Page last updated: 2024-09-05

tolvaptan and relcovaptan

tolvaptan has been researched along with relcovaptan in 5 studies

Compound Research Comparison

Studies
(tolvaptan)
Trials
(tolvaptan)
Recent Studies (post-2010)
(tolvaptan)
Studies
(relcovaptan)
Trials
(relcovaptan)
Recent Studies (post-2010) (relcovaptan)
967172786120940

Protein Interaction Comparison

ProteinTaxonomytolvaptan (IC50)relcovaptan (IC50)
Vasopressin V1a receptorHomo sapiens (human)0.013

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (60.00)29.6817
2010's2 (40.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Streefkerk, JO; van Zwieten, PA1
Kamyar, M; Lemmens-Gruber, R1
Haass, M1
Fuentes, J; Mancera, JM; MartínezRodríguez, G; Martos-Sitcha, JA1
García-Arroyo, FE; Gonzaga, G; Iroz, A; Johnson, RJ; Muñoz-Jiménez, I; Osorio-Alonso, H; Reyes-García, JG; Roncal-Jiménez, CA; Sánchez-Lozada, LG; Tapia, E; Vecchio, M1

Reviews

3 review(s) available for tolvaptan and relcovaptan

ArticleYear
Vasopressin receptor antagonists: pharmacological tools and potential therapeutic agents.
    Autonomic & autacoid pharmacology, 2006, Volume: 26, Issue:2

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Drug Design; Heart Failure; Hormone Antagonists; Humans; Hypertension; Inappropriate ADH Syndrome; Indoles; Presynaptic Terminals; Pyrrolidines; Receptors, Vasopressin; Renal Artery; Sympathetic Nervous System; Synaptic Transmission; Tolvaptan; Vasoconstriction; Vasoconstrictor Agents

2006
Vasopressin antagonists.
    Cellular and molecular life sciences : CMLS, 2006, Volume: 63, Issue:15

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Azepines; Benzamides; Benzazepines; Binding Sites; Cardiovascular Diseases; Clinical Trials as Topic; Hormone Antagonists; Humans; Indoles; Pyrroles; Pyrrolidines; Tolvaptan; Vasopressins; Water-Electrolyte Imbalance

2006
[Vasopressin receptor antagonists and heart failure].
    Therapeutische Umschau. Revue therapeutique, 2009, Volume: 66, Issue:11

    Topics: Administration, Oral; Aged; Antidiuretic Hormone Receptor Antagonists; Azepines; Benzamides; Benzazepines; Controlled Clinical Trials as Topic; Female; Follow-Up Studies; Furosemide; Heart Failure; Hormone Antagonists; Humans; Hyponatremia; Indoles; Male; Morpholines; Platelet Aggregation Inhibitors; Pyrroles; Pyrrolidines; Sodium Potassium Chloride Symporter Inhibitors; Spiro Compounds; Time Factors; Tolvaptan

2009

Other Studies

2 other study(ies) available for tolvaptan and relcovaptan

ArticleYear
AVT and IT regulate ion transport across the opercular epithelium of killifish (Fundulus heteroclitus) and gilthead sea bream (Sparus aurata).
    Comparative biochemistry and physiology. Part A, Molecular & integrative physiology, 2015, Volume: 182

    Topics: Animals; Benzazepines; Bumetanide; Chlorides; Dose-Response Relationship, Drug; Epithelium; Fish Proteins; Fundulidae; Indoles; Ion Transport; Oxytocin; Pyrrolidines; Receptors, Vasopressin; Sea Bream; Tolvaptan; Vasotocin

2015
A Role for Both V1a and V2 Receptors in Renal Heat Stress Injury Amplified by Rehydration with Fructose.
    International journal of molecular sciences, 2019, Nov-16, Volume: 20, Issue:22

    Topics: Animals; Beverages; Fluid Therapy; Fructose; Heat-Shock Response; Hydrocortisone; Immediate-Early Proteins; Indoles; Kidney Cortex; Male; Oxidative Stress; Protein Serine-Threonine Kinases; Pyrrolidines; Rats; Rats, Wistar; Receptors, Vasopressin; Renal Insufficiency, Chronic; Renin-Angiotensin System; Temperature; Tolvaptan; Up-Regulation

2019