tiotidine has been researched along with ranitidine in 33 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 19 (57.58) | 18.7374 |
1990's | 7 (21.21) | 18.2507 |
2000's | 6 (18.18) | 29.6817 |
2010's | 1 (3.03) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Buschauer, A; Elz, S; Hirschfeld, J; Ruat, M; Schunack, W; Schwartz, JC; Traiffort, E | 1 |
Timmerman, H | 1 |
Brown, TH; Ganellin, CR; Griffiths, R; Jones, M; Mitchell, RC; Rana, KK; Saunders, D; Smith, IR; Sore, NE; Young, RC | 1 |
Carrupt, PA; Crivori, P; Cruciani, G; Testa, B | 1 |
Gao, F; Lombardo, F; Shalaeva, MY; Tupper, KA | 1 |
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K | 1 |
Beukers, MW; De Grip, WJ; Klaassen, CH; Leurs, R; Timmerman, H; Verzijl, D | 1 |
Bakker, RA; Leurs, R; Lim, HD; Ling, P; Thurmond, RL; van Rijn, RM | 1 |
Campillo, M; Giraldo, J; Martín, M; Pardo, L | 1 |
Orsetti, M; Sorba, G | 1 |
Krielaart, MJ; van Buuren, KJ; Veenstra, DM | 1 |
Hellstrand, K; Hermodsson, S | 1 |
Jais, AM; Ridzwan, BH; Waton, NG | 1 |
Bast, A; Rekka, E; Sterk, GJ; Timmerman, H | 1 |
Al-Gadi, M; Hill, SJ | 1 |
Hughes, MJ; Kilpatrick, C; Light, KE; Serbus, DC | 1 |
Bast, A; Kroes, BH; Savenije-Chapel, EM | 1 |
Domschke, S; Domschke, W | 1 |
Cheret, AM; Lewin, MJ; Pignal, F | 1 |
Avant, GR; Mitchell, MC; Patwardhan, RV; Schenker, S; Speeg, KV | 1 |
Bertaccini, G; Coruzzi, G | 1 |
Batzri, S; Dyer, J; Harmon, JW; Thompson, WF | 1 |
Buyniski, JP; Cavanagh, RL; Usakewicz, JJ | 1 |
Dinoso, VP | 1 |
Radbil', OS; Sukherova, MI | 1 |
Hirata, Y; Ishii, Y; Yanagisawa, I | 1 |
Lewis, S; Rising, TJ | 1 |
Daly, MJ; Humphray, JM; Stables, R | 1 |
Agut, J; Ortiz, JA; Sacristán, A; Sánchez, JC | 1 |
Asano, T; Fukushima, Y; Kajiwara, T; Katsube, T; Mori, H; Ogawa, K; Ohkawa, SI; Otsuka, H; Saitoh, T; Takahashi, H; Tamai, M | 1 |
Bürckstümmer, T; Buschauer, A; Dove, S; Kelley, MT; Seifert, R; Wenzel-Seifert, K | 1 |
Cannon, KE; Fleck, MW; Hough, LB | 1 |
3 review(s) available for tiotidine and ranitidine
Article | Year |
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Histamine H3 ligands: just pharmacological tools or potential therapeutic agents?
Topics: Animals; Histamine; Histamine Antagonists; Molecular Structure; Neurotransmitter Agents; Receptors, Histamine; Receptors, Histamine H3; Structure-Activity Relationship | 1990 |
New histamine H2-receptor antagonists.
Topics: Animals; Anticoagulants; Chemical Phenomena; Chemistry; Cimetidine; Confusion; Dogs; Drug Interactions; Duodenal Ulcer; Furans; Gastric Juice; Gastric Mucosa; Guanidines; Gynecomastia; Histamine H2 Antagonists; Humans; Imidazoles; Male; Molecular Conformation; Ranitidine; Spermatozoa; Thiazoles | 1980 |
[New generation of histamine H2 receptor blockaders].
