torpedo has been researched along with carbachol in 115 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 66 (57.39) | 18.7374 |
1990's | 39 (33.91) | 18.2507 |
2000's | 8 (6.96) | 29.6817 |
2010's | 1 (0.87) | 24.3611 |
2020's | 1 (0.87) | 2.80 |
Authors | Studies |
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Min, CK; Weiland, GA | 2 |
Arrondo, JL; Castresana, J; Fernandez, AM; Fernandez-Ballester, G; Ferragut, JA; Gonzalez-Ros, JM; Laynez, JL | 1 |
Chen, L; Martin, GB; Rechnitz, GA | 1 |
Arrondo, JL; Castresana, J; Fernandez-Ballester, G; Ferragut, JA; Gonzalez-Ros, JM | 1 |
Barth, A; Görne-Tschelnokow, U; Hucho, F; Mäntele, W; Naumann, D | 1 |
Duvvuri, P; Johnson, DA; Kerr, JA; Valenzuela, CF | 1 |
Baenziger, JE; Miller, KW; Rothschild, KJ | 1 |
Baenziger, JE; McCarthy, MP; Miller, KW; Rothschild, KJ | 1 |
Eterović, VA; Ferchmin, PA; Hann, RM; Szczawinska, K | 1 |
Cohen, JB; White, BH | 1 |
Forman, SA; Miller, KW; Wood, SC | 1 |
Cohen, JB; Cohen, SG; Howard, S; White, BH | 1 |
Chen, XJ; Li, L; McNamee, M; Palma, A; Pappone, P | 1 |
Li, LA; McNamee, MG; Ochoa, EL; Plummer, A | 1 |
Albuquerque, EX; Aracava, Y; Eldefrawi, ME; Sherby, SM; VanMeter, WG; Varanda, WA | 1 |
Aoshima, H; Cash, DJ; Hess, GP; Pasquale, EB | 1 |
Albuquerque, EX; Aronstam, RS; Daly, JW; Feigl, DM; King, CT | 1 |
Aronstam, RS; Hong, JS | 1 |
Fels, G; Maelicke, A; Plümer-Wilk, R; Schreiber, M | 1 |
Diebler, MF; Dolezal, V; Israël, M; Lazereg, S; Tucek, S | 1 |
Eriksson, H; Häggblad, J; Hedlund, B; Heilbronn, E | 1 |
Braswell, LM; Forman, SA; Miller, KW; Roth, SH | 1 |
Fahr, A; Heyn, MP; Hucho, F; Lauffer, L; Schmidt, D | 1 |
Forman, SA; Miller, KW; Righi, DL | 1 |
McCarthy, MP; Stroud, RM | 1 |
McCarthy, MP; Mitra, AK; Stroud, RM | 1 |
Mielke, DL; Wallace, BA | 1 |
Bachy, A; Changeux, JP; Chemouilli, P; Heidmann, T; Morre, M | 1 |
Fong, TM; McNamee, MG | 1 |
Firestone, LL; Forman, SA; Miller, KW | 1 |
Bakry, NM; Eldefrawi, ME; Schweizer, G; Valdes, JJ | 1 |
Abood, LG; Kanne, DB | 1 |
Behling, RW; Jelinski, LW; Navon, G; Sammon, MJ; Yamane, T | 1 |
Mihovilovic, M; Richman, DP | 2 |
Herz, JM; Johnson, DA; Taylor, P | 1 |
Changeux, JP; Dennis, M; Giraudat, J; Haumont, PY; Heidmann, T; Lederer, F | 1 |
Lindstrom, JM; Whiting, PJ | 1 |
Clarke, JH; Martinez-Carrion, M | 1 |
Baumann, H; Hucho, F; Lottspeich, F; Muhn, P; Oberthür, W; Wittmann-Liebold, B | 1 |
Nuske, JH | 1 |
Bigelow, J; Michel, L; Oswald, RE | 1 |
Albuquerque, EX; Eldefrawi, AT; Eldefrawi, ME; Sherby, SM | 1 |
Goeldner, M; Hirth, C; Jaganathen, J; Kotzyba-Hibert, F; Lagenbuch-Cachat, J | 1 |
Raftery, MA; Zabrecky, JR | 1 |
Lindstrom, JM; Wan, KK | 1 |
McNamee, MG; Richardson, CA; Walker, JW | 1 |
Martinez-Carrion, M; Mattingly, JR; Soler, G | 1 |
Huganir, RL; Racker, E | 1 |
Abbassy, MA; Eldefrawi, AT; Eldefrawi, ME | 1 |
McNamee, MG; Takeyasu, K; Walker, JW | 1 |
Abbassy, MA; Ei-Fakahany, EF; Eldefrawi, AT; Eldefrawi, ME; Miller, ER | 1 |
Hucho, F; Muhn, P | 1 |
Kaldany, RR; Karlin, A | 1 |
Lindstrom, J; Montal, M; Suarez-Isla, BA; Wan, K | 1 |
Gonzalez-Ros, JM; Martinez-Carrion, M; Paraschos, A | 2 |
Changeux, JP; Heidmann, T | 1 |
Fredkin, DR; Labarca, P; Montal, M; Suarez-Isla, BA | 1 |
Albuquerque, EX; Aronstam, RS; Daly, JW; Souccar, C; Varanda, WA | 1 |
Oswald, RE | 1 |
Hirose, S; Vieth, WR | 1 |
Farach, MC; Gonzalez-Ros, JM; Martinez-Carrion, M | 1 |
Haring, R; Kloog, Y | 1 |
Haring, R; Kloog, Y; Sokolovsky, M | 1 |
Covarrubias, M; Maelicke, A; Prinz, H | 1 |
Bamberger, MJ; McLaughlin, JT; Oswald, RE | 1 |
Barrantes, FJ; Criado, M; Eibl, H | 1 |
Dalziel, AW; McNamee, MG; Ochoa, EL | 1 |
Sigman, DS; Young, AP | 1 |
Hess, GP; McNamee, MG; Pasquale, EB; Walker, JW | 1 |
Doerge, DR; Ingraham, LL; McNamee, MG | 1 |
Dunn, SM; Raftery, MA | 5 |
Anholt, R; Deerinck, T; Ellisman, M; Fredkin, DR; Lindstrom, J; Montal, M | 1 |
El-Fakahany, EF; Eldefrawi, AT; Eldefrawi, ME | 1 |
Bakry, NM; Eldefrawi, AT; Eldefrawi, ME; Riker, WF | 1 |
Cartaud, J; Changeux, JP; Popot, JL | 1 |
Blanchard, SG; Dunn, SM; Raftery, MA | 1 |
Oshiki, JR; Sigman, DS; Young, AP | 1 |
Min, CK; Owens, J; Weiland, GA | 1 |
Baenziger, JE; McCarthy, MP; Méthot, N | 1 |
Baenziger, JE; Demers, CN; Méthot, N | 1 |
Alifimoff, JK; Bugge, B; Forman, SA; Miller, KW | 1 |
Arias, HR; Johnson, DA | 1 |
Kessler, P; Ménez, A; Servent, D | 1 |
Blanton, MP; Cohen, JB | 1 |
Bugge, B; de Armendi, AJ; Miller, KW; Tonner, PH | 1 |
Hill, WA; Miller, KW; Wood, SC | 1 |
Donnelly-Roberts, DL; Lentz, TL | 1 |
Claudio, T; Wang, YD | 1 |
Aslanian, D; Changeux, JP; Galzi, JL; Grof, P | 1 |
Tasaki, I | 1 |
Ayres, S; Johnson, DA | 1 |
Goeldner, M; Peng, L; Silman, I; Sussman, J | 1 |
Butler, DH; Lasalde, JA; McNamee, MG; Tamamizu, S | 1 |
Dreger, M; Herrmann, A; Hucho, F; Krauss, M | 1 |
Cortes, VI; Eldefrawi, AT; Eldefrawi, ME; Katz, EJ | 1 |
Addona, GH; Bugge, B; Kloczewiak, MA; Miller, KW; Rankin, SE | 1 |
Fairclough, RH; Gudipati, E; Lin, MY; Richman, DP; Twaddle, GM | 1 |
Baenziger, JE; Ryan, SE | 1 |
