Page last updated: 2024-08-23

tiotidine and thiazoles

tiotidine has been researched along with thiazoles in 28 studies

Research

Studies (28)

TimeframeStudies, this research(%)All Research%
pre-199025 (89.29)18.7374
1990's3 (10.71)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Buck, SH; Gilman, DJ; Jones, DF; Wardleworth, JM; Yellin, TO1
Hough, LB; Nalwalk, JW1
Nowak, JZ; Sek, B1
Arrang, JM; Garbarg, M; Schwartz, JC1
Nielsen, ST1
Calcutt, CR; Ganellin, CR; Griffiths, R; Leigh, BK; Maguire, JP; Mitchell, RC; Mylek, ME; Parsons, ME; Smith, IR; Young, RC1
Al-Gadi, M; Hill, SJ1
Coombes, JD; Norris, DB; Rising, TJ; Ross, BC; Steward, A1
Levi, R; Trzeciakowski, JP1
Brater, C; Feldman, M; Richardson, CT; Welborn, J1
Brater, DC; Feldman, M; Kaojarern, S; Richardson, CT1
Domschke, S; Domschke, W1
Douglas, AP; Strecker, RB; Valenzuela, JE1
Cheret, AM; Lewin, MJ; Pignal, F1
Avant, GR; Mitchell, MC; Patwardhan, RV; Schenker, S; Speeg, KV1
Bertaccini, G; Coruzzi, G1
Barker, LA1
Batzri, S; Dyer, J; Harmon, JW; Thompson, WF1
Buyniski, JP; Cavanagh, RL; Usakewicz, JJ1
Dinoso, VP1
Baldwin, JJ; Bolhofer, WA; Cragoe, EJ; Habecker, CN; Hoffman, JM; Lumma, WC; Phillips, BT; Pietruszkiewicz, AM; Torchiana, ML1
Radbil', OS; Sukherova, MI1
Flannery, MC; Johnston, BJ; McIsaac, RL1
Yellin, TO; Zavecz, JH1
Lewis, S; Rising, TJ1
Daly, MJ; Humphray, JM; Stables, R1
Agut, J; Ortiz, JA; Sacristán, A; Sánchez, JC1

Reviews

2 review(s) available for tiotidine and thiazoles

ArticleYear
New histamine H2-receptor antagonists.
    Hepato-gastroenterology, 1980, Volume: 27, Issue:3

    Topics: Animals; Anticoagulants; Chemical Phenomena; Chemistry; Cimetidine; Confusion; Dogs; Drug Interactions; Duodenal Ulcer; Furans; Gastric Juice; Gastric Mucosa; Guanidines; Gynecomastia; Histamine H2 Antagonists; Humans; Imidazoles; Male; Molecular Conformation; Ranitidine; Spermatozoa; Thiazoles

1980
[New generation of histamine H2 receptor blockaders].
    Sovetskaia meditsina, 1982, Issue:12

    Topics: Animals; Anti-Ulcer Agents; Cimetidine; Furans; Guanidines; Histamine H2 Antagonists; Humans; Imidazoles; Ranitidine; Thiazoles

1982

Trials

2 trial(s) available for tiotidine and thiazoles

ArticleYear
Tiotidine, a new long-acting histamine H2-receptor antagonist: comparison with cimetidine.
    Gastroenterology, 1981, Volume: 80, Issue:2

    Topics: Adult; Cimetidine; Duodenal Ulcer; Gastric Acid; Gastric Emptying; Gastrins; Guanidines; Histamine H2 Antagonists; Humans; Middle Aged; Polyethylene Glycols; Thiazoles

1981
Tiotidine, a new H2-receptor antagonist, is a potent inhibitor of nocturnal acid secretion in duodenal ulcer patients.
    Digestive diseases and sciences, 1981, Volume: 26, Issue:5

    Topics: Adult; Cimetidine; Drug Evaluation; Duodenal Ulcer; Gastric Acid; Guanidines; Histamine H2 Antagonists; Humans; Middle Aged; Thiazoles

1981

Other Studies

24 other study(ies) available for tiotidine and thiazoles

ArticleYear
ICI 125,211: a new gastric antisecretory agent acting on histamine H2-receptors.
    Life sciences, 1979, Dec-03, Volume: 25, Issue:23

    Topics: Animals; Cimetidine; Dogs; Female; Gastric Mucosa; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine; Histamine H2 Antagonists; Myocardial Contraction; Thiazoles; Thiourea; Time Factors

1979
Inhibition of morphine antinociception by centrally administered histamine H2 receptor antagonists.
    European journal of pharmacology, 1992, Apr-29, Volume: 215, Issue:1

    Topics: Animals; Benzothiazoles; Brain; Cimetidine; Histamine H2 Antagonists; Injections, Intraventricular; Male; Morphine; Nociceptors; Phenoxypropanolamines; Piperidines; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Thiazoles

