Page last updated: 2024-09-04

tipifarnib and manumycin

tipifarnib has been researched along with manumycin in 3 studies

Compound Research Comparison

Studies
(tipifarnib)
Trials
(tipifarnib)
Recent Studies (post-2010)
(tipifarnib)
Studies
(manumycin)
Trials
(manumycin)
Recent Studies (post-2010) (manumycin)
3099294159047

Protein Interaction Comparison

ProteinTaxonomytipifarnib (IC50)manumycin (IC50)
Thioredoxin reductase 1, cytoplasmicRattus norvegicus (Norway rat)0.81
GTPase KRasHomo sapiens (human)3.58

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (66.67)24.3611
2020's1 (33.33)2.80

Authors

AuthorsStudies
Korzeniecki, C; Priefer, R1
Crovella, S; De Leo, L; Decorti, G; Marcuzzi, A; Pontillo, A; Tommasini, A1
Fang, H; Gao, P; Jiang, X; Qiao, J1

Reviews

1 review(s) available for tipifarnib and manumycin

ArticleYear
Targeting KRAS mutant cancers by preventing signaling transduction in the MAPK pathway.
    European journal of medicinal chemistry, 2021, Feb-05, Volume: 211

    Topics: Humans; Models, Molecular; Molecular Structure; Mutation; Protein Kinase Inhibitors; Proto-Oncogene Proteins p21(ras); Signal Transduction

2021

Other Studies

2 other study(ies) available for tipifarnib and manumycin

ArticleYear
The farnesyltransferase inhibitors tipifarnib and lonafarnib inhibit cytokines secretion in a cellular model of mevalonate kinase deficiency.
    Pediatric research, 2011, Volume: 70, Issue:1

    Topics: Acyclic Monoterpenes; Alendronate; Animals; Anti-Inflammatory Agents; Cell Line; Child; Child, Preschool; Cholesterol; Cytokines; Dose-Response Relationship, Drug; Enzyme Inhibitors; Farnesyltranstransferase; Humans; Inflammation Mediators; Lovastatin; Male; Mevalonate Kinase Deficiency; Mice; Monocytes; Phosphotransferases (Alcohol Group Acceptor); Piperidines; Polyenes; Polyisoprenyl Phosphates; Polyunsaturated Alkamides; Pyridines; Quinolones; Terpenes

2011
In vitro antifungal activity of farnesyltransferase inhibitors against clinical isolates of Aspergillus and Candida.
    Annals of clinical microbiology and antimicrobials, 2013, Dec-05, Volume: 12

    Topics: Antifungal Agents; Aspergillosis; Aspergillus; Candida; Candidiasis; Enzyme Inhibitors; Farnesyltranstransferase; Humans; Microbial Sensitivity Tests; Polyenes; Polyunsaturated Alkamides; Quinolones

2013