Baenziger, JE; Nguyen, HP; Ryan, SE | 1 |
Pedersen, SE; Song, XZ | 1 |
Biscoglio de Jiménez Bonino, MJ; Cortez, LM; del Canto, SG; Testai, FD | 1 |
Chiara, DC; Cohen, JB; Dangott, LJ; Eckenhoff, RG | 1 |
Braekman, JC; Kem, WR; LeFrancois, S; Marszalec, W; Raja, M; Wildeboer, K | 1 |
Ivorra, I; Morales, A; Olivera-Bravo, S | 1 |
Martin, JL; Négrerie, M; Nghiêm, HO | 1 |
Chuang, AR; Doniach, S; Fairclough, RH; Lee, TE; Marek, MS | 1 |
Barrantes, FJ; Bonini, IC; Diaz, C; Maza, E; Pissinis, DE; Salvarezza, RC; Schilardi, PL | 1 |
Hibbs, RE; Karlin, A; Lee, M; Noviello, CM; Rahman, MM; Stowell, MHB; Teng, J; Worrell, BT | 1 |
1 review(s) available for torpedo and carbachol
Article | Year |
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Acetylcholine-receptor-mediated ion fluxes in Electrophorus electricus and Torpedo california membrane vesicles.
Topics: Acetylcholine; Animals; Biological Transport; Calcium; Carbachol; Cations, Monovalent; Cell Membrane; Cell Membrane Permeability; Electric Conductivity; Electric Organ; Electrophorus; Electrophysiology; Ion Channels; Kinetics; Lithium; Mathematics; Models, Biological; Muscles; Potassium; Radioisotopes; Receptors, Cholinergic; Rubidium; Sodium; Torpedo | 1985 |
114 other study(ies) available for torpedo and carbachol
Article | Year |
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Substance P inhibits carbamylcholine-stimulated 22Na+ efflux from acetylcholine receptor-enriched Torpedo electroplaque membrane vesicles.
Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Kinetics; Receptors, Nicotinic; Sodium; Sodium Radioisotopes; Substance P; Torpedo | 1992 |
Protein structural effects of agonist binding to the nicotinic acetylcholine receptor.
Topics: Animals; Calorimetry, Differential Scanning; Carbachol; Fourier Analysis; Hot Temperature; Protein Structure, Secondary; Receptors, Nicotinic; Spectrophotometry, Infrared; Torpedo | 1992 |
Microtiter plate binding assay for cholinergic compounds utilizing the nicotinic acetylcholine receptor.
Topics: Animals; Avidin; Binding, Competitive; Biotin; Bungarotoxins; Carbachol; Enzyme-Linked Immunosorbent Assay; Horseradish Peroxidase; Parasympathomimetics; Receptors, Nicotinic; Torpedo | 1992 |
Protein stability and interaction of the nicotinic acetylcholine receptor with cholinergic ligands studied by Fourier-transform infrared spectroscopy.
Topics: Amides; Animals; Carbachol; Detergents; Fourier Analysis; In Vitro Techniques; Ligands; Protein Denaturation; Protein Structure, Secondary; Receptors, Nicotinic; Spectrophotometry, Infrared; Temperature; Torpedo; Trehalose; Tubocurarine | 1992 |
Fourier transform infrared (FTIR) spectroscopic investigation of the nicotinic acetylcholine receptor (nAChR). Investigation of agonist binding and receptor conformational changes by flash-induced release of 'caged' carbamoylcholine.
Topics: Animals; Carbachol; Fourier Analysis; Protein Conformation; Receptors, Nicotinic; Spectrophotometry, Infrared; Torpedo | 1992 |
Modulation of phencyclidine-sensitive ethidium binding to the Torpedo acetylcholine receptor: interaction of noncompetitive inhibitors with carbamylcholine and cobra alpha-toxin.
Topics: Anesthetics; Animals; Barbiturates; Binding Sites; Binding, Competitive; Carbachol; Cholinergic Antagonists; Cobra Neurotoxin Proteins; Drug Interactions; Ethidium; Phencyclidine; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo | 1992 |
Incorporation of the nicotinic acetylcholine receptor into planar multilamellar films: characterization by fluorescence and Fourier transform infrared difference spectroscopy.
Topics: Animals; Biophysical Phenomena; Biophysics; Carbachol; Ethidium; Fourier Analysis; Membranes, Artificial; Protein Conformation; Receptors, Nicotinic; Spectrometry, Fluorescence; Spectrophotometry, Infrared; Torpedo | 1992 |
Probing conformational changes in the nicotinic acetylcholine receptor by Fourier transform infrared difference spectroscopy.
Topics: Animals; Biophysical Phenomena; Biophysics; Carbachol; In Vitro Techniques; Kinetics; Membranes, Artificial; Protein Conformation; Receptors, Nicotinic; Spectrophotometry, Infrared; Torpedo | 1992 |
Electric organ polyamines and their effects on the acetylcholine receptor.
Topics: Animals; Binding, Competitive; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Polyamines; Receptors, Cholinergic; Rubidium; Spermine; Torpedo | 1992 |
Agonist-induced changes in the structure of the acetylcholine receptor M2 regions revealed by photoincorporation of an uncharged nicotinic noncompetitive antagonist.
Topics: Amino Acid Sequence; Animals; Azirines; Binding Sites; Carbachol; Cell Membrane; Cyanogen Bromide; Electric Organ; Iodine Radioisotopes; Macromolecular Substances; Models, Structural; Molecular Sequence Data; Peptide Fragments; Protein Conformation; Receptors, Nicotinic; Torpedo; Trypsin | 1992 |
Short chain and long chain alkanols have different sites of action on nicotinic acetylcholine receptor channels from Torpedo.
