Weight; Phencyclidine; Photochemistry; Receptors, Nicotinic; Torpedo

1984
Ligand-specific state transitions of the membrane-bound acetylcholine receptor.
    FEBS letters, 1984, Apr-24, Volume: 169, Issue:2

    Topics: 4-Chloro-7-nitrobenzofurazan; Acetylcholine; Anesthetics, Local; Animals; Binding, Competitive; Carbachol; Fluorescence; Gallamine Triethiodide; Receptors, Cholinergic; Time Factors; Torpedo

1984
Mechanism of phencyclidine binding to the acetylcholine receptor from Torpedo electroplaque.
    Molecular pharmacology, 1984, Volume: 25, Issue:3

    Topics: Animals; Carbachol; Cell Membrane; Electric Organ; Glycerol; Kinetics; Phencyclidine; Receptors, Cholinergic; Temperature; Thermodynamics; Torpedo

1984
Functional properties of the acetylcholine receptor incorporated in model lipid membranes. Differential effects of chain length and head group of phospholipids on receptor affinity states and receptor-mediated ion translocation.
    The Journal of biological chemistry, 1984, Jul-25, Volume: 259, Issue:14

    Topics: Animals; Carbachol; Cell Membrane; Cholesterol Esters; Electric Organ; Kinetics; Liposomes; Microscopy, Electron; Models, Biological; Phospholipids; Receptors, Cholinergic; Sodium; Structure-Activity Relationship; Torpedo

1984
Reconstitution of acetylcholine receptor function in lipid vesicles of defined composition.
    Biochimica et biophysica acta, 1983, Jan-05, Volume: 727, Issue:1

    Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Kinetics; Liposomes; Phosphatidylcholines; Phosphatidylserines; Receptors, Cholinergic; Torpedo

1983
Conformational effects of volatile anesthetics on the membrane-bound acetylcholine receptor protein: facilitation of the agonist-induced affinity conversion.
    Biochemistry, 1983, Apr-26, Volume: 22, Issue:9

    Topics: Animals; Carbachol; Cell Membrane; Chloroform; Halothane; Kinetics; Mathematics; Protein Binding; Protein Conformation; Receptors, Cholinergic; Torpedo

1983
Comparison of acetylcholine receptor-controlled cation flux in membrane vesicles from Torpedo californica and Electrophorus electricus: chemical kinetic measurements in the millisecond region.
    Proceedings of the National Academy of Sciences of the United States of America, 1982, Volume: 79, Issue:4

    Topics: Animals; Biological Transport; Carbachol; Cations; Electric Organ; Electrophorus; Kinetics; Membranes; Receptors, Cholinergic; Rubidium; Torpedo

1982
Some neurochemical properties of thiamin.
    Annals of the New York Academy of Sciences, 1982, Volume: 378

    Topics: Anesthetics, Local; Animals; Binding, Competitive; Bungarotoxins; Carbachol; Cell Membrane Permeability; Dose-Response Relationship, Drug; Electric Organ; Potassium Radioisotopes; Receptors, Cholinergic; Sodium Radioisotopes; Thiamine; Thiamine Pyrophosphate; Torpedo

1982
Activation and desensitization of Torpedo acetylcholine receptor: evidence for separate binding sites.
    Proceedings of the National Academy of Sciences of the United States of America, 1982, Volume: 79, Issue:22

    Topics: Acetylcholine; Animals; Binding, Competitive; Carbachol; Cell Membrane; Kinetics; Oxadiazoles; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo

1982
Incorporation of acetylcholine receptors into liposomes. Vesicle structure and acetylcholine receptor function.
    The Journal of biological chemistry, 1982, Jun-25, Volume: 257, Issue:12

    Topics: Animals; Biological Transport, Active; Carbachol; Cell Membrane; Cholesterol; Electric Organ; Freeze Fracturing; Kinetics; Liposomes; Microscopy, Electron; Receptors, Cholinergic; Sodium; Torpedo

1982
Nicotinic acetylcholine receptor desensitization studied by [3H]perhydrohistrionicotoxin binding.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 221, Issue:3

    Topics: Acetylcholinesterase; Amphibian Venoms; Animals; Carbachol; In Vitro Techniques; Isoflurophate; Membranes; Receptors, Cholinergic; Receptors, Nicotinic; Time Factors; Torpedo; Tubocurarine