1992
Cyclic AMP generating systems in vertebrate retina: effects of histamine and an established retinal modulator, dopamine.
    Agents and actions, 1991, Volume: 33, Issue:1-2

    Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Chickens; Cimetidine; Colforsin; Cyclic AMP; Dimaprit; Dopamine; Female; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; Male; Methylhistamines; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Retina; Thiazoles; Thiourea

1991
Autoinhibition of histamine synthesis mediated by presynaptic H3-receptors.
    Neuroscience, 1987, Volume: 23, Issue:1

    Topics: Animals; Burimamide; Cerebral Cortex; Cimetidine; Histamine; Histamine Release; Hypothalamus; Hypothalamus, Posterior; Imidazoles; Impromidine; Male; Potassium; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Histamine; Receptors, Histamine H3; Synaptosomes; Thiazoles

1987
Tiotidine and ICIA 5165 inhibit central and peripheral H2 receptors with equal potency.
    Pharmacology, 1987, Volume: 34, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Animals; Cimetidine; Guanidines; Guinea Pigs; Heart Rate; Hippocampus; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Thiazoles

1987
Zolantidine (SK&F 95282) is a potent selective brain-penetrating histamine H2-receptor antagonist.
    British journal of pharmacology, 1988, Volume: 93, Issue:1

    Topics: Animals; Benzothiazoles; Binding, Competitive; Brain Chemistry; Cimetidine; Cyclic AMP; Female; Guinea Pigs; Hippocampus; Histamine H2 Antagonists; In Vitro Techniques; Male; Phenoxypropanolamines; Piperidines; Rats; Thiazoles; Uterus

1988
Characterization of histamine receptors mediating the stimulation of cyclic AMP accumulation in rabbit cerebral cortical slices.
    British journal of pharmacology, 1985, Volume: 85, Issue:4

    Topics: Adenosine; Animals; Cerebral Cortex; Chlorpheniramine; Cimetidine; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; Imidazoles; Impromidine; Kinetics; Mathematics; Metiamide; Rabbits; Ranitidine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles

1985
In vitro histamine H2-antagonist activity of the novel compound HUK 978.
    Life sciences, 1985, Nov-04, Volume: 37, Issue:18

    Topics: Adenylyl Cyclases; Animals; Cerebral Cortex; Cimetidine; Dose-Response Relationship, Drug; Gastric Mucosa; Guanidines; Guinea Pigs; Histamine; Ileum; Receptors, Histamine; Receptors, Histamine H2; Thiazoles

1985
The cardiac pharmacology of tiotidine (LCL 125, 211): a new histamine H2-receptor antagonist.
    The Journal of pharmacology and experimental therapeutics, 1980, Volume: 214, Issue:3

    Topics: Animals; Arrhythmias, Cardiac; Atrioventricular Node; Cimetidine; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Male; Myocardial Contraction; Thiazoles

1980
New drugs for peptic ulcer.
    British medical journal, 1980, Jul-12, Volume: 281, Issue:6233

    Topics: Benzamides; Benzodiazepinones; Cimetidine; Furans; Guanidines; Histamine H2 Antagonists; Humans; Morpholines; Parasympatholytics; Pepsin A; Peptic Ulcer; Piperazines; Pirenzepine; Prostaglandins E, Synthetic; Ranitidine; Thiazoles; Trimipramine

1980
Tiotidine and cimetidine--kinetics and dynamics.
    Clinical pharmacology and therapeutics, 1981, Volume: 29, Issue:2

    Topics: Adult; Cimetidine; Dose-Response Relationship, Drug; Female; Guanidines; Histamine H2 Antagonists; Humans; Intestinal Absorption; Male; Metabolic Clearance Rate; Middle Aged; Thiazoles; Time Factors

1981
Effects of H2-receptor antagonists cimetidine, ranitidine, and ICI 125,211 on histamine-stimulated adenylate cyclase activity in guinea pig gastric mucosa.
    Molecular pharmacology, 1981, Volume: 20, Issue:2

    Topics: Adenylyl Cyclases; Animals; Cimetidine; Furans; Gastric Mucosa; Guanidines; Guinea Pigs; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Kinetics; Ranitidine; Structure-Activity Relationship; Thiazoles

1981
Inhibition of microsomal drug metabolism by histamine H2-receptor antagonists studied in vivo and in vitro in rodents.
    Gastroenterology, 1982, Volume: 82, Issue:1

    Topics: Aminopyrine; Aminopyrine N-Demethylase; Animals; Breath Tests; Cimetidine; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Furans; Guanidines; Histamine H2 Antagonists; Male; Mice; Mice, Inbred ICR; Microsomes, Liver; Ranitidine; Rats; Rats, Inbred Strains; Thiazoles; Time Factors