Topics: Acetylcholine; Alcohols; Animals; Carbachol; Dose-Response Relationship, Drug; In Vitro Techniques; Ion Channel Gating; Ion Channels; Receptors, Nicotinic; Rubidium; Structure-Activity Relationship; Synaptic Membranes; Torpedo | 1991 |
The hydrophobic photoreagent 3-(trifluoromethyl)-3-m-([125I] iodophenyl) diazirine is a novel noncompetitive antagonist of the nicotinic acetylcholine receptor.
Topics: Affinity Labels; Amphibian Venoms; Animals; Azirines; Carbachol; Cell Membrane; Electric Organ; Iodine Radioisotopes; Kinetics; Macromolecular Substances; Nicotinic Antagonists; Phencyclidine; Receptors, Nicotinic; Sodium; Torpedo | 1991 |
Effects of pH on acetylcholine receptor function.
Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane Permeability; Electric Conductivity; Electrophysiology; Hydrogen-Ion Concentration; Ion Channel Gating; Liposomes; Membrane Potentials; Microelectrodes; Oocytes; Receptors, Nicotinic; RNA, Messenger; Torpedo; Xenopus laevis | 1991 |
Direct effects of thymopentin (Arg-Lys-Asp-Val-Tyr) on cholinergic agonist-induced slow inactivation of nicotinic acetylcholine receptor function.
Topics: Animals; Bungarotoxins; Calcitonin Gene-Related Peptide; Calcium; Carbachol; In Vitro Techniques; Parasympathomimetics; Phencyclidine; Receptors, Nicotinic; Thymopentin; Thymopoietins; Torpedo; Xenopus laevis | 1990 |
The acetylcholine receptor of the neuromuscular junction recognizes mecamylamine as a noncompetitive antagonist.
Topics: Amphibian Venoms; Animals; Bungarotoxins; Carbachol; Electric Conductivity; In Vitro Techniques; Ion Channels; Mecamylamine; Muscle Contraction; Neuromuscular Junction; Rana pipiens; Receptors, Nicotinic; Synaptic Transmission; Torpedo; Tubocurarine | 1985 |
Binding of [3H]perhydrohistrionicotoxin and [3H]phencyclidine to the nicotinic receptor-ion channel complex of Torpedo electroplax. Inhibition by histrionicotoxins and derivatives.
Topics: Amphibian Venoms; Animals; Binding, Competitive; Carbachol; Chemical Phenomena; Chemistry; Electric Organ; In Vitro Techniques; Ion Channels; Phencyclidine; Receptors, Nicotinic; Structure-Activity Relationship; Torpedo | 1985 |
Interactions of chlordecone (kepone) and mirex with the nicotinic acetylcholine receptor--ion channel complex.
Topics: Allosteric Regulation; Amphibian Venoms; Animals; Bungarotoxins; Carbachol; Chlordecone; Electric Organ; In Vitro Techniques; Insecticides; Ion Channels; Mirex; Phencyclidine; Receptors, Nicotinic; Torpedo | 1986 |
A monoclonal antibody interfering with binding and response of the acetylcholine receptor.
Topics: Acetylcholine; Animals; Antibodies, Monoclonal; Antibody Affinity; Antibody Specificity; Binding, Competitive; Carbachol; Cobra Neurotoxin Proteins; Enzyme-Linked Immunosorbent Assay; Hybridomas; Ion Channels; Kinetics; Mice; Parasympathomimetics; Receptors, Nicotinic; Torpedo | 1986 |
Calcium-independent release of acetylcholine from electric organ synaptosomes and its changes by depolarization and cholinergic drugs.
Topics: Acetylcholine; Acetylcholinesterase; Animals; Calcimycin; Calcium; Carbachol; Choline; Electric Organ; Electrophysiology; Gramicidin; Hydrogen-Ion Concentration; Luminescent Measurements; Potassium; Synaptosomes; Torpedo; Valinomycin | 1988 |
Forskolin blocks carbachol-mediated ion-permeability of chick myotube nicotinic receptors and inhibits binding of 3H-phencyclidine to Torpedo microsac nicotinic receptors.
Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Chick Embryo; Cholera Toxin; Colforsin; Ethidium; In Vitro Techniques; Ion Channels; Microtubules; Phencyclidine; Receptors, Nicotinic; Rubidium Radioisotopes; Torpedo | 1987 |
Actions of pentobarbital enantiomers on nicotinic cholinergic receptors.
Topics: Acetylcholine; Allosteric Regulation; Animals; Binding Sites; Carbachol; In Vitro Techniques; Ion Channels; Pentobarbital; Receptors, GABA-A; Receptors, Nicotinic; Rubidium; Stereoisomerism; Torpedo | 1989 |
Covalent labeling of functional states of the acetylcholine receptor. Effects of antagonists on the receptor conformation.
Topics: Acetylcholine; Affinity Labels; Animals; Carbachol; Chemical Phenomena; Chemistry; Choline; Electric Organ; Gallamine Triethiodide; Hexamethonium; Hexamethonium Compounds; In Vitro Techniques; Ion Channels; Kinetics; Lasers; Onium Compounds; Photochemistry; Protein Conformation; Receptors, Cholinergic; Torpedo; Trityl Compounds; Tubocurarine | 1985 |
Ethanol increases agonist affinity for nicotinic receptors from Torpedo.
Topics: Acetylcholine; Animals; Carbachol; Ethanol; Receptors, Nicotinic; Rubidium Radioisotopes; Synaptic Membranes; Torpedo | 1989 |
Conformational states of the nicotinic acetylcholine receptor from Torpedo californica induced by the binding of agonists, antagonists, and local anesthetics. Equilibrium measurements using tritium-hydrogen exchange.
Topics: Animals; Binding, Competitive; Bungarotoxins; Carbachol; Electric Organ; Hydrogen; In Vitro Techniques; Procaine; Protein Conformation; Receptors, Nicotinic; Tetracaine; Torpedo; Tritium | 1989 |
Three-dimensional structure of the nicotinic acetylcholine receptor and location of the major associated 43-kD cytoskeletal protein, determined at 22 A by low dose electron microscopy and x-ray diffraction to 12.5 A.
Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Crystallization; Cytoplasm; Cytoskeletal Proteins; Electric Organ; Image Processing, Computer-Assisted; Lipids; Microscopy, Electron; Molecular Structure; Molecular Weight; Receptors, Cholinergic; Receptors, Nicotinic; Torpedo; X-Ray Diffraction | 1989 |
Secondary structural analyses of the nicotinic acetylcholine receptor as a test of molecular models.
Topics: Animals; Carbachol; Cholic Acid; Cholic Acids; Circular Dichroism; Electrophoresis, Polyacrylamide Gel; Hexamethonium; Hexamethonium Compounds; Liposomes; Protein Conformation; Receptors, Nicotinic; Solubility; Torpedo | 1988 |
Allosteric effects of diprobutine on acetylcholine receptors.
Topics: Allosteric Site; Animals; Antiparkinson Agents; Binding, Competitive; Brain; Butylamines; Carbachol; Electric Organ; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Permeability; Rats; Receptors, Cholinergic; Receptors, Neurotransmitter; Receptors, Nicotinic; Receptors, Phencyclidine; Sodium; Torpedo | 1985 |
Correlation between acetylcholine receptor function and structural properties of membranes.