1982
Interactions of quaternary ammonium drugs with acetylcholinesterase and acetylcholine receptor of Torpedo electric organ.
    Molecular pharmacology, 1982, Volume: 22, Issue:1

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Carbachol; Electric Organ; In Vitro Techniques; Kinetics; Membranes; Quaternary Ammonium Compounds; Receptors, Cholinergic; Sodium; Time Factors; Torpedo

1982
Acetylcholine receptor from Torpedo. Preferential solubilization and efficient reintegration into lipid vesicles.
    Biochimica et biophysica acta, 1982, Oct-07, Volume: 691, Issue:2

    Topics: Animals; Bungarotoxins; Carbachol; Electric Organ; Glucosides; Liposomes; Membrane Lipids; Receptors, Cholinergic; Sodium; Solubility; Torpedo

1982
Multiple binding sites for agonists on Torpedo californica acetylcholine receptor.
    Biochemistry, 1982, Nov-23, Volume: 21, Issue:24

    Topics: Acetylcholine; Animals; Carbachol; Cell Membrane; Choline; Electric Organ; Kinetics; Mathematics; Nicotine; Oxadiazoles; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo

1982
Reconstitution of a functional acetylcholine receptor. Incorporation into artificial lipid vesicles and pharmacology of the agonist-controlled permeability changes.
    European journal of biochemistry, 1981, Volume: 118, Issue:2

    Topics: Acetylcholine; Animals; Carbachol; Cell Membrane Permeability; Cesium; Electric Organ; Hydrogen-Ion Concentration; Membranes, Artificial; Microscopy, Electron; Molecular Weight; Receptors, Cholinergic; Receptors, Nicotinic; Sodium; Torpedo

1981
Effects of local anesthetics and histrionicotoxin on the binding of carbamoylcholine to membrane-bound acetylcholine receptor.
    Biochemistry, 1981, Sep-15, Volume: 20, Issue:19

    Topics: Amphibian Venoms; Anesthetics, Local; Animals; Binding, Competitive; Carbachol; Cell Membrane; Kinetics; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo

1981
Allosteric effects of volatile anesthetics on the membrane-bound acetylcholine receptor protein.
    Molecular pharmacology, 1981, Volume: 20, Issue:3

    Topics: Alcohols; Allosteric Site; alpha7 Nicotinic Acetylcholine Receptor; Anesthetics; Animals; Carbachol; Electric Organ; Halothane; In Vitro Techniques; Kinetics; Membranes; Receptors, Cholinergic; Receptors, Nicotinic; Torpedo

1981
Characterization of the binding of [3H]substance P to the nicotinic acetylcholine receptor of Torpedo electroplaque.
    Molecular pharmacology, 1994, Volume: 45, Issue:2

    Topics: Affinity Labels; Animals; Atropine; Autoradiography; Binding Sites; Bungarotoxins; Carbachol; Cross-Linking Reagents; Electric Organ; Electrophoresis, Polyacrylamide Gel; Nicotinic Antagonists; Phenylalanine; Receptors, Nicotinic; Substance P; Torpedo; Tubocurarine

1994
Secondary structure of the nicotinic acetylcholine receptor: implications for structural models of a ligand-gated ion channel.
    Biochemistry, 1994, Jun-21, Volume: 33, Issue:24

    Topics: Animals; Carbachol; Electric Organ; Ion Channel Gating; Ion Channels; Models, Molecular; Protein Conformation; Protein Structure, Secondary; Receptors, Nicotinic; Spectrometry, Fluorescence; Spectrophotometry, Infrared; Spectroscopy, Fourier Transform Infrared; Tetracaine; Torpedo

1994
Structure of both the ligand- and lipid-dependent channel-inactive states of the nicotinic acetylcholine receptor probed by FTIR spectroscopy and hydrogen exchange.
    Biochemistry, 1995, Nov-21, Volume: 34, Issue:46

    Topics: Animals; Carbachol; Cholesterol; Deuterium; Hydrogen; Hydrogen Bonding; Ion Channels; Lipid Bilayers; Membrane Lipids; Phosphatidic Acids; Phosphatidylcholines; Protein Structure, Secondary; Receptors, Nicotinic; Spectrophotometry; Spectroscopy, Fourier Transform Infrared; Tetracaine; Torpedo

