Page last updated: 2024-09-04

tipifarnib and incb-018424

tipifarnib has been researched along with incb-018424 in 2 studies

Compound Research Comparison

Studies
(tipifarnib)
Trials
(tipifarnib)
Recent Studies (post-2010)
(tipifarnib)
Studies
(incb-018424)
Trials
(incb-018424)
Recent Studies (post-2010) (incb-018424)
30992941,4871851,451

Protein Interaction Comparison

ProteinTaxonomytipifarnib (IC50)incb-018424 (IC50)
Cyclin-G-associated kinaseHomo sapiens (human)0.12
Tyrosine-protein kinase JAK2Homo sapiens (human)0.0573
Cytochrome P450 1A2Homo sapiens (human)0.0001
Tyrosine-protein kinase JAK1Homo sapiens (human)0.0327
Non-receptor tyrosine-protein kinase TYK2Homo sapiens (human)0.0962
Tyrosine-protein kinase JAK3Homo sapiens (human)0.3547
AP2-associated protein kinase 1Homo sapiens (human)0.1
Histone deacetylase 6Homo sapiens (human)0.015

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davis, MI; Khan, J; Li, SQ; Patel, PR; Shen, M; Sun, H; Thomas, CJ1
Barosi, G; Rosti, V1

Reviews

1 review(s) available for tipifarnib and incb-018424

ArticleYear
Novel strategies for patients with chronic myeloproliferative disorders.
    Current opinion in hematology, 2009, Volume: 16, Issue:2

    Topics: Chronic Disease; Humans; Interferon alpha-2; Interferon-alpha; Janus Kinase 2; Mutation; Myeloproliferative Disorders; Nitriles; Primary Myelofibrosis; Pyrazoles; Pyrimidines; Quinolones; Recombinant Proteins; Thalidomide

2009

Other Studies

1 other study(ies) available for tipifarnib and incb-018424

ArticleYear
Identification of potent Yes1 kinase inhibitors using a library screening approach.
    Bioorganic & medicinal chemistry letters, 2013, Aug-01, Volume: 23, Issue:15

    Topics: Binding Sites; Cell Line; Cell Survival; Drug Design; Humans; Hydrogen Bonding; Molecular Docking Simulation; Protein Kinase Inhibitors; Protein Structure, Tertiary; Proto-Oncogene Proteins c-yes; Small Molecule Libraries; Structure-Activity Relationship

2013