Topics: Animals; Biological Transport, Active; Bungarotoxins; Carbachol; Cell Membrane; Chromatography, Affinity; Electric Organ; Electron Spin Resonance Spectroscopy; Kinetics; Membrane Fluidity; Membrane Lipids; Membrane Proteins; Phospholipids; Receptors, Cholinergic; Rubidium; Torpedo | 1986 |
Is agonist self-inhibition at the nicotinic acetylcholine receptor a nonspecific action?
Topics: Acetylcholine; Animals; Carbachol; Choline; Electric Organ; Electron Spin Resonance Spectroscopy; Isoflurophate; Kinetics; Nicotine; Quaternary Ammonium Compounds; Receptors, Nicotinic; Rubidium; Synaptic Membranes; Torpedo | 1987 |
Desensitization of the nicotinic acetylcholine receptor by diisopropylfluorophosphate.
Topics: Acetylcholine; Acetylcholinesterase; Animals; Bungarotoxins; Carbachol; Electric Organ; Isoflurophate; Kinetics; Phencyclidine; Receptors, Nicotinic; Torpedo | 1988 |
Synthesis and biological characterization of pyridohomotropanes. Structure-activity relationships of conformationally restricted nicotinoids.
Topics: Animals; Brain; Carbachol; Electric Organ; Ganglionic Stimulants; In Vitro Techniques; Nicotine; Pyridines; Rats; Receptors, Nicotinic; Structure-Activity Relationship; Torpedo; Tropanes | 1988 |
Measuring relative acetylcholine receptor agonist binding by selective proton nuclear magnetic resonance relaxation experiments.
Topics: Acetylcholine; Animals; Binding, Competitive; Carbachol; Cell Membrane; Electric Organ; Magnetic Resonance Spectroscopy; Muscarine; Nicotine; Receptors, Cholinergic; Torpedo | 1988 |
Monoclonal antibodies as probes of the alpha-bungarotoxin and cholinergic binding regions of the acetylcholine receptor.
Topics: Animals; Antibodies, Monoclonal; Binding Sites; Bungarotoxins; Carbachol; Centrifugation, Density Gradient; Enzyme-Linked Immunosorbent Assay; Molecular Weight; Receptors, Cholinergic; Torpedo; Tubocurarine | 1987 |
Interaction of noncompetitive inhibitors with the acetylcholine receptor. The site specificity and spectroscopic properties of ethidium binding.
Topics: Acetylcholine; Allosteric Site; Animals; Binding Sites; Binding, Competitive; Carbachol; Cell Membrane; Electric Organ; Ethidium; Fluorescence; Fluorescence Polarization; Phencyclidine; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo | 1987 |
Structure of the high-affinity binding site for noncompetitive blockers of the acetylcholine receptor: [3H]chlorpromazine labels homologous residues in the beta and delta chains.
Topics: Amino Acid Sequence; Amino Acids; Animals; Carbachol; Cell Membrane; Chlorpromazine; Macromolecular Substances; Models, Molecular; Peptide Fragments; Phencyclidine; Receptors, Cholinergic; Torpedo | 1987 |
Purification and characterization of a nicotinic acetylcholine receptor from chick brain.
Topics: Acetylcholine; Animals; Antibodies, Monoclonal; Antigen-Antibody Complex; Brain; Bungarotoxins; Carbachol; Chick Embryo; Chickens; Chromatography, Affinity; Electric Organ; Kinetics; Macromolecular Substances; Molecular Weight; Muscles; Peptide Fragments; Receptors, Nicotinic; Torpedo | 1986 |
Labeling of functionally sensitive sulfhydryl-containing domains of acetylcholine receptor from Torpedo californica membranes.
Topics: Alkylation; Animals; Binding, Competitive; Bungarotoxins; Carbachol; Cell Membrane; Cell Membrane Permeability; Cysteine; Electric Organ; Ethylmaleimide; Fluorescent Dyes; Humans; Hydrogen-Ion Concentration; Maleimides; Receptors, Cholinergic; Spectrometry, Fluorescence; Sulfhydryl Compounds; Sulfhydryl Reagents; Torpedo | 1986 |
The reaction site of a non-competitive antagonist in the delta-subunit of the nicotinic acetylcholine receptor.
Topics: Amino Acid Sequence; Amphibian Venoms; Animals; Binding Sites; Carbachol; Electric Organ; Kinetics; Macromolecular Substances; Onium Compounds; Receptors, Nicotinic; Torpedo; Trityl Compounds | 1986 |
Stimulation of protein methylase II from Torpedo marmorata by cholinergic effectors.
Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Cytosol; Electric Organ; Gallamine Triethiodide; Kinetics; Methylation; Phosphates; Phospholipases A; Phospholipases A2; Protein Methyltransferases; Protein O-Methyltransferase; Receptors, Cholinergic; S-Adenosylmethionine; Torpedo | 1986 |
Mechanism of binding of a benzomorphan opiate to the acetylcholine receptor from Torpedo electroplaque.
Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Carbachol; Decamethonium Compounds; In Vitro Techniques; Kinetics; Phenazocine; Phencyclidine; Receptors, Cholinergic; Structure-Activity Relationship; Tetracaine; Torpedo; Tritium; Tubocurarine | 1986 |
Comparison of the actions of carbamate anticholinesterases on the nicotinic acetylcholine receptor.
Topics: Acetylcholine; Amphibian Venoms; Animals; Binding, Competitive; Bungarotoxins; Carbachol; Electric Organ; Kinetics; Neostigmine; Physostigmine; Pyridostigmine Bromide; Receptors, Cholinergic; Torpedo | 1985 |
Aryldiazonium salts as photoaffinity labels of the nicotinic acetylcholine receptor PCP binding site.
Topics: Affinity Labels; Animals; Binding Sites; Bungarotoxins; Carbachol; Diazonium Compounds; Electric Organ; Phencyclidine; Photochemistry; Receptors, Nicotinic; Torpedo | 1985 |
The role of lipids in the function of the acetylcholine receptor.
Topics: Animals; Carbachol; Cholesterol; In Vitro Techniques; Kinetics; Liposomes; Membrane Fusion; Membrane Lipids; Microscopy, Electron; Phospholipids; Receptors, Cholinergic; Torpedo | 1985 |
Effects of monoclonal antibodies on the function of acetylcholine receptors purified from Torpedo californica and reconstituted into vesicles.
Topics: Animals; Antibodies, Monoclonal; Binding, Competitive; Bungarotoxins; Carbachol; Cell Line; Electric Organ; Immunoglobulin Fab Fragments; Kinetics; Mice; Plasmacytoma; Rats; Receptors, Cholinergic; Torpedo | 1985 |
Effects of thio-group modifications of Torpedo californica acetylcholine receptor on ion flux activation and inactivation kinetics.
Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Disulfides; Dithiothreitol; Electric Organ; Electrophorus; Ion Channels; Kinetics; Receptors, Cholinergic; Rubidium; Torpedo | 1984 |
Effects of heating on the ion-gating function and structural domains of the acetylcholine receptor.
Topics: Animals; Carbachol; Cell Membrane; Electric Organ; Hot Temperature; Ion Channels; Kinetics; Macromolecular Substances; Molecular Weight; Receptors, Cholinergic; Thermodynamics; Torpedo | 1984 |
Properties of proteoliposomes reconstituted with acetylcholine receptor from Torpedo californica.
Topics: Animals; Biological Transport; Bungarotoxins; Carbachol; Centrifugation, Density Gradient; Electric Organ; Ion Channels; Kinetics; Liposomes; Receptors, Cholinergic; Torpedo | 1982 |
Allethrin interactions with the nicotinic acetylcholine receptor channel.
Topics: Acetylcholine; Allethrins; Allosteric Site; Amphibian Venoms; Animals; Binding, Competitive; Carbachol; Electric Organ; Ion Channels; Neurotoxins; Parasympatholytics; Receptors, Cholinergic; Receptors, Nicotinic; Temperature; Torpedo | 1982 |
Activation and inactivation kinetics of Torpedo californica acetylcholine receptor in reconstituted membranes.
Topics: Acetylcholine; Animals; Carbachol; Cations; Dose-Response Relationship, Drug; In Vitro Techniques; Ion Channels; Kinetics; Liposomes; Receptors, Cholinergic; Rubidium; Torpedo | 1982 |
Alcohol modulation of drug binding to the channel sites of the nicotinic acetylcholine receptor.
Topics: Alcohols; Amphibian Venoms; Animals; Carbachol; Drug Interactions; Imipramine; Ion Channels; Membranes; Naphthols; Phencyclidine; Receptors, Cholinergic; Torpedo | 1983 |
Covalent labeling of the acetylcholine receptor from Torpedo electric tissue with the channel blocker [3H]triphenylmethylphosphonium by ultraviolet irradiation.
Topics: Acetylcholine; Affinity Labels; Animals; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Hydrogen-Ion Concentration; Ion Channels; Macromolecular Substances; Onium Compounds; Receptors, Cholinergic; Torpedo; Trityl Compounds; Tubocurarine; Ultraviolet Rays | 1983 |
Reaction of quinacrine mustard with the acetylcholine receptor from Torpedo californica.
Topics: Animals; Carbachol; Cell Membrane Permeability; Cobra Neurotoxin Proteins; Electric Organ; Ion Channels; Proadifen; Quinacrine; Quinacrine Mustard; Radioisotopes; Receptors, Cholinergic; Rubidium; Torpedo; Tritium; Tubocurarine | 1983 |
Single-channel recordings from purified acetylcholine receptors reconstituted in bilayers formed at the tip of patch pipets.
Topics: Acetylcholine; Animals; Carbachol; Choline; Electric Conductivity; Electric Organ; Ion Channels; Lipid Bilayers; Methods; Receptors, Cholinergic; Torpedo | 1983 |
Absorption filtration. A tool for the measurement of ion tracer flux in native membranes and reconstituted lipid vesicles.
Topics: Absorption; Animals; Carbachol; Cell Membrane; Electric Organ; Ion Channels; Kinetics; Liposomes; Receptors, Cholinergic; Sodium; Torpedo | 1983 |
Time-resolved photolabeling by the noncompetitive blocker chlorpromazine of the acetylcholine receptor in its transiently open and closed ion channel conformations.
Topics: Acetylcholine; Animals; Carbachol; Chlorpromazine; Ion Channels; Kinetics; Photochemistry; Receptors, Cholinergic; Torpedo; Tubocurarine | 1984 |
Channel properties of the purified acetylcholine receptor from Torpedo californica reconstituted in planar lipid bilayer membranes.
Topics: Animals; Carbachol; Electric Organ; Ion Channels; Lipid Bilayers; Membrane Potentials; Receptors, Nicotinic; Software; Torpedo | 1984 |
Interactions of gephyrotoxin with the acetylcholine receptor-ionic channel complex. II. Enhancement of desensitization.
Topics: Acetylcholine; Alkaloids; Amphibian Venoms; Animals; Carbachol; Drug Synergism; Electric Organ; Evoked Potentials; Ion Channels; Kinetics; Motor Endplate; Muscle Denervation; Muscles; Ranidae; Rats; Receptors, Nicotinic; Torpedo | 1984 |
Effects of calcium on the binding of phencyclidine to acetylcholine receptor-rich membrane fragments from Torpedo californica electroplaque.
Topics: Animals; Calcium; Carbachol; Cations, Divalent; Cell Membrane; Egtazic Acid; Electric Organ; Phencyclidine; Receptors, Cholinergic; Torpedo | 1983 |
Transport of acetylcholine in a membrane. Laminate model of the neuromuscular junction.
Topics: Acetylcholine; Animals; Biological Transport, Active; Carbachol; Collagen; Electric Organ; Kinetics; Membranes, Artificial; Models, Neurological; Neuromuscular Junction; Sodium; Synaptic Membranes; Torpedo | 1984 |
Modification of alpha-bungarotoxin and cholinergic ligand-binding properties of Torpedo acetylcholine receptor by a monoclonal anti-acetylcholine receptor antibody.
Topics: Animals; Antibodies, Monoclonal; Antigen-Antibody Complex; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Kinetics; Ligands; Receptors, Cholinergic; Torpedo; Tubocurarine | 1984 |
Ligand-induced effects at regions of acetylcholine receptor accessible to membrane lipids.
Topics: Animals; Azides; Carbachol; Cell Membrane; Electric Organ; Kinetics; Ligands; Membrane Lipids; Methane; Nitroparaffins; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo | 1983 |
Multiple binding sites for phencyclidine on the nicotinic acetylcholine receptor from Torpedo ocellata electric organ.
Topics: Acetylcholine; Animals; Binding Sites; Bungarotoxins; Carbachol; Dibucaine; Electric Organ; Kinetics; Phencyclidine; Receptors, Cholinergic; Tetracaine; Torpedo; Tubocurarine | 1984 |
Localization of phencyclidine binding sites on alpha and beta subunits of the nicotinic acetylcholine receptor from Torpedo ocellata electric organ using azido phencyclidine.
Topics: Affinity Labels; Animals; Azides; Binding Sites; Binding, Competitive; Carbachol; Cell Membrane; Electric Organ; Macromolecular Substances; Molecular Weight; Phencyclidine; Photochemistry; Receptors, Nicotinic; Torpedo | 1984 |
Ligand-specific state transitions of the membrane-bound acetylcholine receptor.
Topics: 4-Chloro-7-nitrobenzofurazan; Acetylcholine; Anesthetics, Local; Animals; Binding, Competitive; Carbachol; Fluorescence; Gallamine Triethiodide; Receptors, Cholinergic; Time Factors; Torpedo | 1984 |
Mechanism of phencyclidine binding to the acetylcholine receptor from Torpedo electroplaque.
