tolvaptan has been researched along with opc 21268 in 2 studies
Studies (tolvaptan) | Trials (tolvaptan) | Recent Studies (post-2010) (tolvaptan) | Studies (opc 21268) | Trials (opc 21268) | Recent Studies (post-2010) (opc 21268) |
---|---|---|---|---|---|
967 | 172 | 786 | 133 | 3 | 6 |
Protein | Taxonomy | tolvaptan (IC50) | opc 21268 (IC50) |
---|---|---|---|
Vasopressin V1a receptor | Rattus norvegicus (Norway rat) | 0.44 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 1 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Hirano, T; Itai, A; Kan, K; Kondo, K; Kurimura, M; Mori, T; Nakamura, S; Ogawa, H; Shinohara, T; Tanada, Y; Tominaga, M; Yamamura, Y; Yamashita, H | 1 |
Akahoshi, Y; Fujiki, H; Ikeda, T; Iwanaga, Y; Miyazaki, S; Morooka, H; Watanabe, H | 1 |
2 other study(ies) available for tolvaptan and opc 21268
Article | Year |
---|---|
Novel design of nonpeptide AVP V(2) receptor agonists: structural requirements for an agonist having 1-(4-aminobenzoyl)-2,3,4, 5-tetrahydro-1H-1-benzazepine as a template.
Topics: Administration, Oral; Animals; Arginine Vasopressin; Benzazepines; Cyclic AMP; Diuresis; Drug Design; Female; HeLa Cells; Humans; Models, Molecular; Molecular Conformation; Radioligand Assay; Rats; Receptors, Vasopressin; Structure-Activity Relationship | 2000 |
Effects of Long-term Blockade of Vasopressin Receptor Types 1a and 2 on Cardiac and Renal Damage in a Rat Model of Hypertensive Heart Failure.
Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Disease Models, Animal; Drug Therapy, Combination; Fibrosis; Gene Expression Regulation; Heart Failure; Heart Ventricles; Hemodynamics; Hypertension; Hypertrophy, Left Ventricular; Kidney; Kidney Diseases; Male; Piperidines; Quinolones; Rats, Inbred Dahl; Receptors, Vasopressin; Time Factors; Tolvaptan; Ventricular Function, Left; Ventricular Remodeling | 2015 |