Page last updated: 2024-09-04

torcetrapib and niacin

torcetrapib has been researched along with niacin in 13 studies

Compound Research Comparison

Studies
(torcetrapib)
Trials
(torcetrapib)
Recent Studies (post-2010)
(torcetrapib)
Studies
(niacin)
Trials
(niacin)
Recent Studies (post-2010) (niacin)
273288311,9744621,488

Protein Interaction Comparison

ProteinTaxonomytorcetrapib (IC50)niacin (IC50)
Cholesteryl ester transfer proteinHomo sapiens (human)0.14
Cytochrome P450 2C9 Homo sapiens (human)0.14
Hydroxycarboxylic acid receptor 2Homo sapiens (human)0.1726
Hydroxycarboxylic acid receptor 2Mus musculus (house mouse)0.14

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (38.46)29.6817
2010's8 (61.54)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ansell, BJ1
Bloomgarden, ZT1
Suckling, K1
Tan, KC1
Rosenson, RS1
Rizzoni, D; Rossi, GP1
Schaefer, JR1
Kaski, JC1
Abdallah, M; Abi Rafeh, N; Bhat, T; El-Sayegh, S; Kalantar-Zadeh, K; Khoueiry, G; Lafferty, J; Raza, M; Saiful, F1
Taylor, J1
Francis, DP; Keene, D; Price, C; Shun-Shin, MJ1
McCullough, PA; Shin, HJ1

Reviews

6 review(s) available for torcetrapib and niacin

ArticleYear
Rationale for combination therapy with statin drugs in the treatment of dyslipidemia.
    Current atherosclerosis reports, 2005, Volume: 7, Issue:1

    Topics: Anion Exchange Resins; Antihypertensive Agents; Azetidines; Benzenesulfonates; Clofibric Acid; Drug Therapy, Combination; Ezetimibe; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hyperlipidemias; Hypoglycemic Agents; Hypolipidemic Agents; Niacin; Quinolines

2005
Reverse cholesterol transport in type 2 diabetes mellitus.
    Diabetes, obesity & metabolism, 2009, Volume: 11, Issue:6

    Topics: Animals; Anticholesteremic Agents; Apolipoprotein A-I; ATP-Binding Cassette Transporters; Biological Transport; Cholesterol Ester Transfer Proteins; Cholesterol Esters; Diabetes Mellitus, Type 2; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypolipidemic Agents; Lipoproteins, HDL; Liver; Liver X Receptors; Mice; Niacin; Orphan Nuclear Receptors; Peroxisome Proliferator-Activated Receptors; Quinolines; Rabbits; Scavenger Receptors, Class B; Thiazolidinediones

2009
[HDL level or HDL function as the primary target in preventive cardiology].
    Herz, 2012, Volume: 37, Issue:1

    Topics: Anticholesteremic Agents; Atherosclerosis; Atorvastatin; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Cholesterol, LDL; Clinical Trials as Topic; Drug Therapy, Combination; Early Termination of Clinical Trials; Female; Fluorobenzenes; Heptanoic Acids; Humans; Male; Membrane Transport Proteins; Myocardial Infarction; Niacin; Pyrimidines; Pyrroles; Quinolines; Randomized Controlled Trials as Topic; Reference Values; Rosuvastatin Calcium; Scavenger Receptors, Class B; Sulfonamides; Survival Rate; Up-Regulation

2012
High-density lipoprotein in uremic patients: metabolism, impairment, and therapy.
    International urology and nephrology, 2014, Volume: 46, Issue:1

    Topics: Acetamides; Acetates; Acetyl-CoA C-Acetyltransferase; Anti-Inflammatory Agents; Anticholesteremic Agents; Antioxidants; Apolipoprotein A-I; Atherosclerosis; Cholesterol; Cholesterol Ester Transfer Proteins; Dyslipidemias; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypolipidemic Agents; Lipoproteins, HDL; Niacin; PPAR alpha; Quinolines; Renal Insufficiency, Chronic; Sulfonamides; Sulfonic Acids; Uremia