Topics: Animals; Carbachol; Cell Membrane; Electric Organ; Glycerol; Kinetics; Phencyclidine; Receptors, Cholinergic; Temperature; Thermodynamics; Torpedo | 1984 |
Functional properties of the acetylcholine receptor incorporated in model lipid membranes. Differential effects of chain length and head group of phospholipids on receptor affinity states and receptor-mediated ion translocation.
Topics: Animals; Carbachol; Cell Membrane; Cholesterol Esters; Electric Organ; Kinetics; Liposomes; Microscopy, Electron; Models, Biological; Phospholipids; Receptors, Cholinergic; Sodium; Structure-Activity Relationship; Torpedo | 1984 |
Reconstitution of acetylcholine receptor function in lipid vesicles of defined composition.
Topics: Animals; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Kinetics; Liposomes; Phosphatidylcholines; Phosphatidylserines; Receptors, Cholinergic; Torpedo | 1983 |
Conformational effects of volatile anesthetics on the membrane-bound acetylcholine receptor protein: facilitation of the agonist-induced affinity conversion.
Topics: Animals; Carbachol; Cell Membrane; Chloroform; Halothane; Kinetics; Mathematics; Protein Binding; Protein Conformation; Receptors, Cholinergic; Torpedo | 1983 |
Comparison of acetylcholine receptor-controlled cation flux in membrane vesicles from Torpedo californica and Electrophorus electricus: chemical kinetic measurements in the millisecond region.
Topics: Animals; Biological Transport; Carbachol; Cations; Electric Organ; Electrophorus; Kinetics; Membranes; Receptors, Cholinergic; Rubidium; Torpedo | 1982 |
Some neurochemical properties of thiamin.
Topics: Anesthetics, Local; Animals; Binding, Competitive; Bungarotoxins; Carbachol; Cell Membrane Permeability; Dose-Response Relationship, Drug; Electric Organ; Potassium Radioisotopes; Receptors, Cholinergic; Sodium Radioisotopes; Thiamine; Thiamine Pyrophosphate; Torpedo | 1982 |
Activation and desensitization of Torpedo acetylcholine receptor: evidence for separate binding sites.
Topics: Acetylcholine; Animals; Binding, Competitive; Carbachol; Cell Membrane; Kinetics; Oxadiazoles; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo | 1982 |
Incorporation of acetylcholine receptors into liposomes. Vesicle structure and acetylcholine receptor function.
Topics: Animals; Biological Transport, Active; Carbachol; Cell Membrane; Cholesterol; Electric Organ; Freeze Fracturing; Kinetics; Liposomes; Microscopy, Electron; Receptors, Cholinergic; Sodium; Torpedo | 1982 |
Nicotinic acetylcholine receptor desensitization studied by [3H]perhydrohistrionicotoxin binding.
Topics: Acetylcholinesterase; Amphibian Venoms; Animals; Carbachol; In Vitro Techniques; Isoflurophate; Membranes; Receptors, Cholinergic; Receptors, Nicotinic; Time Factors; Torpedo; Tubocurarine | 1982 |
Interactions of quaternary ammonium drugs with acetylcholinesterase and acetylcholine receptor of Torpedo electric organ.
Topics: Acetylcholine; Acetylcholinesterase; Animals; Carbachol; Electric Organ; In Vitro Techniques; Kinetics; Membranes; Quaternary Ammonium Compounds; Receptors, Cholinergic; Sodium; Time Factors; Torpedo | 1982 |
Acetylcholine receptor from Torpedo. Preferential solubilization and efficient reintegration into lipid vesicles.
Topics: Animals; Bungarotoxins; Carbachol; Electric Organ; Glucosides; Liposomes; Membrane Lipids; Receptors, Cholinergic; Sodium; Solubility; Torpedo | 1982 |
Multiple binding sites for agonists on Torpedo californica acetylcholine receptor.
Topics: Acetylcholine; Animals; Carbachol; Cell Membrane; Choline; Electric Organ; Kinetics; Mathematics; Nicotine; Oxadiazoles; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo | 1982 |
Reconstitution of a functional acetylcholine receptor. Incorporation into artificial lipid vesicles and pharmacology of the agonist-controlled permeability changes.
Topics: Acetylcholine; Animals; Carbachol; Cell Membrane Permeability; Cesium; Electric Organ; Hydrogen-Ion Concentration; Membranes, Artificial; Microscopy, Electron; Molecular Weight; Receptors, Cholinergic; Receptors, Nicotinic; Sodium; Torpedo | 1981 |
Effects of local anesthetics and histrionicotoxin on the binding of carbamoylcholine to membrane-bound acetylcholine receptor.
Topics: Amphibian Venoms; Anesthetics, Local; Animals; Binding, Competitive; Carbachol; Cell Membrane; Kinetics; Receptors, Cholinergic; Spectrometry, Fluorescence; Torpedo | 1981 |
Allosteric effects of volatile anesthetics on the membrane-bound acetylcholine receptor protein.
Topics: Alcohols; Allosteric Site; alpha7 Nicotinic Acetylcholine Receptor; Anesthetics; Animals; Carbachol; Electric Organ; Halothane; In Vitro Techniques; Kinetics; Membranes; Receptors, Cholinergic; Receptors, Nicotinic; Torpedo | 1981 |
Characterization of the binding of [3H]substance P to the nicotinic acetylcholine receptor of Torpedo electroplaque.
Topics: Affinity Labels; Animals; Atropine; Autoradiography; Binding Sites; Bungarotoxins; Carbachol; Cross-Linking Reagents; Electric Organ; Electrophoresis, Polyacrylamide Gel; Nicotinic Antagonists; Phenylalanine; Receptors, Nicotinic; Substance P; Torpedo; Tubocurarine | 1994 |
Secondary structure of the nicotinic acetylcholine receptor: implications for structural models of a ligand-gated ion channel.
Topics: Animals; Carbachol; Electric Organ; Ion Channel Gating; Ion Channels; Models, Molecular; Protein Conformation; Protein Structure, Secondary; Receptors, Nicotinic; Spectrometry, Fluorescence; Spectrophotometry, Infrared; Spectroscopy, Fourier Transform Infrared; Tetracaine; Torpedo | 1994 |
Structure of both the ligand- and lipid-dependent channel-inactive states of the nicotinic acetylcholine receptor probed by FTIR spectroscopy and hydrogen exchange.
Topics: Animals; Carbachol; Cholesterol; Deuterium; Hydrogen; Hydrogen Bonding; Ion Channels; Lipid Bilayers; Membrane Lipids; Phosphatidic Acids; Phosphatidylcholines; Protein Structure, Secondary; Receptors, Nicotinic; Spectrophotometry; Spectroscopy, Fourier Transform Infrared; Tetracaine; Torpedo | 1995 |
Effects of substance P on the binding of agonists to the nicotinic acetylcholine receptor of Torpedo electroplaque.