1995
Effects of substance P on the binding of agonists to the nicotinic acetylcholine receptor of Torpedo electroplaque.
    Journal of neurochemistry, 1993, Volume: 60, Issue:6

    Topics: Acetylcholine; Animals; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Kinetics; Least-Squares Analysis; Mathematics; Models, Theoretical; Phencyclidine; Receptors, Nicotinic; Substance P; Time Factors; Torpedo

1993
Stereoselectivity of channel inhibition by secondary alkanol enantiomers at nicotinic acetylcholine receptors.
    Anesthesiology, 1993, Volume: 79, Issue:1

    Topics: Alcohols; Animals; Binding Sites; Carbachol; Ion Channels; Kinetics; Membranes; Models, Biological; Nicotinic Antagonists; Receptors, Nicotinic; Rubidium; Rubidium Radioisotopes; Stereoisomerism; Stimulation, Chemical; Structure-Activity Relationship; Torpedo

1993
Differential agonist-induced displacement of quinacrine and ethidium from their respective histrionicotoxin-sensitive binding sites on the Torpedo acetylcholine receptor.
    Biochemistry, 1995, Feb-07, Volume: 34, Issue:5

    Topics: Acetylcholine; Amphibian Venoms; Animals; Binding Sites; Binding, Competitive; Carbachol; Choline; Cholinergic Agonists; Cholinergic Antagonists; Ethidium; Quinacrine; Receptors, Cholinergic; Torpedo

1995
Site-directed disulfide reduction using an affinity reagent: application on the nicotinic acetylcholine receptor.
    FEBS letters, 1995, Mar-06, Volume: 360, Issue:3

    Topics: Affinity Labels; Animals; Binding Sites; Carbachol; Disulfides; In Vitro Techniques; Kinetics; Oxidation-Reduction; Receptors, Nicotinic; Sulfhydryl Compounds; Torpedo

1995
Cholinergic binding sites on the pentameric acetylcholine receptor of Torpedo californica.
    Biochemistry, 1993, Aug-24, Volume: 32, Issue:33

    Topics: Acetylcholine; Animals; Binding Sites; Carbachol; Cell Membrane; Electric Organ; Fluorescent Dyes; Hexamethonium; Hexamethonium Compounds; Kinetics; Macromolecular Substances; Mathematics; Oxadiazoles; Receptors, Cholinergic; Sulfhydryl Reagents; Torpedo

1993
Identifying the lipid-protein interface of the Torpedo nicotinic acetylcholine receptor: secondary structure implications.
    Biochemistry, 1994, Mar-15, Volume: 33, Issue:10

    Topics: Amino Acid Sequence; Animals; Azirines; Binding Sites; Carbachol; Cell Membrane; Chromatography, High Pressure Liquid; Cross-Linking Reagents; Electric Organ; Electrophoresis, Polyacrylamide Gel; Lipid Metabolism; Models, Molecular; Molecular Sequence Data; Peptide Fragments; Peptide Mapping; Protein Structure, Secondary; Receptors, Nicotinic; Torpedo

1994
Barbiturate action is dependent on the conformational state of the acetylcholine receptor.
    Anesthesiology, 1993, Volume: 79, Issue:5

    Topics: Animals; Barbiturates; Carbachol; Molecular Conformation; Receptors, Cholinergic; Torpedo

1993
Cycloalkanemethanols discriminate between volume- and length-dependent loss of activity of alkanols at the Torpedo nicotinic acetylcholine receptor.
    Molecular pharmacology, 1993, Volume: 44, Issue:6

    Topics: Alcohols; Animals; Carbachol; Dose-Response Relationship, Drug; Methanol; Receptors, Nicotinic; Torpedo

1993
Sodium dodecyl sulfate- and carbamylcholine-induced changes in circular dichroism spectra of acetylcholine receptor synthetic peptides.
    Brain research. Molecular brain research, 1993, Volume: 19, Issue:1-2