1982
Effect of some new Histamine H2-receptor antagonists on the guinea-pig papillary muscle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1981, Volume: 317, Issue:3

    Topics: Animals; Cimetidine; Furans; Guanidines; Guinea Pigs; Histamine Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Myocardial Contraction; Papillary Muscles; Ranitidine; Thiazoles

1981
Histamine H1- and muscarinic receptor antagonist activity of cimetidine and tiotidine in the guinea pig isolated ileum.
    Agents and actions, 1981, Volume: 11, Issue:6-7

    Topics: Animals; Carbachol; Cimetidine; Guanidines; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Thiazoles

1981
Interaction of histamine with gastric mucosal cells. Effect of histamine H2 antagonists on binding and biological response.
    Molecular pharmacology, 1982, Volume: 22, Issue:1

    Topics: Animals; Cimetidine; Cyclic AMP; Furans; Gastric Mucosa; Guanidines; Guinea Pigs; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Ranitidine; Receptors, Histamine; Thiazoles

1982
A comparison of some of the pharmacological properties of etintidine, a new histamine H2-receptor antagonist, with those of cimetidine, ranitidine and tiotidine.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 224, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Cimetidine; Dogs; Female; Furans; Gastric Juice; Guanidines; Guinea Pigs; Heart Rate; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; In Vitro Techniques; Male; Myocardial Contraction; Parasympatholytics; Ranitidine; Rats; Rats, Inbred Strains; Thiazoles; Uterine Contraction

1983
The role of antagonists to acid secretion.
    Comprehensive therapy, 1982, Volume: 8, Issue:12

    Topics: 16,16-Dimethylprostaglandin E2; Benzodiazepinones; Cimetidine; Furans; Gastric Acid; Gastrointestinal Diseases; Guanidines; Histamine H2 Antagonists; Humans; Pirenzepine; Proglumide; Ranitidine; Somatostatin; Thiazoles

1982
Conformational requirements for histamine H2-receptor inhibitors: a structure-activity study of phenylene analogues related to cimetidine and tiotidine.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:2

    Topics: Animals; Benzene Derivatives; Biological Assay; Cimetidine; Dogs; Folic Acid; Gastric Juice; Guanidines; Guinea Pigs; Heart Atria; Histamine H2 Antagonists; Indicators and Reagents; Myocardial Contraction; Receptors, Histamine; Receptors, Histamine H2; Structure-Activity Relationship; Thiazoles

1983
Dose-response curve analysis of gastric secretory responses in the dog and man to impromidine: a new histamine-H2-receptor agonist.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 225, Issue:1

    Topics: Adult; Animals; Binding, Competitive; Cimetidine; Dogs; Dose-Response Relationship, Drug; Female; Gastric Acid; Guanidines; Histamine H2 Antagonists; Humans; Imidazoles; Impromidine; Receptors, Histamine; Receptors, Histamine H2; Thiazoles

1983
Interaction of alpha-adrenergic imidazolines with cardiac histamine H2-receptors.
    European journal of pharmacology, 1981, May-08, Volume: 71, Issue:2-3

    Topics: Animals; Cimetidine; Dose-Response Relationship, Drug; Drug Interactions; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine Release; Imidazoles; In Vitro Techniques; Male; Myocardial Contraction; Receptors, Histamine; Receptors, Histamine H2; Stereoisomerism; Sympathomimetics; Tetrahydronaphthalenes; Thiazoles; Tolazoline

1981
A species comparison of the histamine H2-receptor on mast cells and basophils.
    Agents and actions, 1982, Volume: 12, Issue:3

    Topics: Animals; Basophils; Cimetidine; Female; Furans; Guanidines; Guinea Pigs; Histamine H2 Antagonists; Histamine Release; Humans; In Vitro Techniques; Lung; Male; Mast Cells; Ranitidine; Rats; Receptors, Histamine; Receptors, Histamine H2; Species Specificity; Thiazoles

1982
Pharmacological interactions between ranitidine, cimetidine, metiamide and tiotidine at histamine H2-receptor sites in guinea-pig atria.
    Agents and actions, 1982, Volume: 12, Issue:1-2

    Topics: Animals; Cimetidine; Dimaprit; Drug Interactions; Furans; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine; In Vitro Techniques; Metiamide; Ranitidine; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Thiourea

1982
Action of ebrotidine, ranitidine and cimetidine on the specific binding to histamine H1- and H2-receptors.
    Arzneimittel-Forschung, 1997, Volume: 47, Issue:4A

    Topics: Animals; Benzenesulfonates; Cell Membrane; Cerebellum; Cerebral Cortex; Cimetidine; Depression, Chemical; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Isotope Labeling; Male; Protein Binding; Pyrilamine; Ranitidine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Tritium

1997