Topics: Animals; Anti-Ulcer Agents; Cimetidine; Furans; Guanidines; Histamine H2 Antagonists; Humans; Imidazoles; Ranitidine; Thiazoles | 1982 |
30 other study(ies) available for tiotidine and ranitidine
Article | Year |
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Iodoaminopotentidine and related compounds: a new class of ligands with high affinity and selectivity for the histamine H2 receptor.
Topics: Aniline Compounds; Animals; Atrial Function; Azides; Guanidines; Guinea Pigs; Heart Atria; Heart Rate; Iodine Radioisotopes; Male; Muscle Contraction; Receptors, Histamine H2; Structure-Activity Relationship; Sulfonamides; Vasoconstriction | 1992 |
Development of a new physicochemical model for brain penetration and its application to the design of centrally acting H2 receptor histamine antagonists.
Topics: Algorithms; Animals; Blood-Brain Barrier; Brain; Chemical Phenomena; Chemistry, Physical; Clonidine; Guinea Pigs; Histamine H2 Antagonists; Imipramine; Pyrilamine; Structure-Activity Relationship | 1988 |
Predicting blood-brain barrier permeation from three-dimensional molecular structure.
Topics: Blood-Brain Barrier; Databases, Factual; Models, Chemical; Molecular Conformation; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship | 2000 |
ElogD(oct): a tool for lipophilicity determination in drug discovery. 2. Basic and neutral compounds.
Topics: 1-Octanol; Chromatography, High Pressure Liquid; Pharmaceutical Preparations; Solubility; Water | 2001 |
QSAR-based permeability model for drug-like compounds.
Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship | 2011 |
Heterologous expression of rat epitope-tagged histamine H2 receptors in insect Sf9 cells.
Topics: Adenylyl Cyclases; Animals; Baculoviridae; beta-Cyclodextrins; Blotting, Western; Cell Line, Transformed; Cholesterol; Cimetidine; Cyclic AMP; Cyclodextrins; Epitopes; Fluorescent Antibody Technique; Guanidines; Histamine H2 Antagonists; Histidine; Insecta; Microscopy, Confocal; Oligonucleotides; Piperidines; Ranitidine; Rats; Receptors, Histamine H2; Transfection | 1997 |
Evaluation of histamine H1-, H2-, and H3-receptor ligands at the human histamine H4 receptor: identification of 4-methylhistamine as the first potent and selective H4 receptor agonist.
Topics: Cell Line; Histamine Agonists; Humans; Imidazoles; Indoles; Isothiuronium; Ligands; Methylhistamines; Piperazines; Radioligand Assay; Receptors, G-Protein-Coupled; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Receptors, Histamine H3; Receptors, Histamine H4 | 2005 |
Theoretical studies on the histamine H2 receptor: molecular mechanism of action of antagonists.
Topics: Cimetidine; Computer Simulation; Guanidines; Histamine H1 Antagonists; Histamine H2 Antagonists; Kinetics; Models, Chemical; Molecular Conformation; Ranitidine; Receptors, Histamine H1; Structure-Activity Relationship | 1992 |
Characterization of an accessory binding area in the histamine H2 receptor.
Topics: Animals; Binding Sites; Cerebral Cortex; Cimetidine; Guinea Pigs; Heart Atria; Histamine H2 Antagonists; Ileum; Male; Piperidines; Ranitidine; Receptors, Histamine H2; Structure-Activity Relationship; Triazoles | 1991 |
Mechanism of action of H2-antagonists on histamine- or dimaprit-stimulated H2-receptors of spontaneously beating guinea-pig atrium.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Cimetidine; Dimaprit; Famotidine; Female; Guinea Pigs; Heart; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Radioligand Assay; Ranitidine; Receptors, Histamine H2; Thiourea | 1990 |
Differential effects of histamine receptor antagonists on human natural killer cell activity.