    Topics: Amino Acid Sequence; Animals; Bungarotoxins; Carbachol; Circular Dichroism; Macromolecular Substances; Molecular Sequence Data; Peptide Fragments; Peptides; Protein Structure, Secondary; Receptors, Cholinergic; Sodium Dodecyl Sulfate; Torpedo

1993
Xenopus muscle acetylcholine receptor alpha subunits bind ligands with different affinities.
    The Journal of biological chemistry, 1993, Sep-05, Volume: 268, Issue:25

    Topics: 3T3 Cells; Acetylcholine; Animals; Bungarotoxins; Carbachol; Gene Expression; Immunoblotting; Immunosorbent Techniques; Kinetics; Macromolecular Substances; Mice; Muscles; Receptors, Cholinergic; Sodium; Sodium Channels; Torpedo; Transfection; Xenopus laevis

1993
A Raman spectroscopic study of acetylcholine receptor-rich membranes from Torpedo marmorata. Interaction of the receptor with carbamylcholine and (+)-tubocurarine.
    Biochimica et biophysica acta, 1993, Jun-05, Volume: 1148, Issue:2

    Topics: Animals; Carbachol; Cell Membrane; Membrane Lipids; Protein Structure, Secondary; Receptors, Cholinergic; Spectrum Analysis, Raman; Torpedo; Tubocurarine

1993
Rapid changes in light-scattering in the prism of Torpedo electric organ slice associated with the production of postsynaptic potentials.
    Biochemical and biophysical research communications, 1996, Jan-05, Volume: 218, Issue:1

    Topics: Animals; Calcium; Carbachol; Electric Organ; Electric Stimulation; Electrophysiology; In Vitro Techniques; Light; Physostigmine; Scattering, Radiation; Synaptic Transmission; Time Factors; Torpedo; Tubocurarine

1996
Quinacrine noncompetitive inhibitor binding site localized on the Torpedo acetylcholine receptor in the open state.
    Biochemistry, 1996, May-21, Volume: 35, Issue:20

    Topics: Animals; Binding Sites; Carbachol; Cyclic N-Oxides; Dansyl Compounds; Electric Organ; Fluorescent Dyes; In Vitro Techniques; Kinetics; Lipid Bilayers; Nicotinic Antagonists; Protein Conformation; Quaternary Ammonium Compounds; Quinacrine; Receptors, Nicotinic; Spin Labels; Torpedo

1996
Biochemical evaluation of photolabile precursors of choline and of carbamylcholine for potential time-resolved crystallographic studies on cholinesterases.
    Biochemistry, 1996, Aug-20, Volume: 35, Issue:33

    Topics: Acetylcholinesterase; Animals; Butyrylcholinesterase; Carbachol; Choline; Cholinesterase Inhibitors; Crystallography, X-Ray; Edrophonium; Humans; Photochemistry; Torpedo

1996
Effects of antibody binding on structural transitions of the nicotinic acetylcholine receptor.
    Biochemistry, 1996, Sep-10, Volume: 35, Issue:36

    Topics: Affinity Labels; Animals; Antibodies, Monoclonal; Antigen-Antibody Complex; Azirines; Bungarotoxins; Carbachol; Cross-Linking Reagents; Curare; Electrophoresis, Polyacrylamide Gel; Gene Expression; Immunoglobulin Fab Fragments; Oocytes; Patch-Clamp Techniques; Receptors, Nicotinic; Torpedo; Xenopus laevis

1996
Interactions of the nicotinic acetylcholine receptor transmembrane segments with the lipid bilayer in native receptor-rich membranes.
    Biochemistry, 1997, Jan-28, Volume: 36, Issue:4

    Topics: Animals; Binding Sites; Carbachol; Cell Membrane; Cholesterol; Electric Organ; Electron Spin Resonance Spectroscopy; Endopeptidase K; In Vitro Techniques; Ion Channels; Lipid Bilayers; Phospholipids; Phosphorylation; Receptors, Nicotinic; Signal Transduction; Spin Labels; Torpedo; Tyrosine

1997
Agonist binding to the Torpedo acetylcholine receptor. 1. Complexities revealed by dissociation kinetics.
    Biochemistry, 1997, Apr-01, Volume: 36, Issue:13

