Page last updated: 2024-09-05

tolvaptan and bumetanide

tolvaptan has been researched along with bumetanide in 3 studies

Compound Research Comparison

Studies
(tolvaptan)
Trials
(tolvaptan)
Recent Studies (post-2010)
(tolvaptan)
Studies
(bumetanide)
Trials
(bumetanide)
Recent Studies (post-2010) (bumetanide)
9671727862,033150354

Protein Interaction Comparison

ProteinTaxonomytolvaptan (IC50)bumetanide (IC50)
Solute carrier family 12 member 2Homo sapiens (human)0.8

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's3 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Fuentes, J; Mancera, JM; MartínezRodríguez, G; Martos-Sitcha, JA1

Reviews

1 review(s) available for tolvaptan and bumetanide

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

2 other study(ies) available for tolvaptan and bumetanide

ArticleYear
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
AVT and IT regulate ion transport across the opercular epithelium of killifish (Fundulus heteroclitus) and gilthead sea bream (Sparus aurata).
    Comparative biochemistry and physiology. Part A, Molecular & integrative physiology, 2015, Volume: 182

    Topics: Animals; Benzazepines; Bumetanide; Chlorides; Dose-Response Relationship, Drug; Epithelium; Fish Proteins; Fundulidae; Indoles; Ion Transport; Oxytocin; Pyrrolidines; Receptors, Vasopressin; Sea Bream; Tolvaptan; Vasotocin

2015