tolvaptan has been researched along with relcovaptan in 5 studies
Studies (tolvaptan) | Trials (tolvaptan) | Recent Studies (post-2010) (tolvaptan) | Studies (relcovaptan) | Trials (relcovaptan) | Recent Studies (post-2010) (relcovaptan) |
---|---|---|---|---|---|
967 | 172 | 786 | 120 | 9 | 40 |
Protein | Taxonomy | tolvaptan (IC50) | relcovaptan (IC50) |
---|---|---|---|
Vasopressin V1a receptor | Homo sapiens (human) | 0.013 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 3 (60.00) | 29.6817 |
2010's | 2 (40.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Streefkerk, JO; van Zwieten, PA | 1 |
Kamyar, M; Lemmens-Gruber, R | 1 |
Haass, M | 1 |
Fuentes, J; Mancera, JM; MartínezRodríguez, G; Martos-Sitcha, JA | 1 |
García-Arroyo, FE; Gonzaga, G; Iroz, A; Johnson, RJ; Muñoz-Jiménez, I; Osorio-Alonso, H; Reyes-García, JG; Roncal-Jiménez, CA; Sánchez-Lozada, LG; Tapia, E; Vecchio, M | 1 |
3 review(s) available for tolvaptan and relcovaptan
Article | Year |
---|---|
Vasopressin receptor antagonists: pharmacological tools and potential therapeutic agents.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Drug Design; Heart Failure; Hormone Antagonists; Humans; Hypertension; Inappropriate ADH Syndrome; Indoles; Presynaptic Terminals; Pyrrolidines; Receptors, Vasopressin; Renal Artery; Sympathetic Nervous System; Synaptic Transmission; Tolvaptan; Vasoconstriction; Vasoconstrictor Agents | 2006 |
Vasopressin antagonists.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Azepines; Benzamides; Benzazepines; Binding Sites; Cardiovascular Diseases; Clinical Trials as Topic; Hormone Antagonists; Humans; Indoles; Pyrroles; Pyrrolidines; Tolvaptan; Vasopressins; Water-Electrolyte Imbalance | 2006 |
[Vasopressin receptor antagonists and heart failure].
Topics: Administration, Oral; Aged; Antidiuretic Hormone Receptor Antagonists; Azepines; Benzamides; Benzazepines; Controlled Clinical Trials as Topic; Female; Follow-Up Studies; Furosemide; Heart Failure; Hormone Antagonists; Humans; Hyponatremia; Indoles; Male; Morpholines; Platelet Aggregation Inhibitors; Pyrroles; Pyrrolidines; Sodium Potassium Chloride Symporter Inhibitors; Spiro Compounds; Time Factors; Tolvaptan | 2009 |
2 other study(ies) available for tolvaptan and relcovaptan
Article | Year |
---|---|
AVT and IT regulate ion transport across the opercular epithelium of killifish (Fundulus heteroclitus) and gilthead sea bream (Sparus aurata).
Topics: Animals; Benzazepines; Bumetanide; Chlorides; Dose-Response Relationship, Drug; Epithelium; Fish Proteins; Fundulidae; Indoles; Ion Transport; Oxytocin; Pyrrolidines; Receptors, Vasopressin; Sea Bream; Tolvaptan; Vasotocin | 2015 |
A Role for Both V1a and V2 Receptors in Renal Heat Stress Injury Amplified by Rehydration with Fructose.
Topics: Animals; Beverages; Fluid Therapy; Fructose; Heat-Shock Response; Hydrocortisone; Immediate-Early Proteins; Indoles; Kidney Cortex; Male; Oxidative Stress; Protein Serine-Threonine Kinases; Pyrrolidines; Rats; Rats, Wistar; Receptors, Vasopressin; Renal Insufficiency, Chronic; Renin-Angiotensin System; Temperature; Tolvaptan; Up-Regulation | 2019 |