Topics: Cell Survival; Cimetidine; Cytotoxicity, Immunologic; Dose-Response Relationship, Drug; Histamine H1 Antagonists; Histamine H2 Antagonists; Interferons; Killer Cells, Natural; Leukocytes, Mononuclear; Ranitidine | 1987 |
Anti-acid secretion activity of drugs cimetidine, ranitidine, tiotidine D 15,144 in dogs fixed with gastric fistulae.
Topics: Animals; Cimetidine; Dogs; Female; Gastric Acid; Gastric Fistula; Histamine H2 Antagonists; Ranitidine; Time Factors | 1989 |
Identification of structural characteristics of some potential H2-receptor antagonists that determine the interaction with rat hepatic P-450.
Topics: Animals; Cimetidine; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Histamine H2 Antagonists; Male; Microsomes, Liver; Molecular Structure; NADP; Ranitidine; Rats; Rats, Inbred Strains; Structure-Activity Relationship | 1988 |
Characterization of histamine receptors mediating the stimulation of cyclic AMP accumulation in rabbit cerebral cortical slices.
Topics: Adenosine; Animals; Cerebral Cortex; Chlorpheniramine; Cimetidine; Cyclic AMP; Dose-Response Relationship, Drug; Drug Synergism; Imidazoles; Impromidine; Kinetics; Mathematics; Metiamide; Rabbits; Ranitidine; Receptors, Histamine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles | 1985 |
Antagonistic activity of tiotidine and ranitidine on guinea-pig and rabbit atria.
Topics: Animals; Cimetidine; Female; Guinea Pigs; Heart Rate; Histamine Antagonists; In Vitro Techniques; Kinetics; Male; Myocardial Contraction; Rabbits; Ranitidine | 1986 |
Inhibition of mono-oxygenase and oxidase activity of rat-hepatic cytochrome P-450 by H2-receptor blockers.
Topics: Animals; Cimetidine; Cytochrome P-450 Enzyme Inhibitors; Imidazoles; Male; Methylcholanthrene; Microsomes, Liver; Oxidoreductases; Phenobarbital; Ranitidine; Rats; Rats, Inbred Strains; Safrole | 1984 |
New drugs for peptic ulcer.
Topics: Benzamides; Benzodiazepinones; Cimetidine; Furans; Guanidines; Histamine H2 Antagonists; Humans; Morpholines; Parasympatholytics; Pepsin A; Peptic Ulcer; Piperazines; Pirenzepine; Prostaglandins E, Synthetic; Ranitidine; Thiazoles; Trimipramine | 1980 |
Effects of H2-receptor antagonists cimetidine, ranitidine, and ICI 125,211 on histamine-stimulated adenylate cyclase activity in guinea pig gastric mucosa.
Topics: Adenylyl Cyclases; Animals; Cimetidine; Furans; Gastric Mucosa; Guanidines; Guinea Pigs; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Kinetics; Ranitidine; Structure-Activity Relationship; Thiazoles | 1981 |
Inhibition of microsomal drug metabolism by histamine H2-receptor antagonists studied in vivo and in vitro in rodents.
Topics: Aminopyrine; Aminopyrine N-Demethylase; Animals; Breath Tests; Cimetidine; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Furans; Guanidines; Histamine H2 Antagonists; Male; Mice; Mice, Inbred ICR; Microsomes, Liver; Ranitidine; Rats; Rats, Inbred Strains; Thiazoles; Time Factors | 1982 |
Effect of some new Histamine H2-receptor antagonists on the guinea-pig papillary muscle.
Topics: Animals; Cimetidine; Furans; Guanidines; Guinea Pigs; Histamine Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Myocardial Contraction; Papillary Muscles; Ranitidine; Thiazoles | 1981 |
Interaction of histamine with gastric mucosal cells. Effect of histamine H2 antagonists on binding and biological response.
Topics: Animals; Cimetidine; Cyclic AMP; Furans; Gastric Mucosa; Guanidines; Guinea Pigs; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Ranitidine; Receptors, Histamine; Thiazoles | 1982 |
A comparison of some of the pharmacological properties of etintidine, a new histamine H2-receptor antagonist, with those of cimetidine, ranitidine and tiotidine.