    Topics: Acetylcholine; Alkaloids; Animals; Binding Sites; Binding, Competitive; Bungarotoxins; Carbachol; Cell Membrane; Choline; Cholinergic Agonists; Dihydro-beta-Erythroidine; Kinetics; Ligands; Membrane Proteins; Protein Binding; Receptors, Cholinergic; Torpedo; Tubocurarine

1997
Chlorpyrifos, parathion, and their oxons bind to and desensitize a nicotinic acetylcholine receptor: relevance to their toxicities.
    Toxicology and applied pharmacology, 1997, Volume: 146, Issue:2

    Topics: Animals; Binding, Competitive; Bungarotoxins; Carbachol; Chlorpyrifos; Cholinesterase Inhibitors; Cholinesterases; Dose-Response Relationship, Drug; Insecticides; Iodine Radioisotopes; Lethal Dose 50; Nicotinic Agonists; Paraoxon; Parathion; Phencyclidine; Receptors, Nicotinic; Structure-Activity Relationship; Torpedo; Tritium

1997
The cholesterol dependence of activation and fast desensitization of the nicotinic acetylcholine receptor.
    Biophysical journal, 1997, Volume: 73, Issue:5

    Topics: Animals; Carbachol; Cholesterol; Ethidium; Fluorescent Dyes; Fluorometry; Kinetics; Lipid Bilayers; Liposomes; Nicotinic Agonists; Phosphatidylcholines; Phospholipids; Receptors, Nicotinic; Torpedo

1997
Differential surface accessibility of alpha(187-199) in the Torpedo acetylcholine receptor alpha subunits.
    Journal of molecular biology, 1998, Sep-18, Volume: 282, Issue:2

    Topics: Animals; Antibodies, Monoclonal; Binding Sites; Bungarotoxins; Carbachol; Epitopes; Kinetics; Membrane Proteins; Octoxynol; Receptors, Nicotinic; Titrimetry; Torpedo; Tubocurarine

1998
A structure-based approach to nicotinic receptor pharmacology.
    Molecular pharmacology, 1999, Volume: 55, Issue:2

    Topics: Anesthetics, Local; Animals; Binding Sites; Binding, Competitive; Carbachol; Dibucaine; Lidocaine; Neurotransmitter Agents; Prilocaine; Protein Conformation; Receptors, Nicotinic; Spectroscopy, Fourier Transform Infrared; Tetracaine; Torpedo

1999
Anesthetic-induced structural changes in the nicotinic acetylcholine receptor.
    Toxicology letters, 1998, Nov-23, Volume: 100-101

    Topics: Anesthetics; Animals; Carbachol; Electric Organ; In Vitro Techniques; Parasympathomimetics; Protein Conformation; Receptors, Nicotinic; Spectroscopy, Fourier Transform Infrared; Torpedo

1998
Electrostatic interactions regulate desensitization of the nicotinic acetylcholine receptor.
    Biophysical journal, 2000, Volume: 78, Issue:3

    Topics: Animals; Binding Sites; Carbachol; Cell Membrane; Dansyl Compounds; Electric Organ; Ethidium; Fluorescent Dyes; Kinetics; Models, Chemical; Models, Molecular; Nicotinic Agonists; Nicotinic Antagonists; Osmolar Concentration; Protein Conformation; Quaternary Ammonium Compounds; Radioligand Assay; Receptors, Nicotinic; Static Electricity; Torpedo

2000
Roles of agonist-binding sites in nicotinic acetylcholine receptor function.
    Biochemical and biophysical research communications, 2000, Dec-20, Volume: 279, Issue:2

    Topics: Animals; Binding Sites; Biological Transport; Carbachol; Cell Membrane; Electric Organ; Ion Channel Gating; Kinetics; Models, Biological; Nicotinic Agonists; Receptors, Nicotinic; Thallium; Torpedo

2000
Conotoxin MI inhibits the alpha-delta acetylcholine binding site of the Torpedo marmorata receptor.
    Biochemical and biophysical research communications, 2002, Jul-26, Volume: 295, Issue:4

    Topics: Acetylcholine; Animals; Binding Sites; Binding, Competitive; Bungarotoxins; Carbachol; Conotoxins; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Protein Binding; Receptors, Nicotinic; Species Specificity; Torpedo