2014
Effect on cardiovascular risk of high density lipoprotein targeted drug treatments niacin, fibrates, and CETP inhibitors: meta-analysis of randomised controlled trials including 117,411 patients.
    BMJ (Clinical research ed.), 2014, Jul-18, Volume: 349

    Topics: Amides; Anticholesteremic Agents; Cholesterol Ester Transfer Proteins; Coronary Disease; Esters; Fibric Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Lipoproteins, HDL; Myocardial Infarction; Niacin; Oxazolidinones; Quinolines; Randomized Controlled Trials as Topic; Stroke; Sulfhydryl Compounds

2014
Focus on lipids: high-density lipoprotein cholesterol and its associated lipoproteins in cardiac and renal disease.
    Nephron. Clinical practice, 2014, Volume: 127, Issue:1-4

    Topics: Amides; Apolipoprotein A-I; Benzodiazepines; Black or African American; Cholesterol Ester Transfer Proteins; Cholesterol Esters; Cholesterol, HDL; Cholesterol, LDL; Cohort Studies; Esters; Heart Diseases; Humans; Hyperlipoproteinemias; Kidney Diseases; Liver; Niacin; Observational Studies as Topic; Oxazolidinones; Prospective Studies; Quinolines; Randomized Controlled Trials as Topic; Risk; Sulfhydryl Compounds; Triglycerides; White People

2014

Other Studies

7 other study(ies) available for torcetrapib and niacin

ArticleYear
2nd International Symposium on Triglycerides and HDL: lipid abnormalities and their treatment.
    Diabetes care, 2005, Volume: 28, Issue:11

    Topics: Anticholesteremic Agents; Cholesterol, HDL; Drug Therapy, Combination; Gemfibrozil; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypolipidemic Agents; Niacin; Quinolines; Simvastatin; Triglycerides

2005
Niacin into the void. Failure of HDL cholesterol drug may B this vitamin's big chance.
    Harvard health letter, 2007, Volume: 32, Issue:6

    Topics: Cholesterol, HDL; Flushing; Humans; Hypolipidemic Agents; Niacin; Quinolines; Treatment Failure

2007
The continuing complexities of high-density lipoprotein metabolism in drug discovery and development.
    Expert opinion on therapeutic targets, 2007, Volume: 11, Issue:9

    Topics: Animals; Anticholesteremic Agents; Atherosclerosis; Blood Pressure; Cholesterol Ester Transfer Proteins; Clinical Trials, Phase III as Topic; Drug Design; Humans; Lipoproteins, HDL; Niacin; Quinolines

2007
Functional assessment of HDL: Moving beyond static measures for risk assessment.
    Cardiovascular drugs and therapy, 2010, Volume: 24, Issue:1

    Topics: Amides; Animals; Anticholesteremic Agents; Azetidines; Cardiovascular Diseases; Cholesterol; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Cholesterol, LDL; Clinical Trials as Topic; Esters; Ezetimibe; Glucose; Humans; Insulin; Lipase; Lipoproteins, HDL; Niacin; Quinolines; Risk Assessment; Risk Factors; Sulfhydryl Compounds

2010
Therapy: raising HDL cholesterol levels: a flight of Icarus?
    Nature reviews. Endocrinology, 2010, Volume: 6, Issue:5

    Topics: Atherosclerosis; Azetidines; Carotid Arteries; Cholesterol, HDL; Cholesterol, LDL; Clinical Trials as Topic; Ezetimibe; Humans; Niacin; Quinolines

2010
HDL- cholesterol: a nut too hard to crack?
    Cardiovascular drugs and therapy, 2012, Volume: 26, Issue:5

    Topics: Anticholesteremic Agents; Atherosclerosis; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Cholesterol, LDL; Humans; Niacin; Quinolines

2012
CardioPulse: is raising HDL a valid treatment target? : epidemiological studies show a relationship between high HDL and lower cardiovascular events but subsequent research casts doubt on treatment benefit.
    European heart journal, 2013, Volume: 34, Issue:16

    Topics: Amides; Anticholesteremic Agents; Cardiovascular Diseases; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Esters; Fibric Acids; Humans; Hypolipidemic Agents; Niacin; Quinolines; Sulfhydryl Compounds

2013