Topics: Adrenergic beta-Antagonists; Animals; Cimetidine; Dogs; Female; Furans; Gastric Juice; Guanidines; Guinea Pigs; Heart Rate; Histamine H1 Antagonists; Histamine H2 Antagonists; Imidazoles; In Vitro Techniques; Male; Myocardial Contraction; Parasympatholytics; Ranitidine; Rats; Rats, Inbred Strains; Thiazoles; Uterine Contraction | 1983 |
The role of antagonists to acid secretion.
Topics: 16,16-Dimethylprostaglandin E2; Benzodiazepinones; Cimetidine; Furans; Gastric Acid; Gastrointestinal Diseases; Guanidines; Histamine H2 Antagonists; Humans; Pirenzepine; Proglumide; Ranitidine; Somatostatin; Thiazoles | 1982 |
Histamine H2 receptor antagonists. 1. Synthesis of N-cyano and N-carbamoyl amidine derivatives and their biological activities.
Topics: Amidines; Animals; Carbamates; Cimetidine; Dogs; Histamine; Histamine H2 Antagonists; Nitriles; Ranitidine; Structure-Activity Relationship | 1984 |
A species comparison of the histamine H2-receptor on mast cells and basophils.
Topics: Animals; Basophils; Cimetidine; Female; Furans; Guanidines; Guinea Pigs; Histamine H2 Antagonists; Histamine Release; Humans; In Vitro Techniques; Lung; Male; Mast Cells; Ranitidine; Rats; Receptors, Histamine; Receptors, Histamine H2; Species Specificity; Thiazoles | 1982 |
Pharmacological interactions between ranitidine, cimetidine, metiamide and tiotidine at histamine H2-receptor sites in guinea-pig atria.
Topics: Animals; Cimetidine; Dimaprit; Drug Interactions; Furans; Guanidines; Guinea Pigs; Heart; Heart Rate; Histamine; In Vitro Techniques; Metiamide; Ranitidine; Receptors, Histamine; Receptors, Histamine H2; Thiazoles; Thiourea | 1982 |
Action of ebrotidine, ranitidine and cimetidine on the specific binding to histamine H1- and H2-receptors.
Topics: Animals; Benzenesulfonates; Cell Membrane; Cerebellum; Cerebral Cortex; Cimetidine; Depression, Chemical; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Isotope Labeling; Male; Protein Binding; Pyrilamine; Ranitidine; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Tritium | 1997 |
Long-lasting binding of IT-066 to human histamine H2 receptor.
Topics: Animals; Anti-Ulcer Agents; CHO Cells; Cimetidine; Cricetinae; Cyclic AMP; Famotidine; Fixatives; Formaldehyde; Histamine H2 Antagonists; Piperidines; Polymers; Protein Binding; Pyridines; Ranitidine; Receptors, Histamine H2 | 2000 |
Distinct interaction of human and guinea pig histamine H2-receptor with guanidine-type agonists.
Topics: Alternative Splicing; Amino Acid Sequence; Animals; Binding Sites; Cell Membrane; Cells, Cultured; Cimetidine; GTP-Binding Protein alpha Subunits, Gs; Guanidine; Guanidines; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Histamine Agonists; Humans; Insecta; Models, Molecular; Molecular Sequence Data; Piperidines; Protein Conformation; Protein Isoforms; Ranitidine; Receptors, Histamine H2; Sequence Homology, Amino Acid; Species Specificity; Structure-Activity Relationship; Sulfur Radioisotopes; Tritium | 2001 |
Effects of cimetidine-like drugs on recombinant GABAA receptors.
Topics: Cell Line; Cimetidine; Dose-Response Relationship, Drug; Famotidine; Fibroblasts; Histamine H2 Antagonists; Humans; Patch-Clamp Techniques; Ranitidine; Receptors, GABA-A; Recombinant Proteins | 2004 |