Page last updated: 2024-09-04

tipifarnib and fti 276

tipifarnib has been researched along with fti 276 in 3 studies

Compound Research Comparison

Studies
(tipifarnib)
Trials
(tipifarnib)
Recent Studies (post-2010)
(tipifarnib)
Studies
(fti 276)
Trials
(fti 276)
Recent Studies (post-2010) (fti 276)
309929430013

Protein Interaction Comparison

ProteinTaxonomytipifarnib (IC50)fti 276 (IC50)
Protein farnesyltransferase subunit betaSaccharomyces cerevisiae S288C0.0008
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaBos taurus (cattle)0.0005
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaSaccharomyces cerevisiae S288C0.0008
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaHomo sapiens (human)0.0067
Protein farnesyltransferase subunit betaBos taurus (cattle)0.0005
Protein farnesyltransferase subunit betaHomo sapiens (human)0.0033
Geranylgeranyl transferase type-1 subunit betaHomo sapiens (human)0.05
Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alphaMus musculus (house mouse)1
Protein farnesyltransferase subunit betaMus musculus (house mouse)1

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bell, IM1
Distefano, MD; Ochocki, JD1
Buuh, ZY; Lyu, Z; Wang, RE1

Reviews

2 review(s) available for tipifarnib and fti 276

ArticleYear
Inhibitors of farnesyltransferase: a rational approach to cancer chemotherapy?
    Journal of medicinal chemistry, 2004, Apr-08, Volume: 47, Issue:8

    Topics: Alkyl and Aryl Transferases; Animals; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Clinical Trials as Topic; Drug Design; Farnesyltranstransferase; Genes, ras; Humans; Neoplasms

2004
Interrogating the Roles of Post-Translational Modifications of Non-Histone Proteins.
    Journal of medicinal chemistry, 2018, 04-26, Volume: 61, Issue:8

    Topics: Acetylation; Animals; Citrullination; Enzyme Inhibitors; Glycosylation; Humans; Methylation; Phosphorylation; Protein Prenylation; Protein Processing, Post-Translational; Proteins; Ubiquitination

2018

Other Studies

1 other study(ies) available for tipifarnib and fti 276

ArticleYear
Prenyltransferase Inhibitors: Treating Human Ailments from Cancer to Parasitic Infections.
    MedChemComm, 2013, Volume: 4, Issue:3

    Topics:

2013