Topics: Acetylcholine; Animals; Bungarotoxins; Carbachol; Cell Membrane; Electric Organ; Kinetics; Least-Squares Analysis; Mathematics; Models, Theoretical; Phencyclidine; Receptors, Nicotinic; Substance P; Time Factors; Torpedo | 1993 |
Stereoselectivity of channel inhibition by secondary alkanol enantiomers at nicotinic acetylcholine receptors.
Topics: Alcohols; Animals; Binding Sites; Carbachol; Ion Channels; Kinetics; Membranes; Models, Biological; Nicotinic Antagonists; Receptors, Nicotinic; Rubidium; Rubidium Radioisotopes; Stereoisomerism; Stimulation, Chemical; Structure-Activity Relationship; Torpedo | 1993 |
Differential agonist-induced displacement of quinacrine and ethidium from their respective histrionicotoxin-sensitive binding sites on the Torpedo acetylcholine receptor.
Topics: Acetylcholine; Amphibian Venoms; Animals; Binding Sites; Binding, Competitive; Carbachol; Choline; Cholinergic Agonists; Cholinergic Antagonists; Ethidium; Quinacrine; Receptors, Cholinergic; Torpedo | 1995 |
Site-directed disulfide reduction using an affinity reagent: application on the nicotinic acetylcholine receptor.
Topics: Affinity Labels; Animals; Binding Sites; Carbachol; Disulfides; In Vitro Techniques; Kinetics; Oxidation-Reduction; Receptors, Nicotinic; Sulfhydryl Compounds; Torpedo | 1995 |
Cholinergic binding sites on the pentameric acetylcholine receptor of Torpedo californica.
Topics: Acetylcholine; Animals; Binding Sites; Carbachol; Cell Membrane; Electric Organ; Fluorescent Dyes; Hexamethonium; Hexamethonium Compounds; Kinetics; Macromolecular Substances; Mathematics; Oxadiazoles; Receptors, Cholinergic; Sulfhydryl Reagents; Torpedo | 1993 |
Identifying the lipid-protein interface of the Torpedo nicotinic acetylcholine receptor: secondary structure implications.
Topics: Amino Acid Sequence; Animals; Azirines; Binding Sites; Carbachol; Cell Membrane; Chromatography, High Pressure Liquid; Cross-Linking Reagents; Electric Organ; Electrophoresis, Polyacrylamide Gel; Lipid Metabolism; Models, Molecular; Molecular Sequence Data; Peptide Fragments; Peptide Mapping; Protein Structure, Secondary; Receptors, Nicotinic; Torpedo | 1994 |
Barbiturate action is dependent on the conformational state of the acetylcholine receptor.
Topics: Animals; Barbiturates; Carbachol; Molecular Conformation; Receptors, Cholinergic; Torpedo | 1993 |
Cycloalkanemethanols discriminate between volume- and length-dependent loss of activity of alkanols at the Torpedo nicotinic acetylcholine receptor.
Topics: Alcohols; Animals; Carbachol; Dose-Response Relationship, Drug; Methanol; Receptors, Nicotinic; Torpedo | 1993 |
Sodium dodecyl sulfate- and carbamylcholine-induced changes in circular dichroism spectra of acetylcholine receptor synthetic peptides.
Topics: Amino Acid Sequence; Animals; Bungarotoxins; Carbachol; Circular Dichroism; Macromolecular Substances; Molecular Sequence Data; Peptide Fragments; Peptides; Protein Structure, Secondary; Receptors, Cholinergic; Sodium Dodecyl Sulfate; Torpedo | 1993 |
Xenopus muscle acetylcholine receptor alpha subunits bind ligands with different affinities.
Topics: 3T3 Cells; Acetylcholine; Animals; Bungarotoxins; Carbachol; Gene Expression; Immunoblotting; Immunosorbent Techniques; Kinetics; Macromolecular Substances; Mice; Muscles; Receptors, Cholinergic; Sodium; Sodium Channels; Torpedo; Transfection; Xenopus laevis | 1993 |
A Raman spectroscopic study of acetylcholine receptor-rich membranes from Torpedo marmorata. Interaction of the receptor with carbamylcholine and (+)-tubocurarine.
Topics: Animals; Carbachol; Cell Membrane; Membrane Lipids; Protein Structure, Secondary; Receptors, Cholinergic; Spectrum Analysis, Raman; Torpedo; Tubocurarine | 1993 |
Rapid changes in light-scattering in the prism of Torpedo electric organ slice associated with the production of postsynaptic potentials.
Topics: Animals; Calcium; Carbachol; Electric Organ; Electric Stimulation; Electrophysiology; In Vitro Techniques; Light; Physostigmine; Scattering, Radiation; Synaptic Transmission; Time Factors; Torpedo; Tubocurarine | 1996 |
Quinacrine noncompetitive inhibitor binding site localized on the Torpedo acetylcholine receptor in the open state.
Topics: Animals; Binding Sites; Carbachol; Cyclic N-Oxides; Dansyl Compounds; Electric Organ; Fluorescent Dyes; In Vitro Techniques; Kinetics; Lipid Bilayers; Nicotinic Antagonists; Protein Conformation; Quaternary Ammonium Compounds; Quinacrine; Receptors, Nicotinic; Spin Labels; Torpedo | 1996 |
Biochemical evaluation of photolabile precursors of choline and of carbamylcholine for potential time-resolved crystallographic studies on cholinesterases.
Topics: Acetylcholinesterase; Animals; Butyrylcholinesterase; Carbachol; Choline; Cholinesterase Inhibitors; Crystallography, X-Ray; Edrophonium; Humans; Photochemistry; Torpedo | 1996 |
Effects of antibody binding on structural transitions of the nicotinic acetylcholine receptor.
Topics: Affinity Labels; Animals; Antibodies, Monoclonal; Antigen-Antibody Complex; Azirines; Bungarotoxins; Carbachol; Cross-Linking Reagents; Curare; Electrophoresis, Polyacrylamide Gel; Gene Expression; Immunoglobulin Fab Fragments; Oocytes; Patch-Clamp Techniques; Receptors, Nicotinic; Torpedo; Xenopus laevis | 1996 |
Interactions of the nicotinic acetylcholine receptor transmembrane segments with the lipid bilayer in native receptor-rich membranes.
Topics: Animals; Binding Sites; Carbachol; Cell Membrane; Cholesterol; Electric Organ; Electron Spin Resonance Spectroscopy; Endopeptidase K; In Vitro Techniques; Ion Channels; Lipid Bilayers; Phospholipids; Phosphorylation; Receptors, Nicotinic; Signal Transduction; Spin Labels; Torpedo; Tyrosine | 1997 |
Agonist binding to the Torpedo acetylcholine receptor. 1. Complexities revealed by dissociation kinetics.
Topics: Acetylcholine; Alkaloids; Animals; Binding Sites; Binding, Competitive; Bungarotoxins; Carbachol; Cell Membrane; Choline; Cholinergic Agonists; Dihydro-beta-Erythroidine; Kinetics; Ligands; Membrane Proteins; Protein Binding; Receptors, Cholinergic; Torpedo; Tubocurarine | 1997 |
Chlorpyrifos, parathion, and their oxons bind to and desensitize a nicotinic acetylcholine receptor: relevance to their toxicities.