2002
Identification of nicotinic acetylcholine receptor amino acids photolabeled by the volatile anesthetic halothane.
    Biochemistry, 2003, Nov-25, Volume: 42, Issue:46

    Topics: Amino Acid Sequence; Anesthetics, Inhalation; Animals; Binding Sites; Binding, Competitive; Carbachol; Carbon Radioisotopes; Halothane; Isoflurane; Models, Molecular; Molecular Sequence Data; Peptide Fragments; Photoaffinity Labels; Protein Subunits; Receptors, Nicotinic; Sequence Analysis, Protein; Sodium-Potassium-Exchanging ATPase; Torpedo; Tryptophan; Tubocurarine; Tyrosine

2003
Nicotinic receptor inhibition by Tetraponera ant alkaloids.
    Cellular and molecular neurobiology, 2004, Volume: 24, Issue:4

    Topics: Alkaloids; Animals; Ants; Anura; Binding Sites; Binding, Competitive; Brain; Carbachol; Cells, Cultured; Fetus; Ganglia, Autonomic; Heterocyclic Compounds, 3-Ring; Ion Channels; Membrane Potentials; Molecular Structure; Muscle Contraction; Neural Inhibition; Neuromuscular Junction; Patch-Clamp Techniques; PC12 Cells; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Synaptic Transmission; Torpedo; Venoms

2004
The acetylcholinesterase inhibitor BW284c51 is a potent blocker of Torpedo nicotinic AchRs incorporated into the Xenopus oocyte membrane.
    British journal of pharmacology, 2005, Volume: 144, Issue:1

    Topics: Acetylcholine; Animals; Benzenaminium, 4,4'-(3-oxo-1,5-pentanediyl)bis(N,N-dimethyl-N-2-propenyl-), Dibromide; Carbachol; Cell Membrane; Cholinergic Agents; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Electric Conductivity; Female; Inhibitory Concentration 50; Kinetics; Membrane Proteins; Microinjections; Molecular Structure; Neurotransmitter Agents; Nicotinic Antagonists; Oocytes; Patch-Clamp Techniques; Receptors, Muscarinic; Receptors, Nicotinic; Tacrine; Torpedo; Xenopus

2005
Functionality of nitrated acetylcholine receptor: the two-step formation of nitrotyrosines reveals their differential role in effectors binding.
    FEBS letters, 2005, May-09, Volume: 579, Issue:12

    Topics: Acetylcholine; Animals; Autoradiography; Binding Sites; Binding, Competitive; Bungarotoxins; Carbachol; Carbon Radioisotopes; Cell Membrane; Dose-Response Relationship, Drug; Iodine Radioisotopes; Kinetics; Nicotinic Agonists; Protein Binding; Receptors, Nicotinic; Spectrophotometry; Tetranitromethane; Torpedo; Tubocurarine; Tyrosine

2005
Redistribution of terbium ions across acetylcholine receptor-enriched membranes induced by agonist desensitization.
    Biophysical journal, 2009, Apr-08, Volume: 96, Issue:7

    Topics: Animals; Carbachol; Cell Membrane; Cholinergic Agonists; Ion Channel Gating; Ion Channels; Phase Transition; Porosity; Protein Stability; Protein Structure, Tertiary; Receptors, Cholinergic; Scattering, Small Angle; Terbium; Titrimetry; Torpedo; X-Ray Diffraction

2009
Functional nicotinic acetylcholine receptor reconstitution in Au(111)-supported thiolipid monolayers.
    Nanoscale, 2015, Oct-14, Volume: 7, Issue:38

    Topics: Animals; Carbachol; Fish Proteins; Gold; Microscopy, Atomic Force; Receptors, Nicotinic; Sulfhydryl Compounds; Torpedo

2015
Structure of the Native Muscle-type Nicotinic Receptor and Inhibition by Snake Venom Toxins.
    Neuron, 2020, 06-17, Volume: 106, Issue:6

    Topics: Animals; Binding Sites; Bungarotoxins; Carbachol; Cryoelectron Microscopy; Electric Organ; Molecular Conformation; Nicotinic Agonists; Nicotinic Antagonists; Patch-Clamp Techniques; Protein Conformation; Receptors, Nicotinic; Torpedo

2020