Page last updated: 2024-08-25

topsentin and oxadiazoles

topsentin has been researched along with oxadiazoles in 2 studies

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's2 (100.00)2.80

Authors

AuthorsStudies
Auriemma, G; Carbone, D; Cascioferro, S; Cirrincione, G; Cusimano, MG; Deng, D; Di Sarno, V; Diana, P; Giovannetti, E; Musella, S; Parrino, B; Pecoraro, C; Schillaci, D1
Avan, A; Carbone, D; Cascioferro, S; Diana, P; Giovannetti, E; Parrino, B; Pecoraro, C; Peters, GJ; Puerta, A1

Other Studies

2 other study(ies) available for topsentin and oxadiazoles

ArticleYear
1,2,4-Oxadiazole topsentin analogs as staphylococcal biofilm inhibitors targeting the bacterial transpeptidase sortase A.
    European journal of medicinal chemistry, 2021, Jan-01, Volume: 209

    Topics: Aminoacyltransferases; Anti-Bacterial Agents; Bacterial Proteins; Biofilms; Cell Line; Cysteine Endopeptidases; Humans; Imidazoles; Indoles; Oxadiazoles; Pseudomonas aeruginosa; Pseudomonas Infections; Staphylococcal Infections; Staphylococcus aureus

2021
A New Oxadiazole-Based Topsentin Derivative Modulates Cyclin-Dependent Kinase 1 Expression and Exerts Cytotoxic Effects on Pancreatic Cancer Cells.
    Molecules (Basel, Switzerland), 2021, Dec-21, Volume: 27, Issue:1

    Topics: Antineoplastic Agents; Apoptosis; Carcinoma, Pancreatic Ductal; Catalytic Domain; CDC2 Protein Kinase; Cell Line, Tumor; Cell Proliferation; Drug Screening Assays, Antitumor; Humans; Imidazoles; Indoles; Molecular Docking Simulation; Oxadiazoles; Pancreatic Neoplasms; Protein Binding; Protein Kinase Inhibitors; Signal Transduction; Structure-Activity Relationship

2021