Topics: Animals; Binding, Competitive; Bungarotoxins; Carbachol; Chlorpyrifos; Cholinesterase Inhibitors; Cholinesterases; Dose-Response Relationship, Drug; Insecticides; Iodine Radioisotopes; Lethal Dose 50; Nicotinic Agonists; Paraoxon; Parathion; Phencyclidine; Receptors, Nicotinic; Structure-Activity Relationship; Torpedo; Tritium | 1997 |
The cholesterol dependence of activation and fast desensitization of the nicotinic acetylcholine receptor.
Topics: Animals; Carbachol; Cholesterol; Ethidium; Fluorescent Dyes; Fluorometry; Kinetics; Lipid Bilayers; Liposomes; Nicotinic Agonists; Phosphatidylcholines; Phospholipids; Receptors, Nicotinic; Torpedo | 1997 |
Differential surface accessibility of alpha(187-199) in the Torpedo acetylcholine receptor alpha subunits.
Topics: Animals; Antibodies, Monoclonal; Binding Sites; Bungarotoxins; Carbachol; Epitopes; Kinetics; Membrane Proteins; Octoxynol; Receptors, Nicotinic; Titrimetry; Torpedo; Tubocurarine | 1998 |
A structure-based approach to nicotinic receptor pharmacology.
Topics: Anesthetics, Local; Animals; Binding Sites; Binding, Competitive; Carbachol; Dibucaine; Lidocaine; Neurotransmitter Agents; Prilocaine; Protein Conformation; Receptors, Nicotinic; Spectroscopy, Fourier Transform Infrared; Tetracaine; Torpedo | 1999 |
Anesthetic-induced structural changes in the nicotinic acetylcholine receptor.
Topics: Anesthetics; Animals; Carbachol; Electric Organ; In Vitro Techniques; Parasympathomimetics; Protein Conformation; Receptors, Nicotinic; Spectroscopy, Fourier Transform Infrared; Torpedo | 1998 |
Electrostatic interactions regulate desensitization of the nicotinic acetylcholine receptor.
Topics: Animals; Binding Sites; Carbachol; Cell Membrane; Dansyl Compounds; Electric Organ; Ethidium; Fluorescent Dyes; Kinetics; Models, Chemical; Models, Molecular; Nicotinic Agonists; Nicotinic Antagonists; Osmolar Concentration; Protein Conformation; Quaternary Ammonium Compounds; Radioligand Assay; Receptors, Nicotinic; Static Electricity; Torpedo | 2000 |
Roles of agonist-binding sites in nicotinic acetylcholine receptor function.
Topics: Animals; Binding Sites; Biological Transport; Carbachol; Cell Membrane; Electric Organ; Ion Channel Gating; Kinetics; Models, Biological; Nicotinic Agonists; Receptors, Nicotinic; Thallium; Torpedo | 2000 |
Conotoxin MI inhibits the alpha-delta acetylcholine binding site of the Torpedo marmorata receptor.
Topics: Acetylcholine; Animals; Binding Sites; Binding, Competitive; Bungarotoxins; Carbachol; Conotoxins; Dose-Response Relationship, Drug; Electrophoresis, Polyacrylamide Gel; Protein Binding; Receptors, Nicotinic; Species Specificity; Torpedo | 2002 |
Identification of nicotinic acetylcholine receptor amino acids photolabeled by the volatile anesthetic halothane.
Topics: Amino Acid Sequence; Anesthetics, Inhalation; Animals; Binding Sites; Binding, Competitive; Carbachol; Carbon Radioisotopes; Halothane; Isoflurane; Models, Molecular; Molecular Sequence Data; Peptide Fragments; Photoaffinity Labels; Protein Subunits; Receptors, Nicotinic; Sequence Analysis, Protein; Sodium-Potassium-Exchanging ATPase; Torpedo; Tryptophan; Tubocurarine; Tyrosine | 2003 |
Nicotinic receptor inhibition by Tetraponera ant alkaloids.
Topics: Alkaloids; Animals; Ants; Anura; Binding Sites; Binding, Competitive; Brain; Carbachol; Cells, Cultured; Fetus; Ganglia, Autonomic; Heterocyclic Compounds, 3-Ring; Ion Channels; Membrane Potentials; Molecular Structure; Muscle Contraction; Neural Inhibition; Neuromuscular Junction; Patch-Clamp Techniques; PC12 Cells; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Synaptic Transmission; Torpedo; Venoms | 2004 |
The acetylcholinesterase inhibitor BW284c51 is a potent blocker of Torpedo nicotinic AchRs incorporated into the Xenopus oocyte membrane.
Topics: Acetylcholine; Animals; Benzenaminium, 4,4'-(3-oxo-1,5-pentanediyl)bis(N,N-dimethyl-N-2-propenyl-), Dibromide; Carbachol; Cell Membrane; Cholinergic Agents; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Electric Conductivity; Female; Inhibitory Concentration 50; Kinetics; Membrane Proteins; Microinjections; Molecular Structure; Neurotransmitter Agents; Nicotinic Antagonists; Oocytes; Patch-Clamp Techniques; Receptors, Muscarinic; Receptors, Nicotinic; Tacrine; Torpedo; Xenopus | 2005 |
Functionality of nitrated acetylcholine receptor: the two-step formation of nitrotyrosines reveals their differential role in effectors binding.
Topics: Acetylcholine; Animals; Autoradiography; Binding Sites; Binding, Competitive; Bungarotoxins; Carbachol; Carbon Radioisotopes; Cell Membrane; Dose-Response Relationship, Drug; Iodine Radioisotopes; Kinetics; Nicotinic Agonists; Protein Binding; Receptors, Nicotinic; Spectrophotometry; Tetranitromethane; Torpedo; Tubocurarine; Tyrosine | 2005 |
Redistribution of terbium ions across acetylcholine receptor-enriched membranes induced by agonist desensitization.
Topics: Animals; Carbachol; Cell Membrane; Cholinergic Agonists; Ion Channel Gating; Ion Channels; Phase Transition; Porosity; Protein Stability; Protein Structure, Tertiary; Receptors, Cholinergic; Scattering, Small Angle; Terbium; Titrimetry; Torpedo; X-Ray Diffraction | 2009 |
Functional nicotinic acetylcholine receptor reconstitution in Au(111)-supported thiolipid monolayers.
Topics: Animals; Carbachol; Fish Proteins; Gold; Microscopy, Atomic Force; Receptors, Nicotinic; Sulfhydryl Compounds; Torpedo | 2015 |
Structure of the Native Muscle-type Nicotinic Receptor and Inhibition by Snake Venom Toxins.
Topics: Animals; Binding Sites; Bungarotoxins; Carbachol; Cryoelectron Microscopy; Electric Organ; Molecular Conformation; Nicotinic Agonists; Nicotinic Antagonists; Patch-Clamp Techniques; Protein Conformation; Receptors, Nicotinic; Torpedo | 2020 |